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中文名称 英文名称 CAS号 化学式 结构式图片
—— (8S)-11-(4-fluorophenyl)-N-prop-2-ynyl-5-pyridin-4-yl-2-thia-4,6,7,13-tetrazatricyclo[7.4.0.03,7]trideca-1(9),3,5,10,12-pentaen-8-amine —— C22H15FN6S
(8S)-11-(4-fluorophenyl)-N-prop-2-ynyl-5-pyridin-4-yl-2-thia-4,6,7,13-tetrazatricyclo[7.4.0.03,7]trideca-1(9),3,5,10,12-pentaen-8-amine
—— 8-ethoxy-3-(furan-2-ylmethyl)-4H-[1,3]oxazino[6,5-b]quinolin-2-one —— C18H16N2O4
8-ethoxy-3-(furan-2-ylmethyl)-4H-[1,3]oxazino[6,5-b]quinolin-2-one
—— (8S)-11-(4-fluorophenyl)-5-pyridin-4-yl-2-thia-4,6,7,13-tetrazatricyclo[7.4.0.03,7]trideca-1(9),3,5,10,12-pentaen-8-ol —— C19H12FN5OS
(8S)-11-(4-fluorophenyl)-5-pyridin-4-yl-2-thia-4,6,7,13-tetrazatricyclo[7.4.0.03,7]trideca-1(9),3,5,10,12-pentaen-8-ol
—— (8R)-11-(4-fluorophenyl)-N-prop-2-ynyl-5-pyridin-4-yl-2-thia-4,6,7,13-tetrazatricyclo[7.4.0.03,7]trideca-1(9),3,5,10,12-pentaen-8-amine —— C22H15FN6S
(8R)-11-(4-fluorophenyl)-N-prop-2-ynyl-5-pyridin-4-yl-2-thia-4,6,7,13-tetrazatricyclo[7.4.0.03,7]trideca-1(9),3,5,10,12-pentaen-8-amine
—— (8R)-11-(4-fluorophenyl)-5-pyridin-3-yl-8-pyrrolidin-1-yl-2-thia-4,6,7,13-tetrazatricyclo[7.4.0.03,7]trideca-1(9),3,5,10,12-pentaene —— C23H19FN6S
(8R)-11-(4-fluorophenyl)-5-pyridin-3-yl-8-pyrrolidin-1-yl-2-thia-4,6,7,13-tetrazatricyclo[7.4.0.03,7]trideca-1(9),3,5,10,12-pentaene
—— (8S)-11-phenyl-N,N-bis(prop-2-enyl)-5-pyridin-3-yl-2-thia-4,6,7,13-tetrazatricyclo[7.4.0.03,7]trideca-1(9),3,5,10,12-pentaen-8-amine —— C25H22N6S
(8S)-11-phenyl-N,N-bis(prop-2-enyl)-5-pyridin-3-yl-2-thia-4,6,7,13-tetrazatricyclo[7.4.0.03,7]trideca-1(9),3,5,10,12-pentaen-8-amine
—— (8R)-11-(4-fluorophenyl)-N-prop-2-enyl-5-pyridin-4-yl-2-thia-4,6,7,13-tetrazatricyclo[7.4.0.03,7]trideca-1(9),3,5,10,12-pentaen-8-amine —— C22H17FN6S
(8R)-11-(4-fluorophenyl)-N-prop-2-enyl-5-pyridin-4-yl-2-thia-4,6,7,13-tetrazatricyclo[7.4.0.03,7]trideca-1(9),3,5,10,12-pentaen-8-amine
—— (8R)-11-(4-fluorophenyl)-5-pyridin-4-yl-8-pyrrolidin-1-yl-2-thia-4,6,7,13-tetrazatricyclo[7.4.0.03,7]trideca-1(9),3,5,10,12-pentaene —— C23H19FN6S
(8R)-11-(4-fluorophenyl)-5-pyridin-4-yl-8-pyrrolidin-1-yl-2-thia-4,6,7,13-tetrazatricyclo[7.4.0.03,7]trideca-1(9),3,5,10,12-pentaene
—— (8R)-11-phenyl-5-pyridin-3-yl-8-pyrrolidin-1-yl-2-thia-4,6,7,13-tetrazatricyclo[7.4.0.03,7]trideca-1(9),3,5,10,12-pentaene —— C23H20N6S
