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二氮杂卓

中文名称 英文名称 CAS号 化学式 结构式图片
—— [(3R)-oxolan-3-yl]-[4-[(1-propan-2-ylpyrazol-4-yl)methyl]-1,4-diazepan-1-yl]methanone —— C17H28N4O2
[(3R)-oxolan-3-yl]-[4-[(1-propan-2-ylpyrazol-4-yl)methyl]-1,4-diazepan-1-yl]methanone
—— (2S)-1-[4-[(2-methyl-1,3-thiazol-4-yl)methyl]-1,4-diazepan-1-yl]-2-pyrazol-1-ylpropan-1-one —— C16H23N5OS
(2S)-1-[4-[(2-methyl-1,3-thiazol-4-yl)methyl]-1,4-diazepan-1-yl]-2-pyrazol-1-ylpropan-1-one
—— [(3S)-oxolan-3-yl]-[4-[(1-propan-2-ylpyrazol-4-yl)methyl]-1,4-diazepan-1-yl]methanone —— C17H28N4O2
[(3S)-oxolan-3-yl]-[4-[(1-propan-2-ylpyrazol-4-yl)methyl]-1,4-diazepan-1-yl]methanone
—— (2R)-1-[4-[(2-methyl-1,3-thiazol-4-yl)methyl]-1,4-diazepan-1-yl]-2-pyrazol-1-ylpropan-1-one —— C16H23N5OS
(2R)-1-[4-[(2-methyl-1,3-thiazol-4-yl)methyl]-1,4-diazepan-1-yl]-2-pyrazol-1-ylpropan-1-one
—— (2S)-2-(cyclopropylmethoxy)-1-[4-(1,3-thiazol-4-ylmethyl)-1,4-diazepan-1-yl]propan-1-one —— C16H25N3O2S
(2S)-2-(cyclopropylmethoxy)-1-[4-(1,3-thiazol-4-ylmethyl)-1,4-diazepan-1-yl]propan-1-one
—— (2R)-2-(cyclopropylmethoxy)-1-[4-(1,3-thiazol-4-ylmethyl)-1,4-diazepan-1-yl]propan-1-one —— C16H25N3O2S
(2R)-2-(cyclopropylmethoxy)-1-[4-(1,3-thiazol-4-ylmethyl)-1,4-diazepan-1-yl]propan-1-one
—— [(1R,2S)-2-pyridin-3-ylcyclopropyl]-[4-(1,3-thiazol-4-ylmethyl)-1,4-diazepan-1-yl]methanone —— C18H22N4OS
[(1R,2S)-2-pyridin-3-ylcyclopropyl]-[4-(1,3-thiazol-4-ylmethyl)-1,4-diazepan-1-yl]methanone
—— [(1R,2R)-2-pyridin-3-ylcyclopropyl]-[4-(1,3-thiazol-4-ylmethyl)-1,4-diazepan-1-yl]methanone —— C18H22N4OS
[(1R,2R)-2-pyridin-3-ylcyclopropyl]-[4-(1,3-thiazol-4-ylmethyl)-1,4-diazepan-1-yl]methanone
—— [(1S,2R)-2-pyridin-3-ylcyclopropyl]-[4-(1,3-thiazol-4-ylmethyl)-1,4-diazepan-1-yl]methanone —— C18H22N4OS
[(1S,2R)-2-pyridin-3-ylcyclopropyl]-[4-(1,3-thiazol-4-ylmethyl)-1,4-diazepan-1-yl]methanone
—— [(1S,2S)-2-pyridin-3-ylcyclopropyl]-[4-(1,3-thiazol-4-ylmethyl)-1,4-diazepan-1-yl]methanone —— C18H22N4OS
[(1S,2S)-2-pyridin-3-ylcyclopropyl]-[4-(1,3-thiazol-4-ylmethyl)-1,4-diazepan-1-yl]methanone
—— (2S)-1-[4-(1,3-thiazol-4-ylmethyl)-1,4-diazepan-1-yl]-2-(1,2,4-triazol-1-yl)propan-1-one —— C14H20N6OS
(2S)-1-[4-(1,3-thiazol-4-ylmethyl)-1,4-diazepan-1-yl]-2-(1,2,4-triazol-1-yl)propan-1-one
—— (2R)-1-[4-(1,3-thiazol-4-ylmethyl)-1,4-diazepan-1-yl]-2-(1,2,4-triazol-1-yl)propan-1-one —— C14H20N6OS
(2R)-1-[4-(1,3-thiazol-4-ylmethyl)-1,4-diazepan-1-yl]-2-(1,2,4-triazol-1-yl)propan-1-one
