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—— (8R)-11-methyl-10-oxo-5-thia-11,12-diazatricyclo[6.4.0.02,6]dodeca-1(12),2(6),3-triene-4-carboxylic acid —— C11H10N2O3S
(8R)-11-methyl-10-oxo-5-thia-11,12-diazatricyclo[6.4.0.02,6]dodeca-1(12),2(6),3-triene-4-carboxylic acid
—— (8R)-8-piperidin-4-yl-6-azaspiro[3.5]nonane-5,7,9-trione —— C13H18N2O3
(8R)-8-piperidin-4-yl-6-azaspiro[3.5]nonane-5,7,9-trione
—— (8S)-8-(1,3-thiazol-4-yl)-5,6,7,8-tetrahydroimidazo[1,5-a]pyrazine-1-carboxylic acid —— C10H10N4O2S
(8S)-8-(1,3-thiazol-4-yl)-5,6,7,8-tetrahydroimidazo[1,5-a]pyrazine-1-carboxylic acid
—— (8S)-11-methyl-10-oxo-5-thia-11,12-diazatricyclo[6.4.0.02,6]dodeca-1(12),2(6),3-triene-4-carboxylic acid —— C11H10N2O3S
(8S)-11-methyl-10-oxo-5-thia-11,12-diazatricyclo[6.4.0.02,6]dodeca-1(12),2(6),3-triene-4-carboxylic acid
—— (8S)-8-(pyrrolidin-1-ylmethyl)-5,6,7,8-tetrahydroimidazo[1,5-a]pyrazine-1-carboxylic acid —— C12H18N4O2
(8S)-8-(pyrrolidin-1-ylmethyl)-5,6,7,8-tetrahydroimidazo[1,5-a]pyrazine-1-carboxylic acid
—— (8R)-8-(1,3-thiazol-4-yl)-5,6,7,8-tetrahydroimidazo[1,5-a]pyrazine-1-carboxylic acid —— C10H10N4O2S
(8R)-8-(1,3-thiazol-4-yl)-5,6,7,8-tetrahydroimidazo[1,5-a]pyrazine-1-carboxylic acid
—— (8R)-8-(pyrrolidin-1-ylmethyl)-5,6,7,8-tetrahydroimidazo[1,5-a]pyrazine-1-carboxylic acid —— C12H18N4O2
(8R)-8-(pyrrolidin-1-ylmethyl)-5,6,7,8-tetrahydroimidazo[1,5-a]pyrazine-1-carboxylic acid
—— 8-chloro-7,9-dimethyl-4,5-dihydro-[1,3]thiazolo[5,4-c]quinoline —— C12H11ClN2S
8-chloro-7,9-dimethyl-4,5-dihydro-[1,3]thiazolo[5,4-c]quinoline
—— 8-chloro-2-methyl-5,10-dihydro-4H-[1,3]thiazolo[5,4-c][1]benzazepine —— C12H11ClN2S
8-chloro-2-methyl-5,10-dihydro-4H-[1,3]thiazolo[5,4-c][1]benzazepine
—— 8-chloro-2,5-dimethyl-4,9-dihydro-[1,3]thiazolo[5,4-b]quinoline —— C12H11ClN2S
8-chloro-2,5-dimethyl-4,9-dihydro-[1,3]thiazolo[5,4-b]quinoline
—— 8-chloro-7-methyl-5,6-dihydro-4H-[1,3]thiazolo[5,4-d][1]benzazepine —— C12H11ClN2S
8-chloro-7-methyl-5,6-dihydro-4H-[1,3]thiazolo[5,4-d][1]benzazepine
—— 8-bromo-4,5-dihydro-[1,2]oxazolo[5,4-c]quinoline —— C10H7BrN2O
8-bromo-4,5-dihydro-[1,2]oxazolo[5,4-c]quinoline
—— (8S)-8-(4-chloro-3-fluorophenyl)-5,6,7,8-tetrahydroimidazo[1,5-a]pyrazine —— C12H11ClFN3
(8S)-8-(4-chloro-3-fluorophenyl)-5,6,7,8-tetrahydroimidazo[1,5-a]pyrazine
—— (8R)-8-(4-chloro-3-fluorophenyl)-5,6,7,8-tetrahydroimidazo[1,5-a]pyrazine —— C12H11ClFN3
(8R)-8-(4-chloro-3-fluorophenyl)-5,6,7,8-tetrahydroimidazo[1,5-a]pyrazine
—— (8S)-8-(2-chloro-5-fluorophenyl)-5,6,7,8-tetrahydroimidazo[1,5-a]pyrazine —— C12H11ClFN3
(8S)-8-(2-chloro-5-fluorophenyl)-5,6,7,8-tetrahydroimidazo[1,5-a]pyrazine
—— (8R)-8-(2-chloro-5-fluorophenyl)-5,6,7,8-tetrahydroimidazo[1,5-a]pyrazine —— C12H11ClFN3
(8R)-8-(2-chloro-5-fluorophenyl)-5,6,7,8-tetrahydroimidazo[1,5-a]pyrazine
