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二氮杂卓

中文名称 英文名称 CAS号 化学式 结构式图片
—— (3S)-4-(cyclopropylmethyl)-3-propan-2-yl-1-[1-(pyrazol-1-ylmethyl)cyclopropanecarbonyl]-1,4-diazepan-5-one —— C20H30N4O2
(3S)-4-(cyclopropylmethyl)-3-propan-2-yl-1-[1-(pyrazol-1-ylmethyl)cyclopropanecarbonyl]-1,4-diazepan-5-one
—— (3R)-4-(cyclopropylmethyl)-3-propan-2-yl-1-[1-(pyrazol-1-ylmethyl)cyclopropanecarbonyl]-1,4-diazepan-5-one —— C20H30N4O2
(3R)-4-(cyclopropylmethyl)-3-propan-2-yl-1-[1-(pyrazol-1-ylmethyl)cyclopropanecarbonyl]-1,4-diazepan-5-one
—— (3R)-4-[(4-fluorophenyl)methyl]-3-propan-2-yl-1-[(3-propan-2-ylimidazol-4-yl)methyl]-1,4-diazepan-5-one —— C22H31FN4O
(3R)-4-[(4-fluorophenyl)methyl]-3-propan-2-yl-1-[(3-propan-2-ylimidazol-4-yl)methyl]-1,4-diazepan-5-one
—— (3S)-4-[(4-fluorophenyl)methyl]-3-propan-2-yl-1-[(3-propan-2-ylimidazol-4-yl)methyl]-1,4-diazepan-5-one —— C22H31FN4O
(3S)-4-[(4-fluorophenyl)methyl]-3-propan-2-yl-1-[(3-propan-2-ylimidazol-4-yl)methyl]-1,4-diazepan-5-one
—— 1-[[(3S)-oxolan-3-yl]methyl]-4-(pyridin-3-ylmethyl)-1,4-diazepane —— C16H25N3O
1-[[(3S)-oxolan-3-yl]methyl]-4-(pyridin-3-ylmethyl)-1,4-diazepane
—— (3R)-4-[(4-fluorophenyl)methyl]-3-propan-2-yl-1-(2-propoxyacetyl)-1,4-diazepan-5-one —— C20H29FN2O3
(3R)-4-[(4-fluorophenyl)methyl]-3-propan-2-yl-1-(2-propoxyacetyl)-1,4-diazepan-5-one
—— 1-[3-[(3S)-4-(cyclopropylmethyl)-3-propan-2-yl-1,4-diazepan-1-yl]-3-oxopropyl]-6-methylpyridin-2-one —— C21H33N3O2
1-[3-[(3S)-4-(cyclopropylmethyl)-3-propan-2-yl-1,4-diazepan-1-yl]-3-oxopropyl]-6-methylpyridin-2-one
—— (3S)-4-[(4-fluorophenyl)methyl]-3-propan-2-yl-1-(2-propoxyacetyl)-1,4-diazepan-5-one —— C20H29FN2O3
(3S)-4-[(4-fluorophenyl)methyl]-3-propan-2-yl-1-(2-propoxyacetyl)-1,4-diazepan-5-one
—— 1-(2-Pyridin-4-ylethyl)-1,4-diazepane-1,4-diium —— C12H21N3+2
1-(2-Pyridin-4-ylethyl)-1,4-diazepane-1,4-diium
—— 1-(2-Pyridin-2-ylethyl)-1,4-diazepane-1,4-diium —— C12H21N3+2
1-(2-Pyridin-2-ylethyl)-1,4-diazepane-1,4-diium
—— N-benzyl-4-[(2R)-oxolane-2-carbonyl]-1,4-diazepane-1-sulfonamide —— C17H25N3O4S
N-benzyl-4-[(2R)-oxolane-2-carbonyl]-1,4-diazepane-1-sulfonamide
—— N-benzyl-4-[(2S)-oxolane-2-carbonyl]-1,4-diazepane-1-sulfonamide —— C17H25N3O4S
N-benzyl-4-[(2S)-oxolane-2-carbonyl]-1,4-diazepane-1-sulfonamide
—— 1-[(3R)-3-(5-methylfuran-2-yl)butyl]-4-(pyridin-3-ylmethyl)-1,4-diazepane —— C20H29N3O
1-[(3R)-3-(5-methylfuran-2-yl)butyl]-4-(pyridin-3-ylmethyl)-1,4-diazepane
—— (3S)-4-(cyclopropylmethyl)-3-propan-2-yl-1-(2-pyridin-3-ylacetyl)-1,4-diazepan-5-one —— C19H27N3O2
(3S)-4-(cyclopropylmethyl)-3-propan-2-yl-1-(2-pyridin-3-ylacetyl)-1,4-diazepan-5-one
—— 2-[2-[(3S)-4-[(4-fluorophenyl)methyl]-5-oxo-3-propan-2-yl-1,4-diazepan-1-yl]-2-oxoethoxy]acetamide —— C19H26FN3O4
2-[2-[(3S)-4-[(4-fluorophenyl)methyl]-5-oxo-3-propan-2-yl-1,4-diazepan-1-yl]-2-oxoethoxy]acetamide
—— 2-[2-[(3R)-4-[(4-fluorophenyl)methyl]-5-oxo-3-propan-2-yl-1,4-diazepan-1-yl]-2-oxoethoxy]acetamide —— C19H26FN3O4
2-[2-[(3R)-4-[(4-fluorophenyl)methyl]-5-oxo-3-propan-2-yl-1,4-diazepan-1-yl]-2-oxoethoxy]acetamide
