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—— (8S,9R,13S,14R,17E)-17-[(Z)-(1-ethyl-5-methylpyrazol-4-yl)methylidenehydrazinylidene]-13-methyl-7,8,9,11,12,14,15,16-octahydro-6H-cyclopenta[a]phenanthren-3-ol —— C25H32N4O
(8S,9R,13S,14R,17E)-17-[(Z)-(1-ethyl-5-methylpyrazol-4-yl)methylidenehydrazinylidene]-13-methyl-7,8,9,11,12,14,15,16-octahydro-6H-cyclopenta[a]phenanthren-3-ol
—— (8S,9R,13S,14S,17E)-13-methyl-17-[(E)-(2-propylpyrazol-3-yl)methylidenehydrazinylidene]-7,8,9,11,12,14,15,16-octahydro-6H-cyclopenta[a]phenanthren-3-ol —— C25H32N4O
(8S,9R,13S,14S,17E)-13-methyl-17-[(E)-(2-propylpyrazol-3-yl)methylidenehydrazinylidene]-7,8,9,11,12,14,15,16-octahydro-6H-cyclopenta[a]phenanthren-3-ol
—— (8S,8aS)-6-amino-8-[2-[(2-chlorophenyl)methoxy]phenyl]-1,3,8,8a-tetrahydroisochromene-5,7,7-tricarbonitrile —— C25H19ClN4O2
(8S,8aS)-6-amino-8-[2-[(2-chlorophenyl)methoxy]phenyl]-1,3,8,8a-tetrahydroisochromene-5,7,7-tricarbonitrile
—— (8R,9R,13S,14R,16E)-16-[(1,5-dimethylpyrazol-4-yl)methylidene]-3-hydroxy-13-methyl-6,7,8,9,11,12,14,15-octahydrocyclopenta[a]phenanthren-17-one —— C24H28N2O2
(8R,9R,13S,14R,16E)-16-[(1,5-dimethylpyrazol-4-yl)methylidene]-3-hydroxy-13-methyl-6,7,8,9,11,12,14,15-octahydrocyclopenta[a]phenanthren-17-one
—— (8S,9R,13S,14R,17E)-13-methyl-17-[(Z)-(1,3,5-trimethylpyrazol-4-yl)methylidenehydrazinylidene]-7,8,9,11,12,14,15,16-octahydro-6H-cyclopenta[a]phenanthren-3-ol —— C25H32N4O
(8S,9R,13S,14R,17E)-13-methyl-17-[(Z)-(1,3,5-trimethylpyrazol-4-yl)methylidenehydrazinylidene]-7,8,9,11,12,14,15,16-octahydro-6H-cyclopenta[a]phenanthren-3-ol
—— (8S,9R,13R,14S,17E)-17-[(Z)-(1-ethyl-5-methylpyrazol-4-yl)methylidenehydrazinylidene]-13-methyl-7,8,9,11,12,14,15,16-octahydro-6H-cyclopenta[a]phenanthren-3-ol —— C25H32N4O
(8S,9R,13R,14S,17E)-17-[(Z)-(1-ethyl-5-methylpyrazol-4-yl)methylidenehydrazinylidene]-13-methyl-7,8,9,11,12,14,15,16-octahydro-6H-cyclopenta[a]phenanthren-3-ol
—— (8S,9R,13R,14R,17E)-17-[(Z)-(1-ethyl-5-methylpyrazol-4-yl)methylidenehydrazinylidene]-13-methyl-7,8,9,11,12,14,15,16-octahydro-6H-cyclopenta[a]phenanthren-3-ol —— C25H32N4O
