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—— 8-(1H-imidazol-2-ylmethyl)-3-[(2S)-2-phenylpropyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one —— C20H26N4O2
8-(1H-imidazol-2-ylmethyl)-3-[(2S)-2-phenylpropyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
—— 8-(1H-imidazol-2-ylmethyl)-3-[(2R)-2-phenylpropyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one —— C20H26N4O2
8-(1H-imidazol-2-ylmethyl)-3-[(2R)-2-phenylpropyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
—— 8-[(2R)-1-imidazol-1-ylpropan-2-yl]-3-(2-phenoxyethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one —— C21H28N4O3
8-[(2R)-1-imidazol-1-ylpropan-2-yl]-3-(2-phenoxyethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
—— 8-[5-(hydroxymethyl)furan-2-carbonyl]-3-[(2S)-pentan-2-yl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one —— C18H26N2O5
8-[5-(hydroxymethyl)furan-2-carbonyl]-3-[(2S)-pentan-2-yl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
—— 8-[5-(hydroxymethyl)furan-2-carbonyl]-3-[(2R)-pentan-2-yl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one —— C18H26N2O5
8-[5-(hydroxymethyl)furan-2-carbonyl]-3-[(2R)-pentan-2-yl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
—— 8-(6-aminopyridine-3-carbonyl)-3-[(2S)-pentan-2-yl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one —— C18H26N4O3
8-(6-aminopyridine-3-carbonyl)-3-[(2S)-pentan-2-yl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
—— 8-(6-aminopyridine-3-carbonyl)-3-[(2R)-pentan-2-yl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one —— C18H26N4O3
8-(6-aminopyridine-3-carbonyl)-3-[(2R)-pentan-2-yl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
—— 8-[(3S)-oxan-3-yl]-3-(2-phenoxyethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one —— C20H28N2O4
8-[(3S)-oxan-3-yl]-3-(2-phenoxyethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
—— 8-[(3R)-oxan-3-yl]-3-(2-phenoxyethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one —— C20H28N2O4
8-[(3R)-oxan-3-yl]-3-(2-phenoxyethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
—— 8-(2-methyl-6-oxo-1H-pyrimidine-5-carbonyl)-3-[(2S)-pentan-2-yl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one —— C18H26N4O4
8-(2-methyl-6-oxo-1H-pyrimidine-5-carbonyl)-3-[(2S)-pentan-2-yl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
—— 8-[(2S)-2-(2-chloro-4-fluorophenoxy)propanoyl]-2-ethyl-2,8-diazaspiro[4.5]decan-3-one —— C19H24ClFN2O3
8-[(2S)-2-(2-chloro-4-fluorophenoxy)propanoyl]-2-ethyl-2,8-diazaspiro[4.5]decan-3-one
—— 8-[(2-aminopyridin-3-yl)methyl]-3-[3-[(3S)-3-(dimethylamino)pyrrolidin-1-yl]propyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one —— C22H36N6O2
8-[(2-aminopyridin-3-yl)methyl]-3-[3-[(3S)-3-(dimethylamino)pyrrolidin-1-yl]propyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
—— 8-(2-methyl-6-oxo-1H-pyrimidine-5-carbonyl)-3-[(2R)-pentan-2-yl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one —— C18H26N4O4