—— (2R)-2-(2,5-dimethylfuran-3-yl)-1-[4-[(1-methylpyrazol-4-yl)methyl]-1,4-diazepan-1-yl]propan-1-one —— C19H28N4O2
(2R)-2-(2,5-dimethylfuran-3-yl)-1-[4-[(1-methylpyrazol-4-yl)methyl]-1,4-diazepan-1-yl]propan-1-one
—— (2S)-2-(2,5-dimethylfuran-3-yl)-1-[4-[(1-methylpyrazol-4-yl)methyl]-1,4-diazepan-1-yl]propan-1-one —— C19H28N4O2
(2S)-2-(2,5-dimethylfuran-3-yl)-1-[4-[(1-methylpyrazol-4-yl)methyl]-1,4-diazepan-1-yl]propan-1-one
—— [(2R)-oxolan-2-yl]-[4-(1,3-thiazol-4-ylmethyl)-1,4-diazepan-1-yl]methanone —— C14H21N3O2S
[(2R)-oxolan-2-yl]-[4-(1,3-thiazol-4-ylmethyl)-1,4-diazepan-1-yl]methanone
—— [4-[(1-ethylimidazol-2-yl)methyl]-1,4-diazepan-1-yl]-[(2S)-oxolan-2-yl]methanone —— C16H26N4O2
[4-[(1-ethylimidazol-2-yl)methyl]-1,4-diazepan-1-yl]-[(2S)-oxolan-2-yl]methanone
—— [(2S)-oxolan-2-yl]-[4-(1,3-thiazol-4-ylmethyl)-1,4-diazepan-1-yl]methanone —— C14H21N3O2S
[(2S)-oxolan-2-yl]-[4-(1,3-thiazol-4-ylmethyl)-1,4-diazepan-1-yl]methanone
—— 2-[(1S)-cyclopent-2-en-1-yl]-1-[4-[(1-ethylimidazol-2-yl)methyl]-1,4-diazepan-1-yl]ethanone —— C18H28N4O
2-[(1S)-cyclopent-2-en-1-yl]-1-[4-[(1-ethylimidazol-2-yl)methyl]-1,4-diazepan-1-yl]ethanone
—— [4-[(2-methyl-1,3-thiazol-4-yl)methyl]-1,4-diazepan-1-yl]-[(3S)-oxolan-3-yl]methanone —— C15H23N3O2S
[4-[(2-methyl-1,3-thiazol-4-yl)methyl]-1,4-diazepan-1-yl]-[(3S)-oxolan-3-yl]methanone
—— [4-[(1-ethylimidazol-2-yl)methyl]-1,4-diazepan-1-yl]-[(1R,2S)-2-(furan-2-yl)cyclopropyl]methanone —— C19H26N4O2
[4-[(1-ethylimidazol-2-yl)methyl]-1,4-diazepan-1-yl]-[(1R,2S)-2-(furan-2-yl)cyclopropyl]methanone
—— 2-[(1R)-cyclopent-2-en-1-yl]-1-[4-[(1-ethylimidazol-2-yl)methyl]-1,4-diazepan-1-yl]ethanone —— C18H28N4O
2-[(1R)-cyclopent-2-en-1-yl]-1-[4-[(1-ethylimidazol-2-yl)methyl]-1,4-diazepan-1-yl]ethanone
—— [4-[(2-methyl-1,3-thiazol-4-yl)methyl]-1,4-diazepan-1-yl]-[(3R)-oxolan-3-yl]methanone —— C15H23N3O2S
[4-[(2-methyl-1,3-thiazol-4-yl)methyl]-1,4-diazepan-1-yl]-[(3R)-oxolan-3-yl]methanone
—— [(1S,2S)-2-(furan-2-yl)cyclopropyl]-[4-[(1-methylpyrazol-4-yl)methyl]-1,4-diazepan-1-yl]methanone —— C18H24N4O2
[(1S,2S)-2-(furan-2-yl)cyclopropyl]-[4-[(1-methylpyrazol-4-yl)methyl]-1,4-diazepan-1-yl]methanone
—— 1-[(3S,5R)-3,5-dimethylpiperidin-1-yl]sulfonyl-4-ethyl-1,4-diazepane —— C14H29N3O2S
1-[(3S,5R)-3,5-dimethylpiperidin-1-yl]sulfonyl-4-ethyl-1,4-diazepane
—— [(1R)-cyclohex-3-en-1-yl]-[4-(1,3-thiazol-4-ylmethyl)-1,4-diazepan-1-yl]methanone —— C16H23N3OS
