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中文名称 英文名称 CAS号 化学式 结构式图片
—— 8-(Azepan-1-yl)-2-[(3-methylphenyl)methyl]-[1,2,4]triazolo[4,3-a]pyrazin-3-one —— C19H23N5O
8-(Azepan-1-yl)-2-[(3-methylphenyl)methyl]-[1,2,4]triazolo[4,3-a]pyrazin-3-one
—— 8-(Azepan-1-yl)-2-[[3-(4-methylsulfanylphenyl)-1,2,4-oxadiazol-5-yl]methyl]-[1,2,4]triazolo[4,3-a]pyrazin-3-one —— C21H23N7O2S
8-(Azepan-1-yl)-2-[[3-(4-methylsulfanylphenyl)-1,2,4-oxadiazol-5-yl]methyl]-[1,2,4]triazolo[4,3-a]pyrazin-3-one
—— 8-(3,4-dihydro-1H-isoquinolin-2-yl)-2-[(3-methoxyphenyl)methyl]-[1,2,4]triazolo[4,3-a]pyrazin-3-one —— C22H21N5O2
8-(3,4-dihydro-1H-isoquinolin-2-yl)-2-[(3-methoxyphenyl)methyl]-[1,2,4]triazolo[4,3-a]pyrazin-3-one
—— 8-(3,4-dihydro-1H-isoquinolin-2-yl)-2-[(3-fluoro-4-methoxyphenyl)methyl]-[1,2,4]triazolo[4,3-a]pyrazin-3-one —— C22H20FN5O2
8-(3,4-dihydro-1H-isoquinolin-2-yl)-2-[(3-fluoro-4-methoxyphenyl)methyl]-[1,2,4]triazolo[4,3-a]pyrazin-3-one
—— 8-(3,4-dihydro-1H-isoquinolin-2-yl)-2-[[3-(4-methylsulfanylphenyl)-1,2,4-oxadiazol-5-yl]methyl]-[1,2,4]triazolo[4,3-a]pyrazin-3-one —— C24H21N7O2S
8-(3,4-dihydro-1H-isoquinolin-2-yl)-2-[[3-(4-methylsulfanylphenyl)-1,2,4-oxadiazol-5-yl]methyl]-[1,2,4]triazolo[4,3-a]pyrazin-3-one
—— 8-(3,4-dihydro-1H-isoquinolin-2-yl)-2-[2-(4-fluorophenyl)-2-oxoethyl]-[1,2,4]triazolo[4,3-a]pyrazin-3-one —— C22H18FN5O2
8-(3,4-dihydro-1H-isoquinolin-2-yl)-2-[2-(4-fluorophenyl)-2-oxoethyl]-[1,2,4]triazolo[4,3-a]pyrazin-3-one
—— 8-(3,4-dihydro-1H-isoquinolin-2-yl)-2-[[3-[3-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl]methyl]-[1,2,4]triazolo[4,3-a]pyrazin-3-one —— C24H18F3N7O2
8-(3,4-dihydro-1H-isoquinolin-2-yl)-2-[[3-[3-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl]methyl]-[1,2,4]triazolo[4,3-a]pyrazin-3-one
—— 8-(3,4-dihydro-1H-isoquinolin-2-yl)-2-[(5-methyl-2-phenyl-1,3-oxazol-4-yl)methyl]-[1,2,4]triazolo[4,3-a]pyrazin-3-one —— C25H22N6O2
8-(3,4-dihydro-1H-isoquinolin-2-yl)-2-[(5-methyl-2-phenyl-1,3-oxazol-4-yl)methyl]-[1,2,4]triazolo[4,3-a]pyrazin-3-one
—— 8-(3,4-dihydro-1H-isoquinolin-2-yl)-2-[[3-(2,3-dimethoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl]-[1,2,4]triazolo[4,3-a]pyrazin-3-one —— C25H23N7O4
