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二氮杂卓

中文名称 英文名称 CAS号 化学式 结构式图片
—— 4-(2,2,2-trifluoroethyl)-N-[(3R)-4,4,4-trifluoro-3-hydroxy-3-(1-methylimidazol-2-yl)butyl]-1,4-diazepane-1-carboxamide —— C16H23F6N5O2
4-(2,2,2-trifluoroethyl)-N-[(3R)-4,4,4-trifluoro-3-hydroxy-3-(1-methylimidazol-2-yl)butyl]-1,4-diazepane-1-carboxamide
—— 4-(2,2,2-trifluoroethyl)-N-[(3S)-4,4,4-trifluoro-3-hydroxy-3-(1-methylimidazol-2-yl)butyl]-1,4-diazepane-1-carboxamide —— C16H23F6N5O2
4-(2,2,2-trifluoroethyl)-N-[(3S)-4,4,4-trifluoro-3-hydroxy-3-(1-methylimidazol-2-yl)butyl]-1,4-diazepane-1-carboxamide
—— N-[(2S)-2-(diethylamino)-4-methylpentyl]-4-(2,2,2-trifluoroethyl)-1,4-diazepane-1-carboxamide —— C18H35F3N4O
N-[(2S)-2-(diethylamino)-4-methylpentyl]-4-(2,2,2-trifluoroethyl)-1,4-diazepane-1-carboxamide
—— N-[(2S)-3-ethyl-2-morpholin-4-ylpentyl]-4-(2,2,2-trifluoroethyl)-1,4-diazepane-1-carboxamide —— C19H35F3N4O2
N-[(2S)-3-ethyl-2-morpholin-4-ylpentyl]-4-(2,2,2-trifluoroethyl)-1,4-diazepane-1-carboxamide
—— N-[(2R)-2-(diethylamino)-4-methylpentyl]-4-(2,2,2-trifluoroethyl)-1,4-diazepane-1-carboxamide —— C18H35F3N4O
N-[(2R)-2-(diethylamino)-4-methylpentyl]-4-(2,2,2-trifluoroethyl)-1,4-diazepane-1-carboxamide
—— N-[2-[(2R,6R)-2,6-dimethylmorpholin-4-yl]-2-methylpropyl]-4-(2,2,2-trifluoroethyl)-1,4-diazepane-1-carboxamide —— C18H33F3N4O2
N-[2-[(2R,6R)-2,6-dimethylmorpholin-4-yl]-2-methylpropyl]-4-(2,2,2-trifluoroethyl)-1,4-diazepane-1-carboxamide
—— N-[(2R)-3-ethyl-2-morpholin-4-ylpentyl]-4-(2,2,2-trifluoroethyl)-1,4-diazepane-1-carboxamide —— C19H35F3N4O2
N-[(2R)-3-ethyl-2-morpholin-4-ylpentyl]-4-(2,2,2-trifluoroethyl)-1,4-diazepane-1-carboxamide
—— N-[2-[(2S,6S)-2,6-dimethylmorpholin-4-yl]-2-methylpropyl]-4-(2,2,2-trifluoroethyl)-1,4-diazepane-1-carboxamide —— C18H33F3N4O2
N-[2-[(2S,6S)-2,6-dimethylmorpholin-4-yl]-2-methylpropyl]-4-(2,2,2-trifluoroethyl)-1,4-diazepane-1-carboxamide
—— N-[2-[(2S,6R)-2,6-dimethylmorpholin-4-yl]-2-methylpropyl]-4-(2,2,2-trifluoroethyl)-1,4-diazepane-1-carboxamide —— C18H33F3N4O2
N-[2-[(2S,6R)-2,6-dimethylmorpholin-4-yl]-2-methylpropyl]-4-(2,2,2-trifluoroethyl)-1,4-diazepane-1-carboxamide
—— N-[(2R)-2-(5-methylfuran-2-yl)-2-morpholin-4-ylethyl]-4-(2,2,2-trifluoroethyl)-1,4-diazepane-1-carboxamide —— C19H29F3N4O3
N-[(2R)-2-(5-methylfuran-2-yl)-2-morpholin-4-ylethyl]-4-(2,2,2-trifluoroethyl)-1,4-diazepane-1-carboxamide
—— N-[(2S)-2-(5-methylfuran-2-yl)-2-morpholin-4-ylethyl]-4-(2,2,2-trifluoroethyl)-1,4-diazepane-1-carboxamide —— C19H29F3N4O3
