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—— (6R)-6-N-cyclopentyl-1-N-[(2-ethoxyphenyl)methyl]-7-ethyl-6-methyl-8-oxo-5H-imidazo[1,5-a]pyrazine-1,6-dicarboxamide —— C25H33N5O4
(6R)-6-N-cyclopentyl-1-N-[(2-ethoxyphenyl)methyl]-7-ethyl-6-methyl-8-oxo-5H-imidazo[1,5-a]pyrazine-1,6-dicarboxamide
—— (6S)-6-N-cyclopentyl-7-ethyl-6-methyl-8-oxo-1-N-(2-phenylethyl)-5H-imidazo[1,5-a]pyrazine-1,6-dicarboxamide —— C24H31N5O3
(6S)-6-N-cyclopentyl-7-ethyl-6-methyl-8-oxo-1-N-(2-phenylethyl)-5H-imidazo[1,5-a]pyrazine-1,6-dicarboxamide
—— (6S)-6-N-cyclopentyl-1-N-[(3,4-dimethoxyphenyl)methyl]-7-ethyl-6-methyl-8-oxo-5H-imidazo[1,5-a]pyrazine-1,6-dicarboxamide —— C25H33N5O5
(6S)-6-N-cyclopentyl-1-N-[(3,4-dimethoxyphenyl)methyl]-7-ethyl-6-methyl-8-oxo-5H-imidazo[1,5-a]pyrazine-1,6-dicarboxamide
—— (6S)-6-N-cyclopentyl-7-ethyl-6-methyl-8-oxo-1-N-(3-phenylpropyl)-5H-imidazo[1,5-a]pyrazine-1,6-dicarboxamide —— C25H33N5O3
(6S)-6-N-cyclopentyl-7-ethyl-6-methyl-8-oxo-1-N-(3-phenylpropyl)-5H-imidazo[1,5-a]pyrazine-1,6-dicarboxamide
—— (6R)-6-N-cyclopentyl-1-N-[(3-ethoxy-4-methoxyphenyl)methyl]-7-ethyl-6-methyl-8-oxo-5H-imidazo[1,5-a]pyrazine-1,6-dicarboxamide —— C26H35N5O5
(6R)-6-N-cyclopentyl-1-N-[(3-ethoxy-4-methoxyphenyl)methyl]-7-ethyl-6-methyl-8-oxo-5H-imidazo[1,5-a]pyrazine-1,6-dicarboxamide
—— (6R)-6-N-cyclopentyl-7-ethyl-1-N-[(2-methoxyphenyl)methyl]-6-methyl-8-oxo-5H-imidazo[1,5-a]pyrazine-1,6-dicarboxamide —— C24H31N5O4
(6R)-6-N-cyclopentyl-7-ethyl-1-N-[(2-methoxyphenyl)methyl]-6-methyl-8-oxo-5H-imidazo[1,5-a]pyrazine-1,6-dicarboxamide
—— (6S)-6-N-cyclopentyl-7-ethyl-6-methyl-1-N-[2-(4-methylphenyl)ethyl]-8-oxo-5H-imidazo[1,5-a]pyrazine-1,6-dicarboxamide —— C25H33N5O3
(6S)-6-N-cyclopentyl-7-ethyl-6-methyl-1-N-[2-(4-methylphenyl)ethyl]-8-oxo-5H-imidazo[1,5-a]pyrazine-1,6-dicarboxamide
—— (6R)-6-N-cyclopentyl-7-ethyl-1-N-(furan-2-ylmethyl)-6-methyl-8-oxo-5H-imidazo[1,5-a]pyrazine-1,6-dicarboxamide —— C21H27N5O4
(6R)-6-N-cyclopentyl-7-ethyl-1-N-(furan-2-ylmethyl)-6-methyl-8-oxo-5H-imidazo[1,5-a]pyrazine-1,6-dicarboxamide
—— (6R)-6-N-cyclopentyl-7-ethyl-6-methyl-8-oxo-1-N-propan-2-yl-5H-imidazo[1,5-a]pyrazine-1,6-dicarboxamide —— C19H29N5O3
(6R)-6-N-cyclopentyl-7-ethyl-6-methyl-8-oxo-1-N-propan-2-yl-5H-imidazo[1,5-a]pyrazine-1,6-dicarboxamide
—— 6a-(4-chlorophenyl)-2-[4-(dimethylamino)-3,5-dinitrophenyl]-8-(4-fluoroanilino)-6-(2-hydroxy-6-methoxyphenyl)-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-1,3,7,9-tetrone —— C41H34ClFN6O10