8-(3,4-dihydro-1H-isoquinolin-2-yl)-2-[[3-(2,3-dimethoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl]-[1,2,4]triazolo[4,3-a]pyrazin-3-one
—— 8-(2-Ethylphenyl)sulfanyl-2-[[3-[3-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl]methyl]-[1,2,4]triazolo[4,3-a]pyrazin-3-one —— C23H17F3N6O2S
8-(2-Ethylphenyl)sulfanyl-2-[[3-[3-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl]methyl]-[1,2,4]triazolo[4,3-a]pyrazin-3-one
—— 8-(3,4-dihydro-1H-isoquinolin-2-yl)-2-[[3-(3-fluorophenyl)-1,2,4-oxadiazol-5-yl]methyl]-[1,2,4]triazolo[4,3-a]pyrazin-3-one —— C23H18FN7O2
8-(3,4-dihydro-1H-isoquinolin-2-yl)-2-[[3-(3-fluorophenyl)-1,2,4-oxadiazol-5-yl]methyl]-[1,2,4]triazolo[4,3-a]pyrazin-3-one
—— 8-(Azepan-1-yl)-2-[(3-fluorophenyl)methyl]-[1,2,4]triazolo[4,3-a]pyrazin-3-one —— C18H20FN5O
8-(Azepan-1-yl)-2-[(3-fluorophenyl)methyl]-[1,2,4]triazolo[4,3-a]pyrazin-3-one
—— 8-(Azepan-1-yl)-2-[(3-methoxyphenyl)methyl]-[1,2,4]triazolo[4,3-a]pyrazin-3-one —— C19H23N5O2
8-(Azepan-1-yl)-2-[(3-methoxyphenyl)methyl]-[1,2,4]triazolo[4,3-a]pyrazin-3-one
—— 8-(Azepan-1-yl)-2-[(4-methylphenyl)methyl]-[1,2,4]triazolo[4,3-a]pyrazin-3-one —— C19H23N5O
8-(Azepan-1-yl)-2-[(4-methylphenyl)methyl]-[1,2,4]triazolo[4,3-a]pyrazin-3-one
—— 8-(Azepan-1-yl)-2-[(2,5-difluorophenyl)methyl]-[1,2,4]triazolo[4,3-a]pyrazin-3-one —— C18H19F2N5O
8-(Azepan-1-yl)-2-[(2,5-difluorophenyl)methyl]-[1,2,4]triazolo[4,3-a]pyrazin-3-one
—— 8-(3,4-dihydro-1H-isoquinolin-2-yl)-2-[(3-fluorophenyl)methyl]-[1,2,4]triazolo[4,3-a]pyrazin-3-one —— C21H18FN5O
8-(3,4-dihydro-1H-isoquinolin-2-yl)-2-[(3-fluorophenyl)methyl]-[1,2,4]triazolo[4,3-a]pyrazin-3-one
—— 8-[4-(4-Methylphenyl)piperazin-1-yl]-2-[[3-(4-methylsulfanylphenyl)-1,2,4-oxadiazol-5-yl]methyl]-[1,2,4]triazolo[4,3-a]pyrazin-3-one —— C26H26N8O2S
8-[4-(4-Methylphenyl)piperazin-1-yl]-2-[[3-(4-methylsulfanylphenyl)-1,2,4-oxadiazol-5-yl]methyl]-[1,2,4]triazolo[4,3-a]pyrazin-3-one
—— 8-Benzylsulfanyl-2-[[3-[3-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl]methyl]-[1,2,4]triazolo[4,3-a]pyrazin-3-one —— C22H15F3N6O2S
8-Benzylsulfanyl-2-[[3-[3-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl]methyl]-[1,2,4]triazolo[4,3-a]pyrazin-3-one
—— 8-(Azepan-1-yl)-2-[(5-methyl-2-phenyl-1,3-oxazol-4-yl)methyl]-[1,2,4]triazolo[4,3-a]pyrazin-3-one —— C22H24N6O2
