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中文名称 英文名称 CAS号 化学式 结构式图片
—— (8aS)-4-amino-8a-phenyl-2-pyrrolidin-1-yl-7,8-dihydropyrrolo[1,2-a][1,3,5]triazin-6-one —— C16H19N5O
(8aS)-4-amino-8a-phenyl-2-pyrrolidin-1-yl-7,8-dihydropyrrolo[1,2-a][1,3,5]triazin-6-one
—— (8S)-3-cyclohexyl-8-(2-methoxynaphthalen-1-yl)-6-oxo-2,4,7,8-tetrahydropyrido[2,1-b][1,3,5]thiadiazine-9-carbonitrile —— C25H27N3O2S
(8S)-3-cyclohexyl-8-(2-methoxynaphthalen-1-yl)-6-oxo-2,4,7,8-tetrahydropyrido[2,1-b][1,3,5]thiadiazine-9-carbonitrile
—— (8R)-3-(furan-2-ylmethyl)-6-oxo-8-phenyl-2,4,7,8-tetrahydropyrido[2,1-b][1,3,5]thiadiazine-9-carbonitrile —— C19H17N3O2S
(8R)-3-(furan-2-ylmethyl)-6-oxo-8-phenyl-2,4,7,8-tetrahydropyrido[2,1-b][1,3,5]thiadiazine-9-carbonitrile
—— (8R)-8-(4-methoxyphenyl)-3-methyl-6-oxo-2,4,7,8-tetrahydropyrido[2,1-b][1,3,5]thiadiazine-9-carbonitrile —— C16H17N3O2S
(8R)-8-(4-methoxyphenyl)-3-methyl-6-oxo-2,4,7,8-tetrahydropyrido[2,1-b][1,3,5]thiadiazine-9-carbonitrile
—— (8S)-8-(3-bromophenyl)-3-methyl-6-oxo-2,4,7,8-tetrahydropyrido[2,1-b][1,3,5]thiadiazine-9-carbonitrile —— C15H14BrN3OS
(8S)-8-(3-bromophenyl)-3-methyl-6-oxo-2,4,7,8-tetrahydropyrido[2,1-b][1,3,5]thiadiazine-9-carbonitrile
—— (8S)-3-methyl-8-(4-methylsulfanylphenyl)-6-oxo-2,4,7,8-tetrahydropyrido[2,1-b][1,3,5]thiadiazine-9-carbonitrile —— C16H17N3OS2
(8S)-3-methyl-8-(4-methylsulfanylphenyl)-6-oxo-2,4,7,8-tetrahydropyrido[2,1-b][1,3,5]thiadiazine-9-carbonitrile
—— (8R)-3-(3-chlorophenyl)-8-(3-nitrophenyl)-6-oxo-2,4,7,8-tetrahydropyrido[2,1-b][1,3,5]thiadiazine-9-carbonitrile —— C20H15ClN4O3S
(8R)-3-(3-chlorophenyl)-8-(3-nitrophenyl)-6-oxo-2,4,7,8-tetrahydropyrido[2,1-b][1,3,5]thiadiazine-9-carbonitrile
—— 8-nitro-2-[(E)-2-(1,3,5-trimethylpyrazol-4-yl)ethenyl]quinoline —— C17H16N4O2
8-nitro-2-[(E)-2-(1,3,5-trimethylpyrazol-4-yl)ethenyl]quinoline
—— 8-[[(2S,6S)-2,6-dimethylmorpholin-4-yl]methyl]-1,3-dimethyl-7-phenacylpurine-2,6-dione —— C22H27N5O4
8-[[(2S,6S)-2,6-dimethylmorpholin-4-yl]methyl]-1,3-dimethyl-7-phenacylpurine-2,6-dione
—— 8-nitro-2-[(E)-2-thiophen-2-ylethenyl]quinoline —— C15H10N2O2S
8-nitro-2-[(E)-2-thiophen-2-ylethenyl]quinoline
—— 8-chloro-1,3-dimethyl-7-[(3Z)-2-oxo-3-(1,3,3-trimethylindol-2-ylidene)propyl]purine-2,6-dione —— C21H22ClN5O3
8-chloro-1,3-dimethyl-7-[(3Z)-2-oxo-3-(1,3,3-trimethylindol-2-ylidene)propyl]purine-2,6-dione
—— 8-chloro-N-[3-[(2R)-2-ethylpiperidin-1-yl]propyl]-6-methylbenzo[b][1,4]benzothiazepine-3-carboxamide —— C25H30ClN3OS
8-chloro-N-[3-[(2R)-2-ethylpiperidin-1-yl]propyl]-6-methylbenzo[b][1,4]benzothiazepine-3-carboxamide
—— 8-chloro-N-[3-[(2R,6R)-2,6-dimethylpiperidin-1-yl]propyl]-6-methylbenzo[b][1,4]benzothiazepine-3-carboxamide —— C25H30ClN3OS
8-chloro-N-[3-[(2R,6R)-2,6-dimethylpiperidin-1-yl]propyl]-6-methylbenzo[b][1,4]benzothiazepine-3-carboxamide
—— (8S)-6-amino-8-[3-(4-fluorophenyl)-1,2-oxazol-4-yl]-2-(hydroxymethyl)-4-oxo-5,8-dihydropyrano[3,2-b]pyridine-7-carbonitrile —— C19H13FN4O4
