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二氮杂卓

中文名称 英文名称 CAS号 化学式 结构式图片
—— (6R)-1-(cyclobutanecarbonyl)-4-methyl-6-[(4-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one —— C22H26N2O2S
(6R)-1-(cyclobutanecarbonyl)-4-methyl-6-[(4-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6S)-1-(cyclopentanecarbonyl)-4-methyl-6-[(4-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one —— C23H28N2O2S
(6S)-1-(cyclopentanecarbonyl)-4-methyl-6-[(4-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one
—— Ethyl 9-methyl-4-oxo-5,6-diazatricyclo[5.2.0.02,5]non-8-ene-6-carboxylate —— C11H14N2O3
Ethyl 9-methyl-4-oxo-5,6-diazatricyclo[5.2.0.02,5]non-8-ene-6-carboxylate
—— (6S)-4-ethyl-1-[(1-ethylimidazol-2-yl)methyl]-6-[(4-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one —— C24H30N4OS
(6S)-4-ethyl-1-[(1-ethylimidazol-2-yl)methyl]-6-[(4-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6R)-4-ethyl-1-[(1-ethylimidazol-2-yl)methyl]-6-[(4-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one —— C24H30N4OS
(6R)-4-ethyl-1-[(1-ethylimidazol-2-yl)methyl]-6-[(4-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6R)-1-[(5-methoxy-1,3-dimethylpyrazol-4-yl)methyl]-4-methyl-6-[(4-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one —— C24H30N4O2S
(6R)-1-[(5-methoxy-1,3-dimethylpyrazol-4-yl)methyl]-4-methyl-6-[(4-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6S)-1-[(5-methoxy-1,3-dimethylpyrazol-4-yl)methyl]-4-methyl-6-[(4-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one —— C24H30N4O2S
(6S)-1-[(5-methoxy-1,3-dimethylpyrazol-4-yl)methyl]-4-methyl-6-[(4-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6R)-4-ethyl-1-(3-pyridin-4-ylpropanoyl)-6-[(2-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one —— C26H29N3O2S
(6R)-4-ethyl-1-(3-pyridin-4-ylpropanoyl)-6-[(2-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6R)-4-ethyl-1-(3-methoxypropanoyl)-6-[(2-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one —— C22H28N2O3S
(6R)-4-ethyl-1-(3-methoxypropanoyl)-6-[(2-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6S)-4-ethyl-1-(2-pyrazol-1-ylacetyl)-6-[(2-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one —— C23H26N4O2S
(6S)-4-ethyl-1-(2-pyrazol-1-ylacetyl)-6-[(2-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6S)-1-(cyclobutanecarbonyl)-4-ethyl-6-[(2-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one —— C23H28N2O2S
(6S)-1-(cyclobutanecarbonyl)-4-ethyl-6-[(2-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6S)-4-ethyl-1-(2-pyridin-2-yloxyacetyl)-6-[(2-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one —— C25H27N3O3S
(6S)-4-ethyl-1-(2-pyridin-2-yloxyacetyl)-6-[(2-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6R)-4-ethyl-1-(2-pyrazol-1-ylacetyl)-6-[(2-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one —— C23H26N4O2S
(6R)-4-ethyl-1-(2-pyrazol-1-ylacetyl)-6-[(2-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6S)-4-ethyl-1-(3-methoxypropanoyl)-6-[(2-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one —— C22H28N2O3S
(6S)-4-ethyl-1-(3-methoxypropanoyl)-6-[(2-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6S)-4-ethyl-1-(3-pyridin-4-ylpropanoyl)-6-[(2-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one —— C26H29N3O2S
(6S)-4-ethyl-1-(3-pyridin-4-ylpropanoyl)-6-[(2-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6R)-4-ethyl-1-[3-[(2R)-oxolan-2-yl]propanoyl]-6-[(4-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one —— C25H32N2O3S