8-(Azepan-1-yl)-2-[(5-methyl-2-phenyl-1,3-oxazol-4-yl)methyl]-[1,2,4]triazolo[4,3-a]pyrazin-3-one
—— 8-(Azepan-1-yl)-2-[(3,4-difluorophenyl)methyl]-[1,2,4]triazolo[4,3-a]pyrazin-3-one —— C18H19F2N5O
8-(Azepan-1-yl)-2-[(3,4-difluorophenyl)methyl]-[1,2,4]triazolo[4,3-a]pyrazin-3-one
—— 8-Benzylsulfanyl-2-[[3-(4-tert-butylphenyl)-1,2,4-oxadiazol-5-yl]methyl]-[1,2,4]triazolo[4,3-a]pyrazin-3-one —— C25H24N6O2S
8-Benzylsulfanyl-2-[[3-(4-tert-butylphenyl)-1,2,4-oxadiazol-5-yl]methyl]-[1,2,4]triazolo[4,3-a]pyrazin-3-one
—— 8-(Azepan-1-yl)-2-(1,3-benzodioxol-5-ylmethyl)-[1,2,4]triazolo[4,3-a]pyrazin-3-one —— C19H21N5O3
8-(Azepan-1-yl)-2-(1,3-benzodioxol-5-ylmethyl)-[1,2,4]triazolo[4,3-a]pyrazin-3-one
—— 8-Benzylsulfanyl-2-[(2,5-difluorophenyl)methyl]-[1,2,4]triazolo[4,3-a]pyrazin-3-one —— C19H14F2N4OS
8-Benzylsulfanyl-2-[(2,5-difluorophenyl)methyl]-[1,2,4]triazolo[4,3-a]pyrazin-3-one
—— 8-Benzylsulfanyl-2-[(3-methoxyphenyl)methyl]-[1,2,4]triazolo[4,3-a]pyrazin-3-one —— C20H18N4O2S
8-Benzylsulfanyl-2-[(3-methoxyphenyl)methyl]-[1,2,4]triazolo[4,3-a]pyrazin-3-one
—— 8-(Azepan-1-yl)-2-[2-(4-chlorophenyl)-2-oxoethyl]-[1,2,4]triazolo[4,3-a]pyrazin-3-one —— C19H20ClN5O2
8-(Azepan-1-yl)-2-[2-(4-chlorophenyl)-2-oxoethyl]-[1,2,4]triazolo[4,3-a]pyrazin-3-one
—— 8-Benzylsulfanyl-2-[(3,4-difluorophenyl)methyl]-[1,2,4]triazolo[4,3-a]pyrazin-3-one —— C19H14F2N4OS
8-Benzylsulfanyl-2-[(3,4-difluorophenyl)methyl]-[1,2,4]triazolo[4,3-a]pyrazin-3-one
—— 8-(Azepan-1-yl)-2-[[3-[3-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl]methyl]-[1,2,4]triazolo[4,3-a]pyrazin-3-one —— C21H20F3N7O2
8-(Azepan-1-yl)-2-[[3-[3-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl]methyl]-[1,2,4]triazolo[4,3-a]pyrazin-3-one
—— 8-(Azepan-1-yl)-2-[[3-(3-fluorophenyl)-1,2,4-oxadiazol-5-yl]methyl]-[1,2,4]triazolo[4,3-a]pyrazin-3-one —— C20H20FN7O2
8-(Azepan-1-yl)-2-[[3-(3-fluorophenyl)-1,2,4-oxadiazol-5-yl]methyl]-[1,2,4]triazolo[4,3-a]pyrazin-3-one
—— 8-(Azepan-1-yl)-2-[(3-fluoro-4-methoxyphenyl)methyl]-[1,2,4]triazolo[4,3-a]pyrazin-3-one —— C19H22FN5O2
8-(Azepan-1-yl)-2-[(3-fluoro-4-methoxyphenyl)methyl]-[1,2,4]triazolo[4,3-a]pyrazin-3-one
—— 8-Benzylsulfanyl-2-[[3-(4-methylsulfanylphenyl)-1,2,4-oxadiazol-5-yl]methyl]-[1,2,4]triazolo[4,3-a]pyrazin-3-one —— C22H18N6O2S2