8-(2-methyl-6-oxo-1H-pyrimidine-5-carbonyl)-3-[(2R)-pentan-2-yl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
—— 8-[(2-aminopyridin-3-yl)methyl]-3-[3-[(3R)-3-(dimethylamino)pyrrolidin-1-yl]propyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one —— C22H36N6O2
8-[(2-aminopyridin-3-yl)methyl]-3-[3-[(3R)-3-(dimethylamino)pyrrolidin-1-yl]propyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
—— 8-[(2R)-2-(2-chloro-4-fluorophenoxy)propanoyl]-2-ethyl-2,8-diazaspiro[4.5]decan-3-one —— C19H24ClFN2O3
8-[(2R)-2-(2-chloro-4-fluorophenoxy)propanoyl]-2-ethyl-2,8-diazaspiro[4.5]decan-3-one
—— 8-(2-amino-6-propan-2-ylpyrimidine-4-carbonyl)-3-[(2S)-pentan-2-yl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one —— C20H31N5O3
8-(2-amino-6-propan-2-ylpyrimidine-4-carbonyl)-3-[(2S)-pentan-2-yl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
—— 8-(2-amino-6-propan-2-ylpyrimidine-4-carbonyl)-3-[(2R)-pentan-2-yl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one —— C20H31N5O3
8-(2-amino-6-propan-2-ylpyrimidine-4-carbonyl)-3-[(2R)-pentan-2-yl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
—— 8-[5-methylsulfonyl-4-[(3S)-piperidin-3-yl]pyrimidin-2-yl]-2,8-diazaspiro[4.5]decan-3-one —— C18H27N5O3S
8-[5-methylsulfonyl-4-[(3S)-piperidin-3-yl]pyrimidin-2-yl]-2,8-diazaspiro[4.5]decan-3-one
—— 8-[(2S)-4-hydroxy-4-methylpentan-2-yl]-3-(2-phenoxyethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one —— C21H32N2O4
8-[(2S)-4-hydroxy-4-methylpentan-2-yl]-3-(2-phenoxyethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
—— 8-[(2R)-4-hydroxy-4-methylpentan-2-yl]-3-(2-phenoxyethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one —— C21H32N2O4
8-[(2R)-4-hydroxy-4-methylpentan-2-yl]-3-(2-phenoxyethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
—— 8-[5-methylsulfonyl-4-[(3R)-piperidin-3-yl]pyrimidin-2-yl]-2,8-diazaspiro[4.5]decan-3-one —— C18H27N5O3S
8-[5-methylsulfonyl-4-[(3R)-piperidin-3-yl]pyrimidin-2-yl]-2,8-diazaspiro[4.5]decan-3-one
—— (8R)-2-(2,3-dihydro-1,4-benzodioxin-6-ylmethylsulfanyl)-8-methyl-6,7,8,9-tetrahydro-[1,2,4]triazolo[1,5-a]quinazoline —— C19H20N4O2S
(8R)-2-(2,3-dihydro-1,4-benzodioxin-6-ylmethylsulfanyl)-8-methyl-6,7,8,9-tetrahydro-[1,2,4]triazolo[1,5-a]quinazoline
—— 8-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-2-[(1R,2R,3S)-2,3-dimethylcyclohexyl]pyrido[4,3-b][1,6]naphthyridine-1,9-dione —— C28H29N3O4
8-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-2-[(1R,2R,3S)-2,3-dimethylcyclohexyl]pyrido[4,3-b][1,6]naphthyridine-1,9-dione
—— 8-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-2-[(1S,2R,3S)-2,3-dimethylcyclohexyl]pyrido[4,3-b][1,6]naphthyridine-1,9-dione —— C28H29N3O4
8-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-2-[(1S,2R,3S)-2,3-dimethylcyclohexyl]pyrido[4,3-b][1,6]naphthyridine-1,9-dione
—— 8-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-2-[(1S,2S)-2-methylcyclohexyl]pyrido[4,3-b][1,6]naphthyridine-1,9-dione —— C27H27N3O4
