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中文名称 英文名称 CAS号 化学式 结构式图片
—— 8-chloro-N-[(1R)-2-methoxy-1-(2-methylpyrazol-3-yl)ethyl]quinoline-2-carboxamide —— C17H17ClN4O2
8-chloro-N-[(1R)-2-methoxy-1-(2-methylpyrazol-3-yl)ethyl]quinoline-2-carboxamide
—— 8-[2-[(1S)-2,3-dihydro-1H-inden-1-yl]acetyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one —— C18H22N2O3
8-[2-[(1S)-2,3-dihydro-1H-inden-1-yl]acetyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
—— (8R)-2-(dimethylamino)-8-[4-(3-hydroxy-3-methylbut-1-ynyl)phenyl]-4,5,7,8-tetrahydro-[1,3]thiazolo[4,5-c]azepin-6-one —— C20H23N3O2S
(8R)-2-(dimethylamino)-8-[4-(3-hydroxy-3-methylbut-1-ynyl)phenyl]-4,5,7,8-tetrahydro-[1,3]thiazolo[4,5-c]azepin-6-one
—— 8-[2-[(1R)-2,3-dihydro-1H-inden-1-yl]acetyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one —— C18H22N2O3
8-[2-[(1R)-2,3-dihydro-1H-inden-1-yl]acetyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
—— (8S)-8-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)-7,8-dihydro-5H-[1,3]dioxolo[4,5-g]quinolin-6-one —— C21H19N3O4
(8S)-8-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)-7,8-dihydro-5H-[1,3]dioxolo[4,5-g]quinolin-6-one
—— (8R)-8-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)-7,8-dihydro-5H-[1,3]dioxolo[4,5-g]quinolin-6-one —— C21H19N3O4
(8R)-8-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)-7,8-dihydro-5H-[1,3]dioxolo[4,5-g]quinolin-6-one
—— (8S)-2-(dimethylamino)-8-[4-(3-hydroxy-3-methylbut-1-ynyl)phenyl]-4,5,7,8-tetrahydro-[1,3]thiazolo[4,5-c]azepin-6-one —— C20H23N3O2S
(8S)-2-(dimethylamino)-8-[4-(3-hydroxy-3-methylbut-1-ynyl)phenyl]-4,5,7,8-tetrahydro-[1,3]thiazolo[4,5-c]azepin-6-one
—— (8S)-2-amino-8-[5-(3-hydroxy-3-methylbut-1-ynyl)thiophen-2-yl]-4,5,7,8-tetrahydro-[1,3]thiazolo[4,5-c]azepin-6-one —— C16H17N3O2S2
(8S)-2-amino-8-[5-(3-hydroxy-3-methylbut-1-ynyl)thiophen-2-yl]-4,5,7,8-tetrahydro-[1,3]thiazolo[4,5-c]azepin-6-one
—— (8R)-2-amino-8-[5-(3-hydroxy-3-methylbut-1-ynyl)thiophen-2-yl]-4,5,7,8-tetrahydro-[1,3]thiazolo[4,5-c]azepin-6-one —— C16H17N3O2S2
(8R)-2-amino-8-[5-(3-hydroxy-3-methylbut-1-ynyl)thiophen-2-yl]-4,5,7,8-tetrahydro-[1,3]thiazolo[4,5-c]azepin-6-one