(6R)-4-ethyl-1-[3-[(2R)-oxolan-2-yl]propanoyl]-6-[(4-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6R)-4-ethyl-1-(3-pyrazol-1-ylpropanoyl)-6-[(4-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one —— C24H28N4O2S
(6R)-4-ethyl-1-(3-pyrazol-1-ylpropanoyl)-6-[(4-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6R)-4-ethyl-1-(2-pyrazol-1-ylacetyl)-6-[(4-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one —— C23H26N4O2S
(6R)-4-ethyl-1-(2-pyrazol-1-ylacetyl)-6-[(4-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6R)-4-ethyl-1-[3-[(2S)-oxolan-2-yl]propanoyl]-6-[(4-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one —— C25H32N2O3S
(6R)-4-ethyl-1-[3-[(2S)-oxolan-2-yl]propanoyl]-6-[(4-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6R)-1-(cyclobutanecarbonyl)-4-ethyl-6-[(2-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one —— C23H28N2O2S
(6R)-1-(cyclobutanecarbonyl)-4-ethyl-6-[(2-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6S)-4-ethyl-1-(2-pyrazol-1-ylacetyl)-6-[(4-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one —— C23H26N4O2S
(6S)-4-ethyl-1-(2-pyrazol-1-ylacetyl)-6-[(4-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6S)-4-ethyl-1-(3-pyrazol-1-ylpropanoyl)-6-[(4-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one —— C24H28N4O2S
(6S)-4-ethyl-1-(3-pyrazol-1-ylpropanoyl)-6-[(4-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6S)-4-ethyl-1-[3-[(2S)-oxolan-2-yl]propanoyl]-6-[(4-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one —— C25H32N2O3S
(6S)-4-ethyl-1-[3-[(2S)-oxolan-2-yl]propanoyl]-6-[(4-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6S)-4-propyl-6-[(2-thiophen-2-ylphenyl)methyl]-1-[2-(1,2,4-triazol-1-yl)acetyl]-1,4-diazepan-5-one —— C23H27N5O2S
(6S)-4-propyl-6-[(2-thiophen-2-ylphenyl)methyl]-1-[2-(1,2,4-triazol-1-yl)acetyl]-1,4-diazepan-5-one
—— (6R)-4-propyl-6-[(2-thiophen-2-ylphenyl)methyl]-1-[2-(1,2,4-triazol-1-yl)acetyl]-1,4-diazepan-5-one —— C23H27N5O2S
(6R)-4-propyl-6-[(2-thiophen-2-ylphenyl)methyl]-1-[2-(1,2,4-triazol-1-yl)acetyl]-1,4-diazepan-5-one
—— (6R)-4-propyl-1-(2-pyridin-3-ylacetyl)-6-[(4-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one —— C26H29N3O2S
(6R)-4-propyl-1-(2-pyridin-3-ylacetyl)-6-[(4-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6R)-4-propyl-1-(2-pyrazol-1-ylacetyl)-6-[(2-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one —— C24H28N4O2S
(6R)-4-propyl-1-(2-pyrazol-1-ylacetyl)-6-[(2-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6R)-4-propyl-6-[(3-thiophen-2-ylphenyl)methyl]-1-[2-(1,2,4-triazol-1-yl)acetyl]-1,4-diazepan-5-one —— C23H27N5O2S
(6R)-4-propyl-6-[(3-thiophen-2-ylphenyl)methyl]-1-[2-(1,2,4-triazol-1-yl)acetyl]-1,4-diazepan-5-one
—— (6S)-4-propyl-6-[(4-thiophen-2-ylphenyl)methyl]-1-[2-(1,2,4-triazol-1-yl)acetyl]-1,4-diazepan-5-one —— C23H27N5O2S
(6S)-4-propyl-6-[(4-thiophen-2-ylphenyl)methyl]-1-[2-(1,2,4-triazol-1-yl)acetyl]-1,4-diazepan-5-one
—— (6S)-1-(2-methoxyacetyl)-4-propyl-6-[(4-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one —— C22H28N2O3S
(6S)-1-(2-methoxyacetyl)-4-propyl-6-[(4-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6S)-4-propyl-1-(2-pyridin-3-ylacetyl)-6-[(4-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one —— C26H29N3O2S
(6S)-4-propyl-1-(2-pyridin-3-ylacetyl)-6-[(4-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6S)-4-propyl-6-[(3-thiophen-2-ylphenyl)methyl]-1-[2-(1,2,4-triazol-1-yl)acetyl]-1,4-diazepan-5-one —— C23H27N5O2S
