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中文名称 英文名称 CAS号 化学式 结构式图片
—— 8-(azepan-1-ium-1-ylmethyl)-3-(1,3-dihydrobenzimidazol-2-ylidene)chromene-2,7-dione —— C23H24N3O3+
8-(azepan-1-ium-1-ylmethyl)-3-(1,3-dihydrobenzimidazol-2-ylidene)chromene-2,7-dione
—— 8-(Azepan-1-ium-1-ylmethyl)-3-(2,3-dihydro-1,4-benzodioxin-6-yl)-7-hydroxychromen-4-one —— C24H26NO5+
8-(Azepan-1-ium-1-ylmethyl)-3-(2,3-dihydro-1,4-benzodioxin-6-yl)-7-hydroxychromen-4-one
—— 8-(cyclopropylmethyl)-4-methyl-2-[(3S)-1-[(1-methylpyrazol-4-yl)methyl]piperidin-3-yl]-6,7-dihydro-5H-pyrido[2,3-d]pyrimidine —— C22H32N6
8-(cyclopropylmethyl)-4-methyl-2-[(3S)-1-[(1-methylpyrazol-4-yl)methyl]piperidin-3-yl]-6,7-dihydro-5H-pyrido[2,3-d]pyrimidine
—— 8-[(4-methoxyphenyl)methyl]-4-methyl-2-[(3R)-1-methylsulfonylpiperidin-3-yl]-6,7-dihydro-5H-pyrido[2,3-d]pyrimidine —— C22H30N4O3S
8-[(4-methoxyphenyl)methyl]-4-methyl-2-[(3R)-1-methylsulfonylpiperidin-3-yl]-6,7-dihydro-5H-pyrido[2,3-d]pyrimidine
—— 8-benzyl-2-[(3S)-1-ethylsulfonylpiperidin-3-yl]-4-methyl-6,7-dihydro-5H-pyrido[2,3-d]pyrimidine —— C22H30N4O2S
8-benzyl-2-[(3S)-1-ethylsulfonylpiperidin-3-yl]-4-methyl-6,7-dihydro-5H-pyrido[2,3-d]pyrimidine
—— 8-benzyl-2-[(2S)-1-(3-methoxypropanoyl)piperidin-2-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C24H30N4O3
8-benzyl-2-[(2S)-1-(3-methoxypropanoyl)piperidin-2-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-benzyl-4-methyl-2-[(2R)-1-methylsulfonylpiperidin-2-yl]-6,7-dihydro-5H-pyrido[2,3-d]pyrimidine —— C21H28N4O2S
8-benzyl-4-methyl-2-[(2R)-1-methylsulfonylpiperidin-2-yl]-6,7-dihydro-5H-pyrido[2,3-d]pyrimidine
—— 8-benzyl-4-methyl-2-[(2S)-1-(oxan-4-yl)piperidin-2-yl]-6,7-dihydro-5H-pyrido[2,3-d]pyrimidine —— C25H34N4O
8-benzyl-4-methyl-2-[(2S)-1-(oxan-4-yl)piperidin-2-yl]-6,7-dihydro-5H-pyrido[2,3-d]pyrimidine
—— 8-benzyl-2-[(2R)-1-[(4-fluorophenyl)methyl]piperidin-2-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C27H29FN4O
8-benzyl-2-[(2R)-1-[(4-fluorophenyl)methyl]piperidin-2-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-(cyclopropylmethyl)-2-[(2R)-1-[(3,5-dimethyl-1H-pyrazol-4-yl)sulfonyl]piperidin-2-yl]-4-methyl-6,7-dihydro-5H-pyrido[2,3-d]pyrimidine —— C22H32N6O2S
8-(cyclopropylmethyl)-2-[(2R)-1-[(3,5-dimethyl-1H-pyrazol-4-yl)sulfonyl]piperidin-2-yl]-4-methyl-6,7-dihydro-5H-pyrido[2,3-d]pyrimidine
—— 8-[(4-fluorophenyl)methyl]-4-methyl-2-[[methyl-[(3S)-3-phenylbutyl]amino]methyl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C27H31FN4O
8-[(4-fluorophenyl)methyl]-4-methyl-2-[[methyl-[(3S)-3-phenylbutyl]amino]methyl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-methyl-2-[(E)-2-[5-(2-nitrophenyl)furan-2-yl]ethenyl]quinoline-4-carboxylic acid —— C23H16N2O5
8-methyl-2-[(E)-2-[5-(2-nitrophenyl)furan-2-yl]ethenyl]quinoline-4-carboxylic acid
—— 8-[(4-Fluorophenyl)methyl]-4-methyl-2-[[methyl-[(2-propan-2-ylpyrimidin-5-yl)methyl]amino]methyl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C25H29FN6O
