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中文名称 英文名称 CAS号 化学式 结构式图片
—— (E)-3-(3,4-dihydroxyphenyl)-N-[5-(o-tolylsulfamoyl)-1-naphthyl]prop-2-enamide —— C26H22N2O5S
(E)-3-(3,4-dihydroxyphenyl)-N-[5-(o-tolylsulfamoyl)-1-naphthyl]prop-2-enamide
—— (E)-N-(5-{[3-(1H-imidazol-1-yl)propyl]amino}-1,3,4-thiadiazol-2-yl)-3-phenyl-2-propenamide —— C17H18N6OS
(E)-N-(5-{[3-(1H-imidazol-1-yl)propyl]amino}-1,3,4-thiadiazol-2-yl)-3-phenyl-2-propenamide
—— (E)-5-(1,3-dichloro-6,12-dioxo-indolo[2,1-b]quinazolin-8-yl)-2-(9H-fluoren-9-ylmethoxycarbonylamino)pent-4-enoic acid —— C35H23Cl2N3O6
(E)-5-(1,3-dichloro-6,12-dioxo-indolo[2,1-b]quinazolin-8-yl)-2-(9H-fluoren-9-ylmethoxycarbonylamino)pent-4-enoic acid
—— (E)-3-(3,4-dihydroxyphenyl)-N-[5-(p-tolylsulfamoyl)-1-naphthyl]prop-2-enamide —— C26H22N2O5S
(E)-3-(3,4-dihydroxyphenyl)-N-[5-(p-tolylsulfamoyl)-1-naphthyl]prop-2-enamide
—— (E)-3-(3,4-dihydroxyphenyl)-N-[5-(phenylsulfamoyl)-1-naphthyl]prop-2-enamide —— C25H20N2O5S
(E)-3-(3,4-dihydroxyphenyl)-N-[5-(phenylsulfamoyl)-1-naphthyl]prop-2-enamide
—— (E)-N-{5-[(4-fluorobenzyl)amino]-1,3,4-thiadiazol-2-yl}-9-octadecenamide —— C27H41FN4OS
(E)-N-{5-[(4-fluorobenzyl)amino]-1,3,4-thiadiazol-2-yl}-9-octadecenamide
—— (E)-3-(2-chlorophenyl)-N-{5-[(4-fluorobenzyl)amino]-1,3,4-thiadiazol-2-yl}-2-propenamide —— C18H14ClFN4OS
(E)-3-(2-chlorophenyl)-N-{5-[(4-fluorobenzyl)amino]-1,3,4-thiadiazol-2-yl}-2-propenamide
—— (E)-(S)-4-((S)-2-{3-[(5-Methyl-isoxazole-3-carbonyl)-amino]-2-oxo-2H-pyridin-1-yl}-butyrylamino)-5-((S)-2-oxo-pyrrolidin-3-yl)-pent-2-enoic acid isopropyl ester —— C26H33N5O7
(E)-(S)-4-((S)-2-{3-[(5-Methyl-isoxazole-3-carbonyl)-amino]-2-oxo-2H-pyridin-1-yl}-butyrylamino)-5-((S)-2-oxo-pyrrolidin-3-yl)-pent-2-enoic acid isopropyl ester
—— (E)-(S)-6-Carbamoyl-4-[(2R,5S)-5-cyclopentylsulfanylcarbonylamino-6-methyl-2-(4-methyl-benzyl)-4-oxo-heptanoylamino]-hex-2-enoic acid ethyl ester —— C31H45N3O6S
(E)-(S)-6-Carbamoyl-4-[(2R,5S)-5-cyclopentylsulfanylcarbonylamino-6-methyl-2-(4-methyl-benzyl)-4-oxo-heptanoylamino]-hex-2-enoic acid ethyl ester
—— (E)-2-(2-hydroxyphenyl)sulfanyl-3-phenyl-prop-2-enenitrile —— C15H11NOS