(8S,9R,13R,14R,17E)-17-[(Z)-(1-ethyl-5-methylpyrazol-4-yl)methylidenehydrazinylidene]-13-methyl-7,8,9,11,12,14,15,16-octahydro-6H-cyclopenta[a]phenanthren-3-ol
—— (8S,9S,13R,14S,16Z)-3-methoxy-16-[(4-methoxyphenyl)methylidene]-13-methyl-6,7,8,9,11,12,14,15-octahydrocyclopenta[a]phenanthren-17-one —— C27H30O3
(8S,9S,13R,14S,16Z)-3-methoxy-16-[(4-methoxyphenyl)methylidene]-13-methyl-6,7,8,9,11,12,14,15-octahydrocyclopenta[a]phenanthren-17-one
—— (8S,9R,13S,14S,17Z)-13-methyl-17-[(E)-(2-propylpyrazol-3-yl)methylidenehydrazinylidene]-7,8,9,11,12,14,15,16-octahydro-6H-cyclopenta[a]phenanthren-3-ol —— C25H32N4O
(8S,9R,13S,14S,17Z)-13-methyl-17-[(E)-(2-propylpyrazol-3-yl)methylidenehydrazinylidene]-7,8,9,11,12,14,15,16-octahydro-6H-cyclopenta[a]phenanthren-3-ol
—— (8S,9R,13R,14R,17E)-13-methyl-17-[(Z)-(1,3,5-trimethylpyrazol-4-yl)methylidenehydrazinylidene]-7,8,9,11,12,14,15,16-octahydro-6H-cyclopenta[a]phenanthren-3-ol —— C25H32N4O
(8S,9R,13R,14R,17E)-13-methyl-17-[(Z)-(1,3,5-trimethylpyrazol-4-yl)methylidenehydrazinylidene]-7,8,9,11,12,14,15,16-octahydro-6H-cyclopenta[a]phenanthren-3-ol
—— (8R,9R,13S,14S,16Z)-16-[(1,5-dimethylpyrazol-4-yl)methylidene]-3-methoxy-13-methyl-6,7,8,9,11,12,14,15-octahydrocyclopenta[a]phenanthren-17-one —— C25H30N2O2
(8R,9R,13S,14S,16Z)-16-[(1,5-dimethylpyrazol-4-yl)methylidene]-3-methoxy-13-methyl-6,7,8,9,11,12,14,15-octahydrocyclopenta[a]phenanthren-17-one
—— (8S,9S,13S,14S,16Z)-3-methoxy-16-[(4-methoxyphenyl)methylidene]-13-methyl-6,7,8,9,11,12,14,15-octahydrocyclopenta[a]phenanthren-17-one —— C27H30O3
(8S,9S,13S,14S,16Z)-3-methoxy-16-[(4-methoxyphenyl)methylidene]-13-methyl-6,7,8,9,11,12,14,15-octahydrocyclopenta[a]phenanthren-17-one
—— (8R,9R,13S,14R,16Z)-3-methoxy-13-methyl-16-[(2-propylpyrazol-3-yl)methylidene]-6,7,8,9,11,12,14,15-octahydrocyclopenta[a]phenanthren-17-one —— C26H32N2O2
(8R,9R,13S,14R,16Z)-3-methoxy-13-methyl-16-[(2-propylpyrazol-3-yl)methylidene]-6,7,8,9,11,12,14,15-octahydrocyclopenta[a]phenanthren-17-one
—— (8R,9R,13S,14S,16E)-16-[(1,5-dimethylpyrazol-4-yl)methylidene]-3-hydroxy-13-methyl-6,7,8,9,11,12,14,15-octahydrocyclopenta[a]phenanthren-17-one —— C24H28N2O2
(8R,9R,13S,14S,16E)-16-[(1,5-dimethylpyrazol-4-yl)methylidene]-3-hydroxy-13-methyl-6,7,8,9,11,12,14,15-octahydrocyclopenta[a]phenanthren-17-one
