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—— (9aR)-8-(5-cyclopropylpyrazin-2-yl)oxy-2-[3-(trifluoromethyl)benzoyl]-3,4,7,8,9,9a-hexahydro-1H-pyrrolo[1,2-a][1,4]diazepin-5-one —— C23H23F3N4O3
(9aR)-8-(5-cyclopropylpyrazin-2-yl)oxy-2-[3-(trifluoromethyl)benzoyl]-3,4,7,8,9,9a-hexahydro-1H-pyrrolo[1,2-a][1,4]diazepin-5-one
—— 9-Bromo-3-[ethoxy(trimethylsilyl)methyl]-1-methyl-8-(trifluoromethyl)-1,5-dihydro-[1,2,4]triazino[3,4-c][1,4]benzoxazin-2-one —— C18H23BrF3N3O3Si
9-Bromo-3-[ethoxy(trimethylsilyl)methyl]-1-methyl-8-(trifluoromethyl)-1,5-dihydro-[1,2,4]triazino[3,4-c][1,4]benzoxazin-2-one
—— 9-(1,3-dimethylpiperidin-4-yl)-8-(2-fluoro-3-methoxyphenyl)-1-methyl-3,5-dihydro-1H-[1,2,4]triazino[3,4-c][1,4]benzoxazin-2-one —— C25H29FN4O3
9-(1,3-dimethylpiperidin-4-yl)-8-(2-fluoro-3-methoxyphenyl)-1-methyl-3,5-dihydro-1H-[1,2,4]triazino[3,4-c][1,4]benzoxazin-2-one
—— 9-[1-(1,3-dimethylazetidin-3-yl)ethyl]-8-[2-(2-hydroxypropan-2-yl)phenyl]-1-methyl-3,5-dihydro-1H-[1,2,4]triazino[3,4-c][1,4]benzoxazin-2-one —— C27H34N4O3
9-[1-(1,3-dimethylazetidin-3-yl)ethyl]-8-[2-(2-hydroxypropan-2-yl)phenyl]-1-methyl-3,5-dihydro-1H-[1,2,4]triazino[3,4-c][1,4]benzoxazin-2-one
—— 9-[azetidin-3-yl(methyl)arsanyl]-8-fluoro-1-methyl-3,5-dihydro-1H-[1,2,4]triazino[3,4-c][1,4]benzoxazin-2-one —— C15H18AsFN4O2
9-[azetidin-3-yl(methyl)arsanyl]-8-fluoro-1-methyl-3,5-dihydro-1H-[1,2,4]triazino[3,4-c][1,4]benzoxazin-2-one
—— 9H-fluoren-9-one O-{[(3-chlorophenyl)amino]carbonyl}oxime —— C20H13ClN2O2
9H-fluoren-9-one O-{[(3-chlorophenyl)amino]carbonyl}oxime
—— 9-[azetidin-3-yl(methyl)amino]-8-fluoro-1-methyl-3,5-dihydro-1H-[1,2,4]triazino[3,4-c][1,4]benzoxazin-2-one —— C15H18FN5O2
9-[azetidin-3-yl(methyl)amino]-8-fluoro-1-methyl-3,5-dihydro-1H-[1,2,4]triazino[3,4-c][1,4]benzoxazin-2-one
—— 9-(azetidin-3-ylamino)-1-methyl-8-[(2R)-1,1,1-trifluoropropan-2-yl]-3,5-dihydro-1H-[1,2,4]triazino[3,4-c][1,4]benzoxazin-2-one —— C17H20F3N5O2
9-(azetidin-3-ylamino)-1-methyl-8-[(2R)-1,1,1-trifluoropropan-2-yl]-3,5-dihydro-1H-[1,2,4]triazino[3,4-c][1,4]benzoxazin-2-one
—— [9-[(1,3-Dimethylazetidin-3-yl)amino]-1-methyl-2-oxo-8-(trifluoromethyl)-1,3,4a,5-tetrahydro-[1,2,4]triazino[3,4-c][1,4]benzoxazin-4-yl] 2,2,2-trifluoroacetate —— C19H21F6N5O4
[9-[(1,3-Dimethylazetidin-3-yl)amino]-1-methyl-2-oxo-8-(trifluoromethyl)-1,3,4a,5-tetrahydro-[1,2,4]triazino[3,4-c][1,4]benzoxazin-4-yl] 2,2,2-trifluoroacetate
—— 9-(azetidin-3-ylamino)-8-(2-fluorophenyl)-1-methyl-5,10b-dihydro-3H-chromeno[4,3-e][1,2,4]triazin-2-one —— C20H20FN5O2