—— (8R)-3-methyl-8-(5-propylfuran-2-yl)-7,8-dihydro-5H-[1,3]oxazolo[5,4-g]quinoline-2,6-dione —— C18H18N2O4
(8R)-3-methyl-8-(5-propylfuran-2-yl)-7,8-dihydro-5H-[1,3]oxazolo[5,4-g]quinoline-2,6-dione
—— (8S)-3-methyl-8-(5-propylfuran-2-yl)-7,8-dihydro-5H-[1,3]oxazolo[5,4-g]quinoline-2,6-dione —— C18H18N2O4
(8S)-3-methyl-8-(5-propylfuran-2-yl)-7,8-dihydro-5H-[1,3]oxazolo[5,4-g]quinoline-2,6-dione
—— (8S)-2-amino-8-[4-(3,4-dimethylphenoxy)phenyl]-4,5,7,8-tetrahydro-[1,3]thiazolo[4,5-c]azepin-6-one —— C21H21N3O2S
(8S)-2-amino-8-[4-(3,4-dimethylphenoxy)phenyl]-4,5,7,8-tetrahydro-[1,3]thiazolo[4,5-c]azepin-6-one
—— (8R)-2-amino-8-[1-(3-methylphenyl)pyrazol-4-yl]-4,5,7,8-tetrahydro-[1,3]thiazolo[4,5-c]azepin-6-one —— C17H17N5OS
(8R)-2-amino-8-[1-(3-methylphenyl)pyrazol-4-yl]-4,5,7,8-tetrahydro-[1,3]thiazolo[4,5-c]azepin-6-one
—— (8R)-2-amino-8-[4-(3,4-dimethylphenoxy)phenyl]-4,5,7,8-tetrahydro-[1,3]thiazolo[4,5-c]azepin-6-one —— C21H21N3O2S
(8R)-2-amino-8-[4-(3,4-dimethylphenoxy)phenyl]-4,5,7,8-tetrahydro-[1,3]thiazolo[4,5-c]azepin-6-one
—— (8R)-2-amino-8-(2-propoxyphenyl)-4,5,7,8-tetrahydro-[1,3]thiazolo[4,5-c]azepin-6-one —— C16H19N3O2S
(8R)-2-amino-8-(2-propoxyphenyl)-4,5,7,8-tetrahydro-[1,3]thiazolo[4,5-c]azepin-6-one
—— 8-[3-cyclopropyl-5-[(1R)-1-(2-methylimidazol-1-yl)ethyl]-1,2,4-triazol-1-yl]quinoline —— C20H20N6
8-[3-cyclopropyl-5-[(1R)-1-(2-methylimidazol-1-yl)ethyl]-1,2,4-triazol-1-yl]quinoline
—— (8S)-2-amino-8-(2-propoxyphenyl)-4,5,7,8-tetrahydro-[1,3]thiazolo[4,5-c]azepin-6-one —— C16H19N3O2S
(8S)-2-amino-8-(2-propoxyphenyl)-4,5,7,8-tetrahydro-[1,3]thiazolo[4,5-c]azepin-6-one
—— (8S)-8-(3-ethoxyphenyl)-2-pyrrolidin-1-yl-4,5,7,8-tetrahydro-[1,3]thiazolo[4,5-c]azepin-6-one —— C19H23N3O2S
(8S)-8-(3-ethoxyphenyl)-2-pyrrolidin-1-yl-4,5,7,8-tetrahydro-[1,3]thiazolo[4,5-c]azepin-6-one
—— (8S)-2-amino-8-(5-fluoro-2-pyrazol-1-ylphenyl)-4,5,7,8-tetrahydro-[1,3]thiazolo[4,5-c]azepin-6-one —— C16H14FN5OS
(8S)-2-amino-8-(5-fluoro-2-pyrazol-1-ylphenyl)-4,5,7,8-tetrahydro-[1,3]thiazolo[4,5-c]azepin-6-one
—— (8R)-2-amino-8-(5-fluoro-2-pyrazol-1-ylphenyl)-4,5,7,8-tetrahydro-[1,3]thiazolo[4,5-c]azepin-6-one —— C16H14FN5OS