8-[(4-Fluorophenyl)methyl]-4-methyl-2-[[methyl-[(2-propan-2-ylpyrimidin-5-yl)methyl]amino]methyl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-cyclopropyl-2-[(2R)-1-(2-methoxyacetyl)piperidin-2-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C19H26N4O3
8-cyclopropyl-2-[(2R)-1-(2-methoxyacetyl)piperidin-2-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-[(3-Methoxyphenyl)methyl]-4-methyl-2-[[methyl-[(2-methyl-1,3-thiazol-5-yl)methyl]amino]methyl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C23H27N5O2S
8-[(3-Methoxyphenyl)methyl]-4-methyl-2-[[methyl-[(2-methyl-1,3-thiazol-5-yl)methyl]amino]methyl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— (8Z)-8-[(4-methoxyphenyl)methylidene]-2,4-diphenyl-6,7-dihydro-5H-quinoline —— C29H25NO
(8Z)-8-[(4-methoxyphenyl)methylidene]-2,4-diphenyl-6,7-dihydro-5H-quinoline
—— 8-benzyl-4-methyl-2-[[methyl-[[(2S)-2-methyl-2,3-dihydro-1-benzofuran-5-yl]methyl]amino]methyl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C27H30N4O2
8-benzyl-4-methyl-2-[[methyl-[[(2S)-2-methyl-2,3-dihydro-1-benzofuran-5-yl]methyl]amino]methyl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-(Cyclopropylmethyl)-2-[[2-(3-methoxyphenoxy)ethyl-methylamino]methyl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C23H30N4O3
8-(Cyclopropylmethyl)-2-[[2-(3-methoxyphenoxy)ethyl-methylamino]methyl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-(Cyclopropylmethyl)-2-[[2,2-diphenylethyl(methyl)amino]methyl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C28H32N4O
8-(Cyclopropylmethyl)-2-[[2,2-diphenylethyl(methyl)amino]methyl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-benzyl-4-methyl-2-[(2S)-1-(pyridine-2-carbonyl)pyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C25H25N5O2
8-benzyl-4-methyl-2-[(2S)-1-(pyridine-2-carbonyl)pyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-(cyclohexylmethyl)-4-methyl-2-[(3S)-1-(pyridine-4-carbonyl)piperidin-3-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C26H33N5O2
8-(cyclohexylmethyl)-4-methyl-2-[(3S)-1-(pyridine-4-carbonyl)piperidin-3-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-benzyl-4-methyl-2-[(2R)-1-(pyridine-2-carbonyl)pyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C25H25N5O2
8-benzyl-4-methyl-2-[(2R)-1-(pyridine-2-carbonyl)pyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-(cyclohexylmethyl)-4-methyl-2-[(3S)-1-(pyridin-4-ylmethyl)piperidin-3-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C26H35N5O
8-(cyclohexylmethyl)-4-methyl-2-[(3S)-1-(pyridin-4-ylmethyl)piperidin-3-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-(cyclohexylmethyl)-2-[(3S)-1-(cyclopentanecarbonyl)piperidin-3-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C26H38N4O2
8-(cyclohexylmethyl)-2-[(3S)-1-(cyclopentanecarbonyl)piperidin-3-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-benzyl-4-methyl-2-[(2S)-1-(pyridine-3-carbonyl)pyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C25H25N5O2