6a-(4-chlorophenyl)-2-[4-(dimethylamino)-3,5-dinitrophenyl]-8-(4-fluoroanilino)-6-(2-hydroxy-6-methoxyphenyl)-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-1,3,7,9-tetrone
—— 6-(3-fluorophenyl)-5-methylsulfonyl-2-oxo-1H-pyridine-3-carbonitrile —— C13H9FN2O3S
6-(3-fluorophenyl)-5-methylsulfonyl-2-oxo-1H-pyridine-3-carbonitrile
—— (6S)-6-N-cyclopentyl-1-N-[2-(3,4-dimethoxyphenyl)ethyl]-7-ethyl-6-methyl-8-oxo-5H-imidazo[1,5-a]pyrazine-1,6-dicarboxamide —— C26H35N5O5
(6S)-6-N-cyclopentyl-1-N-[2-(3,4-dimethoxyphenyl)ethyl]-7-ethyl-6-methyl-8-oxo-5H-imidazo[1,5-a]pyrazine-1,6-dicarboxamide
—— (6S)-6-N-cyclopentyl-7-ethyl-1-N-[(2-methoxyphenyl)methyl]-6-methyl-8-oxo-5H-imidazo[1,5-a]pyrazine-1,6-dicarboxamide —— C24H31N5O4
(6S)-6-N-cyclopentyl-7-ethyl-1-N-[(2-methoxyphenyl)methyl]-6-methyl-8-oxo-5H-imidazo[1,5-a]pyrazine-1,6-dicarboxamide
—— (6S)-1-N-[2-(cyclohexen-1-yl)ethyl]-6-N-cyclopentyl-7-ethyl-6-methyl-8-oxo-5H-imidazo[1,5-a]pyrazine-1,6-dicarboxamide —— C24H35N5O3
(6S)-1-N-[2-(cyclohexen-1-yl)ethyl]-6-N-cyclopentyl-7-ethyl-6-methyl-8-oxo-5H-imidazo[1,5-a]pyrazine-1,6-dicarboxamide
—— (6S)-6-N-cyclopentyl-7-ethyl-1-N-[(4-fluorophenyl)methyl]-6-methyl-8-oxo-5H-imidazo[1,5-a]pyrazine-1,6-dicarboxamide —— C23H28FN5O3
(6S)-6-N-cyclopentyl-7-ethyl-1-N-[(4-fluorophenyl)methyl]-6-methyl-8-oxo-5H-imidazo[1,5-a]pyrazine-1,6-dicarboxamide
—— 6a-(4-chlorophenyl)-8-(4-fluoroanilino)-6-(4-hydroxynaphthalen-1-yl)-2-phenyl-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-1,3,7,9-tetrone —— C42H31ClFN3O5
6a-(4-chlorophenyl)-8-(4-fluoroanilino)-6-(4-hydroxynaphthalen-1-yl)-2-phenyl-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-1,3,7,9-tetrone
—— 6a-(4-chlorophenyl)-8-[[3-chloro-5-(trifluoromethyl)pyridin-2-yl]amino]-6-(2-hydroxy-4,6-dimethoxyphenyl)-2-(3-nitrophenyl)-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-1,3,7,9-tetrone —— C40H30Cl2F3N5O9
6a-(4-chlorophenyl)-8-[[3-chloro-5-(trifluoromethyl)pyridin-2-yl]amino]-6-(2-hydroxy-4,6-dimethoxyphenyl)-2-(3-nitrophenyl)-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-1,3,7,9-tetrone
—— 6-Ethoxy-2-pyridin-2-ylquinoline-4-carboxylic acid —— C17H14N2O3
6-Ethoxy-2-pyridin-2-ylquinoline-4-carboxylic acid
—— 6-({2-[(4-chloro-2,5-dimethoxyphenyl)amino]-2-oxoethyl}sulfanyl)-5-cyano-2-methyl-N,4-diphenyl-1,4-dihydropyridine-3-carboxamide —— C30H27ClN4O4S