9-(azetidin-3-ylamino)-8-(2-fluorophenyl)-1-methyl-5,10b-dihydro-3H-chromeno[4,3-e][1,2,4]triazin-2-one
—— 9-[(1,3-dimethylpyrrolidin-3-yl)-methylamino]-8-(2-fluorophenyl)-1-methyl-3,5-dihydro-1H-[1,2,4]triazino[3,4-c][1,4]benzoxazin-2-one —— C24H28FN5O2
9-[(1,3-dimethylpyrrolidin-3-yl)-methylamino]-8-(2-fluorophenyl)-1-methyl-3,5-dihydro-1H-[1,2,4]triazino[3,4-c][1,4]benzoxazin-2-one
—— 9-(azetidin-3-ylmethylamino)-8-fluoro-1-methyl-3,5-dihydro-1H-[1,2,4]triazino[3,4-c][1,4]benzoxazin-2-one —— C15H18FN5O2
9-(azetidin-3-ylmethylamino)-8-fluoro-1-methyl-3,5-dihydro-1H-[1,2,4]triazino[3,4-c][1,4]benzoxazin-2-one
—— 9-[(1S)-1-(azetidin-3-yl)ethyl]-1-methyl-3,5-dihydro-1H-[1,2,4]triazino[3,4-c][1,4]benzoxazin-2-one —— C16H20N4O2
9-[(1S)-1-(azetidin-3-yl)ethyl]-1-methyl-3,5-dihydro-1H-[1,2,4]triazino[3,4-c][1,4]benzoxazin-2-one
—— 9-(azetidin-3-ylamino)-8-(3-fluorophenyl)-1-methyl-5,10b-dihydro-3H-chromeno[4,3-e][1,2,4]triazin-2-one —— C20H20FN5O2
9-(azetidin-3-ylamino)-8-(3-fluorophenyl)-1-methyl-5,10b-dihydro-3H-chromeno[4,3-e][1,2,4]triazin-2-one
—— 9-(1,3-dimethylpiperidin-4-yl)-8-(2-fluoro-4-methylphenyl)-1-methyl-3,5-dihydro-1H-[1,2,4]triazino[3,4-c][1,4]benzoxazin-2-one —— C25H29FN4O2
9-(1,3-dimethylpiperidin-4-yl)-8-(2-fluoro-4-methylphenyl)-1-methyl-3,5-dihydro-1H-[1,2,4]triazino[3,4-c][1,4]benzoxazin-2-one
—— 9-[azetidin-3-yl(benzyl)amino]-1-methyl-3,5-dihydro-1H-[1,2,4]triazino[3,4-c][1,4]benzoxazin-2-one —— C21H23N5O2
9-[azetidin-3-yl(benzyl)amino]-1-methyl-3,5-dihydro-1H-[1,2,4]triazino[3,4-c][1,4]benzoxazin-2-one
—— 9-(3,3-dimethylpiperidin-4-yl)-1-methyl-3,5-dihydro-1H-[1,2,4]triazino[3,4-c][1,4]benzoxazin-2-one —— C18H24N4O2
9-(3,3-dimethylpiperidin-4-yl)-1-methyl-3,5-dihydro-1H-[1,2,4]triazino[3,4-c][1,4]benzoxazin-2-one
—— 9-(azetidin-3-ylamino)-8-(4-chlorophenyl)-1-methyl-4,5-dihydro-3H-chromeno[4,3-e][1,2,4]triazin-2-one —— C20H20ClN5O2
9-(azetidin-3-ylamino)-8-(4-chlorophenyl)-1-methyl-4,5-dihydro-3H-chromeno[4,3-e][1,2,4]triazin-2-one
—— 9-[(3R,4R)-1,3-dimethylpiperidin-4-yl]-8-(2-fluoro-4-methoxyphenyl)-1-methyl-3,5-dihydro-1H-[1,2,4]triazino[3,4-c][1,4]benzoxazin-2-one —— C25H29FN4O3
9-[(3R,4R)-1,3-dimethylpiperidin-4-yl]-8-(2-fluoro-4-methoxyphenyl)-1-methyl-3,5-dihydro-1H-[1,2,4]triazino[3,4-c][1,4]benzoxazin-2-one
—— 9-(2-benzylpiperidin-4-yl)-1-methyl-8-(trifluoromethyl)-3,5-dihydrobenzo[5,6][1,4]oxazino[3,4-c][1,2,4]triazin-2(1H)-one trifluoroacetic acid —— (x)C2HF3O2*C24H25F3N4O2
