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—— 8-[2-(1-Benzylindol-3-yl)ethyl]-4-methyl-2-(methylaminomethyl)-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C27H29N5O
8-[2-(1-Benzylindol-3-yl)ethyl]-4-methyl-2-(methylaminomethyl)-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-[2-(3-Methoxyphenyl)ethyl]-4-methyl-2-[[methyl(pyridin-4-ylmethyl)amino]methyl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C25H29N5O2
8-[2-(3-Methoxyphenyl)ethyl]-4-methyl-2-[[methyl(pyridin-4-ylmethyl)amino]methyl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-[2-[1-(Cyclohexylmethyl)indol-3-yl]ethyl]-4-methyl-2-(methylaminomethyl)-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C27H35N5O
8-[2-[1-(Cyclohexylmethyl)indol-3-yl]ethyl]-4-methyl-2-(methylaminomethyl)-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-[(2-Fluorophenyl)methyl]-4-methyl-2-[1-(pyridin-4-ylmethyl)piperidin-4-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C26H28FN5O
8-[(2-Fluorophenyl)methyl]-4-methyl-2-[1-(pyridin-4-ylmethyl)piperidin-4-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-[(4-fluorophenyl)methyl]-4-methyl-2-[(2S)-1-(pyridine-3-carbonyl)pyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C25H24FN5O2
8-[(4-fluorophenyl)methyl]-4-methyl-2-[(2S)-1-(pyridine-3-carbonyl)pyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-(cyclohexylmethyl)-4-methyl-2-[(2R)-1-(pyridine-4-carbonyl)pyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C25H31N5O2
8-(cyclohexylmethyl)-4-methyl-2-[(2R)-1-(pyridine-4-carbonyl)pyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-[(4-fluorophenyl)methyl]-4-methyl-2-[(2R)-1-(1-methylimidazole-2-carbonyl)pyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C24H25FN6O2
8-[(4-fluorophenyl)methyl]-4-methyl-2-[(2R)-1-(1-methylimidazole-2-carbonyl)pyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-[(4-fluorophenyl)methyl]-4-methyl-2-[(2R)-1-(pyridine-3-carbonyl)pyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C25H24FN5O2
8-[(4-fluorophenyl)methyl]-4-methyl-2-[(2R)-1-(pyridine-3-carbonyl)pyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-[(4-fluorophenyl)methyl]-4-methyl-2-[(2S)-1-(pyridine-4-carbonyl)pyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C25H24FN5O2
8-[(4-fluorophenyl)methyl]-4-methyl-2-[(2S)-1-(pyridine-4-carbonyl)pyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-(cyclohexylmethyl)-2-[(2R)-1-[(4-hydroxyphenyl)methyl]pyrrolidin-2-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C26H34N4O2
8-(cyclohexylmethyl)-2-[(2R)-1-[(4-hydroxyphenyl)methyl]pyrrolidin-2-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-(cyclohexylmethyl)-2-[(2S)-1-[(4-hydroxyphenyl)methyl]pyrrolidin-2-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C26H34N4O2
8-(cyclohexylmethyl)-2-[(2S)-1-[(4-hydroxyphenyl)methyl]pyrrolidin-2-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-[(4-fluorophenyl)methyl]-4-methyl-2-[(2R)-1-(pyridine-4-carbonyl)pyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C25H24FN5O2