(8R)-2-amino-8-(5-fluoro-2-pyrazol-1-ylphenyl)-4,5,7,8-tetrahydro-[1,3]thiazolo[4,5-c]azepin-6-one
—— 8-[3-cyclopropyl-5-[(1S)-1-(2-methylimidazol-1-yl)ethyl]-1,2,4-triazol-1-yl]quinoline —— C20H20N6
8-[3-cyclopropyl-5-[(1S)-1-(2-methylimidazol-1-yl)ethyl]-1,2,4-triazol-1-yl]quinoline
—— (8R)-2-(dimethylamino)-8-[4-methoxy-3-(methoxymethyl)phenyl]-4,5,7,8-tetrahydro-[1,3]thiazolo[4,5-c]azepin-6-one —— C18H23N3O3S
(8R)-2-(dimethylamino)-8-[4-methoxy-3-(methoxymethyl)phenyl]-4,5,7,8-tetrahydro-[1,3]thiazolo[4,5-c]azepin-6-one
—— (8S)-2-amino-8-[1-(3-methylphenyl)pyrazol-4-yl]-4,5,7,8-tetrahydro-[1,3]thiazolo[4,5-c]azepin-6-one —— C17H17N5OS
(8S)-2-amino-8-[1-(3-methylphenyl)pyrazol-4-yl]-4,5,7,8-tetrahydro-[1,3]thiazolo[4,5-c]azepin-6-one
—— (8R)-8-(3-ethoxyphenyl)-2-pyrrolidin-1-yl-4,5,7,8-tetrahydro-[1,3]thiazolo[4,5-c]azepin-6-one —— C19H23N3O2S
(8R)-8-(3-ethoxyphenyl)-2-pyrrolidin-1-yl-4,5,7,8-tetrahydro-[1,3]thiazolo[4,5-c]azepin-6-one
—— (8S)-2-(dimethylamino)-8-(2-phenylphenyl)-4,5,7,8-tetrahydro-[1,3]thiazolo[4,5-c]azepin-6-one —— C21H21N3OS
(8S)-2-(dimethylamino)-8-(2-phenylphenyl)-4,5,7,8-tetrahydro-[1,3]thiazolo[4,5-c]azepin-6-one
—— (8R)-2-amino-8-[4-ethoxy-3-(hydroxymethyl)phenyl]-4,5,7,8-tetrahydro-[1,3]thiazolo[4,5-c]azepin-6-one —— C16H19N3O3S
(8R)-2-amino-8-[4-ethoxy-3-(hydroxymethyl)phenyl]-4,5,7,8-tetrahydro-[1,3]thiazolo[4,5-c]azepin-6-one
—— (8S)-2-amino-8-[4-ethoxy-3-(hydroxymethyl)phenyl]-4,5,7,8-tetrahydro-[1,3]thiazolo[4,5-c]azepin-6-one —— C16H19N3O3S
(8S)-2-amino-8-[4-ethoxy-3-(hydroxymethyl)phenyl]-4,5,7,8-tetrahydro-[1,3]thiazolo[4,5-c]azepin-6-one
—— (8S)-2-(dimethylamino)-8-[4-methoxy-3-(methoxymethyl)phenyl]-4,5,7,8-tetrahydro-[1,3]thiazolo[4,5-c]azepin-6-one —— C18H23N3O3S
(8S)-2-(dimethylamino)-8-[4-methoxy-3-(methoxymethyl)phenyl]-4,5,7,8-tetrahydro-[1,3]thiazolo[4,5-c]azepin-6-one
—— 8-[(4S)-4,5,6,7-tetrahydro-1H-imidazo[4,5-c]pyridin-4-yl]quinoline —— C15H14N4
8-[(4S)-4,5,6,7-tetrahydro-1H-imidazo[4,5-c]pyridin-4-yl]quinoline
—— 8-[(4R)-4,5,6,7-tetrahydro-1H-imidazo[4,5-c]pyridin-4-yl]quinoline —— C15H14N4
