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二氮杂卓

中文名称 英文名称 CAS号 化学式 结构式图片
—— (1R,6S)-9-methyl-N-[1-(pyridin-2-ylmethyl)pyrazol-3-yl]-3,9-diazabicyclo[4.2.1]nonane-3-carboxamide —— C18H24N6O
(1R,6S)-9-methyl-N-[1-(pyridin-2-ylmethyl)pyrazol-3-yl]-3,9-diazabicyclo[4.2.1]nonane-3-carboxamide
—— (2S)-1-[2-[(4-acetyl-1,4-diazepan-1-yl)methyl]-6,7-dihydro-4H-pyrazolo[1,5-a]pyrazin-5-yl]-2-hydroxy-3-methylbutan-1-one —— C19H31N5O3
(2S)-1-[2-[(4-acetyl-1,4-diazepan-1-yl)methyl]-6,7-dihydro-4H-pyrazolo[1,5-a]pyrazin-5-yl]-2-hydroxy-3-methylbutan-1-one
—— (2R)-1-[2-[(4-acetyl-1,4-diazepan-1-yl)methyl]-6,7-dihydro-4H-pyrazolo[1,5-a]pyrazin-5-yl]-2-hydroxy-3-methylbutan-1-one —— C19H31N5O3
(2R)-1-[2-[(4-acetyl-1,4-diazepan-1-yl)methyl]-6,7-dihydro-4H-pyrazolo[1,5-a]pyrazin-5-yl]-2-hydroxy-3-methylbutan-1-one
—— 2-(2-methyl-1,3-thiazol-4-yl)-1-[4-[(2S)-oxolane-2-carbonyl]-1,4-diazepan-1-yl]ethanone —— C16H23N3O3S
2-(2-methyl-1,3-thiazol-4-yl)-1-[4-[(2S)-oxolane-2-carbonyl]-1,4-diazepan-1-yl]ethanone
—— 2-(2-methyl-1,3-thiazol-4-yl)-1-[4-[(2R)-oxolane-2-carbonyl]-1,4-diazepan-1-yl]ethanone —— C16H23N3O3S
2-(2-methyl-1,3-thiazol-4-yl)-1-[4-[(2R)-oxolane-2-carbonyl]-1,4-diazepan-1-yl]ethanone
—— (2R)-2-hydroxy-4-methylsulfanyl-1-[4-(pyridin-3-ylmethyl)-1,4-diazepan-1-yl]butan-1-one —— C16H25N3O2S
(2R)-2-hydroxy-4-methylsulfanyl-1-[4-(pyridin-3-ylmethyl)-1,4-diazepan-1-yl]butan-1-one
—— 1-[[(3R)-piperidin-3-yl]methyl]-4-(thiophen-2-ylmethyl)-1,4-diazepane —— C16H27N3S
1-[[(3R)-piperidin-3-yl]methyl]-4-(thiophen-2-ylmethyl)-1,4-diazepane
—— 1-[(2R)-2-(5-fluoropyrimidin-2-yl)oxyhex-5-enyl]-4-methyl-1,4-diazepane —— C16H25FN4O
1-[(2R)-2-(5-fluoropyrimidin-2-yl)oxyhex-5-enyl]-4-methyl-1,4-diazepane
—— 1-[[(1R)-cyclohex-3-en-1-yl]methyl]-4-(pyridin-4-ylmethyl)-1,4-diazepane —— C18H27N3
1-[[(1R)-cyclohex-3-en-1-yl]methyl]-4-(pyridin-4-ylmethyl)-1,4-diazepane
—— 5-[(2R)-1-(4-methyl-1,4-diazepan-1-yl)hex-5-en-2-yl]oxypyridine-2-carbonitrile —— C18H26N4O
5-[(2R)-1-(4-methyl-1,4-diazepan-1-yl)hex-5-en-2-yl]oxypyridine-2-carbonitrile
—— (6S)-1-(3-methoxypropanoyl)-4-prop-2-enyl-6-[(2-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one —— C23H28N2O3S
(6S)-1-(3-methoxypropanoyl)-4-prop-2-enyl-6-[(2-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6S)-1-(3-phenylpropanoyl)-6-[(2-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one —— C25H26N2O2S
