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—— (8S,9R,13S,14S,17Z)-17-[(E)-(1-ethyl-5-methylpyrazol-4-yl)methylidenehydrazinylidene]-13-methyl-7,8,9,11,12,14,15,16-octahydro-6H-cyclopenta[a]phenanthren-3-ol —— C25H32N4O
(8S,9R,13S,14S,17Z)-17-[(E)-(1-ethyl-5-methylpyrazol-4-yl)methylidenehydrazinylidene]-13-methyl-7,8,9,11,12,14,15,16-octahydro-6H-cyclopenta[a]phenanthren-3-ol
—— 8-[(2S)-2-methyl-1,4-oxazepan-4-yl]quinolin-5-amine —— C15H19N3O
8-[(2S)-2-methyl-1,4-oxazepan-4-yl]quinolin-5-amine
—— 8-[(2R)-2-methyl-1,4-oxazepan-4-yl]quinolin-5-amine —— C15H19N3O
8-[(2R)-2-methyl-1,4-oxazepan-4-yl]quinolin-5-amine
—— [(8aR)-3,4,6,7,8,8a-hexahydro-1H-pyrrolo[1,2-a]pyrazin-2-yl]-[(5R,7S)-5-(4-bromophenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-3-yl]methanone —— C21H23BrF3N5O
[(8aR)-3,4,6,7,8,8a-hexahydro-1H-pyrrolo[1,2-a]pyrazin-2-yl]-[(5R,7S)-5-(4-bromophenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-3-yl]methanone
—— (8S,9S,13R,14S)-3-hydroxy-13-methyl-2-(morpholin-4-ylmethyl)-7,8,9,11,12,14,15,16-octahydro-6H-cyclopenta[a]phenanthren-17-one —— C23H31NO3
(8S,9S,13R,14S)-3-hydroxy-13-methyl-2-(morpholin-4-ylmethyl)-7,8,9,11,12,14,15,16-octahydro-6H-cyclopenta[a]phenanthren-17-one
—— (8S,9R,13R,14S)-3-hydroxy-13-methyl-2-(morpholin-4-ylmethyl)-7,8,9,11,12,14,15,16-octahydro-6H-cyclopenta[a]phenanthren-17-one —— C23H31NO3
(8S,9R,13R,14S)-3-hydroxy-13-methyl-2-(morpholin-4-ylmethyl)-7,8,9,11,12,14,15,16-octahydro-6H-cyclopenta[a]phenanthren-17-one
—— (8S,9S,13S,14S)-3-hydroxy-13-methyl-2-(morpholin-4-ylmethyl)-7,8,9,11,12,14,15,16-octahydro-6H-cyclopenta[a]phenanthren-17-one —— C23H31NO3
(8S,9S,13S,14S)-3-hydroxy-13-methyl-2-(morpholin-4-ylmethyl)-7,8,9,11,12,14,15,16-octahydro-6H-cyclopenta[a]phenanthren-17-one
—— (8S,9R,13S,14S)-3-hydroxy-13-methyl-2-(morpholin-4-ylmethyl)-7,8,9,11,12,14,15,16-octahydro-6H-cyclopenta[a]phenanthren-17-one —— C23H31NO3
(8S,9R,13S,14S)-3-hydroxy-13-methyl-2-(morpholin-4-ylmethyl)-7,8,9,11,12,14,15,16-octahydro-6H-cyclopenta[a]phenanthren-17-one
—— (8S,9R,13S,14S,17Z)-17-[(E)-(1,5-dimethylpyrazol-4-yl)methylidenehydrazinylidene]-13-methyl-7,8,9,11,12,14,15,16-octahydro-6H-cyclopenta[a]phenanthren-3-ol —— C24H30N4O
(8S,9R,13S,14S,17Z)-17-[(E)-(1,5-dimethylpyrazol-4-yl)methylidenehydrazinylidene]-13-methyl-7,8,9,11,12,14,15,16-octahydro-6H-cyclopenta[a]phenanthren-3-ol
—— (8S,9R,13S,14S,17E)-13-methyl-17-[(Z)-(1,3,5-trimethylpyrazol-4-yl)methylidenehydrazinylidene]-7,8,9,11,12,14,15,16-octahydro-6H-cyclopenta[a]phenanthren-3-ol —— C25H32N4O
(8S,9R,13S,14S,17E)-13-methyl-17-[(Z)-(1,3,5-trimethylpyrazol-4-yl)methylidenehydrazinylidene]-7,8,9,11,12,14,15,16-octahydro-6H-cyclopenta[a]phenanthren-3-ol