8-[(4R)-4,5,6,7-tetrahydro-1H-imidazo[4,5-c]pyridin-4-yl]quinoline
—— (8R)-2-amino-8-(5-methoxy-2-pyrazol-1-ylphenyl)-4,5,7,8-tetrahydro-[1,3]thiazolo[4,5-c]azepin-6-one —— C17H17N5O2S
(8R)-2-amino-8-(5-methoxy-2-pyrazol-1-ylphenyl)-4,5,7,8-tetrahydro-[1,3]thiazolo[4,5-c]azepin-6-one
—— (8R)-2-amino-8-[5-(1-methylbenzimidazol-2-yl)furan-2-yl]-4,5,7,8-tetrahydro-[1,3]thiazolo[4,5-c]azepin-6-one —— C19H17N5O2S
(8R)-2-amino-8-[5-(1-methylbenzimidazol-2-yl)furan-2-yl]-4,5,7,8-tetrahydro-[1,3]thiazolo[4,5-c]azepin-6-one
—— (8R)-8-isoquinolin-5-yl-2-pyrrolidin-1-yl-4,5,7,8-tetrahydro-[1,3]thiazolo[4,5-c]azepin-6-one —— C20H20N4OS
(8R)-8-isoquinolin-5-yl-2-pyrrolidin-1-yl-4,5,7,8-tetrahydro-[1,3]thiazolo[4,5-c]azepin-6-one
—— (8S)-2-amino-8-(5-methoxy-2-pyrazol-1-ylphenyl)-4,5,7,8-tetrahydro-[1,3]thiazolo[4,5-c]azepin-6-one —— C17H17N5O2S
(8S)-2-amino-8-(5-methoxy-2-pyrazol-1-ylphenyl)-4,5,7,8-tetrahydro-[1,3]thiazolo[4,5-c]azepin-6-one
—— (8S)-2-amino-8-[2-(4-methoxyphenyl)pyrimidin-5-yl]-4,5,7,8-tetrahydro-[1,3]thiazolo[4,5-c]azepin-6-one —— C18H17N5O2S
(8S)-2-amino-8-[2-(4-methoxyphenyl)pyrimidin-5-yl]-4,5,7,8-tetrahydro-[1,3]thiazolo[4,5-c]azepin-6-one
—— (8S)-2-amino-8-[5-(1-methylbenzimidazol-2-yl)furan-2-yl]-4,5,7,8-tetrahydro-[1,3]thiazolo[4,5-c]azepin-6-one —— C19H17N5O2S
(8S)-2-amino-8-[5-(1-methylbenzimidazol-2-yl)furan-2-yl]-4,5,7,8-tetrahydro-[1,3]thiazolo[4,5-c]azepin-6-one
—— (8S)-8-isoquinolin-5-yl-2-pyrrolidin-1-yl-4,5,7,8-tetrahydro-[1,3]thiazolo[4,5-c]azepin-6-one —— C20H20N4OS
(8S)-8-isoquinolin-5-yl-2-pyrrolidin-1-yl-4,5,7,8-tetrahydro-[1,3]thiazolo[4,5-c]azepin-6-one
—— (8R)-2-amino-8-[2-(4-methoxyphenyl)pyrimidin-5-yl]-4,5,7,8-tetrahydro-[1,3]thiazolo[4,5-c]azepin-6-one —— C18H17N5O2S
(8R)-2-amino-8-[2-(4-methoxyphenyl)pyrimidin-5-yl]-4,5,7,8-tetrahydro-[1,3]thiazolo[4,5-c]azepin-6-one
—— (8R)-2-(dimethylamino)-8-(4-methylsulfonylphenyl)-4,5,7,8-tetrahydro-[1,3]thiazolo[4,5-c]azepin-6-one —— C16H19N3O3S2
(8R)-2-(dimethylamino)-8-(4-methylsulfonylphenyl)-4,5,7,8-tetrahydro-[1,3]thiazolo[4,5-c]azepin-6-one
—— (8R)-8-(1-tert-butyl-3,5-dimethylpyrazol-4-yl)-7,8-dihydro-5H-[1,3]dioxolo[4,5-g]quinolin-6-one —— C19H23N3O3