N-[(2S)-2-(5-methylfuran-2-yl)-2-morpholin-4-ylethyl]-4-(2,2,2-trifluoroethyl)-1,4-diazepane-1-carboxamide
—— 4-[(6S)-4-[(2-aminopyrimidin-5-yl)methyl]-6-hydroxy-1,4-diazepan-1-yl]-4-oxobutanoic acid —— C14H21N5O4
4-[(6S)-4-[(2-aminopyrimidin-5-yl)methyl]-6-hydroxy-1,4-diazepan-1-yl]-4-oxobutanoic acid
—— 1-[(6S)-6-hydroxy-4-(2-hydroxyethyl)-1,4-diazepan-1-yl]-3-(4,5,6,7-tetrahydro-1H-indazol-3-yl)propan-1-one —— C17H28N4O3
1-[(6S)-6-hydroxy-4-(2-hydroxyethyl)-1,4-diazepan-1-yl]-3-(4,5,6,7-tetrahydro-1H-indazol-3-yl)propan-1-one
—— 4-[(6R)-4-[(2-aminopyrimidin-5-yl)methyl]-6-hydroxy-1,4-diazepan-1-yl]-4-oxobutanoic acid —— C14H21N5O4
4-[(6R)-4-[(2-aminopyrimidin-5-yl)methyl]-6-hydroxy-1,4-diazepan-1-yl]-4-oxobutanoic acid
—— 1-[(6R)-6-hydroxy-4-(2-hydroxyethyl)-1,4-diazepan-1-yl]-3-(4,5,6,7-tetrahydro-1H-indazol-3-yl)propan-1-one —— C17H28N4O3
1-[(6R)-6-hydroxy-4-(2-hydroxyethyl)-1,4-diazepan-1-yl]-3-(4,5,6,7-tetrahydro-1H-indazol-3-yl)propan-1-one
—— N-[(2S)-2-pyrrolidin-1-yl-2-thiophen-2-ylethyl]-4-(2,2,2-trifluoroethyl)-1,4-diazepane-1-carboxamide —— C18H27F3N4OS
N-[(2S)-2-pyrrolidin-1-yl-2-thiophen-2-ylethyl]-4-(2,2,2-trifluoroethyl)-1,4-diazepane-1-carboxamide
—— N-[(2S)-2-(diethylamino)-2-phenylethyl]-4-(2,2,2-trifluoroethyl)-1,4-diazepane-1-carboxamide —— C20H31F3N4O
N-[(2S)-2-(diethylamino)-2-phenylethyl]-4-(2,2,2-trifluoroethyl)-1,4-diazepane-1-carboxamide
—— N-[(2R)-2-(diethylamino)-2-phenylethyl]-4-(2,2,2-trifluoroethyl)-1,4-diazepane-1-carboxamide —— C20H31F3N4O
N-[(2R)-2-(diethylamino)-2-phenylethyl]-4-(2,2,2-trifluoroethyl)-1,4-diazepane-1-carboxamide
—— N-[(2R)-2-pyrrolidin-1-yl-2-thiophen-2-ylethyl]-4-(2,2,2-trifluoroethyl)-1,4-diazepane-1-carboxamide —— C18H27F3N4OS
N-[(2R)-2-pyrrolidin-1-yl-2-thiophen-2-ylethyl]-4-(2,2,2-trifluoroethyl)-1,4-diazepane-1-carboxamide
—— (6S)-1-cyclopropylsulfonyl-4-(oxan-4-yl)-1,4-diazepane-6-carboxylic acid —— C14H24N2O5S
(6S)-1-cyclopropylsulfonyl-4-(oxan-4-yl)-1,4-diazepane-6-carboxylic acid
—— 1-[(6S)-4-[(1,5-dimethylpyrazol-4-yl)methyl]-6-hydroxy-1,4-diazepan-1-yl]-3-methylbut-2-en-1-one —— C16H26N4O2
1-[(6S)-4-[(1,5-dimethylpyrazol-4-yl)methyl]-6-hydroxy-1,4-diazepan-1-yl]-3-methylbut-2-en-1-one
—— 1-[(6R)-4-[(1,5-dimethylpyrazol-4-yl)methyl]-6-hydroxy-1,4-diazepan-1-yl]-3-methylbut-2-en-1-one —— C16H26N4O2
1-[(6R)-4-[(1,5-dimethylpyrazol-4-yl)methyl]-6-hydroxy-1,4-diazepan-1-yl]-3-methylbut-2-en-1-one