—— (8S,9R,13S,14R,17E)-17-[(Z)-(1,5-dimethylpyrazol-4-yl)methylidenehydrazinylidene]-13-methyl-7,8,9,11,12,14,15,16-octahydro-6H-cyclopenta[a]phenanthren-3-ol —— C24H30N4O
(8S,9R,13S,14R,17E)-17-[(Z)-(1,5-dimethylpyrazol-4-yl)methylidenehydrazinylidene]-13-methyl-7,8,9,11,12,14,15,16-octahydro-6H-cyclopenta[a]phenanthren-3-ol
—— (8R,9R,13S,14R,16Z)-16-[(1,3-dimethylpyrazol-4-yl)methylidene]-3-methoxy-13-methyl-6,7,8,9,11,12,14,15-octahydrocyclopenta[a]phenanthren-17-one —— C25H30N2O2
(8R,9R,13S,14R,16Z)-16-[(1,3-dimethylpyrazol-4-yl)methylidene]-3-methoxy-13-methyl-6,7,8,9,11,12,14,15-octahydrocyclopenta[a]phenanthren-17-one
—— (8S,9R,13S,14S,17E)-13-methyl-17-[(Z)-(2-propylpyrazol-3-yl)methylidenehydrazinylidene]-7,8,9,11,12,14,15,16-octahydro-6H-cyclopenta[a]phenanthren-3-ol —— C25H32N4O
(8S,9R,13S,14S,17E)-13-methyl-17-[(Z)-(2-propylpyrazol-3-yl)methylidenehydrazinylidene]-7,8,9,11,12,14,15,16-octahydro-6H-cyclopenta[a]phenanthren-3-ol
—— (8S,9R,13R,14S,17E)-13-methyl-17-[(Z)-(1,3,5-trimethylpyrazol-4-yl)methylidenehydrazinylidene]-7,8,9,11,12,14,15,16-octahydro-6H-cyclopenta[a]phenanthren-3-ol —— C25H32N4O
(8S,9R,13R,14S,17E)-13-methyl-17-[(Z)-(1,3,5-trimethylpyrazol-4-yl)methylidenehydrazinylidene]-7,8,9,11,12,14,15,16-octahydro-6H-cyclopenta[a]phenanthren-3-ol
—— (8S,9R,13S,14R,17E)-17-[(Z)-(1-ethyl-3-methylpyrazol-4-yl)methylidenehydrazinylidene]-13-methyl-7,8,9,11,12,14,15,16-octahydro-6H-cyclopenta[a]phenanthren-3-ol —— C25H32N4O
(8S,9R,13S,14R,17E)-17-[(Z)-(1-ethyl-3-methylpyrazol-4-yl)methylidenehydrazinylidene]-13-methyl-7,8,9,11,12,14,15,16-octahydro-6H-cyclopenta[a]phenanthren-3-ol
—— (8R,9R,13S,14S,16Z)-3-methoxy-13-methyl-16-[(2-propylpyrazol-3-yl)methylidene]-6,7,8,9,11,12,14,15-octahydrocyclopenta[a]phenanthren-17-one —— C26H32N2O2
(8R,9R,13S,14S,16Z)-3-methoxy-13-methyl-16-[(2-propylpyrazol-3-yl)methylidene]-6,7,8,9,11,12,14,15-octahydrocyclopenta[a]phenanthren-17-one
—— (8S,9R,13R,14S,17E)-17-[(Z)-(1,5-dimethylpyrazol-4-yl)methylidenehydrazinylidene]-13-methyl-7,8,9,11,12,14,15,16-octahydro-6H-cyclopenta[a]phenanthren-3-ol —— C24H30N4O