9-(2-benzylpiperidin-4-yl)-1-methyl-8-(trifluoromethyl)-3,5-dihydrobenzo[5,6][1,4]oxazino[3,4-c][1,2,4]triazin-2(1H)-one trifluoroacetic acid
—— 9-(azetidin-3-ylamino)-1-methyl-3,5-dihydro-1H-[1,2,4]triazino[3,4-c][1,4]benzothiazin-2-one —— C14H17N5OS
9-(azetidin-3-ylamino)-1-methyl-3,5-dihydro-1H-[1,2,4]triazino[3,4-c][1,4]benzothiazin-2-one
—— 9-(azetidin-3-ylamino)-8-cyclopentyl-1-methyl-3,5-dihydro-1H-[1,2,4]triazino[3,4-c][1,4]benzoxazin-2-one —— C19H25N5O2
9-(azetidin-3-ylamino)-8-cyclopentyl-1-methyl-3,5-dihydro-1H-[1,2,4]triazino[3,4-c][1,4]benzoxazin-2-one
—— 9-(azetidin-3-ylamino)-8-(2-chlorophenyl)-1-methyl-4,5-dihydro-3H-chromeno[4,3-e][1,2,4]triazin-2-one —— C20H20ClN5O2
9-(azetidin-3-ylamino)-8-(2-chlorophenyl)-1-methyl-4,5-dihydro-3H-chromeno[4,3-e][1,2,4]triazin-2-one
—— 9-[(1,3-dimethylazetidin-3-yl)amino]-8-[(Z)-2-ethoxyethenyl]-1-methyl-3,5-dihydro-1H-[1,2,4]triazino[3,4-c][1,4]benzoxazin-2-one —— C20H27N5O3
9-[(1,3-dimethylazetidin-3-yl)amino]-8-[(Z)-2-ethoxyethenyl]-1-methyl-3,5-dihydro-1H-[1,2,4]triazino[3,4-c][1,4]benzoxazin-2-one
—— 9-[(1R)-1-(1,3-dimethylazetidin-3-yl)ethyl]-1-methyl-8-propan-2-yl-3,5-dihydro-1H-[1,2,4]triazino[3,4-c][1,4]benzoxazin-2-one —— C21H30N4O2
9-[(1R)-1-(1,3-dimethylazetidin-3-yl)ethyl]-1-methyl-8-propan-2-yl-3,5-dihydro-1H-[1,2,4]triazino[3,4-c][1,4]benzoxazin-2-one
—— 9-[(1-benzyl-3-methylazetidin-3-yl)-methylamino]-1-methyl-8-phenyl-3,5-dihydro-1H-[1,2,4]triazino[3,4-c][1,4]benzoxazin-2-one —— C29H31N5O2
9-[(1-benzyl-3-methylazetidin-3-yl)-methylamino]-1-methyl-8-phenyl-3,5-dihydro-1H-[1,2,4]triazino[3,4-c][1,4]benzoxazin-2-one
—— 9-(azetidin-3-ylamino)-8-ethyl-1-methyl-3,5-dihydro-1H-[1,2,4]triazino[3,4-c][1,4]benzoxazin-2-one —— C16H21N5O2
9-(azetidin-3-ylamino)-8-ethyl-1-methyl-3,5-dihydro-1H-[1,2,4]triazino[3,4-c][1,4]benzoxazin-2-one
—— 9-(azetidin-3-ylamino)-1-methyl-8-propan-2-yl-3,5-dihydro-1H-[1,2,4]triazino[3,4-c][1,4]benzoxazin-2-one —— C17H23N5O2
9-(azetidin-3-ylamino)-1-methyl-8-propan-2-yl-3,5-dihydro-1H-[1,2,4]triazino[3,4-c][1,4]benzoxazin-2-one
—— 9-(Azetidin-3-yloxy)-1,8-dimethyl-3,5-dihydro-[1,2,4]triazino[3,4-c][1,4]benzoxazine —— C15H18N4O2
9-(Azetidin-3-yloxy)-1,8-dimethyl-3,5-dihydro-[1,2,4]triazino[3,4-c][1,4]benzoxazine
—— [9-[(1,3-Dimethylazetidin-3-yl)amino]-1-methyl-2-oxo-8-phenyl-1,3,4a,5-tetrahydro-[1,2,4]triazino[3,4-c][1,4]benzoxazin-4-yl] 2,2,2-trifluoroacetate —— C24H26F3N5O4
[9-[(1,3-Dimethylazetidin-3-yl)amino]-1-methyl-2-oxo-8-phenyl-1,3,4a,5-tetrahydro-[1,2,4]triazino[3,4-c][1,4]benzoxazin-4-yl] 2,2,2-trifluoroacetate