—— [(4R)-2,2-dimethyloxan-4-yl]-[4-(thiophen-2-ylmethyl)-1,4-diazepan-1-yl]methanone —— C18H28N2O2S
[(4R)-2,2-dimethyloxan-4-yl]-[4-(thiophen-2-ylmethyl)-1,4-diazepan-1-yl]methanone
—— [(4S)-2,2-dimethyloxan-4-yl]-[4-(thiophen-2-ylmethyl)-1,4-diazepan-1-yl]methanone —— C18H28N2O2S
[(4S)-2,2-dimethyloxan-4-yl]-[4-(thiophen-2-ylmethyl)-1,4-diazepan-1-yl]methanone
—— (1R,6S)-N-(6-methylpyridin-2-yl)-9-propan-2-yl-3,9-diazabicyclo[4.2.1]nonane-3-carboxamide —— C17H26N4O
(1R,6S)-N-(6-methylpyridin-2-yl)-9-propan-2-yl-3,9-diazabicyclo[4.2.1]nonane-3-carboxamide
—— (1S,6R)-N-(6-methylpyridin-2-yl)-9-propan-2-yl-3,9-diazabicyclo[4.2.1]nonane-3-carboxamide —— C17H26N4O
(1S,6R)-N-(6-methylpyridin-2-yl)-9-propan-2-yl-3,9-diazabicyclo[4.2.1]nonane-3-carboxamide
—— 1-[(2R)-4-(3-fluorophenyl)butan-2-yl]-4-methylsulfonyl-1,4-diazepane —— C16H25FN2O2S
1-[(2R)-4-(3-fluorophenyl)butan-2-yl]-4-methylsulfonyl-1,4-diazepane
—— 4-[(2S)-4-(3-fluorophenyl)butan-2-yl]-1,4-diazepane-1-carboxamide —— C16H24FN3O
4-[(2S)-4-(3-fluorophenyl)butan-2-yl]-1,4-diazepane-1-carboxamide
—— 1-[(2S)-4-(3-fluorophenyl)butan-2-yl]-4-methylsulfonyl-1,4-diazepane —— C16H25FN2O2S
1-[(2S)-4-(3-fluorophenyl)butan-2-yl]-4-methylsulfonyl-1,4-diazepane
—— 1-[(2R)-4-(3-fluorophenyl)butan-2-yl]-1,4-diazepan-5-one —— C15H21FN2O
1-[(2R)-4-(3-fluorophenyl)butan-2-yl]-1,4-diazepan-5-one
—— 1-[(2S)-4-(3-fluorophenyl)butan-2-yl]-1,4-diazepan-5-one —— C15H21FN2O
1-[(2S)-4-(3-fluorophenyl)butan-2-yl]-1,4-diazepan-5-one
—— 1-[(6R)-6-hydroxy-4-[[1-(2-methoxyethyl)imidazol-2-yl]methyl]-1,4-diazepan-1-yl]ethanone —— C14H24N4O3
1-[(6R)-6-hydroxy-4-[[1-(2-methoxyethyl)imidazol-2-yl]methyl]-1,4-diazepan-1-yl]ethanone
—— 1-[(6S)-6-hydroxy-4-[[1-(2-methoxyethyl)imidazol-2-yl]methyl]-1,4-diazepan-1-yl]ethanone —— C14H24N4O3
1-[(6S)-6-hydroxy-4-[[1-(2-methoxyethyl)imidazol-2-yl]methyl]-1,4-diazepan-1-yl]ethanone
—— (6R)-1-[(2,4-dimethylpyrazol-3-yl)methyl]-4-(oxan-4-yl)-1,4-diazepan-6-ol —— C16H28N4O2
(6R)-1-[(2,4-dimethylpyrazol-3-yl)methyl]-4-(oxan-4-yl)-1,4-diazepan-6-ol
—— 3-[[(2S)-oxolan-2-yl]methoxy]-1-[4-(2,2,2-trifluoroethyl)-1,4-diazepan-1-yl]propan-1-one —— C15H25F3N2O3
3-[[(2S)-oxolan-2-yl]methoxy]-1-[4-(2,2,2-trifluoroethyl)-1,4-diazepan-1-yl]propan-1-one
—— (6S)-1-(oxan-4-yl)-4-propanoyl-1,4-diazepane-6-carboxylic acid —— C14H24N2O4
(6S)-1-(oxan-4-yl)-4-propanoyl-1,4-diazepane-6-carboxylic acid
—— (6R)-1-(oxan-4-yl)-4-propanoyl-1,4-diazepane-6-carboxylic acid —— C14H24N2O4