(8S,9R,13R,14S,17E)-17-[(Z)-(1,5-dimethylpyrazol-4-yl)methylidenehydrazinylidene]-13-methyl-7,8,9,11,12,14,15,16-octahydro-6H-cyclopenta[a]phenanthren-3-ol
—— (8S,9R,13R,14S,17E)-17-[(Z)-(1-ethyl-3-methylpyrazol-4-yl)methylidenehydrazinylidene]-13-methyl-7,8,9,11,12,14,15,16-octahydro-6H-cyclopenta[a]phenanthren-3-ol —— C25H32N4O
(8S,9R,13R,14S,17E)-17-[(Z)-(1-ethyl-3-methylpyrazol-4-yl)methylidenehydrazinylidene]-13-methyl-7,8,9,11,12,14,15,16-octahydro-6H-cyclopenta[a]phenanthren-3-ol
—— (8R,9R,13S,14R,16Z)-16-[(1,5-dimethylpyrazol-4-yl)methylidene]-3-methoxy-13-methyl-6,7,8,9,11,12,14,15-octahydrocyclopenta[a]phenanthren-17-one —— C25H30N2O2
(8R,9R,13S,14R,16Z)-16-[(1,5-dimethylpyrazol-4-yl)methylidene]-3-methoxy-13-methyl-6,7,8,9,11,12,14,15-octahydrocyclopenta[a]phenanthren-17-one
—— (8R,9R,13S,14S,16Z)-16-[(1,3-dimethylpyrazol-4-yl)methylidene]-3-methoxy-13-methyl-6,7,8,9,11,12,14,15-octahydrocyclopenta[a]phenanthren-17-one —— C25H30N2O2
(8R,9R,13S,14S,16Z)-16-[(1,3-dimethylpyrazol-4-yl)methylidene]-3-methoxy-13-methyl-6,7,8,9,11,12,14,15-octahydrocyclopenta[a]phenanthren-17-one
—— (8R,8aS)-6-amino-2-propyl-8-[3-(trifluoromethyl)phenyl]-1,3,8,8a-tetrahydroisoquinoline-5,7,7-tricarbonitrile —— C22H20F3N5
(8R,8aS)-6-amino-2-propyl-8-[3-(trifluoromethyl)phenyl]-1,3,8,8a-tetrahydroisoquinoline-5,7,7-tricarbonitrile
—— (8S,11S)-3-benzylsulfanyl-8-methyl-11-propan-2-yl-3-prop-2-enyl-1,5-dioxaspiro[5.5]undecane-2,4-dione —— C23H30O4S
(8S,11S)-3-benzylsulfanyl-8-methyl-11-propan-2-yl-3-prop-2-enyl-1,5-dioxaspiro[5.5]undecane-2,4-dione
—— (8R,11S)-3-benzylsulfanyl-8-methyl-11-propan-2-yl-3-prop-2-enyl-1,5-dioxaspiro[5.5]undecane-2,4-dione —— C23H30O4S
(8R,11S)-3-benzylsulfanyl-8-methyl-11-propan-2-yl-3-prop-2-enyl-1,5-dioxaspiro[5.5]undecane-2,4-dione
—— (8S,11R)-3-benzylsulfanyl-8-methyl-11-propan-2-yl-3-prop-2-enyl-1,5-dioxaspiro[5.5]undecane-2,4-dione —— C23H30O4S
(8S,11R)-3-benzylsulfanyl-8-methyl-11-propan-2-yl-3-prop-2-enyl-1,5-dioxaspiro[5.5]undecane-2,4-dione
—— (8R,11R)-3-benzylsulfanyl-8-methyl-11-propan-2-yl-3-prop-2-enyl-1,5-dioxaspiro[5.5]undecane-2,4-dione —— C23H30O4S
