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—— ethyl 2-[2-[[(2S)-2-(4-fluorophenyl)sulfonylpropanoyl]amino]-1,3-thiazol-4-yl]acetate —— C16H17FN2O5S2
ethyl 2-[2-[[(2S)-2-(4-fluorophenyl)sulfonylpropanoyl]amino]-1,3-thiazol-4-yl]acetate
—— ethyl 2-[2-[[(2R)-2-(4-fluorophenyl)sulfonylpropanoyl]amino]-1,3-thiazol-4-yl]acetate —— C16H17FN2O5S2
ethyl 2-[2-[[(2R)-2-(4-fluorophenyl)sulfonylpropanoyl]amino]-1,3-thiazol-4-yl]acetate
—— ethyl 5-[[(2S)-2-(4-methoxyphenyl)pyrrolidin-1-yl]methyl]-7-oxo-1H-pyrazolo[1,5-a]pyrimidine-3-carboxylate —— C21H24N4O4
ethyl 5-[[(2S)-2-(4-methoxyphenyl)pyrrolidin-1-yl]methyl]-7-oxo-1H-pyrazolo[1,5-a]pyrimidine-3-carboxylate
—— ethyl 6-[[(2R)-2-(3-methyl-1,2-oxazol-5-yl)pyrrolidin-1-yl]methyl]-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C16H22N4O4
ethyl 6-[[(2R)-2-(3-methyl-1,2-oxazol-5-yl)pyrrolidin-1-yl]methyl]-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— ethyl 4-[(2R)-1-(1,3-benzothiazol-2-ylamino)-1-oxopropan-2-yl]piperazine-1-carboxylate —— C17H22N4O3S
ethyl 4-[(2R)-1-(1,3-benzothiazol-2-ylamino)-1-oxopropan-2-yl]piperazine-1-carboxylate
—— (E)-3-(3-chloro-4,5-dimethoxyphenyl)-N-cyclopropyl-N-[(1-methylimidazol-2-yl)methyl]prop-2-enamide —— C19H22ClN3O3
(E)-3-(3-chloro-4,5-dimethoxyphenyl)-N-cyclopropyl-N-[(1-methylimidazol-2-yl)methyl]prop-2-enamide
—— (E)-N-[1-(2-amino-2-oxoethyl)pyrazol-4-yl]-3-[3-[(2-methyl-1,3-thiazol-4-yl)methoxy]phenyl]prop-2-enamide —— C19H19N5O3S
(E)-N-[1-(2-amino-2-oxoethyl)pyrazol-4-yl]-3-[3-[(2-methyl-1,3-thiazol-4-yl)methoxy]phenyl]prop-2-enamide
—— ethyl 2-[[2-[4-[(2S,4S,5R,6R)-4-[(4,5-dichloroimidazol-1-yl)methyl]-6-[4-(hydroxymethyl)phenyl]-5-methyl-1,3-dioxan-2-yl]phenyl]phenyl]methylcarbamoylamino]acetate —— C34H36Cl2N4O6
ethyl 2-[[2-[4-[(2S,4S,5R,6R)-4-[(4,5-dichloroimidazol-1-yl)methyl]-6-[4-(hydroxymethyl)phenyl]-5-methyl-1,3-dioxan-2-yl]phenyl]phenyl]methylcarbamoylamino]acetate
—— (E)-N-[(2R)-1-imidazol-1-ylpropan-2-yl]-3-(3-nitrophenyl)prop-2-enamide —— C15H16N4O3
(E)-N-[(2R)-1-imidazol-1-ylpropan-2-yl]-3-(3-nitrophenyl)prop-2-enamide
—— (E)-N-[1-(2-amino-2-oxoethyl)pyrazol-4-yl]-3-(5-chloro-2,3-dihydro-1,4-benzodioxin-7-yl)prop-2-enamide —— C16H15ClN4O4
(E)-N-[1-(2-amino-2-oxoethyl)pyrazol-4-yl]-3-(5-chloro-2,3-dihydro-1,4-benzodioxin-7-yl)prop-2-enamide
—— (E)-3-(3,5-dichlorophenyl)-N-[2-(5-methyl-1H-1,2,4-triazol-3-yl)phenyl]prop-2-enamide —— C18H14Cl2N4O
(E)-3-(3,5-dichlorophenyl)-N-[2-(5-methyl-1H-1,2,4-triazol-3-yl)phenyl]prop-2-enamide
—— (E)-N-cyclopropyl-3-(2,6-dichlorophenyl)-N-[(1-methylimidazol-2-yl)methyl]prop-2-enamide —— C17H17Cl2N3O