8-[(4-fluorophenyl)methyl]-4-methyl-2-[(2R)-1-(pyridine-4-carbonyl)pyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-[(4-fluorophenyl)methyl]-4-methyl-2-[(2S)-1-(1-methylimidazole-2-carbonyl)pyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C24H25FN6O2
8-[(4-fluorophenyl)methyl]-4-methyl-2-[(2S)-1-(1-methylimidazole-2-carbonyl)pyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-[2-(2-methoxyphenyl)ethyl]-4-methyl-2-[(2S)-1-methylsulfonylpyrrolidin-2-yl]-6,7-dihydro-5H-pyrido[2,3-d]pyrimidine —— C22H30N4O3S
8-[2-(2-methoxyphenyl)ethyl]-4-methyl-2-[(2S)-1-methylsulfonylpyrrolidin-2-yl]-6,7-dihydro-5H-pyrido[2,3-d]pyrimidine
—— 8-[2-(2-methoxyphenyl)ethyl]-4-methyl-2-[(2R)-1-methylsulfonylpyrrolidin-2-yl]-6,7-dihydro-5H-pyrido[2,3-d]pyrimidine —— C22H30N4O3S
8-[2-(2-methoxyphenyl)ethyl]-4-methyl-2-[(2R)-1-methylsulfonylpyrrolidin-2-yl]-6,7-dihydro-5H-pyrido[2,3-d]pyrimidine
—— 8-(cyclohexylmethyl)-4-methyl-2-[(2S)-1-methylsulfonylpyrrolidin-2-yl]-6,7-dihydro-5H-pyrido[2,3-d]pyrimidine —— C20H32N4O2S
8-(cyclohexylmethyl)-4-methyl-2-[(2S)-1-methylsulfonylpyrrolidin-2-yl]-6,7-dihydro-5H-pyrido[2,3-d]pyrimidine
—— 8-(cyclohexylmethyl)-4-methyl-2-[(2R)-1-methylsulfonylpyrrolidin-2-yl]-6,7-dihydro-5H-pyrido[2,3-d]pyrimidine —— C20H32N4O2S
8-(cyclohexylmethyl)-4-methyl-2-[(2R)-1-methylsulfonylpyrrolidin-2-yl]-6,7-dihydro-5H-pyrido[2,3-d]pyrimidine
—— 8-methoxy-3-(2-methoxyethyl)-4H-[1,3]oxazino[6,5-b]quinolin-2-one —— C15H16N2O4
8-methoxy-3-(2-methoxyethyl)-4H-[1,3]oxazino[6,5-b]quinolin-2-one
—— 8-(ethyl)thieno[3',2':4,5]pyrrolo[1,2-d][1,2,4]triazin-5(6H)-one —— C10H9N3OS
8-(ethyl)thieno[3',2':4,5]pyrrolo[1,2-d][1,2,4]triazin-5(6H)-one
—— 8,10-Dimethyl-2,3,4,5-tetrahydro-[1,4]oxazepino[7,6-b]quinoline —— C14H16N2O
8,10-Dimethyl-2,3,4,5-tetrahydro-[1,4]oxazepino[7,6-b]quinoline
—— 8-(cyclopropylmethyl)-2-[(2R)-1-[(1-ethyl-5-methylpyrazol-4-yl)methyl]piperidin-2-yl]-4-methyl-6,7-dihydro-5H-pyrido[2,3-d]pyrimidine —— C24H36N6
8-(cyclopropylmethyl)-2-[(2R)-1-[(1-ethyl-5-methylpyrazol-4-yl)methyl]piperidin-2-yl]-4-methyl-6,7-dihydro-5H-pyrido[2,3-d]pyrimidine
—— 8-(cyclopropylmethyl)-2-[(2S)-1-[(1-ethyl-5-methylpyrazol-4-yl)methyl]piperidin-2-yl]-4-methyl-6,7-dihydro-5H-pyrido[2,3-d]pyrimidine —— C24H36N6
8-(cyclopropylmethyl)-2-[(2S)-1-[(1-ethyl-5-methylpyrazol-4-yl)methyl]piperidin-2-yl]-4-methyl-6,7-dihydro-5H-pyrido[2,3-d]pyrimidine
—— 8-(cyclopropylmethyl)-2-[(2S)-1-[(1-ethyl-3-methylpyrazol-4-yl)methyl]piperidin-2-yl]-4-methyl-6,7-dihydro-5H-pyrido[2,3-d]pyrimidine —— C24H36N6
8-(cyclopropylmethyl)-2-[(2S)-1-[(1-ethyl-3-methylpyrazol-4-yl)methyl]piperidin-2-yl]-4-methyl-6,7-dihydro-5H-pyrido[2,3-d]pyrimidine
—— 8-(cyclopropylmethyl)-2-[(2R)-1-[(1-ethyl-3-methylpyrazol-4-yl)methyl]piperidin-2-yl]-4-methyl-6,7-dihydro-5H-pyrido[2,3-d]pyrimidine —— C24H36N6
8-(cyclopropylmethyl)-2-[(2R)-1-[(1-ethyl-3-methylpyrazol-4-yl)methyl]piperidin-2-yl]-4-methyl-6,7-dihydro-5H-pyrido[2,3-d]pyrimidine
—— 8-(Cyclopropylmethyl)-4-methyl-2-[1-[3-(3-methyl-1,2,4-oxadiazol-5-yl)propanoyl]piperidin-4-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C23H30N6O3
8-(Cyclopropylmethyl)-4-methyl-2-[1-[3-(3-methyl-1,2,4-oxadiazol-5-yl)propanoyl]piperidin-4-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-Benzyl-2-[[(1,5-dimethylpyrazol-4-yl)methyl-methylamino]methyl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C23H28N6O