(6S)-4-propyl-6-[(3-thiophen-2-ylphenyl)methyl]-1-[2-(1,2,4-triazol-1-yl)acetyl]-1,4-diazepan-5-one
—— (6S)-4-propyl-1-(2-pyrazol-1-ylacetyl)-6-[(2-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one —— C24H28N4O2S
(6S)-4-propyl-1-(2-pyrazol-1-ylacetyl)-6-[(2-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6R)-4-ethyl-1-propanoyl-6-[(2-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one —— C21H26N2O2S
(6R)-4-ethyl-1-propanoyl-6-[(2-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6S)-4-methyl-1-propanoyl-6-[(2-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one —— C20H24N2O2S
(6S)-4-methyl-1-propanoyl-6-[(2-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one
—— (1S,6R)-3,9-dimethyl-3,9-diazabicyclo[4.2.1]nonane —— C9H18N2
(1S,6R)-3,9-dimethyl-3,9-diazabicyclo[4.2.1]nonane
—— (6S)-1-(cyclohexanecarbonyl)-6-[(2-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one —— C23H28N2O2S
(6S)-1-(cyclohexanecarbonyl)-6-[(2-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6R)-1-(cyclobutanecarbonyl)-6-[(2-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one —— C21H24N2O2S
(6R)-1-(cyclobutanecarbonyl)-6-[(2-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6R)-1-(cyclohexanecarbonyl)-6-[(2-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one —— C23H28N2O2S
(6R)-1-(cyclohexanecarbonyl)-6-[(2-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6S)-1-(cyclobutanecarbonyl)-6-[(2-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one —— C21H24N2O2S
(6S)-1-(cyclobutanecarbonyl)-6-[(2-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one
—— 4-[(5R)-1,4,6,6-tetramethyl-1,4-diazepan-5-yl]morpholine —— C13H27N3O
4-[(5R)-1,4,6,6-tetramethyl-1,4-diazepan-5-yl]morpholine
—— (6R)-1-[(2S)-oxolane-2-carbonyl]-4-prop-2-enyl-6-[(4-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one —— C24H28N2O3S
(6R)-1-[(2S)-oxolane-2-carbonyl]-4-prop-2-enyl-6-[(4-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6S)-1-[(2S)-oxolane-2-carbonyl]-4-prop-2-enyl-6-[(4-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one —— C24H28N2O3S
(6S)-1-[(2S)-oxolane-2-carbonyl]-4-prop-2-enyl-6-[(4-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6S)-1-[(2R)-oxolane-2-carbonyl]-4-prop-2-enyl-6-[(4-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one —— C24H28N2O3S
(6S)-1-[(2R)-oxolane-2-carbonyl]-4-prop-2-enyl-6-[(4-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6S)-4-prop-2-enyl-1-(2-pyridin-3-ylacetyl)-6-[(4-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one —— C26H27N3O2S
(6S)-4-prop-2-enyl-1-(2-pyridin-3-ylacetyl)-6-[(4-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6R)-4-prop-2-enyl-1-(2-pyridin-3-ylacetyl)-6-[(4-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one —— C26H27N3O2S
(6R)-4-prop-2-enyl-1-(2-pyridin-3-ylacetyl)-6-[(4-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6S)-1-(1H-imidazol-2-ylmethyl)-4-prop-2-enyl-6-[(4-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one —— C23H26N4OS
(6S)-1-(1H-imidazol-2-ylmethyl)-4-prop-2-enyl-6-[(4-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one
—— (1S,6R)-11-methyl-3,11-diazabicyclo[4.4.1]undecan-4-one —— C10H18N2O
(1S,6R)-11-methyl-3,11-diazabicyclo[4.4.1]undecan-4-one
—— (1S,6R)-10-methyl-3,10-diazabicyclo[4.3.1]decan-4-one —— C9H16N2O
(1S,6R)-10-methyl-3,10-diazabicyclo[4.3.1]decan-4-one
—— 2-(4-Methyl-1,4-diazepan-1-yl)-1-phenylethanol —— C14H22N2O
2-(4-Methyl-1,4-diazepan-1-yl)-1-phenylethanol