(6S)-1-(3-phenylpropanoyl)-6-[(2-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6R)-1-(3-phenylpropanoyl)-6-[(2-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one —— C25H26N2O2S
(6R)-1-(3-phenylpropanoyl)-6-[(2-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6R)-1-(3-methoxypropanoyl)-4-prop-2-enyl-6-[(2-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one —— C23H28N2O3S
(6R)-1-(3-methoxypropanoyl)-4-prop-2-enyl-6-[(2-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one
—— 2-hydroxy-1-[(6R)-6-(methoxymethyl)-4-methylsulfonyl-1,4-diazepan-1-yl]ethanone —— C10H20N2O5S
2-hydroxy-1-[(6R)-6-(methoxymethyl)-4-methylsulfonyl-1,4-diazepan-1-yl]ethanone
—— 1-[(6S)-6-(methoxymethyl)-4-methyl-1,4-diazepan-1-yl]ethanone —— C10H20N2O2
1-[(6S)-6-(methoxymethyl)-4-methyl-1,4-diazepan-1-yl]ethanone
—— (6S)-6-(methoxymethyl)-1-methyl-4-(1-methylimidazol-4-yl)sulfonyl-1,4-diazepane —— C12H22N4O3S
(6S)-6-(methoxymethyl)-1-methyl-4-(1-methylimidazol-4-yl)sulfonyl-1,4-diazepane
—— 6-(Methoxymethyl)-1,4-dimethyl-1,4-diazepane —— C9H20N2O
6-(Methoxymethyl)-1,4-dimethyl-1,4-diazepane
—— 1-[(6R)-6-(methoxymethyl)-4-methyl-1,4-diazepan-1-yl]ethanone —— C10H20N2O2
1-[(6R)-6-(methoxymethyl)-4-methyl-1,4-diazepan-1-yl]ethanone
—— 2-hydroxy-1-[(6S)-6-(methoxymethyl)-4-methylsulfonyl-1,4-diazepan-1-yl]ethanone —— C10H20N2O5S
2-hydroxy-1-[(6S)-6-(methoxymethyl)-4-methylsulfonyl-1,4-diazepan-1-yl]ethanone
—— 1-[(6-Hydroxy-1,4-dimethyl-1,4-diazepan-6-yl)methyl]pyrrolidin-2-one —— C12H23N3O2
1-[(6-Hydroxy-1,4-dimethyl-1,4-diazepan-6-yl)methyl]pyrrolidin-2-one
—— (6S)-4-cyclopentyl-N,N-dimethyl-6-(pyridin-2-ylmethyl)-1,4-diazepane-1-sulfonamide —— C18H30N4O2S
(6S)-4-cyclopentyl-N,N-dimethyl-6-(pyridin-2-ylmethyl)-1,4-diazepane-1-sulfonamide
—— 1-[(6R)-4-cyclopentyl-6-(pyridin-2-ylmethyl)-1,4-diazepan-1-yl]-3-(4-fluorophenyl)propan-1-one —— C25H32FN3O
1-[(6R)-4-cyclopentyl-6-(pyridin-2-ylmethyl)-1,4-diazepan-1-yl]-3-(4-fluorophenyl)propan-1-one
—— 1-[(6S)-4-cyclopentyl-6-(pyridin-2-ylmethyl)-1,4-diazepan-1-yl]-4-phenylbutan-1-one —— C26H35N3O
1-[(6S)-4-cyclopentyl-6-(pyridin-2-ylmethyl)-1,4-diazepan-1-yl]-4-phenylbutan-1-one
—— 1-[(6S)-4-[(2-ethylpyrimidin-5-yl)methyl]-6-(pyridin-2-ylmethyl)-1,4-diazepan-1-yl]ethanone —— C20H27N5O
1-[(6S)-4-[(2-ethylpyrimidin-5-yl)methyl]-6-(pyridin-2-ylmethyl)-1,4-diazepan-1-yl]ethanone
—— 1-[(6R)-4-cyclopentyl-6-(pyridin-2-ylmethyl)-1,4-diazepan-1-yl]-2-(3,5-dimethyl-1,2-oxazol-4-yl)ethanone —— C23H32N4O2