—— 9-[(3R,4R)-1,3-dimethylpiperidin-4-yl]-8-(2-fluorophenyl)-1-methyl-3,5-dihydro-1H-[1,2,4]triazino[3,4-c][1,4]benzoxazin-2-one;hydrochloride —— C24H28ClFN4O2
9-[(3R,4R)-1,3-dimethylpiperidin-4-yl]-8-(2-fluorophenyl)-1-methyl-3,5-dihydro-1H-[1,2,4]triazino[3,4-c][1,4]benzoxazin-2-one;hydrochloride
—— 9-(azetidin-3-ylamino)-1-methyl-8-[(2S)-1,1,1-trifluoropropan-2-yl]-3,5-dihydro-1H-[1,2,4]triazino[3,4-c][1,4]benzoxazin-2-one —— C17H20F3N5O2
9-(azetidin-3-ylamino)-1-methyl-8-[(2S)-1,1,1-trifluoropropan-2-yl]-3,5-dihydro-1H-[1,2,4]triazino[3,4-c][1,4]benzoxazin-2-one
—— 9-(azetidin-3-ylamino)-1-methyl-8-(trifluoromethyl)-4,5-dihydro-3H-chromeno[4,3-e][1,2,4]triazin-2-one —— C15H16F3N5O2
9-(azetidin-3-ylamino)-1-methyl-8-(trifluoromethyl)-4,5-dihydro-3H-chromeno[4,3-e][1,2,4]triazin-2-one
—— 9-(azetidin-3-ylamino)-8-(2-chlorophenyl)-1-methyl-5,10b-dihydro-3H-chromeno[4,3-e][1,2,4]triazin-2-one —— C20H20ClN5O2
9-(azetidin-3-ylamino)-8-(2-chlorophenyl)-1-methyl-5,10b-dihydro-3H-chromeno[4,3-e][1,2,4]triazin-2-one
—— 9-[(1R)-1-(azetidin-3-yl)ethyl]-1-methyl-3,5-dihydro-1H-[1,2,4]triazino[3,4-c][1,4]benzoxazin-2-one —— C16H20N4O2
9-[(1R)-1-(azetidin-3-yl)ethyl]-1-methyl-3,5-dihydro-1H-[1,2,4]triazino[3,4-c][1,4]benzoxazin-2-one
—— 9-(azetidin-3-ylamino)-8-(3-fluorophenyl)-1-methyl-4,5-dihydro-3H-chromeno[4,3-e][1,2,4]triazin-2-one —— C20H20FN5O2
9-(azetidin-3-ylamino)-8-(3-fluorophenyl)-1-methyl-4,5-dihydro-3H-chromeno[4,3-e][1,2,4]triazin-2-one
—— 9-(azetidin-3-yloxy)-8-fluoro-1-methyl-3,5-dihydro-1H-[1,2,4]triazino[3,4-c][1,4]benzoxazin-2-one;2,2,2-trifluoroacetic acid —— C16H16F4N4O5
9-(azetidin-3-yloxy)-8-fluoro-1-methyl-3,5-dihydro-1H-[1,2,4]triazino[3,4-c][1,4]benzoxazin-2-one;2,2,2-trifluoroacetic acid
—— 9-(1,7-diazaspiro[3.5]nonan-1-yl)-1,8-dimethyl-3,5-dihydro-1H-[1,2,4]triazino[3,4-c][1,4]benzoxazin-2-one —— C19H25N5O2
9-(1,7-diazaspiro[3.5]nonan-1-yl)-1,8-dimethyl-3,5-dihydro-1H-[1,2,4]triazino[3,4-c][1,4]benzoxazin-2-one
—— 9-[(3R,4R)-1,3-dimethylpiperidin-4-yl]-8-(2-fluoro-5-methoxyphenyl)-1-methyl-3,5-dihydro-1H-[1,2,4]triazino[3,4-c][1,4]benzoxazin-2-one —— C25H29FN4O3
9-[(3R,4R)-1,3-dimethylpiperidin-4-yl]-8-(2-fluoro-5-methoxyphenyl)-1-methyl-3,5-dihydro-1H-[1,2,4]triazino[3,4-c][1,4]benzoxazin-2-one
—— [9-[2-(Aminomethyl)pyrrolidin-1-yl]-1-methyl-2-oxo-1,3,4a,5-tetrahydro-[1,2,4]triazino[3,4-c][1,4]benzoxazin-4-yl] 2,2,2-trifluoroacetate —— C18H22F3N5O4