—— 8-(trifluoromethyl)-1,9-dihydropyrrolo[3,2-h]quinolin-6-one —— C12H7F3N2O
8-(trifluoromethyl)-1,9-dihydropyrrolo[3,2-h]quinolin-6-one
—— (8R)-7,7-dioxo-8-(1H-pyrrol-3-yl)-6,8-dihydro-5H-imidazo[5,1-c][1,4]thiazin-3-amine —— C10H12N4O2S
(8R)-7,7-dioxo-8-(1H-pyrrol-3-yl)-6,8-dihydro-5H-imidazo[5,1-c][1,4]thiazin-3-amine
—— (8aS)-1-oxospiro[2,3,6,7,8,8a-hexahydropyrrolo[1,2-a]pyrazine-4,4'-cyclohexane]-1'-carboxylic acid —— C13H20N2O3
(8aS)-1-oxospiro[2,3,6,7,8,8a-hexahydropyrrolo[1,2-a]pyrazine-4,4'-cyclohexane]-1'-carboxylic acid
—— (8S)-7,7-dioxo-8-(1H-pyrrol-3-yl)-6,8-dihydro-5H-imidazo[5,1-c][1,4]thiazin-3-amine —— C10H12N4O2S
(8S)-7,7-dioxo-8-(1H-pyrrol-3-yl)-6,8-dihydro-5H-imidazo[5,1-c][1,4]thiazin-3-amine
—— (8R,9S)-9-hydroxy-8-piperidin-4-yl-6-azaspiro[3.5]nonane-5,7-dione —— C13H20N2O3
(8R,9S)-9-hydroxy-8-piperidin-4-yl-6-azaspiro[3.5]nonane-5,7-dione
—— (8S,9R)-9-hydroxy-8-piperidin-4-yl-6-azaspiro[3.5]nonane-5,7-dione —— C13H20N2O3
(8S,9R)-9-hydroxy-8-piperidin-4-yl-6-azaspiro[3.5]nonane-5,7-dione
—— (8R,9S)-8-[(4R)-azepan-4-yl]-6-methyl-6-azaspiro[3.5]nonan-9-ol —— C15H28N2O
(8R,9S)-8-[(4R)-azepan-4-yl]-6-methyl-6-azaspiro[3.5]nonan-9-ol
—— (8R,9R)-8-[(4S)-1-methylazepan-4-yl]-6-azaspiro[3.5]nonan-9-ol —— C15H28N2O
(8R,9R)-8-[(4S)-1-methylazepan-4-yl]-6-azaspiro[3.5]nonan-9-ol
—— 8-chloro-5-methoxy-4,9-dihydro-[1,3]thiazolo[5,4-b]quinoline —— C11H9ClN2OS
8-chloro-5-methoxy-4,9-dihydro-[1,3]thiazolo[5,4-b]quinoline
—— (8R,9R)-8-[(4R)-1-methylazepan-4-yl]-6-azaspiro[3.5]nonan-9-ol —— C15H28N2O
(8R,9R)-8-[(4R)-1-methylazepan-4-yl]-6-azaspiro[3.5]nonan-9-ol
—— (8S,9S)-8-[(4R)-azepan-4-yl]-6-methyl-6-azaspiro[3.5]nonan-9-ol —— C15H28N2O
(8S,9S)-8-[(4R)-azepan-4-yl]-6-methyl-6-azaspiro[3.5]nonan-9-ol
—— 8-chloro-7-methoxy-4,9-dihydro-[1,3]thiazolo[5,4-b]quinoline —— C11H9ClN2OS
8-chloro-7-methoxy-4,9-dihydro-[1,3]thiazolo[5,4-b]quinoline
—— 8-bromo-11-methyl-3,4,6,7,11,12-hexazatricyclo[7.3.0.02,6]dodeca-1(12),2,4,7,9-pentaene —— C7H5BrN6
8-bromo-11-methyl-3,4,6,7,11,12-hexazatricyclo[7.3.0.02,6]dodeca-1(12),2,4,7,9-pentaene
—— 8-(trifluoromethyl)-1,4,5,10-tetrahydropyrazolo[4,3-c][1]benzazepine —— C12H10F3N3
8-(trifluoromethyl)-1,4,5,10-tetrahydropyrazolo[4,3-c][1]benzazepine
—— 8-amino-7-bromo-2-methylisoquinolin-1-one —— C10H9BrN2O
8-amino-7-bromo-2-methylisoquinolin-1-one
—— 8-bromo-7-hydroxy-2-methylisoquinolin-1-one —— C10H8BrNO2
8-bromo-7-hydroxy-2-methylisoquinolin-1-one
—— 8-Bromo-5-methylindolizine-3-carboxylic acid —— C10H8BrNO2
8-Bromo-5-methylindolizine-3-carboxylic acid
—— (8S)-5-bromo-8-methyl-3,6,7,8-tetrahydro-2H-furo[2,3-e]isoindole —— C11H12BrNO
(8S)-5-bromo-8-methyl-3,6,7,8-tetrahydro-2H-furo[2,3-e]isoindole