[(1R)-cyclohex-3-en-1-yl]-[4-(1,3-thiazol-4-ylmethyl)-1,4-diazepan-1-yl]methanone
—— [(1S)-cyclohex-3-en-1-yl]-[4-(1,3-thiazol-4-ylmethyl)-1,4-diazepan-1-yl]methanone —— C16H23N3OS
[(1S)-cyclohex-3-en-1-yl]-[4-(1,3-thiazol-4-ylmethyl)-1,4-diazepan-1-yl]methanone
—— 2-[(1S)-cyclopent-2-en-1-yl]-1-[4-[(1-methylpyrazol-4-yl)methyl]-1,4-diazepan-1-yl]ethanone —— C17H26N4O
2-[(1S)-cyclopent-2-en-1-yl]-1-[4-[(1-methylpyrazol-4-yl)methyl]-1,4-diazepan-1-yl]ethanone
—— 2-[(1R)-cyclopent-2-en-1-yl]-1-[4-[(1-methylpyrazol-4-yl)methyl]-1,4-diazepan-1-yl]ethanone —— C17H26N4O
2-[(1R)-cyclopent-2-en-1-yl]-1-[4-[(1-methylpyrazol-4-yl)methyl]-1,4-diazepan-1-yl]ethanone
—— [4-[(1-methylpyrazol-4-yl)methyl]-1,4-diazepan-1-yl]-[(3R)-oxolan-3-yl]methanone —— C15H24N4O2
[4-[(1-methylpyrazol-4-yl)methyl]-1,4-diazepan-1-yl]-[(3R)-oxolan-3-yl]methanone
—— [4-[(1-methylpyrazol-4-yl)methyl]-1,4-diazepan-1-yl]-[(3S)-oxolan-3-yl]methanone —— C15H24N4O2
[4-[(1-methylpyrazol-4-yl)methyl]-1,4-diazepan-1-yl]-[(3S)-oxolan-3-yl]methanone
—— (3R)-1-[4-[(1-ethylimidazol-2-yl)methyl]-1,4-diazepan-1-yl]-3-pyrrol-1-ylbutan-1-one —— C19H29N5O
(3R)-1-[4-[(1-ethylimidazol-2-yl)methyl]-1,4-diazepan-1-yl]-3-pyrrol-1-ylbutan-1-one
—— (3S)-1-[4-[(1-ethylimidazol-2-yl)methyl]-1,4-diazepan-1-yl]-3-pyrrol-1-ylbutan-1-one —— C19H29N5O
(3S)-1-[4-[(1-ethylimidazol-2-yl)methyl]-1,4-diazepan-1-yl]-3-pyrrol-1-ylbutan-1-one
—— 3-[(2R)-oxolan-2-yl]-1-[4-[(1-propan-2-ylpyrazol-4-yl)methyl]-1,4-diazepan-1-yl]propan-1-one —— C19H32N4O2
3-[(2R)-oxolan-2-yl]-1-[4-[(1-propan-2-ylpyrazol-4-yl)methyl]-1,4-diazepan-1-yl]propan-1-one
—— (3S)-1-[4-[(1-methylpyrazol-4-yl)methyl]-1,4-diazepan-1-yl]-3-pyrrol-1-ylbutan-1-one —— C18H27N5O
(3S)-1-[4-[(1-methylpyrazol-4-yl)methyl]-1,4-diazepan-1-yl]-3-pyrrol-1-ylbutan-1-one
—— (2S)-1-[4-[(1-ethylpyrazol-4-yl)methyl]-1,4-diazepan-1-yl]-2-methyl-3-pyrazol-1-ylpropan-1-one —— C18H28N6O
(2S)-1-[4-[(1-ethylpyrazol-4-yl)methyl]-1,4-diazepan-1-yl]-2-methyl-3-pyrazol-1-ylpropan-1-one
—— (2R)-1-[4-[(1-ethylpyrazol-4-yl)methyl]-1,4-diazepan-1-yl]-2-methyl-3-pyrazol-1-ylpropan-1-one —— C18H28N6O
(2R)-1-[4-[(1-ethylpyrazol-4-yl)methyl]-1,4-diazepan-1-yl]-2-methyl-3-pyrazol-1-ylpropan-1-one
—— (3R)-1-[4-[(1-methylpyrazol-4-yl)methyl]-1,4-diazepan-1-yl]-3-pyrrol-1-ylbutan-1-one —— C18H27N5O
(3R)-1-[4-[(1-methylpyrazol-4-yl)methyl]-1,4-diazepan-1-yl]-3-pyrrol-1-ylbutan-1-one
—— (2R)-2-imidazol-1-yl-1-[4-[(1-methylpyrazol-4-yl)methyl]-1,4-diazepan-1-yl]propan-1-one —— C16H24N6O
(2R)-2-imidazol-1-yl-1-[4-[(1-methylpyrazol-4-yl)methyl]-1,4-diazepan-1-yl]propan-1-one
—— (2S)-2-imidazol-1-yl-1-[4-[(1-methylpyrazol-4-yl)methyl]-1,4-diazepan-1-yl]propan-1-one —— C16H24N6O
(2S)-2-imidazol-1-yl-1-[4-[(1-methylpyrazol-4-yl)methyl]-1,4-diazepan-1-yl]propan-1-one
—— [(3R)-oxolan-3-yl]-[4-(1,3-thiazol-4-ylmethyl)-1,4-diazepan-1-yl]methanone —— C14H21N3O2S
[(3R)-oxolan-3-yl]-[4-(1,3-thiazol-4-ylmethyl)-1,4-diazepan-1-yl]methanone
—— [(3S)-oxolan-3-yl]-[4-(1,3-thiazol-4-ylmethyl)-1,4-diazepan-1-yl]methanone —— C14H21N3O2S
[(3S)-oxolan-3-yl]-[4-(1,3-thiazol-4-ylmethyl)-1,4-diazepan-1-yl]methanone
—— 1-[4-[(1-ethylpyrazol-4-yl)methyl]-1,4-diazepan-1-yl]-3-[(2R)-oxolan-2-yl]propan-1-one —— C18H30N4O2
1-[4-[(1-ethylpyrazol-4-yl)methyl]-1,4-diazepan-1-yl]-3-[(2R)-oxolan-2-yl]propan-1-one
—— 1-[4-[(5-Tert-butyl-1,3-oxazol-2-yl)methyl]-1,4-diazepan-1-yl]-2-methylpropan-1-one —— C17H29N3O2
1-[4-[(5-Tert-butyl-1,3-oxazol-2-yl)methyl]-1,4-diazepan-1-yl]-2-methylpropan-1-one
—— 2-Methyl-1-(4-prop-2-enyl-1,4-diazepan-1-yl)propan-1-one —— C12H22N2O
2-Methyl-1-(4-prop-2-enyl-1,4-diazepan-1-yl)propan-1-one
—— 1-[4-[(2-Tert-butyl-1,3-thiazol-4-yl)methyl]-1,4-diazepan-1-yl]-2-methylpropan-1-one —— C17H29N3OS
1-[4-[(2-Tert-butyl-1,3-thiazol-4-yl)methyl]-1,4-diazepan-1-yl]-2-methylpropan-1-one
—— (2S)-1-[4-[(1-propan-2-ylpyrazol-4-yl)methyl]-1,4-diazepan-1-yl]-2-(1,2,4-triazol-1-yl)propan-1-one —— C17H27N7O
(2S)-1-[4-[(1-propan-2-ylpyrazol-4-yl)methyl]-1,4-diazepan-1-yl]-2-(1,2,4-triazol-1-yl)propan-1-one
—— 2-cyclopentyl-1-[4-[(1R)-1-(3-methyl-1,2,4-oxadiazol-5-yl)ethyl]-1,4-diazepan-1-yl]ethanone —— C17H28N4O2
2-cyclopentyl-1-[4-[(1R)-1-(3-methyl-1,2,4-oxadiazol-5-yl)ethyl]-1,4-diazepan-1-yl]ethanone
—— 2-cyclopentyl-1-[4-[(1S)-1-(3-methyl-1,2,4-oxadiazol-5-yl)ethyl]-1,4-diazepan-1-yl]ethanone —— C17H28N4O2
2-cyclopentyl-1-[4-[(1S)-1-(3-methyl-1,2,4-oxadiazol-5-yl)ethyl]-1,4-diazepan-1-yl]ethanone
—— 1-[4-[(1R,2R)-2-(5-methylthiophen-2-yl)cyclopropanecarbonyl]-1,4-diazepan-1-yl]propan-1-one —— C17H24N2O2S
1-[4-[(1R,2R)-2-(5-methylthiophen-2-yl)cyclopropanecarbonyl]-1,4-diazepan-1-yl]propan-1-one
—— 1-[4-[(1R,2S)-2-(5-methylthiophen-2-yl)cyclopropanecarbonyl]-1,4-diazepan-1-yl]propan-1-one —— C17H24N2O2S
1-[4-[(1R,2S)-2-(5-methylthiophen-2-yl)cyclopropanecarbonyl]-1,4-diazepan-1-yl]propan-1-one