8-Benzylsulfanyl-2-[[3-(4-methylsulfanylphenyl)-1,2,4-oxadiazol-5-yl]methyl]-[1,2,4]triazolo[4,3-a]pyrazin-3-one
—— 8-Morpholin-4-yl-2-[[3-[3-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl]methyl]-[1,2,4]triazolo[4,3-a]pyrazin-3-one —— C19H16F3N7O3
8-Morpholin-4-yl-2-[[3-[3-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl]methyl]-[1,2,4]triazolo[4,3-a]pyrazin-3-one
—— 8-(Azepan-1-yl)-2-[2-(4-fluorophenyl)-2-oxoethyl]-[1,2,4]triazolo[4,3-a]pyrazin-3-one —— C19H20FN5O2
8-(Azepan-1-yl)-2-[2-(4-fluorophenyl)-2-oxoethyl]-[1,2,4]triazolo[4,3-a]pyrazin-3-one
—— 8-Benzylsulfanyl-2-[2-(4-fluorophenyl)-2-oxoethyl]-[1,2,4]triazolo[4,3-a]pyrazin-3-one —— C20H15FN4O2S
8-Benzylsulfanyl-2-[2-(4-fluorophenyl)-2-oxoethyl]-[1,2,4]triazolo[4,3-a]pyrazin-3-one
—— 8-Benzylsulfanyl-2-[[3-(3-fluorophenyl)-1,2,4-oxadiazol-5-yl]methyl]-[1,2,4]triazolo[4,3-a]pyrazin-3-one —— C21H15FN6O2S
8-Benzylsulfanyl-2-[[3-(3-fluorophenyl)-1,2,4-oxadiazol-5-yl]methyl]-[1,2,4]triazolo[4,3-a]pyrazin-3-one
—— 8-(2-Ethylphenyl)sulfanyl-2-[(3-fluoro-4-methoxyphenyl)methyl]-[1,2,4]triazolo[4,3-a]pyrazin-3-one —— C21H19FN4O2S
8-(2-Ethylphenyl)sulfanyl-2-[(3-fluoro-4-methoxyphenyl)methyl]-[1,2,4]triazolo[4,3-a]pyrazin-3-one
—— 8-Benzylsulfanyl-2-[(3-fluoro-4-methoxyphenyl)methyl]-[1,2,4]triazolo[4,3-a]pyrazin-3-one —— C20H17FN4O2S
8-Benzylsulfanyl-2-[(3-fluoro-4-methoxyphenyl)methyl]-[1,2,4]triazolo[4,3-a]pyrazin-3-one
—— 8-ethyl-5-(2-fluorophenyl)-7-methyl-2H-[1,2,4]triazolo[4,3-c]pyrimidin-3-one —— C14H13FN4O
8-ethyl-5-(2-fluorophenyl)-7-methyl-2H-[1,2,4]triazolo[4,3-c]pyrimidin-3-one
—— 8-(Azepan-1-yl)-2-benzyl-[1,2,4]triazolo[4,3-a]pyrazin-3-one —— C18H21N5O
8-(Azepan-1-yl)-2-benzyl-[1,2,4]triazolo[4,3-a]pyrazin-3-one
—— 8-ethyl-5-(4-methoxyphenyl)-7-methyl-2H-[1,2,4]triazolo[4,3-c]pyrimidin-3-one —— C15H16N4O2
8-ethyl-5-(4-methoxyphenyl)-7-methyl-2H-[1,2,4]triazolo[4,3-c]pyrimidin-3-one
—— 8-(2-Ethylphenyl)sulfanyl-2-[[3-(3-fluorophenyl)-1,2,4-oxadiazol-5-yl]methyl]-[1,2,4]triazolo[4,3-a]pyrazin-3-one —— C22H17FN6O2S
8-(2-Ethylphenyl)sulfanyl-2-[[3-(3-fluorophenyl)-1,2,4-oxadiazol-5-yl]methyl]-[1,2,4]triazolo[4,3-a]pyrazin-3-one
—— 8-(2-Ethylphenyl)sulfanyl-2-[[3-(4-methylsulfanylphenyl)-1,2,4-oxadiazol-5-yl]methyl]-[1,2,4]triazolo[4,3-a]pyrazin-3-one —— C23H20N6O2S2