8-Benzyl-2-[[(1,5-dimethylpyrazol-4-yl)methyl-methylamino]methyl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-Cyclopentyl-4-methyl-2-[1-(2-methylpropyl)piperidin-4-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C22H34N4O
8-Cyclopentyl-4-methyl-2-[1-(2-methylpropyl)piperidin-4-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-[(3-fluorophenyl)methyl]-4-methyl-2-[(2S)-1-(pyridine-2-carbonyl)pyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C25H24FN5O2
8-[(3-fluorophenyl)methyl]-4-methyl-2-[(2S)-1-(pyridine-2-carbonyl)pyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-[2-(3-Methoxyphenyl)ethyl]-4-methyl-2-[[methyl-[(2-methylphenyl)methyl]amino]methyl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C27H32N4O2
8-[2-(3-Methoxyphenyl)ethyl]-4-methyl-2-[[methyl-[(2-methylphenyl)methyl]amino]methyl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-benzyl-4-methyl-2-[(2S)-1-pyrimidin-2-ylpyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C23H24N6O
8-benzyl-4-methyl-2-[(2S)-1-pyrimidin-2-ylpyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-cyclopentyl-4-methyl-2-[1-[3-[(2S)-oxolan-2-yl]propanoyl]piperidin-4-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C25H36N4O3
8-cyclopentyl-4-methyl-2-[1-[3-[(2S)-oxolan-2-yl]propanoyl]piperidin-4-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-(cyclopropylmethyl)-4-methyl-2-[1-[(2R)-2-pyrrolidin-1-ylpropanoyl]piperidin-4-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C24H35N5O2
8-(cyclopropylmethyl)-4-methyl-2-[1-[(2R)-2-pyrrolidin-1-ylpropanoyl]piperidin-4-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-cyclopentyl-4-methyl-2-[1-[(3R)-1-methyl-5-oxopyrrolidine-3-carbonyl]piperidin-4-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C24H33N5O3
8-cyclopentyl-4-methyl-2-[1-[(3R)-1-methyl-5-oxopyrrolidine-3-carbonyl]piperidin-4-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-[(4-methoxyphenyl)methyl]-4-methyl-2-[(3R)-1-propanoylpiperidin-3-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C24H30N4O3
8-[(4-methoxyphenyl)methyl]-4-methyl-2-[(3R)-1-propanoylpiperidin-3-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-[(4-fluorophenyl)methyl]-2-[(2R)-1-(2-hydroxy-2-methylpropanoyl)pyrrolidin-2-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C23H27FN4O3
8-[(4-fluorophenyl)methyl]-2-[(2R)-1-(2-hydroxy-2-methylpropanoyl)pyrrolidin-2-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-benzyl-4-methyl-2-[(2R)-1-pyrimidin-2-ylpyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C23H24N6O
8-benzyl-4-methyl-2-[(2R)-1-pyrimidin-2-ylpyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-(cyclopropylmethyl)-2-[(3S)-1-[2-(4-fluorophenyl)acetyl]piperidin-3-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C25H29FN4O2
8-(cyclopropylmethyl)-2-[(3S)-1-[2-(4-fluorophenyl)acetyl]piperidin-3-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-[(4-Fluorophenyl)methyl]-4-methyl-2-(1-propan-2-ylpiperidin-4-yl)-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C23H29FN4O