(E)-2-(2-hydroxyphenyl)sulfanyl-3-phenyl-prop-2-enenitrile
—— ethyl (E,4S)-7-amino-4-[[(2R,5S)-5-(cyclopentylsulfanylcarbonylamino)-2-[(4-fluorophenyl)methyl]-4-oxo-6-phenyl-hexanoyl]amino]-7-oxo-hept-2-enoate —— C34H42FN3O6S
ethyl (E,4S)-7-amino-4-[[(2R,5S)-5-(cyclopentylsulfanylcarbonylamino)-2-[(4-fluorophenyl)methyl]-4-oxo-6-phenyl-hexanoyl]amino]-7-oxo-hept-2-enoate
—— (E)-N-{5-[(1,3-benzodioxol-5-ylmethyl)amino]-1,3,4-thiadiazol-2-yl}-3-(2-chlorophenyl)-2-propenamide —— C19H15ClN4O3S
(E)-N-{5-[(1,3-benzodioxol-5-ylmethyl)amino]-1,3,4-thiadiazol-2-yl}-3-(2-chlorophenyl)-2-propenamide
—— (E)-(S)-4-((S)-2-Benzyloxycarbonylamino-3-phenyl-propionylamino)-6-carbamoyl-hex-2-enoic acid ethyl ester —— C26H31N3O6
(E)-(S)-4-((S)-2-Benzyloxycarbonylamino-3-phenyl-propionylamino)-6-carbamoyl-hex-2-enoic acid ethyl ester
—— [(E)-6-(8-chloro-6,12-dioxo-indolo[2,1-b]quinazolin-2-yl)hex-5-enyl] acetate —— C23H19ClN2O4
[(E)-6-(8-chloro-6,12-dioxo-indolo[2,1-b]quinazolin-2-yl)hex-5-enyl] acetate
—— (E)-N-[(S)-1-(5-Methyl-4-oxo-4H-thieno[2,3-d][1,3]oxazin-2-yl)-ethyl]-3-(5-nitro-thiophen-2-yl)-acrylamide —— C16H13N3O5S2
(E)-N-[(S)-1-(5-Methyl-4-oxo-4H-thieno[2,3-d][1,3]oxazin-2-yl)-ethyl]-3-(5-nitro-thiophen-2-yl)-acrylamide
—— (E)-3-(3,4-dihydroxyphenyl)-N-[5-[(4-fluorophenyl)sulfamoyl]-1-naphthyl]prop-2-enamide —— C25H19FN2O5S
(E)-3-(3,4-dihydroxyphenyl)-N-[5-[(4-fluorophenyl)sulfamoyl]-1-naphthyl]prop-2-enamide
—— (E)-(S)-4-((2R,5S)-2-Benzyl-5-cyclopentylsulfanylcarbonylamino-7-methyl-4-oxo-octanoylamino)-6-carbamoyl-hex-2-enoic acid ethyl ester —— C31H45N3O6S
(E)-(S)-4-((2R,5S)-2-Benzyl-5-cyclopentylsulfanylcarbonylamino-7-methyl-4-oxo-octanoylamino)-6-carbamoyl-hex-2-enoic acid ethyl ester
—— [(E)-5-(5-amino-7-oxo-6H-imidazo[4,5-b]pyridin-3-yl)-3-(hydroxymethyl)pent-1-enyl]phosphonic acid —— C12H17N4O5P
[(E)-5-(5-amino-7-oxo-6H-imidazo[4,5-b]pyridin-3-yl)-3-(hydroxymethyl)pent-1-enyl]phosphonic acid
—— (E)-3-(2-Chloro-4-hydroxy-phenyl)-N-[(S)-1-(5-methyl-4-oxo-4H-thieno[2,3-d][1,3]oxazin-2-yl)-ethyl]-acrylamide —— C18H15ClN2O4S
(E)-3-(2-Chloro-4-hydroxy-phenyl)-N-[(S)-1-(5-methyl-4-oxo-4H-thieno[2,3-d][1,3]oxazin-2-yl)-ethyl]-acrylamide
