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中文名称 英文名称 CAS号 化学式 结构式图片
—— (8R)-2-(dimethylamino)-8-[3-[(dimethylamino)methyl]-4-methoxyphenyl]-4,5,7,8-tetrahydro-[1,3]thiazolo[4,5-c]azepin-6-one —— C19H26N4O2S
(8R)-2-(dimethylamino)-8-[3-[(dimethylamino)methyl]-4-methoxyphenyl]-4,5,7,8-tetrahydro-[1,3]thiazolo[4,5-c]azepin-6-one
—— (8R)-2-amino-8-[4-(3-hydroxyprop-1-ynyl)thiophen-2-yl]-4,5,7,8-tetrahydro-[1,3]thiazolo[4,5-c]azepin-6-one —— C14H13N3O2S2
(8R)-2-amino-8-[4-(3-hydroxyprop-1-ynyl)thiophen-2-yl]-4,5,7,8-tetrahydro-[1,3]thiazolo[4,5-c]azepin-6-one
—— (8S,8aS)-2-ethyl-8-(2-fluorophenyl)-6-imino-3,5,8,8a-tetrahydro-1H-isoquinoline-5,7,7-tricarbonitrile —— C20H18FN5
(8S,8aS)-2-ethyl-8-(2-fluorophenyl)-6-imino-3,5,8,8a-tetrahydro-1H-isoquinoline-5,7,7-tricarbonitrile
—— (8S)-8-(2,1,3-benzothiadiazol-4-yl)-2-pyrrolidin-1-yl-4,5,7,8-tetrahydro-[1,3]thiazolo[4,5-c]azepin-6-one —— C17H17N5OS2
(8S)-8-(2,1,3-benzothiadiazol-4-yl)-2-pyrrolidin-1-yl-4,5,7,8-tetrahydro-[1,3]thiazolo[4,5-c]azepin-6-one
—— (8S)-1-methyl-8-[3-(pyrazol-1-ylmethyl)phenyl]-7,8-dihydro-5H-[1,3]oxazolo[4,5-g]quinoline-2,6-dione —— C21H18N4O3
(8S)-1-methyl-8-[3-(pyrazol-1-ylmethyl)phenyl]-7,8-dihydro-5H-[1,3]oxazolo[4,5-g]quinoline-2,6-dione
—— (8S,8aR)-2-ethyl-8-(2-fluorophenyl)-6-imino-3,5,8,8a-tetrahydro-1H-isoquinoline-5,7,7-tricarbonitrile —— C20H18FN5
(8S,8aR)-2-ethyl-8-(2-fluorophenyl)-6-imino-3,5,8,8a-tetrahydro-1H-isoquinoline-5,7,7-tricarbonitrile
—— (8R,8aS)-6-imino-2-methyl-8-naphthalen-1-yl-1,2,3,5,8,8a-hexahydroisoquinolin-2-ium-5,7,7-tricarbonitrile —— C23H20N5+
(8R,8aS)-6-imino-2-methyl-8-naphthalen-1-yl-1,2,3,5,8,8a-hexahydroisoquinolin-2-ium-5,7,7-tricarbonitrile
—— (8R,8aR)-6-imino-2-methyl-8-naphthalen-1-yl-1,2,3,5,8,8a-hexahydroisoquinolin-2-ium-5,7,7-tricarbonitrile —— C23H20N5+
(8R,8aR)-6-imino-2-methyl-8-naphthalen-1-yl-1,2,3,5,8,8a-hexahydroisoquinolin-2-ium-5,7,7-tricarbonitrile
—— 8-[4-[(1S)-1-morpholin-4-ylethyl]phenyl]quinolin-4-amine —— C21H23N3O
8-[4-[(1S)-1-morpholin-4-ylethyl]phenyl]quinolin-4-amine
—— 8-[4-[(1R)-1-morpholin-4-ylethyl]phenyl]quinolin-4-amine —— C21H23N3O
8-[4-[(1R)-1-morpholin-4-ylethyl]phenyl]quinolin-4-amine
—— 8-(Azepan-1-ium-1-ylmethyl)-3-(3,4-dimethoxyphenyl)-7-hydroxy-4-methylchromen-2-one —— C25H30NO5+
8-(Azepan-1-ium-1-ylmethyl)-3-(3,4-dimethoxyphenyl)-7-hydroxy-4-methylchromen-2-one
—— 8-[(4-Ethylpiperazine-1,4-diium-1-yl)methyl]-7-hydroxy-3-phenylchromen-2-one —— C22H26N2O3+2
8-[(4-Ethylpiperazine-1,4-diium-1-yl)methyl]-7-hydroxy-3-phenylchromen-2-one
—— (8R)-3-methyl-8-(2,3,4-trimethoxyphenyl)-7,8-dihydro-5H-[1,3]oxazolo[5,4-g]quinoline-2,6-dione —— C20H20N2O6
(8R)-3-methyl-8-(2,3,4-trimethoxyphenyl)-7,8-dihydro-5H-[1,3]oxazolo[5,4-g]quinoline-2,6-dione
—— (8S)-3-methyl-8-(2,3,4-trimethoxyphenyl)-7,8-dihydro-5H-[1,3]oxazolo[5,4-g]quinoline-2,6-dione —— C20H20N2O6
(8S)-3-methyl-8-(2,3,4-trimethoxyphenyl)-7,8-dihydro-5H-[1,3]oxazolo[5,4-g]quinoline-2,6-dione
—— (8S)-2-amino-8-[3-(2-methylphenyl)phenyl]-4,5,7,8-tetrahydro-[1,3]thiazolo[4,5-c]azepin-6-one —— C20H19N3OS
(8S)-2-amino-8-[3-(2-methylphenyl)phenyl]-4,5,7,8-tetrahydro-[1,3]thiazolo[4,5-c]azepin-6-one
—— (8R)-2-amino-8-[3-(2-methylphenyl)phenyl]-4,5,7,8-tetrahydro-[1,3]thiazolo[4,5-c]azepin-6-one —— C20H19N3OS
(8R)-2-amino-8-[3-(2-methylphenyl)phenyl]-4,5,7,8-tetrahydro-[1,3]thiazolo[4,5-c]azepin-6-one
—— (8S)-2-amino-8-[5-(piperidin-1-ylmethyl)thiophen-2-yl]-4,5,7,8-tetrahydro-[1,3]thiazolo[4,5-c]azepin-6-one —— C17H22N4OS2
(8S)-2-amino-8-[5-(piperidin-1-ylmethyl)thiophen-2-yl]-4,5,7,8-tetrahydro-[1,3]thiazolo[4,5-c]azepin-6-one
—— (8R)-2-amino-8-[5-(piperidin-1-ylmethyl)thiophen-2-yl]-4,5,7,8-tetrahydro-[1,3]thiazolo[4,5-c]azepin-6-one —— C17H22N4OS2
(8R)-2-amino-8-[5-(piperidin-1-ylmethyl)thiophen-2-yl]-4,5,7,8-tetrahydro-[1,3]thiazolo[4,5-c]azepin-6-one
—— (8S)-2-amino-8-(2-chloro-4-fluorophenyl)-4,5,7,8-tetrahydro-[1,3]thiazolo[4,5-c]azepin-6-one —— C13H11ClFN3OS
(8S)-2-amino-8-(2-chloro-4-fluorophenyl)-4,5,7,8-tetrahydro-[1,3]thiazolo[4,5-c]azepin-6-one
—— (8R)-2-amino-8-(2-chloro-4-fluorophenyl)-4,5,7,8-tetrahydro-[1,3]thiazolo[4,5-c]azepin-6-one —— C13H11ClFN3OS
(8R)-2-amino-8-(2-chloro-4-fluorophenyl)-4,5,7,8-tetrahydro-[1,3]thiazolo[4,5-c]azepin-6-one
—— 8-[3-cyclopropyl-5-[(1R)-1-pyrazol-1-ylpropyl]-1,2,4-triazol-1-yl]quinoline —— C20H20N6
8-[3-cyclopropyl-5-[(1R)-1-pyrazol-1-ylpropyl]-1,2,4-triazol-1-yl]quinoline
—— (8R)-2-(dimethylamino)-8-[2-(2-methylphenyl)pyrimidin-5-yl]-4,5,7,8-tetrahydro-[1,3]thiazolo[4,5-c]azepin-6-one —— C20H21N5OS
(8R)-2-(dimethylamino)-8-[2-(2-methylphenyl)pyrimidin-5-yl]-4,5,7,8-tetrahydro-[1,3]thiazolo[4,5-c]azepin-6-one
—— 8-[3-cyclopropyl-5-[(1S)-1-pyrazol-1-ylpropyl]-1,2,4-triazol-1-yl]quinoline —— C20H20N6
8-[3-cyclopropyl-5-[(1S)-1-pyrazol-1-ylpropyl]-1,2,4-triazol-1-yl]quinoline
—— (8R)-8-(4-tert-butylphenyl)-2-morpholin-4-yl-4,5,7,8-tetrahydro-[1,3]thiazolo[4,5-c]azepin-6-one —— C21H27N3O2S
(8R)-8-(4-tert-butylphenyl)-2-morpholin-4-yl-4,5,7,8-tetrahydro-[1,3]thiazolo[4,5-c]azepin-6-one
—— (8S)-8-(4-tert-butylphenyl)-2-morpholin-4-yl-4,5,7,8-tetrahydro-[1,3]thiazolo[4,5-c]azepin-6-one —— C21H27N3O2S
(8S)-8-(4-tert-butylphenyl)-2-morpholin-4-yl-4,5,7,8-tetrahydro-[1,3]thiazolo[4,5-c]azepin-6-one
—— (8S)-8-(4-hydroxy-3,5-dimethylphenyl)-2-morpholin-4-yl-4,5,7,8-tetrahydro-[1,3]thiazolo[4,5-c]azepin-6-one —— C19H23N3O3S
(8S)-8-(4-hydroxy-3,5-dimethylphenyl)-2-morpholin-4-yl-4,5,7,8-tetrahydro-[1,3]thiazolo[4,5-c]azepin-6-one
—— (8R)-8-(4-hydroxy-3,5-dimethylphenyl)-2-morpholin-4-yl-4,5,7,8-tetrahydro-[1,3]thiazolo[4,5-c]azepin-6-one —— C19H23N3O3S
(8R)-8-(4-hydroxy-3,5-dimethylphenyl)-2-morpholin-4-yl-4,5,7,8-tetrahydro-[1,3]thiazolo[4,5-c]azepin-6-one
—— 8-Chloro-4-(4-phenylpiperazin-1-yl)-2-(trifluoromethyl)quinolin-1-ium —— C20H18ClF3N3+
8-Chloro-4-(4-phenylpiperazin-1-yl)-2-(trifluoromethyl)quinolin-1-ium
—— (8S)-8-(2-methoxypyridin-3-yl)-3-methyl-7,8-dihydro-5H-[1,3]oxazolo[5,4-g]quinoline-2,6-dione —— C17H15N3O4
(8S)-8-(2-methoxypyridin-3-yl)-3-methyl-7,8-dihydro-5H-[1,3]oxazolo[5,4-g]quinoline-2,6-dione
—— (8S)-2-amino-8-(2,1,3-benzothiadiazol-4-yl)-4,5,7,8-tetrahydro-[1,3]thiazolo[4,5-c]azepin-6-one —— C13H11N5OS2
(8S)-2-amino-8-(2,1,3-benzothiadiazol-4-yl)-4,5,7,8-tetrahydro-[1,3]thiazolo[4,5-c]azepin-6-one
—— (8R)-8-(2-methoxypyridin-3-yl)-3-methyl-7,8-dihydro-5H-[1,3]oxazolo[5,4-g]quinoline-2,6-dione —— C17H15N3O4
(8R)-8-(2-methoxypyridin-3-yl)-3-methyl-7,8-dihydro-5H-[1,3]oxazolo[5,4-g]quinoline-2,6-dione
—— (8S)-8-(2-ethylsulfanylpyrimidin-5-yl)-2-morpholin-4-yl-4,5,7,8-tetrahydro-[1,3]thiazolo[4,5-c]azepin-6-one —— C17H21N5O2S2
(8S)-8-(2-ethylsulfanylpyrimidin-5-yl)-2-morpholin-4-yl-4,5,7,8-tetrahydro-[1,3]thiazolo[4,5-c]azepin-6-one
—— (8R)-2-amino-8-(2,1,3-benzothiadiazol-4-yl)-4,5,7,8-tetrahydro-[1,3]thiazolo[4,5-c]azepin-6-one —— C13H11N5OS2
(8R)-2-amino-8-(2,1,3-benzothiadiazol-4-yl)-4,5,7,8-tetrahydro-[1,3]thiazolo[4,5-c]azepin-6-one
—— (8R)-8-(2-ethylsulfanylpyrimidin-5-yl)-2-morpholin-4-yl-4,5,7,8-tetrahydro-[1,3]thiazolo[4,5-c]azepin-6-one —— C17H21N5O2S2
(8R)-8-(2-ethylsulfanylpyrimidin-5-yl)-2-morpholin-4-yl-4,5,7,8-tetrahydro-[1,3]thiazolo[4,5-c]azepin-6-one
—— (8R)-8-(3-chloro-5-fluoro-4-methoxyphenyl)-1,5,7,8-tetrahydro-[1,3]oxazolo[4,5-g]quinoline-2,6-dione —— C17H12ClFN2O4
(8R)-8-(3-chloro-5-fluoro-4-methoxyphenyl)-1,5,7,8-tetrahydro-[1,3]oxazolo[4,5-g]quinoline-2,6-dione
—— (8S)-8-(3-chloro-5-fluoro-4-methoxyphenyl)-1,5,7,8-tetrahydro-[1,3]oxazolo[4,5-g]quinoline-2,6-dione —— C17H12ClFN2O4
(8S)-8-(3-chloro-5-fluoro-4-methoxyphenyl)-1,5,7,8-tetrahydro-[1,3]oxazolo[4,5-g]quinoline-2,6-dione
—— (8S)-2-amino-8-[3-(4-methoxyphenoxy)phenyl]-4,5,7,8-tetrahydro-[1,3]thiazolo[4,5-c]azepin-6-one —— C20H19N3O3S
(8S)-2-amino-8-[3-(4-methoxyphenoxy)phenyl]-4,5,7,8-tetrahydro-[1,3]thiazolo[4,5-c]azepin-6-one
—— (8R)-2-amino-8-(3-chloro-4-propoxyphenyl)-4,5,7,8-tetrahydro-[1,3]thiazolo[4,5-c]azepin-6-one —— C16H18ClN3O2S
(8R)-2-amino-8-(3-chloro-4-propoxyphenyl)-4,5,7,8-tetrahydro-[1,3]thiazolo[4,5-c]azepin-6-one
—— (8S)-2-amino-8-(3-chloro-4-propoxyphenyl)-4,5,7,8-tetrahydro-[1,3]thiazolo[4,5-c]azepin-6-one —— C16H18ClN3O2S
(8S)-2-amino-8-(3-chloro-4-propoxyphenyl)-4,5,7,8-tetrahydro-[1,3]thiazolo[4,5-c]azepin-6-one
—— (8R)-2-amino-8-[3-(4-methoxyphenoxy)phenyl]-4,5,7,8-tetrahydro-[1,3]thiazolo[4,5-c]azepin-6-one —— C20H19N3O3S
(8R)-2-amino-8-[3-(4-methoxyphenoxy)phenyl]-4,5,7,8-tetrahydro-[1,3]thiazolo[4,5-c]azepin-6-one