(8R,11R)-3-benzylsulfanyl-8-methyl-11-propan-2-yl-3-prop-2-enyl-1,5-dioxaspiro[5.5]undecane-2,4-dione
—— 8-[(2E)-2-[(E)-2-bromo-3-phenylprop-2-enylidene]hydrazinyl]-7-[(4-chlorophenyl)methyl]-3-methylpurine-2,6-dione —— C22H18BrClN6O2
8-[(2E)-2-[(E)-2-bromo-3-phenylprop-2-enylidene]hydrazinyl]-7-[(4-chlorophenyl)methyl]-3-methylpurine-2,6-dione
—— (8S,8aS)-6-amino-2-methyl-8-(4-nitrothiophen-2-yl)-1,3,8,8a-tetrahydroisoquinoline-5,7,7-tricarbonitrile —— C17H14N6O2S
(8S,8aS)-6-amino-2-methyl-8-(4-nitrothiophen-2-yl)-1,3,8,8a-tetrahydroisoquinoline-5,7,7-tricarbonitrile
—— 8-O-benzyl 6-O-ethyl (1R,2R,3R,7S)-3,10-dimethyl-4-oxo-9-oxa-5,6,8-triazatricyclo[5.2.2.02,5]undec-10-ene-6,8-dicarboxylate —— C20H23N3O6
8-O-benzyl 6-O-ethyl (1R,2R,3R,7S)-3,10-dimethyl-4-oxo-9-oxa-5,6,8-triazatricyclo[5.2.2.02,5]undec-10-ene-6,8-dicarboxylate
—— (8S,8aR)-6-amino-2-methyl-8-(4-nitrothiophen-2-yl)-1,3,8,8a-tetrahydroisoquinoline-5,7,7-tricarbonitrile —— C17H14N6O2S
(8S,8aR)-6-amino-2-methyl-8-(4-nitrothiophen-2-yl)-1,3,8,8a-tetrahydroisoquinoline-5,7,7-tricarbonitrile
—— 8-O-benzyl 6-O-ethyl (1S,2R,3R,7R)-3,10-dimethyl-4-oxo-9-oxa-5,6,8-triazatricyclo[5.2.2.02,5]undec-10-ene-6,8-dicarboxylate —— C20H23N3O6
8-O-benzyl 6-O-ethyl (1S,2R,3R,7R)-3,10-dimethyl-4-oxo-9-oxa-5,6,8-triazatricyclo[5.2.2.02,5]undec-10-ene-6,8-dicarboxylate
—— (8S,9S,13S,14S,17E)-13-methyl-17-(methylhydrazinylidene)-7,8,9,11,12,14,15,16-octahydro-6H-cyclopenta[a]phenanthren-3-ol —— C19H26N2O
(8S,9S,13S,14S,17E)-13-methyl-17-(methylhydrazinylidene)-7,8,9,11,12,14,15,16-octahydro-6H-cyclopenta[a]phenanthren-3-ol
—— 8-methyl-2-[(1-methyltetrazol-5-yl)sulfanylmethyl]-3H-quinazolin-4-one —— C12H12N6OS
8-methyl-2-[(1-methyltetrazol-5-yl)sulfanylmethyl]-3H-quinazolin-4-one
—— 8-(4-Aminopiperidin-1-yl)-2-benzyl-[1,2,4]triazolo[4,3-a]pyrazin-3(2H)-one —— C17H20N6O
8-(4-Aminopiperidin-1-yl)-2-benzyl-[1,2,4]triazolo[4,3-a]pyrazin-3(2H)-one
—— 8-[(3R)-3-aminopyrrolidin-1-yl]-2-[(4-fluorophenyl)methyl]-[1,2,4]triazolo[4,3-a]pyrazin-3-one —— C16H17FN6O
8-[(3R)-3-aminopyrrolidin-1-yl]-2-[(4-fluorophenyl)methyl]-[1,2,4]triazolo[4,3-a]pyrazin-3-one
—— 8-[(3S)-3-aminopyrrolidin-1-yl]-2-benzyl-[1,2,4]triazolo[4,3-a]pyrazin-3-one —— C16H18N6O