8-benzyl-4-methyl-2-[(2S)-1-(pyridine-3-carbonyl)pyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-(cyclohexylmethyl)-2-[(3S)-1-(2-methoxyacetyl)piperidin-3-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C23H34N4O3
8-(cyclohexylmethyl)-2-[(3S)-1-(2-methoxyacetyl)piperidin-3-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-benzyl-4-methyl-2-[(2R)-1-(2-pyridin-4-ylacetyl)pyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C26H27N5O2
8-benzyl-4-methyl-2-[(2R)-1-(2-pyridin-4-ylacetyl)pyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-(Cyclohexylmethyl)-2-[1-[2-(dimethylamino)acetyl]piperidin-4-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C24H37N5O2
8-(Cyclohexylmethyl)-2-[1-[2-(dimethylamino)acetyl]piperidin-4-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-(cyclohexylmethyl)-4-methyl-2-[(3R)-1-(pyridine-4-carbonyl)piperidin-3-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C26H33N5O2
8-(cyclohexylmethyl)-4-methyl-2-[(3R)-1-(pyridine-4-carbonyl)piperidin-3-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-benzyl-4-methyl-2-[(2S)-1-(pyridine-3-carbonyl)piperidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C26H27N5O2
8-benzyl-4-methyl-2-[(2S)-1-(pyridine-3-carbonyl)piperidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-[(2-fluorophenyl)methyl]-4-methyl-2-[(3R)-1-(1H-pyrazole-5-carbonyl)piperidin-3-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C24H25FN6O2
8-[(2-fluorophenyl)methyl]-4-methyl-2-[(3R)-1-(1H-pyrazole-5-carbonyl)piperidin-3-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-methyl-2-[(E)-2-[5-[3-(trifluoromethyl)phenyl]furan-2-yl]ethenyl]quinoline-4-carboxylic acid —— C24H16F3NO3
8-methyl-2-[(E)-2-[5-[3-(trifluoromethyl)phenyl]furan-2-yl]ethenyl]quinoline-4-carboxylic acid
—— 8-methyl-2-[(E)-2-[5-(4-nitrophenyl)furan-2-yl]ethenyl]quinoline-4-carboxylic acid —— C23H16N2O5
8-methyl-2-[(E)-2-[5-(4-nitrophenyl)furan-2-yl]ethenyl]quinoline-4-carboxylic acid
—— 8-methyl-N-[(1S)-1-[3-(3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]imidazo[1,2-a]pyridine-2-carboxamide —— C20H19N5O2
8-methyl-N-[(1S)-1-[3-(3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]imidazo[1,2-a]pyridine-2-carboxamide
—— 8-methoxy-2-methyl-N-[[(2R)-oxolan-2-yl]methyl]-N-(pyridin-2-ylmethyl)quinoline-3-carboxamide —— C23H25N3O3
8-methoxy-2-methyl-N-[[(2R)-oxolan-2-yl]methyl]-N-(pyridin-2-ylmethyl)quinoline-3-carboxamide
—— 8-chloro-2-[[(3S)-3-[(2-methylimidazol-1-yl)methyl]piperidin-1-yl]methyl]quinoline —— C20H23ClN4
8-chloro-2-[[(3S)-3-[(2-methylimidazol-1-yl)methyl]piperidin-1-yl]methyl]quinoline
—— 8-chloro-4-[2-[(2R)-2-ethyl-3-oxopiperazin-1-yl]-2-oxoethyl]-1,4-benzoxazin-3-one —— C16H18ClN3O4
8-chloro-4-[2-[(2R)-2-ethyl-3-oxopiperazin-1-yl]-2-oxoethyl]-1,4-benzoxazin-3-one
—— (8aR)-1-[[1-(4-fluorophenyl)pyrazol-4-yl]methyl]-8a-methyl-3,4,7,8-tetrahydro-2H-pyrrolo[1,2-a]pyrimidin-6-one —— C18H21FN4O
(8aR)-1-[[1-(4-fluorophenyl)pyrazol-4-yl]methyl]-8a-methyl-3,4,7,8-tetrahydro-2H-pyrrolo[1,2-a]pyrimidin-6-one