(8S)-6-amino-8-[3-(4-fluorophenyl)-1,2-oxazol-4-yl]-2-(hydroxymethyl)-4-oxo-5,8-dihydropyrano[3,2-b]pyridine-7-carbonitrile
—— 8-[[5-(2-Methoxyphenyl)-1,3,4-oxadiazol-2-yl]carbamoyl]naphthalene-1-carboxylic acid —— C21H15N3O5
8-[[5-(2-Methoxyphenyl)-1,3,4-oxadiazol-2-yl]carbamoyl]naphthalene-1-carboxylic acid
—— 8-[(2S)-1-naphthalen-2-ylsulfonylpropan-2-yl]-1,4-dioxa-8-azaspiro[4.5]decane —— C20H25NO4S
8-[(2S)-1-naphthalen-2-ylsulfonylpropan-2-yl]-1,4-dioxa-8-azaspiro[4.5]decane
—— (8R,8aR)-6-amino-8-(2-ethoxyphenyl)-2-methyl-1,3,8,8a-tetrahydroisoquinoline-5,7,7-tricarbonitrile —— C21H21N5O
(8R,8aR)-6-amino-8-(2-ethoxyphenyl)-2-methyl-1,3,8,8a-tetrahydroisoquinoline-5,7,7-tricarbonitrile
—— (8S,8aS)-6-amino-8-[4-(dimethylamino)phenyl]-2-methyl-1,3,8,8a-tetrahydroisoquinoline-5,7,7-tricarbonitrile —— C21H22N6
(8S,8aS)-6-amino-8-[4-(dimethylamino)phenyl]-2-methyl-1,3,8,8a-tetrahydroisoquinoline-5,7,7-tricarbonitrile
—— 8-(cyclopropylmethyl)-2-[(3S)-1-[(1,5-dimethylpyrazol-4-yl)methyl]piperidin-3-yl]-4-methyl-6,7-dihydro-5H-pyrido[2,3-d]pyrimidine —— C23H34N6
8-(cyclopropylmethyl)-2-[(3S)-1-[(1,5-dimethylpyrazol-4-yl)methyl]piperidin-3-yl]-4-methyl-6,7-dihydro-5H-pyrido[2,3-d]pyrimidine
—— 8-methyl-N-[(1R)-6-morpholin-4-ylsulfonyl-2,3-dihydro-1H-inden-1-yl]imidazo[1,2-a]pyridine-2-carboxamide —— C22H24N4O4S
8-methyl-N-[(1R)-6-morpholin-4-ylsulfonyl-2,3-dihydro-1H-inden-1-yl]imidazo[1,2-a]pyridine-2-carboxamide
—— (8-methylimidazo[1,2-a]pyridin-2-yl)-[(2S)-2-methyl-2-(morpholine-4-carbonyl)pyrrolidin-1-yl]methanone —— C19H24N4O3
(8-methylimidazo[1,2-a]pyridin-2-yl)-[(2S)-2-methyl-2-(morpholine-4-carbonyl)pyrrolidin-1-yl]methanone
—— 8-methyl-N-[1-[2-oxo-2-[[(2S)-oxolan-2-yl]methylamino]ethyl]pyrazol-4-yl]imidazo[1,2-a]pyridine-2-carboxamide —— C19H22N6O3
8-methyl-N-[1-[2-oxo-2-[[(2S)-oxolan-2-yl]methylamino]ethyl]pyrazol-4-yl]imidazo[1,2-a]pyridine-2-carboxamide
—— 8-methyl-N-[1-[2-oxo-2-[3-(trifluoromethyl)anilino]ethyl]pyrazol-4-yl]imidazo[1,2-a]pyridine-2-carboxamide —— C21H17F3N6O2
8-methyl-N-[1-[2-oxo-2-[3-(trifluoromethyl)anilino]ethyl]pyrazol-4-yl]imidazo[1,2-a]pyridine-2-carboxamide
—— 8-(cyclohexylmethyl)-4-methyl-2-[(2S)-1-(2-phenylacetyl)pyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C27H34N4O2
8-(cyclohexylmethyl)-4-methyl-2-[(2S)-1-(2-phenylacetyl)pyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-[(4-fluorophenyl)methyl]-4-methyl-2-[(2R)-1-(1H-pyrazole-5-carbonyl)pyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C23H23FN6O2
8-[(4-fluorophenyl)methyl]-4-methyl-2-[(2R)-1-(1H-pyrazole-5-carbonyl)pyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-(cyclohexylmethyl)-2-[(2R)-1-(2-cyclopentylacetyl)pyrrolidin-2-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C26H38N4O2
8-(cyclohexylmethyl)-2-[(2R)-1-(2-cyclopentylacetyl)pyrrolidin-2-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-[(2-methoxyphenyl)methyl]-4-methyl-2-[(2S)-1-[(1-methylpyrazol-4-yl)methyl]pyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C25H30N6O2