—— (E)-(R)-4-[(S)-2-((S)-2-Benzyloxycarbonylamino-4-methyl-pentanoylamino)-3-phenyl-propionylamino]-5-(2-oxo-imidazolidin-1-yl)-pent-2-enoic acid ethyl ester —— C33H43N5O7
(E)-(R)-4-[(S)-2-((S)-2-Benzyloxycarbonylamino-4-methyl-pentanoylamino)-3-phenyl-propionylamino]-5-(2-oxo-imidazolidin-1-yl)-pent-2-enoic acid ethyl ester
—— (E)-3-{3-[2-((S)-4,4-Difluoro-2-{[(2S,4S)-1-((S)-2-isobutoxycarbonylamino-3-methyl-butyryl)-4-phenyl-pyrrolidine-2-carbonyl]-amino}-butyrylamino)-ethyl]-phenyl}-acrylic acid ethyl ester —— C38H50F2N4O7
(E)-3-{3-[2-((S)-4,4-Difluoro-2-{[(2S,4S)-1-((S)-2-isobutoxycarbonylamino-3-methyl-butyryl)-4-phenyl-pyrrolidine-2-carbonyl]-amino}-butyrylamino)-ethyl]-phenyl}-acrylic acid ethyl ester
—— (E)-N-[5-(benzylsulfamoyl)-1-naphthyl]-3-(3,4-dihydroxyphenyl)prop-2-enamide —— C26H22N2O5S
(E)-N-[5-(benzylsulfamoyl)-1-naphthyl]-3-(3,4-dihydroxyphenyl)prop-2-enamide
—— (E)-N-[(S)-1-(5-Methyl-4-oxo-4H-thieno[2,3-d][1,3]oxazin-2-yl)-ethyl]-3-(1-methyl-1H-pyrrol-2-yl)-acrylamide —— C17H17N3O3S
(E)-N-[(S)-1-(5-Methyl-4-oxo-4H-thieno[2,3-d][1,3]oxazin-2-yl)-ethyl]-3-(1-methyl-1H-pyrrol-2-yl)-acrylamide
—— (E)-3-[3,4-bis[(4-fluorophenyl)methoxy]phenyl]-N-[2-oxo-2-[2-(6-thioxocyclohexa-1,3-dien-1-yl)ethylamino]ethyl]prop-2-enamide —— C33H30F2N2O4S
(E)-3-[3,4-bis[(4-fluorophenyl)methoxy]phenyl]-N-[2-oxo-2-[2-(6-thioxocyclohexa-1,3-dien-1-yl)ethylamino]ethyl]prop-2-enamide
—— ethyl (E,4S)-7-amino-4-[[(2S)-2-[[(2S)-2-(benzyloxycarbonylamino)-4-methyl-pentanoyl]amino]-3-(4-cyanophenyl)propanoyl]amino]-7-oxo-hept-2-enoate —— C33H41N5O7
ethyl (E,4S)-7-amino-4-[[(2S)-2-[[(2S)-2-(benzyloxycarbonylamino)-4-methyl-pentanoyl]amino]-3-(4-cyanophenyl)propanoyl]amino]-7-oxo-hept-2-enoate
—— ethyl (E,4S)-4-[[(2S)-2-[[(2S)-2-[[(2S)-2-acetamidopropanoyl]amino]-4-methyl-pentanoyl]amino]-3-phenyl-propanoyl]amino]-7-amino-7-oxo-hept-2-enoate —— C29H43N5O7
ethyl (E,4S)-4-[[(2S)-2-[[(2S)-2-[[(2S)-2-acetamidopropanoyl]amino]-4-methyl-pentanoyl]amino]-3-phenyl-propanoyl]amino]-7-amino-7-oxo-hept-2-enoate
—— (E)-(S)-6-Carbamoyl-4-[(S)-2-((S)-4-methyl-2-methylsulfanylcarbonylamino-pentanoylamino)-3-phenyl-propionylamino]-hex-2-enoic acid ethyl ester —— C26H38N4O6S