(E)-N-cyclopropyl-3-(2,6-dichlorophenyl)-N-[(1-methylimidazol-2-yl)methyl]prop-2-enamide
—— (E)-3-(2,3-dichlorophenyl)-1-[4-[(3,5-dimethyl-1,2-oxazol-4-yl)methyl]piperazin-1-yl]prop-2-en-1-one —— C19H21Cl2N3O2
(E)-3-(2,3-dichlorophenyl)-1-[4-[(3,5-dimethyl-1,2-oxazol-4-yl)methyl]piperazin-1-yl]prop-2-en-1-one
—— (E)-3-(3-chloro-4-ethoxy-5-methoxyphenyl)-N-(6-methylsulfonylpyridin-3-yl)prop-2-enamide —— C18H19ClN2O5S
(E)-3-(3-chloro-4-ethoxy-5-methoxyphenyl)-N-(6-methylsulfonylpyridin-3-yl)prop-2-enamide
—— ethyl (Z)-3-[4-[[1-(2,2,2-trifluoroethyl)piperidine-4-carbonyl]amino]phenyl]prop-2-enoate —— C19H23F3N2O3
ethyl (Z)-3-[4-[[1-(2,2,2-trifluoroethyl)piperidine-4-carbonyl]amino]phenyl]prop-2-enoate
—— ethyl (3S)-1-(4-methyl-2-pyrimidin-2-yl-1,3-thiazole-5-carbonyl)piperidine-3-carboxylate —— C17H20N4O3S
ethyl (3S)-1-(4-methyl-2-pyrimidin-2-yl-1,3-thiazole-5-carbonyl)piperidine-3-carboxylate
—— (E)-N-[2,4-bis(difluoromethoxy)phenyl]-3-(3,5-dimethoxyphenyl)prop-2-enamide —— C19H17F4NO5
(E)-N-[2,4-bis(difluoromethoxy)phenyl]-3-(3,5-dimethoxyphenyl)prop-2-enamide
—— (E)-N-(6-methylsulfonylpyridin-3-yl)-3-(2,4,5-trimethoxyphenyl)prop-2-enamide —— C18H20N2O6S
(E)-N-(6-methylsulfonylpyridin-3-yl)-3-(2,4,5-trimethoxyphenyl)prop-2-enamide
—— (E)-3-(1,3-diphenylpyrazol-4-yl)-N-[2-(ethylamino)-2-oxoethyl]-N-methylprop-2-enamide —— C23H24N4O2
(E)-3-(1,3-diphenylpyrazol-4-yl)-N-[2-(ethylamino)-2-oxoethyl]-N-methylprop-2-enamide
—— (E)-3-(5-bromo-2-methoxyphenyl)-N-[3-(1,2,4-triazol-1-ylmethyl)phenyl]prop-2-enamide —— C19H17BrN4O2
(E)-3-(5-bromo-2-methoxyphenyl)-N-[3-(1,2,4-triazol-1-ylmethyl)phenyl]prop-2-enamide
—— ethyl N-[(2R)-1-[(3R)-3-[(5-chloropyridin-2-yl)carbamoyl]piperidin-1-yl]-3-methyl-1-oxobutan-2-yl]carbamate —— C19H27ClN4O4
ethyl N-[(2R)-1-[(3R)-3-[(5-chloropyridin-2-yl)carbamoyl]piperidin-1-yl]-3-methyl-1-oxobutan-2-yl]carbamate
—— (E)-3-[2-(difluoromethoxy)phenyl]-1-[4-[(3,5-dimethyl-1,2-oxazol-4-yl)methyl]piperazin-1-yl]prop-2-en-1-one —— C20H23F2N3O3
(E)-3-[2-(difluoromethoxy)phenyl]-1-[4-[(3,5-dimethyl-1,2-oxazol-4-yl)methyl]piperazin-1-yl]prop-2-en-1-one
—— (E)-3-(1,3-benzoxazol-2-yl)-N-[[4-[(4-ethylpiperazin-1-yl)methyl]phenyl]methyl]prop-2-enamide —— C24H28N4O2
(E)-3-(1,3-benzoxazol-2-yl)-N-[[4-[(4-ethylpiperazin-1-yl)methyl]phenyl]methyl]prop-2-enamide
—— ethyl 4-[[2-(2-pyrimidin-2-yl-1,3-thiazol-4-yl)acetyl]amino]piperidine-1-carboxylate —— C17H21N5O3S
ethyl 4-[[2-(2-pyrimidin-2-yl-1,3-thiazol-4-yl)acetyl]amino]piperidine-1-carboxylate
—— (E)-3-[4-(cyanomethoxy)-3-methoxyphenyl]-N-cyclopropyl-N-[(1-methylimidazol-2-yl)methyl]prop-2-enamide —— C20H22N4O3