—— (8S,9R,13S,14S,17E)-17-[(Z)-(1,5-dimethylpyrazol-4-yl)methylidenehydrazinylidene]-13-methyl-7,8,9,11,12,14,15,16-octahydro-6H-cyclopenta[a]phenanthren-3-ol —— C24H30N4O
(8S,9R,13S,14S,17E)-17-[(Z)-(1,5-dimethylpyrazol-4-yl)methylidenehydrazinylidene]-13-methyl-7,8,9,11,12,14,15,16-octahydro-6H-cyclopenta[a]phenanthren-3-ol
—— (8S,9R,13S,14S,17Z)-13-methyl-17-[(E)-(1,3,5-trimethylpyrazol-4-yl)methylidenehydrazinylidene]-7,8,9,11,12,14,15,16-octahydro-6H-cyclopenta[a]phenanthren-3-ol —— C25H32N4O
(8S,9R,13S,14S,17Z)-13-methyl-17-[(E)-(1,3,5-trimethylpyrazol-4-yl)methylidenehydrazinylidene]-7,8,9,11,12,14,15,16-octahydro-6H-cyclopenta[a]phenanthren-3-ol
—— [(8aR)-3,4,6,7,8,8a-hexahydro-1H-pyrrolo[1,2-a]pyrazin-2-yl]-[(5S,7R)-5-(4-bromophenyl)-3-chloro-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]methanone —— C21H22BrClF3N5O
[(8aR)-3,4,6,7,8,8a-hexahydro-1H-pyrrolo[1,2-a]pyrazin-2-yl]-[(5S,7R)-5-(4-bromophenyl)-3-chloro-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]methanone
—— [(8aR)-3,4,6,7,8,8a-hexahydro-1H-pyrrolo[1,2-a]pyrazin-2-yl]-[(5S,7S)-3-bromo-5-phenyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]methanone —— C21H23BrF3N5O
[(8aR)-3,4,6,7,8,8a-hexahydro-1H-pyrrolo[1,2-a]pyrazin-2-yl]-[(5S,7S)-3-bromo-5-phenyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]methanone
—— (8R)-3-(5-bromopyridin-2-yl)-8-methyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[4,3-a]pyrazine —— C11H12BrN5
(8R)-3-(5-bromopyridin-2-yl)-8-methyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[4,3-a]pyrazine
—— [(8aR)-3,4,6,7,8,8a-hexahydro-1H-pyrrolo[1,2-a]pyrazin-2-yl]-[(5R,7R)-3-chloro-5-phenyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]methanone —— C21H23ClF3N5O
[(8aR)-3,4,6,7,8,8a-hexahydro-1H-pyrrolo[1,2-a]pyrazin-2-yl]-[(5R,7R)-3-chloro-5-phenyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]methanone
—— (8S)-3-(5-bromopyridin-2-yl)-8-methyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[4,3-a]pyrazine —— C11H12BrN5
(8S)-3-(5-bromopyridin-2-yl)-8-methyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[4,3-a]pyrazine
—— 8-[(diethylamino)methyl]-7-hydroxy-5-methyl-3-(4-methyl-1,3-thiazol-2-yl)-4H-chromen-4-one —— C19H22N2O3S
8-[(diethylamino)methyl]-7-hydroxy-5-methyl-3-(4-methyl-1,3-thiazol-2-yl)-4H-chromen-4-one
—— 8-(azepan-1-ylmethyl)-3-(1,3-dihydrobenzimidazol-2-ylidene)chromene-2,7-dione —— C23H23N3O3
8-(azepan-1-ylmethyl)-3-(1,3-dihydrobenzimidazol-2-ylidene)chromene-2,7-dione
—— 8-[(Dimethylamino)methyl]-3-(4-ethylphenoxy)-7-hydroxy-2-methylchromen-4-one —— C21H23NO4
8-[(Dimethylamino)methyl]-3-(4-ethylphenoxy)-7-hydroxy-2-methylchromen-4-one
—— 8-((Dimethylamino)methyl)-7-hydroxy-2-methyl-3-(2-naphthyloxy)-4H-chromen-4-one —— C23H21NO4