—— (8R)-8-methyl-2-(trifluoromethyl)-5,6,7,8-tetrahydro-1H-pyrrolo[2,3-g]isoquinoline —— C13H13F3N2
(8R)-8-methyl-2-(trifluoromethyl)-5,6,7,8-tetrahydro-1H-pyrrolo[2,3-g]isoquinoline
—— (8R)-8-methyl-2-(trifluoromethyl)-5,6,7,8-tetrahydro-1H-pyrrolo[3,2-g]isoquinoline —— C13H13F3N2
(8R)-8-methyl-2-(trifluoromethyl)-5,6,7,8-tetrahydro-1H-pyrrolo[3,2-g]isoquinoline
—— (8S)-8-methyl-2-(trifluoromethyl)-5,6,7,8-tetrahydro-1H-pyrrolo[3,2-g]isoquinoline —— C13H13F3N2
(8S)-8-methyl-2-(trifluoromethyl)-5,6,7,8-tetrahydro-1H-pyrrolo[3,2-g]isoquinoline
—— 8-amino-5-cyclopropyl-1,1-dioxo-3,4-dihydro-2H-thiopyrano[3,2-b]pyridin-6-one —— C11H14N2O3S
8-amino-5-cyclopropyl-1,1-dioxo-3,4-dihydro-2H-thiopyrano[3,2-b]pyridin-6-one
—— 8-methyl-2-(trifluoromethyl)-4,5-dihydro-[1,2,4]triazolo[1,5-a]quinoxaline —— C11H9F3N4
8-methyl-2-(trifluoromethyl)-4,5-dihydro-[1,2,4]triazolo[1,5-a]quinoxaline
—— (8S)-8-methyl-2-(trifluoromethyl)-5,6,7,8-tetrahydro-1H-pyrrolo[2,3-g]isoquinoline —— C13H13F3N2
(8S)-8-methyl-2-(trifluoromethyl)-5,6,7,8-tetrahydro-1H-pyrrolo[2,3-g]isoquinoline
—— 8,10-dichloro-4,5-dihydro-2H-[1,2]oxazolo[4,5-d][1]benzazepine —— C11H8Cl2N2O
8,10-dichloro-4,5-dihydro-2H-[1,2]oxazolo[4,5-d][1]benzazepine
—— 8-methyl-7-methylsulfonylimidazo[1,2-c]pyrimidine-2-carboxylic acid —— C9H9N3O4S
8-methyl-7-methylsulfonylimidazo[1,2-c]pyrimidine-2-carboxylic acid
—— (8R,9aR)-8-(piperazin-1-ylmethyl)-1,3,4,6,7,8,9,9a-octahydropyrido[2,1-c][1,4]thiazine —— C13H25N3S
(8R,9aR)-8-(piperazin-1-ylmethyl)-1,3,4,6,7,8,9,9a-octahydropyrido[2,1-c][1,4]thiazine
—— 8-(1,3-benzodioxol-5-ylmethyl)-1,2,3,4-tetrahydropyrrolo[1,2-a]pyrazine —— C15H16N2O2
8-(1,3-benzodioxol-5-ylmethyl)-1,2,3,4-tetrahydropyrrolo[1,2-a]pyrazine
—— 8-(trifluoromethyl)-4,5-dihydro-[1,3]thiazolo[5,4-c]quinoline —— C11H7F3N2S
8-(trifluoromethyl)-4,5-dihydro-[1,3]thiazolo[5,4-c]quinoline
—— 8-(1,3-benzodioxol-4-ylmethyl)-1,2,3,4-tetrahydropyrrolo[1,2-a]pyrazine —— C15H16N2O2
8-(1,3-benzodioxol-4-ylmethyl)-1,2,3,4-tetrahydropyrrolo[1,2-a]pyrazine
—— (8R)-1-benzyl-5,6,7,8-tetrahydroimidazo[1,5-a]pyridine-8-carboxylic acid —— C15H16N2O2
(8R)-1-benzyl-5,6,7,8-tetrahydroimidazo[1,5-a]pyridine-8-carboxylic acid
—— (8S)-1-benzyl-5,6,7,8-tetrahydroimidazo[1,5-a]pyridine-8-carboxylic acid —— C15H16N2O2
(8S)-1-benzyl-5,6,7,8-tetrahydroimidazo[1,5-a]pyridine-8-carboxylic acid
—— 8-Chloro-7-[(5-chloro-2,3-dihydro-1,4-benzodioxin-7-yl)methyl]-1,3-dimethylpurine-2,6-dione —— C16H14Cl2N4O4
8-Chloro-7-[(5-chloro-2,3-dihydro-1,4-benzodioxin-7-yl)methyl]-1,3-dimethylpurine-2,6-dione
—— (8S,8aS)-8-(5-bromo-2-fluorophenyl)-6-imino-2-propan-2-yl-3,5,8,8a-tetrahydro-1H-isoquinoline-5,7,7-tricarbonitrile —— C21H19BrFN5
(8S,8aS)-8-(5-bromo-2-fluorophenyl)-6-imino-2-propan-2-yl-3,5,8,8a-tetrahydro-1H-isoquinoline-5,7,7-tricarbonitrile