1-[(6R)-4-cyclopentyl-6-(pyridin-2-ylmethyl)-1,4-diazepan-1-yl]-2-(3,5-dimethyl-1,2-oxazol-4-yl)ethanone
—— 1-[(6R)-4-[(2-ethylpyrimidin-5-yl)methyl]-6-(pyridin-2-ylmethyl)-1,4-diazepan-1-yl]ethanone —— C20H27N5O
1-[(6R)-4-[(2-ethylpyrimidin-5-yl)methyl]-6-(pyridin-2-ylmethyl)-1,4-diazepan-1-yl]ethanone
—— 1-[(6S)-4-cyclopentyl-6-(pyridin-2-ylmethyl)-1,4-diazepan-1-yl]-2-(2-methyl-1,3-thiazol-4-yl)ethanone —— C22H30N4OS
1-[(6S)-4-cyclopentyl-6-(pyridin-2-ylmethyl)-1,4-diazepan-1-yl]-2-(2-methyl-1,3-thiazol-4-yl)ethanone
—— 1-[(6S)-4-cyclopentyl-6-(pyridin-2-ylmethyl)-1,4-diazepan-1-yl]-3-(4-fluorophenyl)propan-1-one —— C25H32FN3O
1-[(6S)-4-cyclopentyl-6-(pyridin-2-ylmethyl)-1,4-diazepan-1-yl]-3-(4-fluorophenyl)propan-1-one
—— 1-[(6S)-4-cyclopentyl-6-(pyridin-2-ylmethyl)-1,4-diazepan-1-yl]-2-(3,5-dimethyl-1,2-oxazol-4-yl)ethanone —— C23H32N4O2
1-[(6S)-4-cyclopentyl-6-(pyridin-2-ylmethyl)-1,4-diazepan-1-yl]-2-(3,5-dimethyl-1,2-oxazol-4-yl)ethanone
—— 1-[(6R)-4-cyclopentyl-6-(pyridin-2-ylmethyl)-1,4-diazepan-1-yl]-4-phenylbutan-1-one —— C26H35N3O
1-[(6R)-4-cyclopentyl-6-(pyridin-2-ylmethyl)-1,4-diazepan-1-yl]-4-phenylbutan-1-one
—— cyclopentyl-[(6S)-4-cyclopentyl-6-(pyridin-2-ylmethyl)-1,4-diazepan-1-yl]methanone —— C22H33N3O
cyclopentyl-[(6S)-4-cyclopentyl-6-(pyridin-2-ylmethyl)-1,4-diazepan-1-yl]methanone
—— cyclopentyl-[(6R)-4-cyclopentyl-6-(pyridin-2-ylmethyl)-1,4-diazepan-1-yl]methanone —— C22H33N3O
cyclopentyl-[(6R)-4-cyclopentyl-6-(pyridin-2-ylmethyl)-1,4-diazepan-1-yl]methanone
—— 1-[(6R)-4-acetyl-6-(pyridin-2-ylmethyl)-1,4-diazepan-1-yl]-3-phenylpropan-1-one —— C22H27N3O2
1-[(6R)-4-acetyl-6-(pyridin-2-ylmethyl)-1,4-diazepan-1-yl]-3-phenylpropan-1-one
—— 1-[(6R)-4-methylsulfonyl-6-(pyridin-2-ylmethyl)-1,4-diazepan-1-yl]-3-phenylpropan-1-one —— C21H27N3O3S
1-[(6R)-4-methylsulfonyl-6-(pyridin-2-ylmethyl)-1,4-diazepan-1-yl]-3-phenylpropan-1-one
—— (6S)-1-cyclopentyl-6-(pyridin-2-ylmethyl)-4-pyrrolidin-1-ylsulfonyl-1,4-diazepane —— C20H32N4O2S
(6S)-1-cyclopentyl-6-(pyridin-2-ylmethyl)-4-pyrrolidin-1-ylsulfonyl-1,4-diazepane
—— 2-cyclopentyl-1-[(6R)-4-cyclopentyl-6-(pyridin-2-ylmethyl)-1,4-diazepan-1-yl]ethanone —— C23H35N3O
2-cyclopentyl-1-[(6R)-4-cyclopentyl-6-(pyridin-2-ylmethyl)-1,4-diazepan-1-yl]ethanone
—— (6R)-1-cyclopentyl-6-(pyridin-2-ylmethyl)-4-pyrrolidin-1-ylsulfonyl-1,4-diazepane —— C20H32N4O2S