8-(2-Ethylphenyl)sulfanyl-2-[[3-(4-methylsulfanylphenyl)-1,2,4-oxadiazol-5-yl]methyl]-[1,2,4]triazolo[4,3-a]pyrazin-3-one
—— 8-(3-Fluorophenyl)sulfanyl-2-[[3-[3-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl]methyl]-[1,2,4]triazolo[4,3-a]pyrazin-3-one —— C21H12F4N6O2S
8-(3-Fluorophenyl)sulfanyl-2-[[3-[3-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl]methyl]-[1,2,4]triazolo[4,3-a]pyrazin-3-one
—— 8-Benzylsulfanyl-2-[(5-methyl-2-phenyl-1,3-oxazol-4-yl)methyl]-[1,2,4]triazolo[4,3-a]pyrazin-3-one —— C23H19N5O2S
8-Benzylsulfanyl-2-[(5-methyl-2-phenyl-1,3-oxazol-4-yl)methyl]-[1,2,4]triazolo[4,3-a]pyrazin-3-one
—— 8-Benzylsulfanyl-2-[(3-fluorophenyl)methyl]-[1,2,4]triazolo[4,3-a]pyrazin-3-one —— C19H15FN4OS
8-Benzylsulfanyl-2-[(3-fluorophenyl)methyl]-[1,2,4]triazolo[4,3-a]pyrazin-3-one
—— 8-(2,4-Dimethylphenyl)sulfanyl-2-[2-(4-fluorophenyl)-2-oxoethyl]-[1,2,4]triazolo[4,3-a]pyrazin-3-one —— C21H17FN4O2S
8-(2,4-Dimethylphenyl)sulfanyl-2-[2-(4-fluorophenyl)-2-oxoethyl]-[1,2,4]triazolo[4,3-a]pyrazin-3-one
—— 8-[(4-Chlorophenyl)methylsulfanyl]-2-[(2,5-difluorophenyl)methyl]-[1,2,4]triazolo[4,3-a]pyrazin-3-one —— C19H13ClF2N4OS
8-[(4-Chlorophenyl)methylsulfanyl]-2-[(2,5-difluorophenyl)methyl]-[1,2,4]triazolo[4,3-a]pyrazin-3-one
—— 8-(2-Ethylphenyl)sulfanyl-2-[2-(4-fluorophenyl)-2-oxoethyl]-[1,2,4]triazolo[4,3-a]pyrazin-3-one —— C21H17FN4O2S
8-(2-Ethylphenyl)sulfanyl-2-[2-(4-fluorophenyl)-2-oxoethyl]-[1,2,4]triazolo[4,3-a]pyrazin-3-one
—— 8-[(4-Chlorophenyl)methylsulfanyl]-2-[2-(4-fluorophenyl)-2-oxoethyl]-[1,2,4]triazolo[4,3-a]pyrazin-3-one —— C20H14ClFN4O2S
8-[(4-Chlorophenyl)methylsulfanyl]-2-[2-(4-fluorophenyl)-2-oxoethyl]-[1,2,4]triazolo[4,3-a]pyrazin-3-one
—— 8-Cyclohexylsulfanyl-2-[[3-[3-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl]methyl]-[1,2,4]triazolo[4,3-a]pyrazin-3-one —— C21H19F3N6O2S
8-Cyclohexylsulfanyl-2-[[3-[3-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl]methyl]-[1,2,4]triazolo[4,3-a]pyrazin-3-one
—— 8-Cyclohexylsulfanyl-2-[2-(4-fluorophenyl)-2-oxoethyl]-[1,2,4]triazolo[4,3-a]pyrazin-3-one —— C19H19FN4O2S
8-Cyclohexylsulfanyl-2-[2-(4-fluorophenyl)-2-oxoethyl]-[1,2,4]triazolo[4,3-a]pyrazin-3-one