(8R)-11-phenyl-5-pyridin-3-yl-8-pyrrolidin-1-yl-2-thia-4,6,7,13-tetrazatricyclo[7.4.0.03,7]trideca-1(9),3,5,10,12-pentaene
—— (8S)-11-(4-fluorophenyl)-5-pyridin-3-yl-2-thia-4,6,7,13-tetrazatricyclo[7.4.0.03,7]trideca-1(9),3,5,10,12-pentaen-8-ol —— C19H12FN5OS
(8S)-11-(4-fluorophenyl)-5-pyridin-3-yl-2-thia-4,6,7,13-tetrazatricyclo[7.4.0.03,7]trideca-1(9),3,5,10,12-pentaen-8-ol
—— (8S)-11-phenyl-5-pyridin-3-yl-8-pyrrolidin-1-yl-2-thia-4,6,7,13-tetrazatricyclo[7.4.0.03,7]trideca-1(9),3,5,10,12-pentaene —— C23H20N6S
(8S)-11-phenyl-5-pyridin-3-yl-8-pyrrolidin-1-yl-2-thia-4,6,7,13-tetrazatricyclo[7.4.0.03,7]trideca-1(9),3,5,10,12-pentaene
—— 8,9-dimethyl-3-(2-morpholin-4-ylethyl)-4H-[1,3]oxazino[6,5-b]quinolin-2-one —— C19H23N3O3
8,9-dimethyl-3-(2-morpholin-4-ylethyl)-4H-[1,3]oxazino[6,5-b]quinolin-2-one
—— (8R)-11-phenyl-N,N-bis(prop-2-enyl)-5-pyridin-3-yl-2-thia-4,6,7,13-tetrazatricyclo[7.4.0.03,7]trideca-1(9),3,5,10,12-pentaen-8-amine —— C25H22N6S
(8R)-11-phenyl-N,N-bis(prop-2-enyl)-5-pyridin-3-yl-2-thia-4,6,7,13-tetrazatricyclo[7.4.0.03,7]trideca-1(9),3,5,10,12-pentaen-8-amine
—— (8S)-8-(4-methylpiperazin-1-yl)-11-phenyl-5-pyridin-3-yl-2-thia-4,6,7,13-tetrazatricyclo[7.4.0.03,7]trideca-1(9),3,5,10,12-pentaene —— C24H23N7S
(8S)-8-(4-methylpiperazin-1-yl)-11-phenyl-5-pyridin-3-yl-2-thia-4,6,7,13-tetrazatricyclo[7.4.0.03,7]trideca-1(9),3,5,10,12-pentaene
—— (8R)-11-phenyl-5-pyridin-4-yl-8-pyrrolidin-1-yl-2-thia-4,6,7,13-tetrazatricyclo[7.4.0.03,7]trideca-1(9),3,5,10,12-pentaene —— C23H20N6S
(8R)-11-phenyl-5-pyridin-4-yl-8-pyrrolidin-1-yl-2-thia-4,6,7,13-tetrazatricyclo[7.4.0.03,7]trideca-1(9),3,5,10,12-pentaene
—— 8,9-dimethyl-3-(3-morpholin-4-ylpropyl)-4H-[1,3]oxazino[6,5-b]quinolin-2-one —— C20H25N3O3
8,9-dimethyl-3-(3-morpholin-4-ylpropyl)-4H-[1,3]oxazino[6,5-b]quinolin-2-one
—— (8R)-8-(4-methylpiperazin-1-yl)-11-phenyl-5-pyridin-3-yl-2-thia-4,6,7,13-tetrazatricyclo[7.4.0.03,7]trideca-1(9),3,5,10,12-pentaene —— C24H23N7S
(8R)-8-(4-methylpiperazin-1-yl)-11-phenyl-5-pyridin-3-yl-2-thia-4,6,7,13-tetrazatricyclo[7.4.0.03,7]trideca-1(9),3,5,10,12-pentaene
—— 8-methyl-3-[[4-(4-methylpiperazin-1-yl)anilino]methyl]-1H-quinolin-2-one —— C22H26N4O
8-methyl-3-[[4-(4-methylpiperazin-1-yl)anilino]methyl]-1H-quinolin-2-one