(8R)-8-(1-tert-butyl-3,5-dimethylpyrazol-4-yl)-7,8-dihydro-5H-[1,3]dioxolo[4,5-g]quinolin-6-one
—— (8S)-2-(dimethylamino)-8-(4-methylsulfonylphenyl)-4,5,7,8-tetrahydro-[1,3]thiazolo[4,5-c]azepin-6-one —— C16H19N3O3S2
(8S)-2-(dimethylamino)-8-(4-methylsulfonylphenyl)-4,5,7,8-tetrahydro-[1,3]thiazolo[4,5-c]azepin-6-one
—— 8-[3-[(1R)-1-(dimethylamino)ethyl]phenyl]quinolin-4-amine —— C19H21N3
8-[3-[(1R)-1-(dimethylamino)ethyl]phenyl]quinolin-4-amine
—— (8R)-2-amino-8-(6-methoxy-1,3-benzodioxol-5-yl)-4,5,7,8-tetrahydro-[1,3]thiazolo[4,5-c]azepin-6-one —— C15H15N3O4S
(8R)-2-amino-8-(6-methoxy-1,3-benzodioxol-5-yl)-4,5,7,8-tetrahydro-[1,3]thiazolo[4,5-c]azepin-6-one
—— (8S)-8-(1-tert-butyl-3,5-dimethylpyrazol-4-yl)-7,8-dihydro-5H-[1,3]dioxolo[4,5-g]quinolin-6-one —— C19H23N3O3
(8S)-8-(1-tert-butyl-3,5-dimethylpyrazol-4-yl)-7,8-dihydro-5H-[1,3]dioxolo[4,5-g]quinolin-6-one
—— (8S)-2-amino-8-(6-methoxy-1,3-benzodioxol-5-yl)-4,5,7,8-tetrahydro-[1,3]thiazolo[4,5-c]azepin-6-one —— C15H15N3O4S
(8S)-2-amino-8-(6-methoxy-1,3-benzodioxol-5-yl)-4,5,7,8-tetrahydro-[1,3]thiazolo[4,5-c]azepin-6-one
—— 8-methoxy-N-[(3R)-2-oxoazepan-3-yl]-3,4-dihydro-2H-quinoline-1-carboxamide —— C17H23N3O3
8-methoxy-N-[(3R)-2-oxoazepan-3-yl]-3,4-dihydro-2H-quinoline-1-carboxamide
—— (8R)-8-(2,1,3-benzothiadiazol-4-yl)-2-pyrrolidin-1-yl-4,5,7,8-tetrahydro-[1,3]thiazolo[4,5-c]azepin-6-one —— C17H17N5OS2
(8R)-8-(2,1,3-benzothiadiazol-4-yl)-2-pyrrolidin-1-yl-4,5,7,8-tetrahydro-[1,3]thiazolo[4,5-c]azepin-6-one
—— (8R)-1-methyl-8-[3-(pyrazol-1-ylmethyl)phenyl]-7,8-dihydro-5H-[1,3]oxazolo[4,5-g]quinoline-2,6-dione —— C21H18N4O3
(8R)-1-methyl-8-[3-(pyrazol-1-ylmethyl)phenyl]-7,8-dihydro-5H-[1,3]oxazolo[4,5-g]quinoline-2,6-dione
—— 8-methoxy-N-[(3S)-2-oxoazepan-3-yl]-3,4-dihydro-2H-quinoline-1-carboxamide —— C17H23N3O3
8-methoxy-N-[(3S)-2-oxoazepan-3-yl]-3,4-dihydro-2H-quinoline-1-carboxamide
—— (8S)-2-amino-8-[4-(3-hydroxyprop-1-ynyl)thiophen-2-yl]-4,5,7,8-tetrahydro-[1,3]thiazolo[4,5-c]azepin-6-one —— C14H13N3O2S2
(8S)-2-amino-8-[4-(3-hydroxyprop-1-ynyl)thiophen-2-yl]-4,5,7,8-tetrahydro-[1,3]thiazolo[4,5-c]azepin-6-one