—— (8S)-8-(2-cyclopentyloxyphenyl)-2-(dimethylamino)-4,5,7,8-tetrahydro-[1,3]thiazolo[4,5-c]azepin-6-one —— C20H25N3O2S
(8S)-8-(2-cyclopentyloxyphenyl)-2-(dimethylamino)-4,5,7,8-tetrahydro-[1,3]thiazolo[4,5-c]azepin-6-one
—— (8R)-8-(2-cyclopentyloxyphenyl)-2-(dimethylamino)-4,5,7,8-tetrahydro-[1,3]thiazolo[4,5-c]azepin-6-one —— C20H25N3O2S
(8R)-8-(2-cyclopentyloxyphenyl)-2-(dimethylamino)-4,5,7,8-tetrahydro-[1,3]thiazolo[4,5-c]azepin-6-one
—— (8S)-2-amino-8-(2-methyl-4-pyrazol-1-ylphenyl)-4,5,7,8-tetrahydro-[1,3]thiazolo[4,5-c]azepin-6-one —— C17H17N5OS
(8S)-2-amino-8-(2-methyl-4-pyrazol-1-ylphenyl)-4,5,7,8-tetrahydro-[1,3]thiazolo[4,5-c]azepin-6-one
—— [8-methyl-2-[4-[(1R)-1-morpholin-4-ylethyl]phenyl]quinolin-3-yl]methanol —— C23H26N2O2
[8-methyl-2-[4-[(1R)-1-morpholin-4-ylethyl]phenyl]quinolin-3-yl]methanol
—— (8R)-3-methyl-8-(2-propan-2-ylpyrimidin-4-yl)-7,8-dihydro-5H-[1,3]oxazolo[5,4-g]quinoline-2,6-dione —— C18H18N4O3
(8R)-3-methyl-8-(2-propan-2-ylpyrimidin-4-yl)-7,8-dihydro-5H-[1,3]oxazolo[5,4-g]quinoline-2,6-dione
—— (8R)-2-amino-8-(2-methyl-4-pyrazol-1-ylphenyl)-4,5,7,8-tetrahydro-[1,3]thiazolo[4,5-c]azepin-6-one —— C17H17N5OS
(8R)-2-amino-8-(2-methyl-4-pyrazol-1-ylphenyl)-4,5,7,8-tetrahydro-[1,3]thiazolo[4,5-c]azepin-6-one
—— (8S)-3-methyl-8-(2-propan-2-ylpyrimidin-4-yl)-7,8-dihydro-5H-[1,3]oxazolo[5,4-g]quinoline-2,6-dione —— C18H18N4O3
(8S)-3-methyl-8-(2-propan-2-ylpyrimidin-4-yl)-7,8-dihydro-5H-[1,3]oxazolo[5,4-g]quinoline-2,6-dione
—— [8-methyl-2-[4-[(1S)-1-morpholin-4-ylethyl]phenyl]quinolin-3-yl]methanol —— C23H26N2O2
[8-methyl-2-[4-[(1S)-1-morpholin-4-ylethyl]phenyl]quinolin-3-yl]methanol
—— (8-chloroquinolin-2-yl)-[(2S)-2-(3-methyl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]methanone —— C17H15ClN4O2
(8-chloroquinolin-2-yl)-[(2S)-2-(3-methyl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]methanone
—— (8R)-8-[2-(methoxymethyl)pyrimidin-5-yl]-2-morpholin-4-yl-4,5,7,8-tetrahydro-[1,3]thiazolo[4,5-c]azepin-6-one —— C17H21N5O3S
(8R)-8-[2-(methoxymethyl)pyrimidin-5-yl]-2-morpholin-4-yl-4,5,7,8-tetrahydro-[1,3]thiazolo[4,5-c]azepin-6-one