(E)-3-[4-(cyanomethoxy)-3-methoxyphenyl]-N-cyclopropyl-N-[(1-methylimidazol-2-yl)methyl]prop-2-enamide
—— (E)-N-[2-(ethylamino)-2-oxoethyl]-N-methyl-3-(1-phenyl-3-pyridin-3-ylpyrazol-4-yl)prop-2-enamide —— C22H23N5O2
(E)-N-[2-(ethylamino)-2-oxoethyl]-N-methyl-3-(1-phenyl-3-pyridin-3-ylpyrazol-4-yl)prop-2-enamide
—— (E)-N-cyclopropyl-3-(2,3-dichlorophenyl)-N-[(1-methylimidazol-2-yl)methyl]prop-2-enamide —— C17H17Cl2N3O
(E)-N-cyclopropyl-3-(2,3-dichlorophenyl)-N-[(1-methylimidazol-2-yl)methyl]prop-2-enamide
—— (E)-3-[4-(methylsulfamoyl)phenyl]-N-[[3-(2-oxo-1,3-oxazolidin-3-yl)phenyl]methyl]prop-2-enamide —— C20H21N3O5S
(E)-3-[4-(methylsulfamoyl)phenyl]-N-[[3-(2-oxo-1,3-oxazolidin-3-yl)phenyl]methyl]prop-2-enamide
—— (E)-N-[(1R)-2-anilino-2-oxo-1-phenylethyl]-3-(4-methoxyphenyl)prop-2-enamide —— C24H22N2O3
(E)-N-[(1R)-2-anilino-2-oxo-1-phenylethyl]-3-(4-methoxyphenyl)prop-2-enamide
—— (E)-N-[2-(dimethylamino)ethyl]-3-(3-nitrophenyl)-N-(2-phenylethyl)prop-2-enamide —— C21H25N3O3
(E)-N-[2-(dimethylamino)ethyl]-3-(3-nitrophenyl)-N-(2-phenylethyl)prop-2-enamide
—— ethyl 2-[[2-[4-[(2S,4R,5R,6S)-4-[4-(hydroxymethyl)phenyl]-5-methyl-6-[(4-methyl-1,2,4-triazol-3-yl)sulfanylmethyl]-1,3-dioxan-2-yl]phenyl]phenyl]methylcarbamoylamino]acetate —— C34H39N5O6S
ethyl 2-[[2-[4-[(2S,4R,5R,6S)-4-[4-(hydroxymethyl)phenyl]-5-methyl-6-[(4-methyl-1,2,4-triazol-3-yl)sulfanylmethyl]-1,3-dioxan-2-yl]phenyl]phenyl]methylcarbamoylamino]acetate
—— (E)-3-(4-chlorophenyl)-N-[[3-(morpholin-4-ylmethyl)phenyl]methyl]prop-2-enamide —— C21H23ClN2O2
(E)-3-(4-chlorophenyl)-N-[[3-(morpholin-4-ylmethyl)phenyl]methyl]prop-2-enamide
—— ethyl 4-[(Z)-3-[[1-(2-amino-2-oxoethyl)pyrazol-4-yl]amino]-3-oxoprop-1-enyl]-1-ethyl-2,5-dimethylpyrrole-3-carboxylate —— C19H25N5O4
ethyl 4-[(Z)-3-[[1-(2-amino-2-oxoethyl)pyrazol-4-yl]amino]-3-oxoprop-1-enyl]-1-ethyl-2,5-dimethylpyrrole-3-carboxylate
—— (E)-3-[4-(2-amino-2-oxoethoxy)-3-methoxyphenyl]-N-[3-[ethylsulfonyl(methyl)amino]propyl]prop-2-enamide —— C18H27N3O6S
(E)-3-[4-(2-amino-2-oxoethoxy)-3-methoxyphenyl]-N-[3-[ethylsulfonyl(methyl)amino]propyl]prop-2-enamide
—— (E)-N-[(1S,8aR)-1,2,3,5,6,7,8,8a-octahydroindolizin-1-yl]-3-(3-nitrophenyl)prop-2-enamide —— C17H21N3O3
(E)-N-[(1S,8aR)-1,2,3,5,6,7,8,8a-octahydroindolizin-1-yl]-3-(3-nitrophenyl)prop-2-enamide
—— (E)-3-(5-bromo-2-fluorophenyl)-N-[3-(1,2,4-triazol-1-ylmethyl)phenyl]prop-2-enamide —— C18H14BrFN4O
(E)-3-(5-bromo-2-fluorophenyl)-N-[3-(1,2,4-triazol-1-ylmethyl)phenyl]prop-2-enamide
—— (E)-3-[4-(methanesulfonamido)phenyl]-N-[(2S)-1-morpholin-4-ylpropan-2-yl]prop-2-enamide —— C17H25N3O4S