(6R)-1-cyclopentyl-6-(pyridin-2-ylmethyl)-4-pyrrolidin-1-ylsulfonyl-1,4-diazepane
—— 1-[(6S)-4-methylsulfonyl-6-(pyridin-2-ylmethyl)-1,4-diazepan-1-yl]-3-phenylpropan-1-one —— C21H27N3O3S
1-[(6S)-4-methylsulfonyl-6-(pyridin-2-ylmethyl)-1,4-diazepan-1-yl]-3-phenylpropan-1-one
—— 1-[(6R)-4-cyclopentyl-6-(pyridin-2-ylmethyl)-1,4-diazepan-1-yl]-2-(2-methyl-1,3-thiazol-4-yl)ethanone —— C22H30N4OS
1-[(6R)-4-cyclopentyl-6-(pyridin-2-ylmethyl)-1,4-diazepan-1-yl]-2-(2-methyl-1,3-thiazol-4-yl)ethanone
—— cyclobutyl-[(6S)-4-cyclopentyl-6-(pyridin-2-ylmethyl)-1,4-diazepan-1-yl]methanone —— C21H31N3O
cyclobutyl-[(6S)-4-cyclopentyl-6-(pyridin-2-ylmethyl)-1,4-diazepan-1-yl]methanone
—— cyclobutyl-[(6R)-4-cyclopentyl-6-(pyridin-2-ylmethyl)-1,4-diazepan-1-yl]methanone —— C21H31N3O
cyclobutyl-[(6R)-4-cyclopentyl-6-(pyridin-2-ylmethyl)-1,4-diazepan-1-yl]methanone
—— 1-[(6S)-4-acetyl-6-(pyridin-2-ylmethyl)-1,4-diazepan-1-yl]-3-phenylpropan-1-one —— C22H27N3O2
1-[(6S)-4-acetyl-6-(pyridin-2-ylmethyl)-1,4-diazepan-1-yl]-3-phenylpropan-1-one
—— cyclohexyl-[(6R)-4-cyclopentyl-6-(pyridin-2-ylmethyl)-1,4-diazepan-1-yl]methanone —— C23H35N3O
cyclohexyl-[(6R)-4-cyclopentyl-6-(pyridin-2-ylmethyl)-1,4-diazepan-1-yl]methanone
—— 2-cyclopentyl-1-[(6S)-4-cyclopentyl-6-(pyridin-2-ylmethyl)-1,4-diazepan-1-yl]ethanone —— C23H35N3O
2-cyclopentyl-1-[(6S)-4-cyclopentyl-6-(pyridin-2-ylmethyl)-1,4-diazepan-1-yl]ethanone
—— 3-(4-fluorophenyl)-1-[(6S)-6-hydroxy-4-methyl-6-(1,2,4-triazol-1-ylmethyl)-1,4-diazepan-1-yl]propan-1-one —— C18H24FN5O2
3-(4-fluorophenyl)-1-[(6S)-6-hydroxy-4-methyl-6-(1,2,4-triazol-1-ylmethyl)-1,4-diazepan-1-yl]propan-1-one
—— 3-(4-fluorophenyl)-1-[(6S)-6-hydroxy-4-methyl-6-[(2-methylimidazol-1-yl)methyl]-1,4-diazepan-1-yl]propan-1-one —— C20H27FN4O2
3-(4-fluorophenyl)-1-[(6S)-6-hydroxy-4-methyl-6-[(2-methylimidazol-1-yl)methyl]-1,4-diazepan-1-yl]propan-1-one
—— 3-(4-fluorophenyl)-1-[(6R)-6-hydroxy-4-methyl-6-(pyrazol-1-ylmethyl)-1,4-diazepan-1-yl]propan-1-one —— C19H25FN4O2
3-(4-fluorophenyl)-1-[(6R)-6-hydroxy-4-methyl-6-(pyrazol-1-ylmethyl)-1,4-diazepan-1-yl]propan-1-one
—— 1-[(6R)-6-hydroxy-4-methyl-6-(pyrazol-1-ylmethyl)-1,4-diazepan-1-yl]-3-phenylpropan-1-one —— C19H26N4O2
1-[(6R)-6-hydroxy-4-methyl-6-(pyrazol-1-ylmethyl)-1,4-diazepan-1-yl]-3-phenylpropan-1-one
—— (6R)-6-(methoxymethyl)-1-(pyridin-3-ylmethyl)-1,4-diazepane —— C13H21N3O
(6R)-6-(methoxymethyl)-1-(pyridin-3-ylmethyl)-1,4-diazepane