8-[(2-methoxyphenyl)methyl]-4-methyl-2-[(2S)-1-[(1-methylpyrazol-4-yl)methyl]pyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-(cyclohexylmethyl)-4-methyl-2-[(2S)-1-(thiadiazole-4-carbonyl)pyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C22H28N6O2S
8-(cyclohexylmethyl)-4-methyl-2-[(2S)-1-(thiadiazole-4-carbonyl)pyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-[(2-fluorophenyl)methyl]-2-[(3R)-1-(2-hydroxyacetyl)piperidin-3-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C22H25FN4O3
8-[(2-fluorophenyl)methyl]-2-[(3R)-1-(2-hydroxyacetyl)piperidin-3-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-benzyl-2-[(2R)-1-[(1,3-dimethylpyrazol-4-yl)methyl]pyrrolidin-2-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C25H30N6O
8-benzyl-2-[(2R)-1-[(1,3-dimethylpyrazol-4-yl)methyl]pyrrolidin-2-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-[(4-fluorophenyl)methyl]-4-methyl-2-[(2S)-1-(5-methyl-1H-pyrazole-4-carbonyl)pyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C24H25FN6O2
8-[(4-fluorophenyl)methyl]-4-methyl-2-[(2S)-1-(5-methyl-1H-pyrazole-4-carbonyl)pyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-benzyl-4-methyl-2-[(3R)-1-(2-propan-2-yloxyacetyl)piperidin-3-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C25H32N4O3
8-benzyl-4-methyl-2-[(3R)-1-(2-propan-2-yloxyacetyl)piperidin-3-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-(cyclopropylmethyl)-4-methyl-2-[(2S)-1-[2-(methylamino)pyridine-4-carbonyl]piperidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C24H30N6O2
8-(cyclopropylmethyl)-4-methyl-2-[(2S)-1-[2-(methylamino)pyridine-4-carbonyl]piperidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-methyl-3-[(3S)-3-phenylpiperidine-1-carbonyl]pyrido[1,2-a]pyrimidin-4-one —— C21H21N3O2
8-methyl-3-[(3S)-3-phenylpiperidine-1-carbonyl]pyrido[1,2-a]pyrimidin-4-one
—— 8-[(4-methoxyphenyl)methyl]-4-methyl-2-[(3S)-1-propylpiperidin-3-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C24H32N4O2
8-[(4-methoxyphenyl)methyl]-4-methyl-2-[(3S)-1-propylpiperidin-3-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-(cyclohexylmethyl)-2-[(2R)-1-(3-methoxypropanoyl)pyrrolidin-2-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C23H34N4O3
8-(cyclohexylmethyl)-2-[(2R)-1-(3-methoxypropanoyl)pyrrolidin-2-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-(cyclopropylmethyl)-2-[(3S)-1-[(1,3-dimethylpyrazol-4-yl)methyl]piperidin-3-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C23H32N6O
8-(cyclopropylmethyl)-2-[(3S)-1-[(1,3-dimethylpyrazol-4-yl)methyl]piperidin-3-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-benzyl-2-[(3S)-1-[2-(diethylamino)acetyl]piperidin-3-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C26H35N5O2
8-benzyl-2-[(3S)-1-[2-(diethylamino)acetyl]piperidin-3-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-[(4-fluorophenyl)methyl]-2-[(2S)-1-(2-methoxy-2-methylpropanoyl)pyrrolidin-2-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C24H29FN4O3