8-[(3S)-3-aminopyrrolidin-1-yl]-2-benzyl-[1,2,4]triazolo[4,3-a]pyrazin-3-one
—— 8-[(3R)-3-aminopyrrolidin-1-yl]-2-[(3-fluorophenyl)methyl]-[1,2,4]triazolo[4,3-a]pyrazin-3-one —— C16H17FN6O
8-[(3R)-3-aminopyrrolidin-1-yl]-2-[(3-fluorophenyl)methyl]-[1,2,4]triazolo[4,3-a]pyrazin-3-one
—— 8-(4-Aminopiperidin-1-yl)-2-ethyl-[1,2,4]triazolo[4,3-a]pyrazin-3(2H)-one —— C12H18N6O
8-(4-Aminopiperidin-1-yl)-2-ethyl-[1,2,4]triazolo[4,3-a]pyrazin-3(2H)-one
—— 8-[(3S)-3-aminopyrrolidin-1-yl]-2-[(2-fluorophenyl)methyl]-[1,2,4]triazolo[4,3-a]pyrazin-3-one —— C16H17FN6O
8-[(3S)-3-aminopyrrolidin-1-yl]-2-[(2-fluorophenyl)methyl]-[1,2,4]triazolo[4,3-a]pyrazin-3-one
—— 8-[(3R)-3-aminopyrrolidin-1-yl]-2-[(2-fluorophenyl)methyl]-[1,2,4]triazolo[4,3-a]pyrazin-3-one —— C16H17FN6O
8-[(3R)-3-aminopyrrolidin-1-yl]-2-[(2-fluorophenyl)methyl]-[1,2,4]triazolo[4,3-a]pyrazin-3-one
—— 8-[(3R)-3-aminopyrrolidin-1-yl]-2-benzyl-[1,2,4]triazolo[4,3-a]pyrazin-3-one —— C16H18N6O
8-[(3R)-3-aminopyrrolidin-1-yl]-2-benzyl-[1,2,4]triazolo[4,3-a]pyrazin-3-one
—— 8-(4-Amino-piperidin-1-yl)-2-(3-fluoro-benzyl)-2H-[1,2,4]triazolo[4,3-a]pyrazin-3-one —— C17H19FN6O
8-(4-Amino-piperidin-1-yl)-2-(3-fluoro-benzyl)-2H-[1,2,4]triazolo[4,3-a]pyrazin-3-one
—— 8-(2-Fluorophenoxy)-[1,2,4]triazolo[4,3-a]pyrazin-3(2H)-one —— C11H7FN4O2
8-(2-Fluorophenoxy)-[1,2,4]triazolo[4,3-a]pyrazin-3(2H)-one
—— 8-[(3S)-3-aminopyrrolidin-1-yl]-2-[(4-fluorophenyl)methyl]-[1,2,4]triazolo[4,3-a]pyrazin-3-one —— C16H17FN6O
8-[(3S)-3-aminopyrrolidin-1-yl]-2-[(4-fluorophenyl)methyl]-[1,2,4]triazolo[4,3-a]pyrazin-3-one
—— 8-[(3S)-3-aminopyrrolidin-1-yl]-2-[(3-fluorophenyl)methyl]-[1,2,4]triazolo[4,3-a]pyrazin-3-one —— C16H17FN6O
8-[(3S)-3-aminopyrrolidin-1-yl]-2-[(3-fluorophenyl)methyl]-[1,2,4]triazolo[4,3-a]pyrazin-3-one
—— 8-(4-Aminopiperidin-1-yl)-2-(4-fluorobenzyl)-[1,2,4]triazolo[4,3-a]pyrazin-3(2H)-one —— C17H19FN6O
8-(4-Aminopiperidin-1-yl)-2-(4-fluorobenzyl)-[1,2,4]triazolo[4,3-a]pyrazin-3(2H)-one
—— [(8S)-8-methyl-6,7,8,9-tetrahydro-[1,2,4]triazolo[4,3-b]cinnolin-3-yl]methanamine —— C11H15N5
[(8S)-8-methyl-6,7,8,9-tetrahydro-[1,2,4]triazolo[4,3-b]cinnolin-3-yl]methanamine