(6R)-1-(oxan-4-yl)-4-propanoyl-1,4-diazepane-6-carboxylic acid
—— (6S)-1-(2-hydroxyethyl)-4-[[5-(1H-pyrazol-5-yl)thiophen-2-yl]methyl]-1,4-diazepan-6-ol —— C15H22N4O2S
(6S)-1-(2-hydroxyethyl)-4-[[5-(1H-pyrazol-5-yl)thiophen-2-yl]methyl]-1,4-diazepan-6-ol
—— (6R)-1-[(2-aminopyridin-3-yl)methyl]-4-(2-hydroxyacetyl)-1,4-diazepane-6-carboxylic acid —— C14H20N4O4
(6R)-1-[(2-aminopyridin-3-yl)methyl]-4-(2-hydroxyacetyl)-1,4-diazepane-6-carboxylic acid
—— (6S)-1-[(2-aminopyridin-3-yl)methyl]-4-(2-hydroxyacetyl)-1,4-diazepane-6-carboxylic acid —— C14H20N4O4
(6S)-1-[(2-aminopyridin-3-yl)methyl]-4-(2-hydroxyacetyl)-1,4-diazepane-6-carboxylic acid
—— 1-[(6S)-4-[[5-(furan-2-yl)-1,3,4-oxadiazol-2-yl]methyl]-6-hydroxy-1,4-diazepan-1-yl]ethanone —— C14H18N4O4
1-[(6S)-4-[[5-(furan-2-yl)-1,3,4-oxadiazol-2-yl]methyl]-6-hydroxy-1,4-diazepan-1-yl]ethanone
—— [(1R,2R)-2-methylcyclopropyl]-[4-(2,2,2-trifluoroethyl)-1,4-diazepan-1-yl]methanone —— C12H19F3N2O
[(1R,2R)-2-methylcyclopropyl]-[4-(2,2,2-trifluoroethyl)-1,4-diazepan-1-yl]methanone
—— (2S)-2-methyl-1-[4-(2,2,2-trifluoroethyl)-1,4-diazepan-1-yl]pentan-1-one —— C13H23F3N2O
(2S)-2-methyl-1-[4-(2,2,2-trifluoroethyl)-1,4-diazepan-1-yl]pentan-1-one
—— 3-[(2S)-oxolan-2-yl]-1-[4-(2,2,2-trifluoroethyl)-1,4-diazepan-1-yl]propan-1-one —— C14H23F3N2O2
3-[(2S)-oxolan-2-yl]-1-[4-(2,2,2-trifluoroethyl)-1,4-diazepan-1-yl]propan-1-one
—— 1-[(6R)-4-[[5-(furan-2-yl)-1,3,4-oxadiazol-2-yl]methyl]-6-hydroxy-1,4-diazepan-1-yl]ethanone —— C14H18N4O4
1-[(6R)-4-[[5-(furan-2-yl)-1,3,4-oxadiazol-2-yl]methyl]-6-hydroxy-1,4-diazepan-1-yl]ethanone
—— 3-[(2R)-oxolan-2-yl]-1-[4-(2,2,2-trifluoroethyl)-1,4-diazepan-1-yl]propan-1-one —— C14H23F3N2O2
3-[(2R)-oxolan-2-yl]-1-[4-(2,2,2-trifluoroethyl)-1,4-diazepan-1-yl]propan-1-one
—— [(1R,2S)-2-methylcyclopropyl]-[4-(2,2,2-trifluoroethyl)-1,4-diazepan-1-yl]methanone —— C12H19F3N2O
[(1R,2S)-2-methylcyclopropyl]-[4-(2,2,2-trifluoroethyl)-1,4-diazepan-1-yl]methanone
—— [(1S,2S)-2-methylcyclopropyl]-[4-(2,2,2-trifluoroethyl)-1,4-diazepan-1-yl]methanone —— C12H19F3N2O
[(1S,2S)-2-methylcyclopropyl]-[4-(2,2,2-trifluoroethyl)-1,4-diazepan-1-yl]methanone
—— [(1S,2R)-2-methylcyclopropyl]-[4-(2,2,2-trifluoroethyl)-1,4-diazepan-1-yl]methanone —— C12H19F3N2O
[(1S,2R)-2-methylcyclopropyl]-[4-(2,2,2-trifluoroethyl)-1,4-diazepan-1-yl]methanone
—— (2R)-2-methyl-1-[4-(2,2,2-trifluoroethyl)-1,4-diazepan-1-yl]pentan-1-one —— C13H23F3N2O
(2R)-2-methyl-1-[4-(2,2,2-trifluoroethyl)-1,4-diazepan-1-yl]pentan-1-one