6-({2-[(4-chloro-2,5-dimethoxyphenyl)amino]-2-oxoethyl}sulfanyl)-5-cyano-2-methyl-N,4-diphenyl-1,4-dihydropyridine-3-carboxamide
—— 6a-(4-chlorophenyl)-8-[[3-chloro-5-(trifluoromethyl)pyridin-2-yl]amino]-2-[[3-chloro-6-(trifluoromethyl)pyridin-2-yl]-methylamino]-6-(2-hydroxy-4-phenylmethoxyphenyl)-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-1,3,7,9-tetrone —— C46H33Cl3F6N6O6
6a-(4-chlorophenyl)-8-[[3-chloro-5-(trifluoromethyl)pyridin-2-yl]amino]-2-[[3-chloro-6-(trifluoromethyl)pyridin-2-yl]-methylamino]-6-(2-hydroxy-4-phenylmethoxyphenyl)-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-1,3,7,9-tetrone
—— 6-(2-methylpiperidine-1-carbonyl)-2H-thiazolo[3,2-a]pyrimidin-5(3H)-one —— C13H17N3O2S
6-(2-methylpiperidine-1-carbonyl)-2H-thiazolo[3,2-a]pyrimidin-5(3H)-one
—— 6-(Dimethylsulfamoyl)-2-(7-methoxy-1-benzofuran-2-yl)quinoline-4-carboxylic acid —— C21H18N2O6S
6-(Dimethylsulfamoyl)-2-(7-methoxy-1-benzofuran-2-yl)quinoline-4-carboxylic acid
—— 6a-(4-chlorophenyl)-8-[[3-chloro-5-(trifluoromethyl)pyridin-2-yl]amino]-2-[4-[[4-(dimethylamino)phenyl]diazenyl]phenyl]-6-(4-hydroxy-3,5-dimethylphenyl)-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-1,3,7,9-tetrone —— C48H40Cl2F3N7O5
6a-(4-chlorophenyl)-8-[[3-chloro-5-(trifluoromethyl)pyridin-2-yl]amino]-2-[4-[[4-(dimethylamino)phenyl]diazenyl]phenyl]-6-(4-hydroxy-3,5-dimethylphenyl)-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-1,3,7,9-tetrone
—— 6-(3-Ethoxy-2-hydroxyphenyl)-8-methyl-2-propyl-3a,4,6,11,11a,11b-hexahydronaphtho[6,7-e]isoindole-1,3,7,10-tetrone —— C28H29NO6
6-(3-Ethoxy-2-hydroxyphenyl)-8-methyl-2-propyl-3a,4,6,11,11a,11b-hexahydronaphtho[6,7-e]isoindole-1,3,7,10-tetrone
—— 6-amino-3-methyl-1-phenyl-4-(2-pyridyl)-4H-pyrano[3,2-d]pyrazole-5-carbonitril e —— C19H15N5O
6-amino-3-methyl-1-phenyl-4-(2-pyridyl)-4H-pyrano[3,2-d]pyrazole-5-carbonitril e
—— 6-(2-Chloro-4-hydroxyphenyl)-2-(4-ethenylphenyl)-8-methyl-3a,4,6,11,11a,11b-hexahydronaphtho[6,7-e]isoindole-1,3,7,10-tetrone —— C31H24ClNO5
6-(2-Chloro-4-hydroxyphenyl)-2-(4-ethenylphenyl)-8-methyl-3a,4,6,11,11a,11b-hexahydronaphtho[6,7-e]isoindole-1,3,7,10-tetrone
—— 6-acetamido-N-[[3-[3-[4-[(4-acetamidophenyl)sulfanylmethyl]-6-[4-(hydroxymethyl)phenyl]-1,3-dioxan-2-yl]phenyl]phenyl]methyl]hexanamide —— C41H47N3O6S
6-acetamido-N-[[3-[3-[4-[(4-acetamidophenyl)sulfanylmethyl]-6-[4-(hydroxymethyl)phenyl]-1,3-dioxan-2-yl]phenyl]phenyl]methyl]hexanamide
—— 6-{3-[(1,3-dioxo-2-phenyl-2,3-dihydro-1H-isoindol-5-yl)oxy]phenyl}-5H-dibenzo[c,e]azepine-5,7(6H)-dione —— C34H20N2O5