8-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-2-[(1S,2S)-2-methylcyclohexyl]pyrido[4,3-b][1,6]naphthyridine-1,9-dione
—— 8-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-2-[(1R,2R,3R)-2,3-dimethylcyclohexyl]pyrido[4,3-b][1,6]naphthyridine-1,9-dione —— C28H29N3O4
8-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-2-[(1R,2R,3R)-2,3-dimethylcyclohexyl]pyrido[4,3-b][1,6]naphthyridine-1,9-dione
—— 8-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-2-[(1S,2R)-2-methylcyclohexyl]pyrido[4,3-b][1,6]naphthyridine-1,9-dione —— C27H27N3O4
8-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-2-[(1S,2R)-2-methylcyclohexyl]pyrido[4,3-b][1,6]naphthyridine-1,9-dione
—— 8-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-2-[(1R,2R)-2-methylcyclohexyl]pyrido[4,3-b][1,6]naphthyridine-1,9-dione —— C27H27N3O4
8-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-2-[(1R,2R)-2-methylcyclohexyl]pyrido[4,3-b][1,6]naphthyridine-1,9-dione
—— 8-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-2-[(1S,2R,3R)-2,3-dimethylcyclohexyl]pyrido[4,3-b][1,6]naphthyridine-1,9-dione —— C28H29N3O4
8-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-2-[(1S,2R,3R)-2,3-dimethylcyclohexyl]pyrido[4,3-b][1,6]naphthyridine-1,9-dione
—— 8-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-2-[(1R,2S)-2-methylcyclohexyl]pyrido[4,3-b][1,6]naphthyridine-1,9-dione —— C27H27N3O4
8-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-2-[(1R,2S)-2-methylcyclohexyl]pyrido[4,3-b][1,6]naphthyridine-1,9-dione
—— 8-(2-hydroxy-3-methoxybenzoyl)-3-[(2R)-pentan-2-yl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one —— C20H28N2O5
8-(2-hydroxy-3-methoxybenzoyl)-3-[(2R)-pentan-2-yl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
—— 8-(2-hydroxy-3-methoxybenzoyl)-3-[(2S)-pentan-2-yl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one —— C20H28N2O5
8-(2-hydroxy-3-methoxybenzoyl)-3-[(2S)-pentan-2-yl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
—— 8-[(3S)-oxan-3-yl]-3-(2-phenylethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one —— C20H28N2O3
8-[(3S)-oxan-3-yl]-3-(2-phenylethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
—— 8-[(3R)-oxan-3-yl]-3-(2-phenylethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one —— C20H28N2O3
8-[(3R)-oxan-3-yl]-3-(2-phenylethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
—— 8-[(3-methylimidazo[1,5-a]pyridin-1-yl)methyl]-3-[(2S)-2-phenylpropyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one —— C25H30N4O2
8-[(3-methylimidazo[1,5-a]pyridin-1-yl)methyl]-3-[(2S)-2-phenylpropyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
—— 8-[(3-methylimidazo[1,5-a]pyridin-1-yl)methyl]-3-[(2R)-2-phenylpropyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one —— C25H30N4O2
8-[(3-methylimidazo[1,5-a]pyridin-1-yl)methyl]-3-[(2R)-2-phenylpropyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