8-((Dimethylamino)methyl)-7-hydroxy-2-methyl-3-(2-naphthyloxy)-4H-chromen-4-one
—— 8-[[(2R)-2-ethylpiperidin-1-yl]methyl]-7-hydroxy-3-phenylchromen-4-one —— C23H25NO3
8-[[(2R)-2-ethylpiperidin-1-yl]methyl]-7-hydroxy-3-phenylchromen-4-one
—— 8-[(dimethylamino)methyl]-2-ethyl-3-(4-fluorophenoxy)-7-hydroxy-4H-chromen-4-one —— C20H20FNO4
8-[(dimethylamino)methyl]-2-ethyl-3-(4-fluorophenoxy)-7-hydroxy-4H-chromen-4-one
—— 8-[[(2S)-2-ethylpiperidin-1-yl]methyl]-7-hydroxy-3-phenylchromen-4-one —— C23H25NO3
8-[[(2S)-2-ethylpiperidin-1-yl]methyl]-7-hydroxy-3-phenylchromen-4-one
—— 8-Piperidinomethyl-7-hydroxy-4-methyl-3-aethyl-cumarin —— C18H23NO3
8-Piperidinomethyl-7-hydroxy-4-methyl-3-aethyl-cumarin
—— (8Z)-8-[(cyclohexylamino)methylidene]-4-methylchromene-2,7-dione —— C17H19NO3
(8Z)-8-[(cyclohexylamino)methylidene]-4-methylchromene-2,7-dione
—— (8R)-8-methyl-2,3,7,8,9,10-hexahydrocyclohepta[g][1,4]benzodioxin-6-one —— C14H16O3
(8R)-8-methyl-2,3,7,8,9,10-hexahydrocyclohepta[g][1,4]benzodioxin-6-one
—— (8S)-8-methyl-2,3,7,8,9,10-hexahydrocyclohepta[g][1,4]benzodioxin-6-one —— C14H16O3
(8S)-8-methyl-2,3,7,8,9,10-hexahydrocyclohepta[g][1,4]benzodioxin-6-one
—— 8-fluoro-3-[(Z)-(4-fluorophenyl)methylideneamino]-5H-pyrimido[5,4-b]indol-4-one —— C17H10F2N4O
8-fluoro-3-[(Z)-(4-fluorophenyl)methylideneamino]-5H-pyrimido[5,4-b]indol-4-one
—— 8-fluoro-3-[(Z)-(3-fluorophenyl)methylideneamino]-5H-pyrimido[5,4-b]indol-4-one —— C17H10F2N4O
8-fluoro-3-[(Z)-(3-fluorophenyl)methylideneamino]-5H-pyrimido[5,4-b]indol-4-one
—— 8-fluoro-3-[(Z)-(2-fluorophenyl)methylideneamino]-2-methyl-5H-pyrimido[5,4-b]indol-4-one —— C18H12F2N4O
8-fluoro-3-[(Z)-(2-fluorophenyl)methylideneamino]-2-methyl-5H-pyrimido[5,4-b]indol-4-one
—— 8-chloro-3-[(Z)-(1-methylpyrrol-2-yl)methylideneamino]-1,5-dihydropyrimido[5,4-b]indole-2,4-dione —— C16H12ClN5O2
8-chloro-3-[(Z)-(1-methylpyrrol-2-yl)methylideneamino]-1,5-dihydropyrimido[5,4-b]indole-2,4-dione
—— 8-chloro-3-[(4-oxocyclohexa-2,5-dien-1-ylidene)methylamino]-5H-pyrimido[5,4-b]indol-4-one —— C17H11ClN4O2
8-chloro-3-[(4-oxocyclohexa-2,5-dien-1-ylidene)methylamino]-5H-pyrimido[5,4-b]indol-4-one
—— 8-methoxy-3-[(Z)-pyridin-3-ylmethylideneamino]-1,5-dihydropyrimido[5,4-b]indole-2,4-dione —— C17H13N5O3
8-methoxy-3-[(Z)-pyridin-3-ylmethylideneamino]-1,5-dihydropyrimido[5,4-b]indole-2,4-dione
—— 8-methoxy-3-[(Z)-pyridin-4-ylmethylideneamino]-1,5-dihydropyrimido[5,4-b]indole-2,4-dione —— C17H13N5O3
8-methoxy-3-[(Z)-pyridin-4-ylmethylideneamino]-1,5-dihydropyrimido[5,4-b]indole-2,4-dione
—— 8-fluoro-3-[(Z)-(4-methylphenyl)methylideneamino]-5H-pyrimido[5,4-b]indol-4-one —— C18H13FN4O
8-fluoro-3-[(Z)-(4-methylphenyl)methylideneamino]-5H-pyrimido[5,4-b]indol-4-one