8-[(4-Fluorophenyl)methyl]-4-methyl-2-(1-propan-2-ylpiperidin-4-yl)-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-Benzyl-2-[1-[2-(diethylamino)acetyl]piperidin-4-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C26H35N5O2
8-Benzyl-2-[1-[2-(diethylamino)acetyl]piperidin-4-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-(Cyclopropylmethyl)-4-methyl-2-[1-(3-morpholin-4-ylpropanoyl)piperidin-4-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C24H35N5O3
8-(Cyclopropylmethyl)-4-methyl-2-[1-(3-morpholin-4-ylpropanoyl)piperidin-4-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-benzyl-4-methyl-2-[1-[2-[(2R)-oxolan-2-yl]acetyl]piperidin-4-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C26H32N4O3
8-benzyl-4-methyl-2-[1-[2-[(2R)-oxolan-2-yl]acetyl]piperidin-4-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-benzyl-4-methyl-2-[1-[2-[(2S)-oxolan-2-yl]acetyl]piperidin-4-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C26H32N4O3
8-benzyl-4-methyl-2-[1-[2-[(2S)-oxolan-2-yl]acetyl]piperidin-4-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-cyclopentyl-4-methyl-2-[1-[3-[(2R)-oxolan-2-yl]propanoyl]piperidin-4-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C25H36N4O3
8-cyclopentyl-4-methyl-2-[1-[3-[(2R)-oxolan-2-yl]propanoyl]piperidin-4-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-(cyclopropylmethyl)-4-methyl-2-[(3S)-1-(3-phenylpropanoyl)piperidin-3-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C26H32N4O2
8-(cyclopropylmethyl)-4-methyl-2-[(3S)-1-(3-phenylpropanoyl)piperidin-3-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-(cyclohexylmethyl)-2-[(2R)-1-(2-hydroxyacetyl)pyrrolidin-2-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C21H30N4O3
8-(cyclohexylmethyl)-2-[(2R)-1-(2-hydroxyacetyl)pyrrolidin-2-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-benzyl-4-methyl-2-[(2R)-1-(2-oxo-2-pyrrolidin-1-ylethyl)pyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C25H31N5O2
8-benzyl-4-methyl-2-[(2R)-1-(2-oxo-2-pyrrolidin-1-ylethyl)pyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-(cyclopropylmethyl)-4-methyl-2-[(3R)-1-(2-phenoxyacetyl)piperidin-3-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C25H30N4O3
8-(cyclopropylmethyl)-4-methyl-2-[(3R)-1-(2-phenoxyacetyl)piperidin-3-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-(cyclopropylmethyl)-4-methyl-2-[(3S)-1-(2-phenoxyacetyl)piperidin-3-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C25H30N4O3
8-(cyclopropylmethyl)-4-methyl-2-[(3S)-1-(2-phenoxyacetyl)piperidin-3-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-(cyclohexylmethyl)-2-[(2R)-1-(2-hydroxy-2-methylpropanoyl)pyrrolidin-2-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C23H34N4O3
8-(cyclohexylmethyl)-2-[(2R)-1-(2-hydroxy-2-methylpropanoyl)pyrrolidin-2-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-(cyclopropylmethyl)-4-methyl-2-[(3S)-1-(5-propyl-1,2-oxazole-3-carbonyl)piperidin-3-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C24H31N5O3
8-(cyclopropylmethyl)-4-methyl-2-[(3S)-1-(5-propyl-1,2-oxazole-3-carbonyl)piperidin-3-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one