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二氮杂卓

中文名称 英文名称 CAS号 化学式 结构式图片
—— 1-[(3S)-4-(cyclopropylmethyl)-3-propan-2-yl-1,4-diazepan-1-yl]-3-(5-methyl-1H-1,2,4-triazol-3-yl)propan-1-one —— C18H31N5O
1-[(3S)-4-(cyclopropylmethyl)-3-propan-2-yl-1,4-diazepan-1-yl]-3-(5-methyl-1H-1,2,4-triazol-3-yl)propan-1-one
—— (3S)-4-(cyclopropylmethyl)-1-(1H-imidazol-5-ylmethyl)-3-propan-2-yl-1,4-diazepan-5-one —— C16H26N4O
(3S)-4-(cyclopropylmethyl)-1-(1H-imidazol-5-ylmethyl)-3-propan-2-yl-1,4-diazepan-5-one
—— (3R)-4-(cyclopropylmethyl)-1-[(1,4-dimethylpiperidin-4-yl)methyl]-3-propan-2-yl-1,4-diazepan-5-one —— C20H37N3O
(3R)-4-(cyclopropylmethyl)-1-[(1,4-dimethylpiperidin-4-yl)methyl]-3-propan-2-yl-1,4-diazepan-5-one
—— (3R)-4-[(4-fluorophenyl)methyl]-1-[(2-methyl-1,3-oxazol-4-yl)methyl]-3-propan-2-yl-1,4-diazepan-5-one —— C20H26FN3O2
(3R)-4-[(4-fluorophenyl)methyl]-1-[(2-methyl-1,3-oxazol-4-yl)methyl]-3-propan-2-yl-1,4-diazepan-5-one
—— (3S)-4-[(4-fluorophenyl)methyl]-1-[3-(5-methyltetrazol-1-yl)propyl]-3-propan-2-yl-1,4-diazepan-5-one —— C20H29FN6O
(3S)-4-[(4-fluorophenyl)methyl]-1-[3-(5-methyltetrazol-1-yl)propyl]-3-propan-2-yl-1,4-diazepan-5-one
—— (3R)-1-[(1-ethyl-3-methylpyrazol-4-yl)methyl]-4-[(4-fluorophenyl)methyl]-3-propan-2-yl-1,4-diazepan-5-one —— C22H31FN4O
(3R)-1-[(1-ethyl-3-methylpyrazol-4-yl)methyl]-4-[(4-fluorophenyl)methyl]-3-propan-2-yl-1,4-diazepan-5-one
—— (3R)-4-[(4-fluorophenyl)methyl]-1-[3-(5-methyltetrazol-1-yl)propyl]-3-propan-2-yl-1,4-diazepan-5-one —— C20H29FN6O
(3R)-4-[(4-fluorophenyl)methyl]-1-[3-(5-methyltetrazol-1-yl)propyl]-3-propan-2-yl-1,4-diazepan-5-one
—— (3R)-4-(cyclopropylmethyl)-3-propan-2-yl-1-(5-propyl-1,2-oxazole-4-carbonyl)-1,4-diazepan-5-one —— C19H29N3O3
(3R)-4-(cyclopropylmethyl)-3-propan-2-yl-1-(5-propyl-1,2-oxazole-4-carbonyl)-1,4-diazepan-5-one
—— (3R)-4-(cyclopropylmethyl)-1-(1H-imidazol-5-ylmethyl)-3-propan-2-yl-1,4-diazepan-5-one —— C16H26N4O
(3R)-4-(cyclopropylmethyl)-1-(1H-imidazol-5-ylmethyl)-3-propan-2-yl-1,4-diazepan-5-one
—— (3S)-4-[(4-fluorophenyl)methyl]-1-[(2-methyl-1,3-oxazol-4-yl)methyl]-3-propan-2-yl-1,4-diazepan-5-one —— C20H26FN3O2
(3S)-4-[(4-fluorophenyl)methyl]-1-[(2-methyl-1,3-oxazol-4-yl)methyl]-3-propan-2-yl-1,4-diazepan-5-one
—— (3S)-4-benzyl-3-ethyl-1-[4-(1H-pyrazol-4-yl)butanoyl]-1,4-diazepan-5-one —— C21H28N4O2
(3S)-4-benzyl-3-ethyl-1-[4-(1H-pyrazol-4-yl)butanoyl]-1,4-diazepan-5-one
—— (3S)-4-(cyclopropylmethyl)-3-propan-2-yl-1-(5-propyl-1,2-oxazole-4-carbonyl)-1,4-diazepan-5-one —— C19H29N3O3
(3S)-4-(cyclopropylmethyl)-3-propan-2-yl-1-(5-propyl-1,2-oxazole-4-carbonyl)-1,4-diazepan-5-one
—— (3R)-4-[(4-fluorophenyl)methyl]-1-[(5-methylfuran-2-yl)methyl]-3-propan-2-yl-1,4-diazepan-5-one —— C21H27FN2O2
(3R)-4-[(4-fluorophenyl)methyl]-1-[(5-methylfuran-2-yl)methyl]-3-propan-2-yl-1,4-diazepan-5-one
—— (3R)-1-[4-(dimethylamino)butanoyl]-4-[(4-fluorophenyl)methyl]-3-propan-2-yl-1,4-diazepan-5-one —— C21H32FN3O2
(3R)-1-[4-(dimethylamino)butanoyl]-4-[(4-fluorophenyl)methyl]-3-propan-2-yl-1,4-diazepan-5-one
—— (3S)-1-[(1-ethyl-3-methylpyrazol-4-yl)methyl]-4-[(4-fluorophenyl)methyl]-3-propan-2-yl-1,4-diazepan-5-one —— C22H31FN4O
(3S)-1-[(1-ethyl-3-methylpyrazol-4-yl)methyl]-4-[(4-fluorophenyl)methyl]-3-propan-2-yl-1,4-diazepan-5-one
—— (3S)-4-[(4-fluorophenyl)methyl]-1-[(5-methylfuran-2-yl)methyl]-3-propan-2-yl-1,4-diazepan-5-one —— C21H27FN2O2
(3S)-4-[(4-fluorophenyl)methyl]-1-[(5-methylfuran-2-yl)methyl]-3-propan-2-yl-1,4-diazepan-5-one
—— (3S)-1-[4-(dimethylamino)butanoyl]-4-[(4-fluorophenyl)methyl]-3-propan-2-yl-1,4-diazepan-5-one —— C21H32FN3O2
(3S)-1-[4-(dimethylamino)butanoyl]-4-[(4-fluorophenyl)methyl]-3-propan-2-yl-1,4-diazepan-5-one
—— (3R)-4-benzyl-3-ethyl-1-[(1-methylpiperidin-4-yl)methyl]-1,4-diazepan-5-one —— C21H33N3O
(3R)-4-benzyl-3-ethyl-1-[(1-methylpiperidin-4-yl)methyl]-1,4-diazepan-5-one
—— (3R)-4-benzyl-3-ethyl-1-[(3-propan-2-ylimidazol-4-yl)methyl]-1,4-diazepan-5-one —— C21H30N4O
(3R)-4-benzyl-3-ethyl-1-[(3-propan-2-ylimidazol-4-yl)methyl]-1,4-diazepan-5-one
—— (3S)-4-benzyl-3-ethyl-1-[(1-methylpiperidin-4-yl)methyl]-1,4-diazepan-5-one —— C21H33N3O
(3S)-4-benzyl-3-ethyl-1-[(1-methylpiperidin-4-yl)methyl]-1,4-diazepan-5-one
—— (3R)-4-(cyclopropylmethyl)-1-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propanoyl]-3-propan-2-yl-1,4-diazepan-5-one —— C20H32N4O2
(3R)-4-(cyclopropylmethyl)-1-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propanoyl]-3-propan-2-yl-1,4-diazepan-5-one
—— (3S)-4-[(4-fluorophenyl)methyl]-3-propan-2-yl-1-[(5-propan-2-yl-1,2,4-oxadiazol-3-yl)methyl]-1,4-diazepan-5-one —— C21H29FN4O2
(3S)-4-[(4-fluorophenyl)methyl]-3-propan-2-yl-1-[(5-propan-2-yl-1,2,4-oxadiazol-3-yl)methyl]-1,4-diazepan-5-one
—— (3R)-4-[(4-fluorophenyl)methyl]-3-propan-2-yl-1-[(5-propan-2-yl-1,2,4-oxadiazol-3-yl)methyl]-1,4-diazepan-5-one —— C21H29FN4O2
(3R)-4-[(4-fluorophenyl)methyl]-3-propan-2-yl-1-[(5-propan-2-yl-1,2,4-oxadiazol-3-yl)methyl]-1,4-diazepan-5-one
—— (3S)-4-(cyclopropylmethyl)-1-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propanoyl]-3-propan-2-yl-1,4-diazepan-5-one —— C20H32N4O2
(3S)-4-(cyclopropylmethyl)-1-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propanoyl]-3-propan-2-yl-1,4-diazepan-5-one
—— (3S)-4-benzyl-3-ethyl-1-[[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl]-1,4-diazepan-5-one —— C20H28N4O3
(3S)-4-benzyl-3-ethyl-1-[[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl]-1,4-diazepan-5-one
—— (3R)-4-benzyl-3-ethyl-1-[[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl]-1,4-diazepan-5-one —— C20H28N4O3
(3R)-4-benzyl-3-ethyl-1-[[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl]-1,4-diazepan-5-one
—— (3S)-4-[(4-fluorophenyl)methyl]-3-propan-2-yl-1-(2-pyrazol-1-ylethyl)-1,4-diazepan-5-one —— C20H27FN4O
(3S)-4-[(4-fluorophenyl)methyl]-3-propan-2-yl-1-(2-pyrazol-1-ylethyl)-1,4-diazepan-5-one
—— (3S)-1-(5-ethyl-1,2-oxazole-4-carbonyl)-4-[(4-fluorophenyl)methyl]-3-propan-2-yl-1,4-diazepan-5-one —— C21H26FN3O3
(3S)-1-(5-ethyl-1,2-oxazole-4-carbonyl)-4-[(4-fluorophenyl)methyl]-3-propan-2-yl-1,4-diazepan-5-one
—— (3R)-4-benzyl-3-ethyl-1-[2-(3-methyl-1,2-oxazol-5-yl)acetyl]-1,4-diazepan-5-one —— C20H25N3O3
(3R)-4-benzyl-3-ethyl-1-[2-(3-methyl-1,2-oxazol-5-yl)acetyl]-1,4-diazepan-5-one
—— (3R)-4-[(4-fluorophenyl)methyl]-3-propan-2-yl-1-(2-pyrazol-1-ylethyl)-1,4-diazepan-5-one —— C20H27FN4O
(3R)-4-[(4-fluorophenyl)methyl]-3-propan-2-yl-1-(2-pyrazol-1-ylethyl)-1,4-diazepan-5-one
—— (3S)-4-[(4-fluorophenyl)methyl]-3-propan-2-yl-1-[2-(1H-pyrazol-4-yl)ethyl]-1,4-diazepan-5-one —— C20H27FN4O
(3S)-4-[(4-fluorophenyl)methyl]-3-propan-2-yl-1-[2-(1H-pyrazol-4-yl)ethyl]-1,4-diazepan-5-one
—— (3S)-4-benzyl-3-ethyl-1-[2-(3-methyl-1,2-oxazol-5-yl)acetyl]-1,4-diazepan-5-one —— C20H25N3O3
(3S)-4-benzyl-3-ethyl-1-[2-(3-methyl-1,2-oxazol-5-yl)acetyl]-1,4-diazepan-5-one
—— (3R)-1-(5-ethyl-1,2-oxazole-4-carbonyl)-4-[(4-fluorophenyl)methyl]-3-propan-2-yl-1,4-diazepan-5-one —— C21H26FN3O3
(3R)-1-(5-ethyl-1,2-oxazole-4-carbonyl)-4-[(4-fluorophenyl)methyl]-3-propan-2-yl-1,4-diazepan-5-one
—— (3R)-4-[(4-fluorophenyl)methyl]-N,N-dimethyl-5-oxo-3-propan-2-yl-1,4-diazepane-1-sulfonamide —— C17H26FN3O3S
(3R)-4-[(4-fluorophenyl)methyl]-N,N-dimethyl-5-oxo-3-propan-2-yl-1,4-diazepane-1-sulfonamide
—— (3S)-4-benzyl-3-ethyl-1-(4-methoxycyclohexanecarbonyl)-1,4-diazepan-5-one —— C22H32N2O3
(3S)-4-benzyl-3-ethyl-1-(4-methoxycyclohexanecarbonyl)-1,4-diazepan-5-one
—— (3S)-4-[(4-fluorophenyl)methyl]-N,N-dimethyl-5-oxo-3-propan-2-yl-1,4-diazepane-1-sulfonamide —— C17H26FN3O3S
(3S)-4-[(4-fluorophenyl)methyl]-N,N-dimethyl-5-oxo-3-propan-2-yl-1,4-diazepane-1-sulfonamide
—— 1-[(3R)-4-(cyclopropylmethyl)-3-propan-2-yl-1,4-diazepan-1-yl]-2-(2-methylimidazol-1-yl)ethanone —— C18H30N4O
1-[(3R)-4-(cyclopropylmethyl)-3-propan-2-yl-1,4-diazepan-1-yl]-2-(2-methylimidazol-1-yl)ethanone
—— 1-[(3S)-4-(cyclopropylmethyl)-3-propan-2-yl-1,4-diazepan-1-yl]-2-(2-methylimidazol-1-yl)ethanone —— C18H30N4O
1-[(3S)-4-(cyclopropylmethyl)-3-propan-2-yl-1,4-diazepan-1-yl]-2-(2-methylimidazol-1-yl)ethanone
—— (2R)-1-(cyclopropylmethyl)-2-propan-2-yl-4-(1,3,5-trimethylpyrazol-4-yl)sulfonyl-1,4-diazepane —— C18H32N4O2S
(2R)-1-(cyclopropylmethyl)-2-propan-2-yl-4-(1,3,5-trimethylpyrazol-4-yl)sulfonyl-1,4-diazepane
—— (3R)-4-(cyclopropylmethyl)-3-propan-2-yl-1-[(1-propan-2-ylimidazol-2-yl)methyl]-1,4-diazepan-5-one —— C19H32N4O
(3R)-4-(cyclopropylmethyl)-3-propan-2-yl-1-[(1-propan-2-ylimidazol-2-yl)methyl]-1,4-diazepan-5-one
—— (3R)-4-benzyl-3-ethyl-1-[3-(1,2,4-triazol-4-yl)propanoyl]-1,4-diazepan-5-one —— C19H25N5O2
(3R)-4-benzyl-3-ethyl-1-[3-(1,2,4-triazol-4-yl)propanoyl]-1,4-diazepan-5-one
—— (3S)-4-(cyclopropylmethyl)-3-propan-2-yl-1-[(1-propan-2-ylimidazol-2-yl)methyl]-1,4-diazepan-5-one —— C19H32N4O
(3S)-4-(cyclopropylmethyl)-3-propan-2-yl-1-[(1-propan-2-ylimidazol-2-yl)methyl]-1,4-diazepan-5-one
—— (3R)-4-(cyclopropylmethyl)-3-propan-2-yl-1-[3-(tetrazol-1-yl)propanoyl]-1,4-diazepan-5-one —— C16H26N6O2
(3R)-4-(cyclopropylmethyl)-3-propan-2-yl-1-[3-(tetrazol-1-yl)propanoyl]-1,4-diazepan-5-one
—— (3S)-4-[(4-fluorophenyl)methyl]-1-[(4-methylthiadiazol-5-yl)methyl]-3-propan-2-yl-1,4-diazepan-5-one —— C19H25FN4OS
(3S)-4-[(4-fluorophenyl)methyl]-1-[(4-methylthiadiazol-5-yl)methyl]-3-propan-2-yl-1,4-diazepan-5-one
—— (3R)-1-(cyclopropanecarbonyl)-4-[(4-fluorophenyl)methyl]-3-propan-2-yl-1,4-diazepan-5-one —— C19H25FN2O2
(3R)-1-(cyclopropanecarbonyl)-4-[(4-fluorophenyl)methyl]-3-propan-2-yl-1,4-diazepan-5-one
—— (3R)-4-[(4-fluorophenyl)methyl]-1-[(4-methylthiadiazol-5-yl)methyl]-3-propan-2-yl-1,4-diazepan-5-one —— C19H25FN4OS
(3R)-4-[(4-fluorophenyl)methyl]-1-[(4-methylthiadiazol-5-yl)methyl]-3-propan-2-yl-1,4-diazepan-5-one
—— (3S)-4-[(4-fluorophenyl)methyl]-1-(3-methoxypropyl)-3-propan-2-yl-1,4-diazepan-5-one —— C19H29FN2O2
(3S)-4-[(4-fluorophenyl)methyl]-1-(3-methoxypropyl)-3-propan-2-yl-1,4-diazepan-5-one
—— (3R)-4-[(4-fluorophenyl)methyl]-1-(3-methoxypropyl)-3-propan-2-yl-1,4-diazepan-5-one —— C19H29FN2O2
(3R)-4-[(4-fluorophenyl)methyl]-1-(3-methoxypropyl)-3-propan-2-yl-1,4-diazepan-5-one
—— (3S)-4-benzyl-3-ethyl-1-[3-(1,2,4-triazol-4-yl)propanoyl]-1,4-diazepan-5-one —— C19H25N5O2
(3S)-4-benzyl-3-ethyl-1-[3-(1,2,4-triazol-4-yl)propanoyl]-1,4-diazepan-5-one
—— (3S)-4-[(4-fluorophenyl)methyl]-1-[(1-methylimidazol-2-yl)methyl]-3-propan-2-yl-1,4-diazepan-5-one —— C20H27FN4O
(3S)-4-[(4-fluorophenyl)methyl]-1-[(1-methylimidazol-2-yl)methyl]-3-propan-2-yl-1,4-diazepan-5-one