(E)-3-[4-(methanesulfonamido)phenyl]-N-[(2S)-1-morpholin-4-ylpropan-2-yl]prop-2-enamide
—— ethyl 3-[4-[(3S)-3-methylpiperidin-1-yl]butylcarbamoyl]-5-nitrobenzoate —— C20H29N3O5
ethyl 3-[4-[(3S)-3-methylpiperidin-1-yl]butylcarbamoyl]-5-nitrobenzoate
—— ethyl N-[(2R)-1-[(1-benzylpyrazol-4-yl)methylamino]-3-methyl-1-oxobutan-2-yl]carbamate —— C19H26N4O3
ethyl N-[(2R)-1-[(1-benzylpyrazol-4-yl)methylamino]-3-methyl-1-oxobutan-2-yl]carbamate
—— (E)-3-[4-(cyanomethoxy)-3-methoxyphenyl]-N-[2-fluoro-5-(tetrazol-1-yl)phenyl]prop-2-enamide —— C19H15FN6O3
(E)-3-[4-(cyanomethoxy)-3-methoxyphenyl]-N-[2-fluoro-5-(tetrazol-1-yl)phenyl]prop-2-enamide
—— (E)-3-(2-ethoxyphenyl)-N-[2-fluoro-5-(tetrazol-1-yl)phenyl]prop-2-enamide —— C18H16FN5O2
(E)-3-(2-ethoxyphenyl)-N-[2-fluoro-5-(tetrazol-1-yl)phenyl]prop-2-enamide
—— (E)-N-cyclopropyl-3-[4-(difluoromethoxy)phenyl]-N-[(1R)-1-pyridin-2-ylethyl]prop-2-enamide —— C20H20F2N2O2
(E)-N-cyclopropyl-3-[4-(difluoromethoxy)phenyl]-N-[(1R)-1-pyridin-2-ylethyl]prop-2-enamide
—— (E)-3-(5-methoxy-2,3-dihydro-1,4-benzodioxin-7-yl)-N-[2-oxo-2-(2,2,2-trifluoroethylamino)ethyl]prop-2-enamide —— C16H17F3N2O5
(E)-3-(5-methoxy-2,3-dihydro-1,4-benzodioxin-7-yl)-N-[2-oxo-2-(2,2,2-trifluoroethylamino)ethyl]prop-2-enamide
—— (E)-3-(7-chloroquinolin-2-yl)-N-[(3S)-2-oxoazepan-3-yl]prop-2-enamide —— C18H18ClN3O2
(E)-3-(7-chloroquinolin-2-yl)-N-[(3S)-2-oxoazepan-3-yl]prop-2-enamide
—— (E)-N-[(1S,2R)-1-(1H-benzimidazol-2-yl)-2-methylbutyl]-3-(1-benzyltriazol-4-yl)prop-2-enamide —— C24H26N6O
(E)-N-[(1S,2R)-1-(1H-benzimidazol-2-yl)-2-methylbutyl]-3-(1-benzyltriazol-4-yl)prop-2-enamide
—— (E)-3-(3,5-dimethyl-1-phenylpyrazol-4-yl)-N-[(3R)-2-oxoazepan-3-yl]prop-2-enamide —— C20H24N4O2
(E)-3-(3,5-dimethyl-1-phenylpyrazol-4-yl)-N-[(3R)-2-oxoazepan-3-yl]prop-2-enamide
—— (E)-3-[3-[(2-methyl-1,3-thiazol-4-yl)methoxy]phenyl]-N-[(3S)-2-oxoazepan-3-yl]prop-2-enamide —— C20H23N3O3S
(E)-3-[3-[(2-methyl-1,3-thiazol-4-yl)methoxy]phenyl]-N-[(3S)-2-oxoazepan-3-yl]prop-2-enamide
—— (E)-N-[(3S)-2-oxoazepan-3-yl]-3-(1-phenyl-3-thiophen-2-ylpyrazol-4-yl)prop-2-enamide —— C22H22N4O2S
(E)-N-[(3S)-2-oxoazepan-3-yl]-3-(1-phenyl-3-thiophen-2-ylpyrazol-4-yl)prop-2-enamide
—— ethyl 4-[(Z)-3-(4-cyanophenyl)-3-oxoprop-1-enyl]-1-phenylpyrazole-3-carboxylate —— C22H17N3O3
ethyl 4-[(Z)-3-(4-cyanophenyl)-3-oxoprop-1-enyl]-1-phenylpyrazole-3-carboxylate
—— ethyl 4-[(E)-2-cyano-3-oxo-3-(propan-2-ylamino)prop-1-enyl]-1-phenylpyrazole-3-carboxylate —— C19H20N4O3
ethyl 4-[(E)-2-cyano-3-oxo-3-(propan-2-ylamino)prop-1-enyl]-1-phenylpyrazole-3-carboxylate