—— 8-fluoro-3-[(Z)-pyridin-3-ylmethylideneamino]-5H-pyrimido[5,4-b]indol-4-one —— C16H10FN5O
8-fluoro-3-[(Z)-pyridin-3-ylmethylideneamino]-5H-pyrimido[5,4-b]indol-4-one
—— 8-fluoro-3-[(Z)-(2-fluorophenyl)methylideneamino]-5H-pyrimido[5,4-b]indol-4-one —— C17H10F2N4O
8-fluoro-3-[(Z)-(2-fluorophenyl)methylideneamino]-5H-pyrimido[5,4-b]indol-4-one
—— (8Z)-1,3-dimethyl-8-(6-oxocyclohexa-2,4-dien-1-ylidene)-7,9-dihydropurine-2,6-dione —— C13H12N4O3
(8Z)-1,3-dimethyl-8-(6-oxocyclohexa-2,4-dien-1-ylidene)-7,9-dihydropurine-2,6-dione
—— 8-[[(2R)-2-ethylpiperidin-1-yl]methyl]-7-hydroxy-4-propylchromen-2-one —— C20H27NO3
8-[[(2R)-2-ethylpiperidin-1-yl]methyl]-7-hydroxy-4-propylchromen-2-one
—— 8-[[(2S)-2-ethylpiperidin-1-yl]methyl]-7-hydroxy-4-propylchromen-2-one —— C20H27NO3
8-[[(2S)-2-ethylpiperidin-1-yl]methyl]-7-hydroxy-4-propylchromen-2-one
—— 8-[[(2S)-2-ethylpiperidin-1-yl]methyl]-7-hydroxy-6-methyl-2,3-dihydro-1H-cyclopenta[c]chromen-4-one —— C21H27NO3
8-[[(2S)-2-ethylpiperidin-1-yl]methyl]-7-hydroxy-6-methyl-2,3-dihydro-1H-cyclopenta[c]chromen-4-one
—— (8E)-8-(3-methoxy-4-oxocyclohexa-2,5-dien-1-ylidene)-1,3-dimethyl-7,9-dihydropurine-2,6-dione —— C14H14N4O4
(8E)-8-(3-methoxy-4-oxocyclohexa-2,5-dien-1-ylidene)-1,3-dimethyl-7,9-dihydropurine-2,6-dione
—— (8Z,10R)-8-hydroxyimino-4,4-dimethyl-1,15-diazatetracyclo[8.7.0.02,7.011,15]heptadeca-2(7),11,13-trien-6-one —— C17H21N3O2
(8Z,10R)-8-hydroxyimino-4,4-dimethyl-1,15-diazatetracyclo[8.7.0.02,7.011,15]heptadeca-2(7),11,13-trien-6-one
—— 8-[[(2R)-2-ethylpiperidin-1-yl]methyl]-7-hydroxy-6-methyl-2,3-dihydro-1H-cyclopenta[c]chromen-4-one —— C21H27NO3
8-[[(2R)-2-ethylpiperidin-1-yl]methyl]-7-hydroxy-6-methyl-2,3-dihydro-1H-cyclopenta[c]chromen-4-one
—— 8-fluoro-3-[(4-oxocyclohexa-2,5-dien-1-ylidene)methylamino]-5H-pyrimido[5,4-b]indol-4-one —— C17H11FN4O2
8-fluoro-3-[(4-oxocyclohexa-2,5-dien-1-ylidene)methylamino]-5H-pyrimido[5,4-b]indol-4-one
—— 8-fluoro-3-[(Z)-(4-fluorophenyl)methylideneamino]-1,5-dihydropyrimido[5,4-b]indole-2,4-dione —— C17H10F2N4O2
8-fluoro-3-[(Z)-(4-fluorophenyl)methylideneamino]-1,5-dihydropyrimido[5,4-b]indole-2,4-dione
—— 8-fluoro-3-[(Z)-(1-methylpyrrol-2-yl)methylideneamino]-1,5-dihydropyrimido[5,4-b]indole-2,4-dione —— C16H12FN5O2
8-fluoro-3-[(Z)-(1-methylpyrrol-2-yl)methylideneamino]-1,5-dihydropyrimido[5,4-b]indole-2,4-dione
—— 8-chloro-3-[(Z)-(4-fluorophenyl)methylideneamino]-5H-pyrimido[5,4-b]indol-4-one —— C17H10ClFN4O
8-chloro-3-[(Z)-(4-fluorophenyl)methylideneamino]-5H-pyrimido[5,4-b]indol-4-one
—— 8-methoxy-3-[(Z)-thiophen-2-ylmethylideneamino]-1,5-dihydropyrimido[5,4-b]indole-2,4-dione —— C16H12N4O3S
8-methoxy-3-[(Z)-thiophen-2-ylmethylideneamino]-1,5-dihydropyrimido[5,4-b]indole-2,4-dione