(E)-(S)-6-Carbamoyl-4-[(S)-2-((S)-4-methyl-2-methylsulfanylcarbonylamino-pentanoylamino)-3-phenyl-propionylamino]-hex-2-enoic acid ethyl ester
—— (E)-4-oxo-4-[(3R)-3-(1H-pyrazol-5-yl)piperidin-1-yl]but-2-enoic acid —— C12H15N3O3
(E)-4-oxo-4-[(3R)-3-(1H-pyrazol-5-yl)piperidin-1-yl]but-2-enoic acid
—— (E)-(S)-4-[(S)-2-((S)-2-Acetylamino-4-methyl-pentanoylamino)-3-phenyl-propionylamino]-6-carbamoyl-hex-2-enoic acid ethyl ester —— C26H38N4O6
(E)-(S)-4-[(S)-2-((S)-2-Acetylamino-4-methyl-pentanoylamino)-3-phenyl-propionylamino]-6-carbamoyl-hex-2-enoic acid ethyl ester
—— ethyl (E,4S)-7-amino-4-[[(2S)-2-[[(2S)-2-(benzyloxycarbonylamino)-4-methyl-pentanoyl]amino]-3-(4-carbamoylphenyl)propanoyl]amino]-7-oxo-hept-2-enoate —— C33H43N5O8
ethyl (E,4S)-7-amino-4-[[(2S)-2-[[(2S)-2-(benzyloxycarbonylamino)-4-methyl-pentanoyl]amino]-3-(4-carbamoylphenyl)propanoyl]amino]-7-oxo-hept-2-enoate
—— (E)-(R)-4-[(S)-2-((S)-2-Benzyloxycarbonylamino-4-methyl-pentanoylamino)-3-phenyl-propionylamino]-5-ureido-pent-2-enoic acid ethyl ester —— C31H41N5O7
(E)-(R)-4-[(S)-2-((S)-2-Benzyloxycarbonylamino-4-methyl-pentanoylamino)-3-phenyl-propionylamino]-5-ureido-pent-2-enoic acid ethyl ester
—— (E)-3-(3-Bromo-thiophen-2-yl)-N-[(S)-1-(5-methyl-4-oxo-4H-thieno[2,3-d][1,3]oxazin-2-yl)-ethyl]-acrylamide —— C16H13BrN2O3S2
(E)-3-(3-Bromo-thiophen-2-yl)-N-[(S)-1-(5-methyl-4-oxo-4H-thieno[2,3-d][1,3]oxazin-2-yl)-ethyl]-acrylamide
—— ethyl (E,4S)-7-amino-4-[[(2S)-2-[[(2S)-2-(benzyloxycarbonylamino)-4-methyl-pentanoyl]amino]pentanoyl]amino]-7-oxo-hept-2-enoate —— C28H42N4O7
ethyl (E,4S)-7-amino-4-[[(2S)-2-[[(2S)-2-(benzyloxycarbonylamino)-4-methyl-pentanoyl]amino]pentanoyl]amino]-7-oxo-hept-2-enoate
—— (E)-4-[(2R,5S)-5-carbamoyl-2-methylpiperidin-1-yl]-4-oxobut-2-enoic acid —— C11H16N2O4
(E)-4-[(2R,5S)-5-carbamoyl-2-methylpiperidin-1-yl]-4-oxobut-2-enoic acid
—— ethyl (E,4S)-4-[[(2S)-2-[[(2S)-2-[[(2S)-2-acetamido-3-methyl-butanoyl]amino]-4-methyl-pentanoyl]amino]-3-phenyl-propanoyl]amino]-7-amino-7-oxo-hept-2-enoate —— C31H47N5O7
ethyl (E,4S)-4-[[(2S)-2-[[(2S)-2-[[(2S)-2-acetamido-3-methyl-butanoyl]amino]-4-methyl-pentanoyl]amino]-3-phenyl-propanoyl]amino]-7-amino-7-oxo-hept-2-enoate