[9-[2-(Aminomethyl)pyrrolidin-1-yl]-1-methyl-2-oxo-1,3,4a,5-tetrahydro-[1,2,4]triazino[3,4-c][1,4]benzoxazin-4-yl] 2,2,2-trifluoroacetate
—— 9-[(3R,4R)-1,3-dimethylpiperidin-4-yl]-8-(2-fluorophenyl)-1-methyl-3,5-dihydro-1H-[1,2,4]triazino[3,4-c][1,4]benzoxazin-2-one —— C24H27FN4O2
9-[(3R,4R)-1,3-dimethylpiperidin-4-yl]-8-(2-fluorophenyl)-1-methyl-3,5-dihydro-1H-[1,2,4]triazino[3,4-c][1,4]benzoxazin-2-one
—— 9-(azetidin-3-ylamino)-8-(2-fluorophenyl)-1-methyl-4,5-dihydro-3H-chromeno[4,3-e][1,2,4]triazin-2-one —— C20H20FN5O2
9-(azetidin-3-ylamino)-8-(2-fluorophenyl)-1-methyl-4,5-dihydro-3H-chromeno[4,3-e][1,2,4]triazin-2-one
—— 9-[(1-acetyl-3-methylazetidin-3-yl)-methylamino]-8-(2-fluorophenyl)-1-methyl-3,5-dihydro-1H-[1,2,4]triazino[3,4-c][1,4]benzoxazin-2-one —— C24H26FN5O3
9-[(1-acetyl-3-methylazetidin-3-yl)-methylamino]-8-(2-fluorophenyl)-1-methyl-3,5-dihydro-1H-[1,2,4]triazino[3,4-c][1,4]benzoxazin-2-one
—— 9-(azetidin-3-ylamino)-8-(4-fluorophenyl)-1-methyl-4,5-dihydro-3H-chromeno[4,3-e][1,2,4]triazin-2-one —— C20H20FN5O2
9-(azetidin-3-ylamino)-8-(4-fluorophenyl)-1-methyl-4,5-dihydro-3H-chromeno[4,3-e][1,2,4]triazin-2-one
—— 9-(azetidin-3-ylamino)-8-(4-fluorophenyl)-1-methyl-5,10b-dihydro-3H-chromeno[4,3-e][1,2,4]triazin-2-one —— C20H20FN5O2
9-(azetidin-3-ylamino)-8-(4-fluorophenyl)-1-methyl-5,10b-dihydro-3H-chromeno[4,3-e][1,2,4]triazin-2-one
—— 9-(azetidin-3-ylamino)-8-chloro-1-methyl-3,5-dihydro-1H-[1,2,4]triazino[3,4-c][1,4]benzoxazin-2-one —— C14H16ClN5O2
9-(azetidin-3-ylamino)-8-chloro-1-methyl-3,5-dihydro-1H-[1,2,4]triazino[3,4-c][1,4]benzoxazin-2-one
—— 9-(azetidin-3-ylamino)-8-(4-chlorophenyl)-1-methyl-5,10b-dihydro-3H-chromeno[4,3-e][1,2,4]triazin-2-one —— C20H20ClN5O2
9-(azetidin-3-ylamino)-8-(4-chlorophenyl)-1-methyl-5,10b-dihydro-3H-chromeno[4,3-e][1,2,4]triazin-2-one
—— 9-[(2S,4S)-2-benzylpiperidin-4-yl]-1-methyl-3,5-dihydro-1H-[1,2,4]triazino[3,4-c][1,4]benzoxazin-2-one —— C23H26N4O2
9-[(2S,4S)-2-benzylpiperidin-4-yl]-1-methyl-3,5-dihydro-1H-[1,2,4]triazino[3,4-c][1,4]benzoxazin-2-one
—— 9-[[(3S)-1,3-dimethylpyrrolidin-3-yl]-methylamino]-8-(2-fluorophenyl)-1-methyl-3,5-dihydro-1H-[1,2,4]triazino[3,4-c][1,4]benzoxazin-2-one —— C24H28FN5O2
9-[[(3S)-1,3-dimethylpyrrolidin-3-yl]-methylamino]-8-(2-fluorophenyl)-1-methyl-3,5-dihydro-1H-[1,2,4]triazino[3,4-c][1,4]benzoxazin-2-one
—— 9-[azetidin-3-yl(cyclopropyl)amino]-3,5-dihydro-1H-[1,2,4]triazino[3,4-c][1,4]benzoxazin-2-one —— C16H19N5O2
9-[azetidin-3-yl(cyclopropyl)amino]-3,5-dihydro-1H-[1,2,4]triazino[3,4-c][1,4]benzoxazin-2-one