6-{3-[(1,3-dioxo-2-phenyl-2,3-dihydro-1H-isoindol-5-yl)oxy]phenyl}-5H-dibenzo[c,e]azepine-5,7(6H)-dione
—— [6-Bromo-2-(4-tert-butylphenyl)quinolin-4-yl][4-(furan-2-ylcarbonyl)piperazin-1-yl]methanone —— C29H28BrN3O3
[6-Bromo-2-(4-tert-butylphenyl)quinolin-4-yl][4-(furan-2-ylcarbonyl)piperazin-1-yl]methanone
—— 6-bromo-N-cyclopentyl-2-(2,5-dimethylphenyl)quinoline-4-carboxamide —— C23H23BrN2O
6-bromo-N-cyclopentyl-2-(2,5-dimethylphenyl)quinoline-4-carboxamide
—— 6-{[4-(3-methoxyphenyl)piperazin-1-yl]methyl}-N-(4-phenoxyphenyl)-1,3,5-triazine-2,4-diamine —— C27H29N7O2
6-{[4-(3-methoxyphenyl)piperazin-1-yl]methyl}-N-(4-phenoxyphenyl)-1,3,5-triazine-2,4-diamine
—— 6-[(2R)-2-ethylpiperidin-1-yl]sulfonyl-3-(3-oxo-3-piperidin-1-ylpropyl)-1,3-benzothiazol-2-one —— C22H31N3O4S2
6-[(2R)-2-ethylpiperidin-1-yl]sulfonyl-3-(3-oxo-3-piperidin-1-ylpropyl)-1,3-benzothiazol-2-one
—— 6-[(2S)-2-methylpiperidin-1-yl]sulfonyl-3-(3-oxo-3-piperidin-1-ylpropyl)-1,3-benzothiazol-2-one —— C21H29N3O4S2
6-[(2S)-2-methylpiperidin-1-yl]sulfonyl-3-(3-oxo-3-piperidin-1-ylpropyl)-1,3-benzothiazol-2-one
—— 6-hexyl-2-thioxotetrahydropyrimidin-4(1H)-one —— C10H18N2OS
6-hexyl-2-thioxotetrahydropyrimidin-4(1H)-one
—— 6-[[3-[3-[4-[4-(Hydroxymethyl)phenyl]-6-(piperidin-1-ylmethyl)-1,3-dioxan-2-yl]phenyl]phenyl]methylamino]-6-oxohexanoic acid —— C36H44N2O6
6-[[3-[3-[4-[4-(Hydroxymethyl)phenyl]-6-(piperidin-1-ylmethyl)-1,3-dioxan-2-yl]phenyl]phenyl]methylamino]-6-oxohexanoic acid
—— 6-ethyl 3-methyl 2-(cyclohexanecarboxamido)-4,5-dihydrothieno[2,3-c]pyridine-3,6(7H)-dicarboxylate —— C19H26N2O5S
6-ethyl 3-methyl 2-(cyclohexanecarboxamido)-4,5-dihydrothieno[2,3-c]pyridine-3,6(7H)-dicarboxylate
—— (6S)-3-benzyl-N-(3,5-dichlorophenyl)-2-(4-fluorophenyl)imino-4-oxo-1,3-thiazinane-6-carboxamide —— C24H18Cl2FN3O2S
(6S)-3-benzyl-N-(3,5-dichlorophenyl)-2-(4-fluorophenyl)imino-4-oxo-1,3-thiazinane-6-carboxamide
—— 6-[[3-Bromo-4-[2-(4-tert-butylphenoxy)ethoxy]-5-methoxyphenyl]methylidene]-2-ethyl-5-imino-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C27H29BrN4O4S
6-[[3-Bromo-4-[2-(4-tert-butylphenoxy)ethoxy]-5-methoxyphenyl]methylidene]-2-ethyl-5-imino-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— 6-Bromo-2-[4-(4-fluorophenyl)-4-oxobutyl]sulfanyl-3-(1-phenylethyl)quinazolin-4-one —— C26H22BrFN2O2S
6-Bromo-2-[4-(4-fluorophenyl)-4-oxobutyl]sulfanyl-3-(1-phenylethyl)quinazolin-4-one