—— (E)-(S)-4-[(S)-2-((S)-2-Benzyloxycarbonylamino-4-carboxy-butyrylamino)-3-phenyl-propionylamino]-6-carbamoyl-hex-2-enoic acid ethyl ester —— C31H38N4O9
(E)-(S)-4-[(S)-2-((S)-2-Benzyloxycarbonylamino-4-carboxy-butyrylamino)-3-phenyl-propionylamino]-6-carbamoyl-hex-2-enoic acid ethyl ester
—— (E)-(S)-4-[(S)-2-((S)-2-Benzyloxycarbonylamino-4-phenyl-butyrylamino)-3-phenyl-propionylamino]-6-carbamoyl-hex-2-enoic acid ethyl ester —— C36H42N4O7
(E)-(S)-4-[(S)-2-((S)-2-Benzyloxycarbonylamino-4-phenyl-butyrylamino)-3-phenyl-propionylamino]-6-carbamoyl-hex-2-enoic acid ethyl ester
—— (E)-(S)-6-Carbamoyl-4-{(S)-2-[(S)-2-(2-chloro-benzyloxycarbonylamino)-4-methyl-pentanoylamino]-3-phenyl-propionylamino}-hex-2-enoic acid ethyl ester —— C32H41ClN4O7
(E)-(S)-6-Carbamoyl-4-{(S)-2-[(S)-2-(2-chloro-benzyloxycarbonylamino)-4-methyl-pentanoylamino]-3-phenyl-propionylamino}-hex-2-enoic acid ethyl ester
—— (E)-(S)-6-Carbamoyl-4-{(S)-2-[(S)-2-(2-hydroxy-acetylamino)-4-methyl-pentanoylamino]-3-phenyl-propionylamino}-hex-2-enoic acid ethyl ester —— C26H38N4O7
(E)-(S)-6-Carbamoyl-4-{(S)-2-[(S)-2-(2-hydroxy-acetylamino)-4-methyl-pentanoylamino]-3-phenyl-propionylamino}-hex-2-enoic acid ethyl ester
—— (E)-3-(5-bromo-2-furyl)-N-[(1S)-1-(5-methyl-4-oxo-thieno[2,3-d][1,3]oxazin-2-yl)ethyl]prop-2-enamide —— C16H13BrN2O4S
(E)-3-(5-bromo-2-furyl)-N-[(1S)-1-(5-methyl-4-oxo-thieno[2,3-d][1,3]oxazin-2-yl)ethyl]prop-2-enamide
—— (E)-(S)-4-[(S)-2-((S)-2-Benzyloxycarbonylamino-4-methyl-pentanoylamino)-3-thiophen-2-yl-propionylamino]-6-carbamoyl-hex-2-enoic acid ethyl ester —— C30H40N4O7S
(E)-(S)-4-[(S)-2-((S)-2-Benzyloxycarbonylamino-4-methyl-pentanoylamino)-3-thiophen-2-yl-propionylamino]-6-carbamoyl-hex-2-enoic acid ethyl ester
—— ethyl (E,4S)-7-amino-4-[[(2S)-2-[[(2S)-2-(benzyloxycarbonylamino)-4-methyl-pentanoyl]amino]-3-cyclohexyl-propanoyl]amino]-7-oxo-hept-2-enoate —— C32H48N4O7
ethyl (E,4S)-7-amino-4-[[(2S)-2-[[(2S)-2-(benzyloxycarbonylamino)-4-methyl-pentanoyl]amino]-3-cyclohexyl-propanoyl]amino]-7-oxo-hept-2-enoate
—— (E)-(S)-4-[(S)-2-((S)-2-Benzyloxycarbonylamino-4-methyl-pentanoylamino)-3-phenyl-propionylamino]-6-methylcarbamoyl-hex-2-enoic acid ethyl ester —— C33H44N4O7