—— 8-[[(3R,8aS)-3-methyl-3,4,6,7,8,8a-hexahydro-1H-pyrrolo[1,2-a]pyrazin-2-yl]methyl]quinoline —— C18H23N3
8-[[(3R,8aS)-3-methyl-3,4,6,7,8,8a-hexahydro-1H-pyrrolo[1,2-a]pyrazin-2-yl]methyl]quinoline
—— 8,9-Dimethoxy-3-[(4-methoxyphenyl)methyl]-1,2,4,5-tetrahydro-[1,4]diazepino[7,1-b]quinazolin-11-one —— C22H25N3O4
8,9-Dimethoxy-3-[(4-methoxyphenyl)methyl]-1,2,4,5-tetrahydro-[1,4]diazepino[7,1-b]quinazolin-11-one
—— 8,9-dimethoxy-3-[2-[(2R)-oxan-2-yl]acetyl]-1,2,4,5-tetrahydro-[1,4]diazepino[7,1-b]quinazolin-11-one —— C21H27N3O5
8,9-dimethoxy-3-[2-[(2R)-oxan-2-yl]acetyl]-1,2,4,5-tetrahydro-[1,4]diazepino[7,1-b]quinazolin-11-one
—— 8,9-Dimethoxy-3-[(3-methyl-1-prop-2-enylpyrazol-4-yl)methyl]-1,2,4,5-tetrahydro-[1,4]diazepino[7,1-b]quinazolin-11-one —— C22H27N5O3
8,9-Dimethoxy-3-[(3-methyl-1-prop-2-enylpyrazol-4-yl)methyl]-1,2,4,5-tetrahydro-[1,4]diazepino[7,1-b]quinazolin-11-one
—— (8S)-1'-(1-ethyl-5-methylpyrazol-4-yl)sulfonyl-2-methylspiro[5,6-dihydropyrano[3,4-d]pyrimidine-8,3'-piperidine] —— C18H25N5O3S
(8S)-1'-(1-ethyl-5-methylpyrazol-4-yl)sulfonyl-2-methylspiro[5,6-dihydropyrano[3,4-d]pyrimidine-8,3'-piperidine]
—— 8-ethyl-3-[(1S,11S)-3,10,12-triazatetracyclo[10.3.1.02,10.04,9]hexadeca-2,4,6,8-tetraen-11-yl]-1H-quinolin-2-one —— C24H24N4O
8-ethyl-3-[(1S,11S)-3,10,12-triazatetracyclo[10.3.1.02,10.04,9]hexadeca-2,4,6,8-tetraen-11-yl]-1H-quinolin-2-one
—— (8R)-1'-ethylsulfonyl-2-methylspiro[5,6-dihydropyrano[3,4-d]pyrimidine-8,3'-piperidine] —— C14H21N3O3S
(8R)-1'-ethylsulfonyl-2-methylspiro[5,6-dihydropyrano[3,4-d]pyrimidine-8,3'-piperidine]
—— 8-[[4-[(3R)-3-methylpiperidin-1-yl]anilino]methyl]-3,6-dihydro-2H-[1,4]dioxino[2,3-g]quinolin-7-one —— C24H27N3O3
8-[[4-[(3R)-3-methylpiperidin-1-yl]anilino]methyl]-3,6-dihydro-2H-[1,4]dioxino[2,3-g]quinolin-7-one
—— 8-[2-[(2S,6R)-2,6-dimethylpiperidin-1-yl]-2-oxoethyl]-10-phenyl-3,6,8,10,11-pentazatricyclo[7.3.0.02,6]dodeca-1(9),2,11-trien-7-one —— C22H26N6O2
8-[2-[(2S,6R)-2,6-dimethylpiperidin-1-yl]-2-oxoethyl]-10-phenyl-3,6,8,10,11-pentazatricyclo[7.3.0.02,6]dodeca-1(9),2,11-trien-7-one
—— 8-[2-[(2S,6S)-2,6-dimethylpiperidin-1-yl]-2-oxoethyl]-10-(4-fluorophenyl)-3,6,8,10,11-pentazatricyclo[7.3.0.02,6]dodeca-1(9),2,11-trien-7-one —— C22H25FN6O2
8-[2-[(2S,6S)-2,6-dimethylpiperidin-1-yl]-2-oxoethyl]-10-(4-fluorophenyl)-3,6,8,10,11-pentazatricyclo[7.3.0.02,6]dodeca-1(9),2,11-trien-7-one
—— 8-[2-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-2-oxoethyl]-10-phenyl-3,6,8,10,11-pentazatricyclo[7.3.0.02,6]dodeca-1(9),2,11-trien-7-one —— C21H24N6O3
8-[2-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-2-oxoethyl]-10-phenyl-3,6,8,10,11-pentazatricyclo[7.3.0.02,6]dodeca-1(9),2,11-trien-7-one
—— (8S)-2-propan-2-yl-1'-pyrrolidin-1-ylsulfonylspiro[5,6-dihydropyrano[3,4-d]pyrimidine-8,3'-piperidine] —— C18H28N4O3S
(8S)-2-propan-2-yl-1'-pyrrolidin-1-ylsulfonylspiro[5,6-dihydropyrano[3,4-d]pyrimidine-8,3'-piperidine]