8-[(4-fluorophenyl)methyl]-2-[(2S)-1-(2-methoxy-2-methylpropanoyl)pyrrolidin-2-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-(cyclopropylmethyl)-4-methyl-2-[(3R)-1-pyrrolidin-1-ylsulfonylpiperidin-3-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C21H31N5O3S
8-(cyclopropylmethyl)-4-methyl-2-[(3R)-1-pyrrolidin-1-ylsulfonylpiperidin-3-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-(cyclopropylmethyl)-4-methyl-2-[(2R)-1-(2-propan-2-yloxyacetyl)piperidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C22H32N4O3
8-(cyclopropylmethyl)-4-methyl-2-[(2R)-1-(2-propan-2-yloxyacetyl)piperidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-benzyl-2-[(2S)-1-(2-methoxy-2-methylpropanoyl)piperidin-2-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C25H32N4O3
8-benzyl-2-[(2S)-1-(2-methoxy-2-methylpropanoyl)piperidin-2-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-(cyclopropylmethyl)-2-[(3S)-1-[2-(3,4-dimethylphenyl)acetyl]piperidin-3-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C27H34N4O2
8-(cyclopropylmethyl)-2-[(3S)-1-[2-(3,4-dimethylphenyl)acetyl]piperidin-3-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-benzyl-4-methyl-2-[(3R)-1-(1-methylpyrazole-4-carbonyl)piperidin-3-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C25H28N6O2
8-benzyl-4-methyl-2-[(3R)-1-(1-methylpyrazole-4-carbonyl)piperidin-3-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-(cyclopropylmethyl)-4-methyl-2-[(2S)-1-[2-(4-methylpiperidin-1-yl)acetyl]piperidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C25H37N5O2
8-(cyclopropylmethyl)-4-methyl-2-[(2S)-1-[2-(4-methylpiperidin-1-yl)acetyl]piperidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-benzyl-2-[(3R)-1-(2-methoxy-2-methylpropanoyl)piperidin-3-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C25H32N4O3
8-benzyl-2-[(3R)-1-(2-methoxy-2-methylpropanoyl)piperidin-3-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-(cyclopropylmethyl)-4-methyl-2-[(2R)-1-(5-propan-2-yl-1H-pyrazole-3-carbonyl)piperidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C24H32N6O2
8-(cyclopropylmethyl)-4-methyl-2-[(2R)-1-(5-propan-2-yl-1H-pyrazole-3-carbonyl)piperidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-(cyclopropylmethyl)-2-[(3R)-1-[(4-methoxyphenyl)methyl]piperidin-3-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C25H32N4O2
8-(cyclopropylmethyl)-2-[(3R)-1-[(4-methoxyphenyl)methyl]piperidin-3-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-[(2-methoxyphenyl)methyl]-4-methyl-2-[(2S)-1-(3-methylbutanoyl)pyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C25H32N4O3
8-[(2-methoxyphenyl)methyl]-4-methyl-2-[(2S)-1-(3-methylbutanoyl)pyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-(cyclopropylmethyl)-4-methyl-2-[(3R)-1-(1-methylimidazol-4-yl)sulfonylpiperidin-3-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C21H28N6O3S
8-(cyclopropylmethyl)-4-methyl-2-[(3R)-1-(1-methylimidazol-4-yl)sulfonylpiperidin-3-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one