—— (8R)-2-(2-methoxyethylsulfanyl)-8-(2-methoxyphenyl)-8,9-dihydro-7H-[1,2,4]triazolo[1,5-a]quinazolin-6-one —— C19H20N4O3S
(8R)-2-(2-methoxyethylsulfanyl)-8-(2-methoxyphenyl)-8,9-dihydro-7H-[1,2,4]triazolo[1,5-a]quinazolin-6-one
—— (8S)-8-(3-chlorophenyl)-8,9-dihydro-7H-[1,2,4]triazolo[1,5-a]quinazolin-6-one —— C15H11ClN4O
(8S)-8-(3-chlorophenyl)-8,9-dihydro-7H-[1,2,4]triazolo[1,5-a]quinazolin-6-one
—— (8R)-8-(3-chlorophenyl)-2-(methoxymethyl)-8,9-dihydro-7H-[1,2,4]triazolo[1,5-a]quinazolin-6-one —— C17H15ClN4O2
(8R)-8-(3-chlorophenyl)-2-(methoxymethyl)-8,9-dihydro-7H-[1,2,4]triazolo[1,5-a]quinazolin-6-one
—— (8R)-8-(3-methylphenyl)-2-pyridin-4-yl-8,9-dihydro-7H-[1,2,4]triazolo[1,5-a]quinazolin-6-one —— C21H17N5O
(8R)-8-(3-methylphenyl)-2-pyridin-4-yl-8,9-dihydro-7H-[1,2,4]triazolo[1,5-a]quinazolin-6-one
—— (8S)-8-(2-methylphenyl)-2-[(3-nitrophenyl)methylsulfanyl]-8,9-dihydro-7H-[1,2,4]triazolo[1,5-a]quinazolin-6-one —— C23H19N5O3S
(8S)-8-(2-methylphenyl)-2-[(3-nitrophenyl)methylsulfanyl]-8,9-dihydro-7H-[1,2,4]triazolo[1,5-a]quinazolin-6-one
—— (8S)-8-(3-methylphenyl)-2-[(3-methylphenyl)methylsulfanyl]-8,9-dihydro-7H-[1,2,4]triazolo[1,5-a]quinazolin-6-one —— C24H22N4OS
(8S)-8-(3-methylphenyl)-2-[(3-methylphenyl)methylsulfanyl]-8,9-dihydro-7H-[1,2,4]triazolo[1,5-a]quinazolin-6-one
—— (8R)-3-acetyl-8-(2-methoxyphenyl)-2-methyl-8,9-dihydro-7H-pyrazolo[1,5-a]quinazolin-6-one —— C20H19N3O3
(8R)-3-acetyl-8-(2-methoxyphenyl)-2-methyl-8,9-dihydro-7H-pyrazolo[1,5-a]quinazolin-6-one
—— (8R)-2-(4-methoxyphenyl)-8-(3-methylphenyl)-8,9-dihydro-7H-[1,2,4]triazolo[1,5-a]quinazolin-6-one —— C23H20N4O2
(8R)-2-(4-methoxyphenyl)-8-(3-methylphenyl)-8,9-dihydro-7H-[1,2,4]triazolo[1,5-a]quinazolin-6-one
—— (8S)-2-methyl-8-(2-methylphenyl)-8,9-dihydro-7H-pyrazolo[1,5-a]quinazolin-6-one —— C18H17N3O
(8S)-2-methyl-8-(2-methylphenyl)-8,9-dihydro-7H-pyrazolo[1,5-a]quinazolin-6-one
—— (8R)-8-(3-chlorophenyl)-2-ethylsulfanyl-8,9-dihydro-7H-[1,2,4]triazolo[1,5-a]quinazolin-6-one —— C17H15ClN4OS
(8R)-8-(3-chlorophenyl)-2-ethylsulfanyl-8,9-dihydro-7H-[1,2,4]triazolo[1,5-a]quinazolin-6-one
—— (8S)-8-(3-methylphenyl)-2-phenyl-8,9-dihydro-7H-[1,2,4]triazolo[1,5-a]quinazolin-6-one —— C22H18N4O
(8S)-8-(3-methylphenyl)-2-phenyl-8,9-dihydro-7H-[1,2,4]triazolo[1,5-a]quinazolin-6-one
—— (8S)-8-(2-methoxyphenyl)-2-methylsulfanyl-8,9-dihydro-7H-[1,2,4]triazolo[1,5-a]quinazolin-6-one —— C17H16N4O2S
(8S)-8-(2-methoxyphenyl)-2-methylsulfanyl-8,9-dihydro-7H-[1,2,4]triazolo[1,5-a]quinazolin-6-one
—— (8S)-8-(2-methoxyphenyl)-2-pyridin-3-yl-8,9-dihydro-7H-[1,2,4]triazolo[1,5-a]quinazolin-6-one —— C21H17N5O2
(8S)-8-(2-methoxyphenyl)-2-pyridin-3-yl-8,9-dihydro-7H-[1,2,4]triazolo[1,5-a]quinazolin-6-one
—— (8R)-2-cyclohexyl-8-(2-methylphenyl)-8,9-dihydro-7H-[1,2,4]triazolo[1,5-a]quinazolin-6-one —— C22H24N4O
(8R)-2-cyclohexyl-8-(2-methylphenyl)-8,9-dihydro-7H-[1,2,4]triazolo[1,5-a]quinazolin-6-one