—— (6R)-2-(3-chlorophenyl)imino-N-(4-fluorophenyl)-3-[(4-methoxyphenyl)methyl]-4-oxo-1,3-thiazinane-6-carboxamide —— C25H21ClFN3O3S
(6R)-2-(3-chlorophenyl)imino-N-(4-fluorophenyl)-3-[(4-methoxyphenyl)methyl]-4-oxo-1,3-thiazinane-6-carboxamide
—— 6,7-dimethoxy-1-((2-methoxyphenoxy)methyl)-N-(m-tolyl)-3,4-dihydroisoquinoline-2(1H)-carboxamide —— C27H30N2O5
6,7-dimethoxy-1-((2-methoxyphenoxy)methyl)-N-(m-tolyl)-3,4-dihydroisoquinoline-2(1H)-carboxamide
—— (6S)-2-(3-chlorophenyl)imino-N-(4-fluorophenyl)-3-[(4-methoxyphenyl)methyl]-4-oxo-1,3-thiazinane-6-carboxamide —— C25H21ClFN3O3S
(6S)-2-(3-chlorophenyl)imino-N-(4-fluorophenyl)-3-[(4-methoxyphenyl)methyl]-4-oxo-1,3-thiazinane-6-carboxamide
—— (6R)-N-(2-fluorophenyl)-3-[2-(4-methoxyphenyl)ethyl]-4-oxo-2-phenylimino-1,3-thiazinane-6-carboxamide —— C26H24FN3O3S
(6R)-N-(2-fluorophenyl)-3-[2-(4-methoxyphenyl)ethyl]-4-oxo-2-phenylimino-1,3-thiazinane-6-carboxamide
—— 6-Methyl-2-[(2-phenylbutanoyl)amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide —— C20H24N2O2S
6-Methyl-2-[(2-phenylbutanoyl)amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide
—— [6-[2-(2-Hydroxyethylcarbamoyl)pyrrolidine-1-carbonyl]-3a,4,5,7a-tetrahydro-1,3-benzodioxol-4-yl] 2-[2-(2-hydroxyethoxy)ethenyl]benzoate —— C26H32N2O9
[6-[2-(2-Hydroxyethylcarbamoyl)pyrrolidine-1-carbonyl]-3a,4,5,7a-tetrahydro-1,3-benzodioxol-4-yl] 2-[2-(2-hydroxyethoxy)ethenyl]benzoate
—— 6-Chloro-8-fluoro-2-(3-methylphenyl)quinoline-4-carboxylic acid —— C17H11ClFNO2
6-Chloro-8-fluoro-2-(3-methylphenyl)quinoline-4-carboxylic acid
—— 6-tert-butyl-2-[(2-chlorobenzoyl)amino]-N-(2-methylphenyl)-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide —— C27H29ClN2O2S
6-tert-butyl-2-[(2-chlorobenzoyl)amino]-N-(2-methylphenyl)-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide
—— 6-[(1E)-2-(4-butoxyphenyl)ethenyl]-4,8-dimethylazulene —— C24H26O
6-[(1E)-2-(4-butoxyphenyl)ethenyl]-4,8-dimethylazulene
—— 6-Hydroxy-5-[(6-hydroxy-2,4-dioxo-1-phenylpyrimidin-5-yl)-[4-methoxy-3-(pyrrolidin-1-ylmethyl)phenyl]methyl]-1-phenylpyrimidine-2,4-dione —— C33H31N5O7
6-Hydroxy-5-[(6-hydroxy-2,4-dioxo-1-phenylpyrimidin-5-yl)-[4-methoxy-3-(pyrrolidin-1-ylmethyl)phenyl]methyl]-1-phenylpyrimidine-2,4-dione
—— (6R)-2-[[(2R)-2-chloropropanoyl]amino]-6-methyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide —— C13H17ClN2O2S
(6R)-2-[[(2R)-2-chloropropanoyl]amino]-6-methyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide