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—— 8-[(3-fluorophenyl)methyl]-4-methyl-2-[(2S)-1-[(1-methylpyrazol-4-yl)methyl]pyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C24H27FN6O
8-[(3-fluorophenyl)methyl]-4-methyl-2-[(2S)-1-[(1-methylpyrazol-4-yl)methyl]pyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-benzyl-4-methyl-2-[(2S)-1-[2-(2-oxopyrrolidin-1-yl)acetyl]pyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C25H29N5O3
8-benzyl-4-methyl-2-[(2S)-1-[2-(2-oxopyrrolidin-1-yl)acetyl]pyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-cyclopropyl-2-[(2R)-1-[2-(4-methoxy-3-methylphenyl)acetyl]piperidin-2-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C26H32N4O3
8-cyclopropyl-2-[(2R)-1-[2-(4-methoxy-3-methylphenyl)acetyl]piperidin-2-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-benzyl-4-methyl-2-[(3R)-1-(oxan-4-yl)piperidin-3-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C25H32N4O2
8-benzyl-4-methyl-2-[(3R)-1-(oxan-4-yl)piperidin-3-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-cyclopropyl-2-[(2R)-1-[4-(methoxymethyl)benzoyl]piperidin-2-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C25H30N4O3
8-cyclopropyl-2-[(2R)-1-[4-(methoxymethyl)benzoyl]piperidin-2-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-(cyclohexylmethyl)-4-methyl-2-[(2R)-1-[(1-methylpyrazol-4-yl)methyl]pyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C24H34N6O
8-(cyclohexylmethyl)-4-methyl-2-[(2R)-1-[(1-methylpyrazol-4-yl)methyl]pyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-benzyl-4-methyl-2-[(2S)-1-(pyrazine-2-carbonyl)piperidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C25H26N6O2
8-benzyl-4-methyl-2-[(2S)-1-(pyrazine-2-carbonyl)piperidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-[(4-fluorophenyl)methyl]-4-methyl-2-[(2R)-1-(2-oxo-2-pyrazol-1-ylethyl)pyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C24H25FN6O2
8-[(4-fluorophenyl)methyl]-4-methyl-2-[(2R)-1-(2-oxo-2-pyrazol-1-ylethyl)pyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-(cyclopropylmethyl)-2-[(3R)-1-[2-(3,4-dimethylphenyl)acetyl]piperidin-3-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C27H34N4O2
8-(cyclopropylmethyl)-2-[(3R)-1-[2-(3,4-dimethylphenyl)acetyl]piperidin-3-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-benzyl-4-methyl-2-[(2S)-1-[2-(2-oxopyrrolidin-1-yl)ethyl]piperidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C26H33N5O2
8-benzyl-4-methyl-2-[(2S)-1-[2-(2-oxopyrrolidin-1-yl)ethyl]piperidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-(cyclopropylmethyl)-4-methyl-2-[(3S)-1-(3-morpholin-4-ylpropanoyl)piperidin-3-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C24H35N5O3
8-(cyclopropylmethyl)-4-methyl-2-[(3S)-1-(3-morpholin-4-ylpropanoyl)piperidin-3-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-benzyl-4-methyl-2-[(2S)-1-(2-pyrrolidin-1-ylacetyl)piperidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C26H33N5O2
8-benzyl-4-methyl-2-[(2S)-1-(2-pyrrolidin-1-ylacetyl)piperidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-(cyclohexylmethyl)-4-methyl-2-[(2S)-1-(2-pyrrolidin-1-ylacetyl)pyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C25H37N5O2
8-(cyclohexylmethyl)-4-methyl-2-[(2S)-1-(2-pyrrolidin-1-ylacetyl)pyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-[(2-fluorophenyl)methyl]-2-[(3S)-1-(2-hydroxyacetyl)piperidin-3-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C22H25FN4O3
8-[(2-fluorophenyl)methyl]-2-[(3S)-1-(2-hydroxyacetyl)piperidin-3-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-benzyl-2-[(2S)-1-(3-ethyl-1,2-oxazole-5-carbonyl)pyrrolidin-2-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C25H27N5O3
8-benzyl-2-[(2S)-1-(3-ethyl-1,2-oxazole-5-carbonyl)pyrrolidin-2-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-[(4-fluorophenyl)methyl]-4-methyl-2-[(2S)-1-(pyrazine-2-carbonyl)pyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C24H23FN6O2
8-[(4-fluorophenyl)methyl]-4-methyl-2-[(2S)-1-(pyrazine-2-carbonyl)pyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-(cyclohexylmethyl)-4-methyl-2-[(2R)-1-(2-propan-2-yloxyacetyl)pyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C24H36N4O3
8-(cyclohexylmethyl)-4-methyl-2-[(2R)-1-(2-propan-2-yloxyacetyl)pyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-benzyl-4-methyl-2-[(2R)-1-[2-(2-oxopyrrolidin-1-yl)acetyl]pyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C25H29N5O3
8-benzyl-4-methyl-2-[(2R)-1-[2-(2-oxopyrrolidin-1-yl)acetyl]pyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-[(4-fluorophenyl)methyl]-2-[(2R)-1-(2-methoxy-2-methylpropanoyl)pyrrolidin-2-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C24H29FN4O3
8-[(4-fluorophenyl)methyl]-2-[(2R)-1-(2-methoxy-2-methylpropanoyl)pyrrolidin-2-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-[(4-fluorophenyl)methyl]-4-methyl-2-[(2S)-1-(2-pyrazol-1-ylacetyl)pyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C24H25FN6O2
8-[(4-fluorophenyl)methyl]-4-methyl-2-[(2S)-1-(2-pyrazol-1-ylacetyl)pyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-[(4-fluorophenyl)methyl]-2-[(3R)-1-(1H-imidazol-2-ylmethyl)piperidin-3-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C24H27FN6O
8-[(4-fluorophenyl)methyl]-2-[(3R)-1-(1H-imidazol-2-ylmethyl)piperidin-3-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-benzyl-4-methyl-2-[(2R)-1-pyrimidin-2-ylpiperidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C24H26N6O
8-benzyl-4-methyl-2-[(2R)-1-pyrimidin-2-ylpiperidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-[(2-fluorophenyl)methyl]-2-[(3S)-1-(3-methoxypropanoyl)piperidin-3-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C24H29FN4O3
8-[(2-fluorophenyl)methyl]-2-[(3S)-1-(3-methoxypropanoyl)piperidin-3-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-(cyclohexylmethyl)-4-methyl-2-[(2R)-1-(thiadiazole-4-carbonyl)pyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C22H28N6O2S
8-(cyclohexylmethyl)-4-methyl-2-[(2R)-1-(thiadiazole-4-carbonyl)pyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-(cyclopropylmethyl)-4-methyl-2-[(3S)-1-(2-propan-2-yloxyacetyl)piperidin-3-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C22H32N4O3
8-(cyclopropylmethyl)-4-methyl-2-[(3S)-1-(2-propan-2-yloxyacetyl)piperidin-3-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-benzyl-2-[(3R)-1-[2-(diethylamino)acetyl]piperidin-3-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C26H35N5O2
8-benzyl-2-[(3R)-1-[2-(diethylamino)acetyl]piperidin-3-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-[(3-fluorophenyl)methyl]-4-methyl-2-[(2S)-1-(2-methylpropanoyl)pyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C23H27FN4O2
8-[(3-fluorophenyl)methyl]-4-methyl-2-[(2S)-1-(2-methylpropanoyl)pyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-(cyclopropylmethyl)-4-methyl-2-[(2S)-1-(2-propan-2-yloxyacetyl)piperidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C22H32N4O3
8-(cyclopropylmethyl)-4-methyl-2-[(2S)-1-(2-propan-2-yloxyacetyl)piperidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-(cyclohexylmethyl)-2-[(2R)-1-[(1-ethylpyrazol-4-yl)methyl]pyrrolidin-2-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C25H36N6O
8-(cyclohexylmethyl)-2-[(2R)-1-[(1-ethylpyrazol-4-yl)methyl]pyrrolidin-2-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-(cyclopropylmethyl)-4-methyl-2-[(2R)-1-[(2-methyl-1,3-thiazol-5-yl)methyl]piperidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C22H29N5OS
8-(cyclopropylmethyl)-4-methyl-2-[(2R)-1-[(2-methyl-1,3-thiazol-5-yl)methyl]piperidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-benzyl-2-[1-[(1R)-cyclohex-3-ene-1-carbonyl]piperidin-4-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C27H32N4O2
8-benzyl-2-[1-[(1R)-cyclohex-3-ene-1-carbonyl]piperidin-4-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-(cyclopropylmethyl)-4-methyl-2-[(3S)-1-pyrrolidin-1-ylsulfonylpiperidin-3-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C21H31N5O3S
8-(cyclopropylmethyl)-4-methyl-2-[(3S)-1-pyrrolidin-1-ylsulfonylpiperidin-3-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-Benzyl-4-methyl-2-[1-[(2-methyl-1,3-thiazol-5-yl)methyl]piperidin-4-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C25H29N5OS
8-Benzyl-4-methyl-2-[1-[(2-methyl-1,3-thiazol-5-yl)methyl]piperidin-4-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-Cyclopentyl-2-[1-(2-methoxybenzoyl)piperidin-4-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C26H32N4O3
8-Cyclopentyl-2-[1-(2-methoxybenzoyl)piperidin-4-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-[(2-methoxyphenyl)methyl]-4-methyl-2-[(2R)-1-[(1-methylpyrazol-4-yl)methyl]pyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C25H30N6O2
8-[(2-methoxyphenyl)methyl]-4-methyl-2-[(2R)-1-[(1-methylpyrazol-4-yl)methyl]pyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-(cyclohexylmethyl)-4-methyl-2-[(3R)-1-methylsulfonylpiperidin-3-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C21H32N4O3S
8-(cyclohexylmethyl)-4-methyl-2-[(3R)-1-methylsulfonylpiperidin-3-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-benzyl-2-[(2S)-1-(2-cyclopentylacetyl)pyrrolidin-2-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C26H32N4O2
8-benzyl-2-[(2S)-1-(2-cyclopentylacetyl)pyrrolidin-2-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-benzyl-2-[(2S)-1-[2-(dimethylamino)acetyl]piperidin-2-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C24H31N5O2
8-benzyl-2-[(2S)-1-[2-(dimethylamino)acetyl]piperidin-2-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-benzyl-4-methyl-2-[(3S)-1-(oxan-4-yl)piperidin-3-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C25H32N4O2
8-benzyl-4-methyl-2-[(3S)-1-(oxan-4-yl)piperidin-3-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-cyclopropyl-2-[(2S)-1-[4-(methoxymethyl)benzoyl]piperidin-2-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C25H30N4O3
8-cyclopropyl-2-[(2S)-1-[4-(methoxymethyl)benzoyl]piperidin-2-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-benzyl-4-methyl-2-[(3S)-1-(2-propan-2-yloxyacetyl)piperidin-3-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C25H32N4O3
8-benzyl-4-methyl-2-[(3S)-1-(2-propan-2-yloxyacetyl)piperidin-3-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-[(2-fluorophenyl)methyl]-2-[(3R)-1-(2-methoxyacetyl)piperidin-3-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C23H27FN4O3
8-[(2-fluorophenyl)methyl]-2-[(3R)-1-(2-methoxyacetyl)piperidin-3-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-(cyclohexylmethyl)-4-methyl-2-[(3R)-1-(pyridine-2-carbonyl)piperidin-3-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C26H33N5O2
8-(cyclohexylmethyl)-4-methyl-2-[(3R)-1-(pyridine-2-carbonyl)piperidin-3-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-benzyl-4-methyl-2-[(2S)-1-(5-methylpyrazine-2-carbonyl)pyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C25H26N6O2
8-benzyl-4-methyl-2-[(2S)-1-(5-methylpyrazine-2-carbonyl)pyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-(Cyclopropylmethyl)-4-methyl-2-[1-(2-phenoxyacetyl)piperidin-4-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C25H30N4O3
8-(Cyclopropylmethyl)-4-methyl-2-[1-(2-phenoxyacetyl)piperidin-4-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-(cyclopropylmethyl)-4-methyl-2-[(2R)-1-(3-methylbutanoyl)piperidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C22H32N4O2
8-(cyclopropylmethyl)-4-methyl-2-[(2R)-1-(3-methylbutanoyl)piperidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-(cyclohexylmethyl)-4-methyl-2-[1-[(2R)-oxolane-2-carbonyl]piperidin-4-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C25H36N4O3
8-(cyclohexylmethyl)-4-methyl-2-[1-[(2R)-oxolane-2-carbonyl]piperidin-4-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-[(4-fluorophenyl)methyl]-2-[(2R)-1-(2-methoxyacetyl)pyrrolidin-2-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C22H25FN4O3
8-[(4-fluorophenyl)methyl]-2-[(2R)-1-(2-methoxyacetyl)pyrrolidin-2-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-(cyclopropylmethyl)-2-[(2S)-1-[(4-fluorophenyl)methyl]piperidin-2-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C24H29FN4O
8-(cyclopropylmethyl)-2-[(2S)-1-[(4-fluorophenyl)methyl]piperidin-2-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-benzyl-4-methyl-2-[(2R)-1-(4-methyl-1,3-thiazole-5-carbonyl)pyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C24H25N5O2S
8-benzyl-4-methyl-2-[(2R)-1-(4-methyl-1,3-thiazole-5-carbonyl)pyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one