—— (8S)-11-(4-fluorophenyl)-N-prop-2-enyl-5-pyridin-4-yl-2-thia-4,6,7,13-tetrazatricyclo[7.4.0.03,7]trideca-1(9),3,5,10,12-pentaen-8-amine —— C22H17FN6S
(8S)-11-(4-fluorophenyl)-N-prop-2-enyl-5-pyridin-4-yl-2-thia-4,6,7,13-tetrazatricyclo[7.4.0.03,7]trideca-1(9),3,5,10,12-pentaen-8-amine
—— (8R)-N-cyclopropyl-11-phenyl-5-pyridin-3-yl-2-thia-4,6,7,13-tetrazatricyclo[7.4.0.03,7]trideca-1(9),3,5,10,12-pentaen-8-amine —— C22H18N6S
(8R)-N-cyclopropyl-11-phenyl-5-pyridin-3-yl-2-thia-4,6,7,13-tetrazatricyclo[7.4.0.03,7]trideca-1(9),3,5,10,12-pentaen-8-amine
—— 8-methyl-3-[(3,4,5-trimethoxyanilino)methyl]-1H-quinolin-2-one —— C20H22N2O4
8-methyl-3-[(3,4,5-trimethoxyanilino)methyl]-1H-quinolin-2-one
—— 8-methoxy-1'-[(3S)-1-(2-methoxyethyl)-5-oxopyrrolidine-3-carbonyl]spiro[3,4-dihydro-1,4-benzoxazepine-2,4'-piperidine]-5-one —— C22H29N3O6
8-methoxy-1'-[(3S)-1-(2-methoxyethyl)-5-oxopyrrolidine-3-carbonyl]spiro[3,4-dihydro-1,4-benzoxazepine-2,4'-piperidine]-5-one
—— 8-methoxy-1'-[(3R)-1-(2-methoxyethyl)-5-oxopyrrolidine-3-carbonyl]spiro[3,4-dihydro-1,4-benzoxazepine-2,4'-piperidine]-5-one —— C22H29N3O6
8-methoxy-1'-[(3R)-1-(2-methoxyethyl)-5-oxopyrrolidine-3-carbonyl]spiro[3,4-dihydro-1,4-benzoxazepine-2,4'-piperidine]-5-one
—— 8-Methoxy-1'-[2-(trifluoromethyl)benzoyl]spiro[3,4-dihydro-1,4-benzoxazepine-2,4'-piperidine]-5-one —— C22H21F3N2O4
8-Methoxy-1'-[2-(trifluoromethyl)benzoyl]spiro[3,4-dihydro-1,4-benzoxazepine-2,4'-piperidine]-5-one
—— 8-Methoxy-1'-[2-(4-methoxyphenoxy)acetyl]spiro[3,4-dihydro-1,4-benzoxazepine-2,4'-piperidine]-5-one —— C23H26N2O6
8-Methoxy-1'-[2-(4-methoxyphenoxy)acetyl]spiro[3,4-dihydro-1,4-benzoxazepine-2,4'-piperidine]-5-one
—— 8-Methoxy-1'-[3-(2-propan-2-ylimidazol-1-yl)propanoyl]spiro[3,4-dihydro-1,4-benzoxazepine-2,4'-piperidine]-5-one —— C23H30N4O4
8-Methoxy-1'-[3-(2-propan-2-ylimidazol-1-yl)propanoyl]spiro[3,4-dihydro-1,4-benzoxazepine-2,4'-piperidine]-5-one
—— 8-Methoxy-1'-[3-(trifluoromethyl)benzoyl]spiro[3,4-dihydro-1,4-benzoxazepine-2,4'-piperidine]-5-one —— C22H21F3N2O4
8-Methoxy-1'-[3-(trifluoromethyl)benzoyl]spiro[3,4-dihydro-1,4-benzoxazepine-2,4'-piperidine]-5-one
—— 8-methyl-4-(thiophen-2-ylmethyl)-3,5-dihydro-2H-[1,4]oxazepino[7,6-b]quinoline —— C18H18N2OS
8-methyl-4-(thiophen-2-ylmethyl)-3,5-dihydro-2H-[1,4]oxazepino[7,6-b]quinoline
—— 8,9-dimethoxy-4-(thiophen-2-ylmethyl)-3,5-dihydro-2H-[1,4]oxazepino[7,6-b]quinoline —— C19H20N2O3S
8,9-dimethoxy-4-(thiophen-2-ylmethyl)-3,5-dihydro-2H-[1,4]oxazepino[7,6-b]quinoline
—— 8-(Azepan-1-ylmethyl)-6-(4-fluorophenyl)tetrazolo[1,5-a]pyridine —— C18H20FN5
8-(Azepan-1-ylmethyl)-6-(4-fluorophenyl)tetrazolo[1,5-a]pyridine
—— 8-[(4-Cyclopentylpiperazin-1-yl)methyl]-6-(4-fluorophenyl)tetrazolo[1,5-a]pyridine —— C21H25FN6
8-[(4-Cyclopentylpiperazin-1-yl)methyl]-6-(4-fluorophenyl)tetrazolo[1,5-a]pyridine
—— 8-[[(8aR)-3,4,6,7,8,8a-hexahydro-1H-pyrrolo[1,2-a]pyrazin-2-yl]methyl]-6-phenyltetrazolo[1,5-a]pyridine —— C19H22N6
8-[[(8aR)-3,4,6,7,8,8a-hexahydro-1H-pyrrolo[1,2-a]pyrazin-2-yl]methyl]-6-phenyltetrazolo[1,5-a]pyridine
—— (8-methoxy-2H-chromen-3-yl)-[2-[(2S)-pyrrolidin-2-yl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-6-yl]methanone —— C22H24N4O3
(8-methoxy-2H-chromen-3-yl)-[2-[(2S)-pyrrolidin-2-yl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-6-yl]methanone
—— (8-methoxy-2H-chromen-3-yl)-[2-[(2R)-pyrrolidin-2-yl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-6-yl]methanone —— C22H24N4O3
(8-methoxy-2H-chromen-3-yl)-[2-[(2R)-pyrrolidin-2-yl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-6-yl]methanone
—— 8-[(3-Bromo-4-methoxyphenyl)methyl]-2,8-diazaspiro[4.5]decan-3-one —— C16H21BrN2O2
8-[(3-Bromo-4-methoxyphenyl)methyl]-2,8-diazaspiro[4.5]decan-3-one
—— 8-ethyl-3-[(1R,11R)-3,10,12-triazatetracyclo[10.3.1.02,10.04,9]hexadeca-2,4,6,8-tetraen-11-yl]-1H-quinolin-2-one —— C24H24N4O
8-ethyl-3-[(1R,11R)-3,10,12-triazatetracyclo[10.3.1.02,10.04,9]hexadeca-2,4,6,8-tetraen-11-yl]-1H-quinolin-2-one
—— 8-methyl-3-[[4-(5-oxo-1,4-diazepan-1-yl)anilino]methyl]-1H-quinolin-2-one —— C22H24N4O2
8-methyl-3-[[4-(5-oxo-1,4-diazepan-1-yl)anilino]methyl]-1H-quinolin-2-one
—— 8-ethyl-3-[(1R,11S)-3,10,12-triazatetracyclo[10.3.1.02,10.04,9]hexadeca-2,4,6,8-tetraen-11-yl]-1H-quinolin-2-one —— C24H24N4O
8-ethyl-3-[(1R,11S)-3,10,12-triazatetracyclo[10.3.1.02,10.04,9]hexadeca-2,4,6,8-tetraen-11-yl]-1H-quinolin-2-one
—— 8,9-Dimethyl-2,3,4,5-tetrahydro-[1,4]oxazepino[7,6-b]quinoline —— C14H16N2O
8,9-Dimethyl-2,3,4,5-tetrahydro-[1,4]oxazepino[7,6-b]quinoline
—— [8-(Benzenesulfonyl)-1-thia-4,8-diazaspiro[4.5]decan-4-yl]-(4-bromophenyl)methanone —— C20H21BrN2O3S2
[8-(Benzenesulfonyl)-1-thia-4,8-diazaspiro[4.5]decan-4-yl]-(4-bromophenyl)methanone
—— 8-[2-(5-chloro-6-oxo-1H-pyridazin-4-yl)hydrazinyl]-2,3-dihydro-[1,4]dioxino[2,3-f]indol-7-one —— C14H10ClN5O4
8-[2-(5-chloro-6-oxo-1H-pyridazin-4-yl)hydrazinyl]-2,3-dihydro-[1,4]dioxino[2,3-f]indol-7-one
—— 8-methyl-2-[[5-(propylamino)-1,3,4-thiadiazol-2-yl]sulfanylmethyl]-3H-quinazolin-4-one —— C15H17N5OS2
8-methyl-2-[[5-(propylamino)-1,3,4-thiadiazol-2-yl]sulfanylmethyl]-3H-quinazolin-4-one
—— 8-[2-(3-Methoxyphenyl)ethyl]-4-methyl-2-[[methyl(pyridin-2-ylmethyl)amino]methyl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C25H29N5O2
8-[2-(3-Methoxyphenyl)ethyl]-4-methyl-2-[[methyl(pyridin-2-ylmethyl)amino]methyl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-(3-Methoxypropyl)-4-methyl-2-[[methyl(quinoxalin-6-ylmethyl)amino]methyl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C23H28N6O2
8-(3-Methoxypropyl)-4-methyl-2-[[methyl(quinoxalin-6-ylmethyl)amino]methyl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-Benzyl-4-methyl-2-[[methyl(3-phenylpropyl)amino]methyl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C26H30N4O
8-Benzyl-4-methyl-2-[[methyl(3-phenylpropyl)amino]methyl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-benzyl-4-methyl-2-[(2S)-1-(pyridin-2-ylmethyl)piperidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C26H29N5O
8-benzyl-4-methyl-2-[(2S)-1-(pyridin-2-ylmethyl)piperidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-(Cyclohexylmethyl)-4-methyl-2-[1-(pyridin-3-ylmethyl)piperidin-4-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C26H35N5O
8-(Cyclohexylmethyl)-4-methyl-2-[1-(pyridin-3-ylmethyl)piperidin-4-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-benzyl-4-methyl-2-[(2S)-1-(pyridin-3-ylmethyl)piperidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C26H29N5O
8-benzyl-4-methyl-2-[(2S)-1-(pyridin-3-ylmethyl)piperidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-benzyl-4-methyl-2-[(2R)-1-(pyridin-3-ylmethyl)piperidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C26H29N5O
8-benzyl-4-methyl-2-[(2R)-1-(pyridin-3-ylmethyl)piperidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-benzyl-4-methyl-2-[(2R)-1-(pyridin-2-ylmethyl)piperidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C26H29N5O
8-benzyl-4-methyl-2-[(2R)-1-(pyridin-2-ylmethyl)piperidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one