(E)-(S)-4-[(S)-2-((S)-2-Benzyloxycarbonylamino-4-methyl-pentanoylamino)-3-phenyl-propionylamino]-6-methylcarbamoyl-hex-2-enoic acid ethyl ester
—— (E)-4-oxo-4-[(3S)-3-pyrrolidin-1-ylpiperidin-1-yl]but-2-enoic acid —— C13H20N2O3
(E)-4-oxo-4-[(3S)-3-pyrrolidin-1-ylpiperidin-1-yl]but-2-enoic acid
—— (E)-(S)-4-[(S)-2-((S)-2-Benzyloxycarbonylamino-3-hydroxy-3-methyl-butyrylamino)-3-phenyl-propionylamino]-6-carbamoyl-hex-2-enoic acid ethyl ester —— C31H40N4O8
(E)-(S)-4-[(S)-2-((S)-2-Benzyloxycarbonylamino-3-hydroxy-3-methyl-butyrylamino)-3-phenyl-propionylamino]-6-carbamoyl-hex-2-enoic acid ethyl ester
—— (E)-(S)-4-[(S)-2-((R)-2-Benzyloxycarbonylamino-3-methylsulfanyl-propionylamino)-3-phenyl-propionylamino]-6-carbamoyl-hex-2-enoic acid ethyl ester —— C30H38N4O7S
(E)-(S)-4-[(S)-2-((R)-2-Benzyloxycarbonylamino-3-methylsulfanyl-propionylamino)-3-phenyl-propionylamino]-6-carbamoyl-hex-2-enoic acid ethyl ester
—— (E)-(S)-4-[(S)-2-((S)-2-Benzyloxycarbonylamino-4-methyl-pentanoylamino)-3-phenyl-propionylamino]-6-methanesulfinyl-hex-2-enoic acid ethyl ester —— C32H43N3O7S
(E)-(S)-4-[(S)-2-((S)-2-Benzyloxycarbonylamino-4-methyl-pentanoylamino)-3-phenyl-propionylamino]-6-methanesulfinyl-hex-2-enoic acid ethyl ester
—— ethyl (E,4S)-7-amino-4-[[(2S)-2-[[(2S)-2-(tert-butoxycarbonylamino)-4-methyl-pentanoyl]amino]-3-phenyl-propanoyl]amino]-7-oxo-hept-2-enoate —— C29H44N4O7
ethyl (E,4S)-7-amino-4-[[(2S)-2-[[(2S)-2-(tert-butoxycarbonylamino)-4-methyl-pentanoyl]amino]-3-phenyl-propanoyl]amino]-7-oxo-hept-2-enoate
—— (E)-(S)-6-Carbamoyl-4-[(S)-2-((S)-2-methoxycarbonylamino-4-methyl-pentanoylamino)-3-phenyl-propionylamino]-hex-2-enoic acid ethyl ester —— C26H38N4O7
(E)-(S)-6-Carbamoyl-4-[(S)-2-((S)-2-methoxycarbonylamino-4-methyl-pentanoylamino)-3-phenyl-propionylamino]-hex-2-enoic acid ethyl ester
—— (E)-(S)-6-Carbamoyl-4-{(S)-2-[(S)-2-(3-hydroxy-propionylamino)-4-methyl-pentanoylamino]-3-phenyl-propionylamino}-hex-2-enoic acid ethyl ester —— C27H40N4O7
(E)-(S)-6-Carbamoyl-4-{(S)-2-[(S)-2-(3-hydroxy-propionylamino)-4-methyl-pentanoylamino]-3-phenyl-propionylamino}-hex-2-enoic acid ethyl ester