—— 1-[(3S)-3-(5-methylfuran-2-yl)butyl]-4-(pyridin-3-ylmethyl)-1,4-diazepane —— C20H29N3O
1-[(3S)-3-(5-methylfuran-2-yl)butyl]-4-(pyridin-3-ylmethyl)-1,4-diazepane
—— methyl 3-[(3R)-4-[(4-fluorophenyl)methyl]-5-oxo-3-propan-2-yl-1,4-diazepan-1-yl]propanoate —— C19H27FN2O3
methyl 3-[(3R)-4-[(4-fluorophenyl)methyl]-5-oxo-3-propan-2-yl-1,4-diazepan-1-yl]propanoate
—— (3R)-4-(cyclopropylmethyl)-3-propan-2-yl-1-[3-(3,4,5-trimethylpyrazol-1-yl)propanoyl]-1,4-diazepan-5-one —— C21H34N4O2
(3R)-4-(cyclopropylmethyl)-3-propan-2-yl-1-[3-(3,4,5-trimethylpyrazol-1-yl)propanoyl]-1,4-diazepan-5-one
—— (3S)-4-(cyclopropylmethyl)-3-propan-2-yl-1-[3-(3,4,5-trimethylpyrazol-1-yl)propanoyl]-1,4-diazepan-5-one —— C21H34N4O2
(3S)-4-(cyclopropylmethyl)-3-propan-2-yl-1-[3-(3,4,5-trimethylpyrazol-1-yl)propanoyl]-1,4-diazepan-5-one
—— (3S)-4-benzyl-3-ethyl-1-[4-(2-methylimidazol-1-yl)butanoyl]-1,4-diazepan-5-one —— C22H30N4O2
(3S)-4-benzyl-3-ethyl-1-[4-(2-methylimidazol-1-yl)butanoyl]-1,4-diazepan-5-one
—— (3R)-4-benzyl-3-ethyl-1-[4-(2-methylimidazol-1-yl)butanoyl]-1,4-diazepan-5-one —— C22H30N4O2
(3R)-4-benzyl-3-ethyl-1-[4-(2-methylimidazol-1-yl)butanoyl]-1,4-diazepan-5-one
—— [(3S)-4-(cyclopropylmethyl)-3-propan-2-yl-1,4-diazepan-1-yl]-[1-(pyrazol-1-ylmethyl)cyclopropyl]methanone —— C20H32N4O
[(3S)-4-(cyclopropylmethyl)-3-propan-2-yl-1,4-diazepan-1-yl]-[1-(pyrazol-1-ylmethyl)cyclopropyl]methanone
—— [(3R)-4-(cyclopropylmethyl)-3-propan-2-yl-1,4-diazepan-1-yl]-[1-(pyrazol-1-ylmethyl)cyclopropyl]methanone —— C20H32N4O
[(3R)-4-(cyclopropylmethyl)-3-propan-2-yl-1,4-diazepan-1-yl]-[1-(pyrazol-1-ylmethyl)cyclopropyl]methanone
—— (3R)-4-(cyclopropylmethyl)-3-propan-2-yl-1-[2-(1,2,4-triazol-1-yl)acetyl]-1,4-diazepan-5-one —— C16H25N5O2
(3R)-4-(cyclopropylmethyl)-3-propan-2-yl-1-[2-(1,2,4-triazol-1-yl)acetyl]-1,4-diazepan-5-one
—— (3S)-4-(cyclopropylmethyl)-3-propan-2-yl-1-[2-(1,2,4-triazol-1-yl)acetyl]-1,4-diazepan-5-one —— C16H25N5O2
(3S)-4-(cyclopropylmethyl)-3-propan-2-yl-1-[2-(1,2,4-triazol-1-yl)acetyl]-1,4-diazepan-5-one
—— (3S)-1-[2-(4-chloropyrazol-1-yl)acetyl]-4-(cyclopropylmethyl)-3-propan-2-yl-1,4-diazepan-5-one —— C17H25ClN4O2
(3S)-1-[2-(4-chloropyrazol-1-yl)acetyl]-4-(cyclopropylmethyl)-3-propan-2-yl-1,4-diazepan-5-one
—— (3R)-1-[2-(4-chloropyrazol-1-yl)acetyl]-4-(cyclopropylmethyl)-3-propan-2-yl-1,4-diazepan-5-one —— C17H25ClN4O2
(3R)-1-[2-(4-chloropyrazol-1-yl)acetyl]-4-(cyclopropylmethyl)-3-propan-2-yl-1,4-diazepan-5-one
—— (3S)-4-benzyl-3-ethyl-1-[(1-propylimidazol-2-yl)methyl]-1,4-diazepan-5-one —— C21H30N4O
(3S)-4-benzyl-3-ethyl-1-[(1-propylimidazol-2-yl)methyl]-1,4-diazepan-5-one
—— (3R)-4-benzyl-3-ethyl-1-[(1-propylimidazol-2-yl)methyl]-1,4-diazepan-5-one —— C21H30N4O
(3R)-4-benzyl-3-ethyl-1-[(1-propylimidazol-2-yl)methyl]-1,4-diazepan-5-one
—— (3R)-4-(cyclopropylmethyl)-1-[2-(2-oxopyrimidin-1-yl)acetyl]-3-propan-2-yl-1,4-diazepan-5-one —— C18H26N4O3
(3R)-4-(cyclopropylmethyl)-1-[2-(2-oxopyrimidin-1-yl)acetyl]-3-propan-2-yl-1,4-diazepan-5-one
—— (3S)-4-(cyclopropylmethyl)-1-[2-(2-oxopyrimidin-1-yl)acetyl]-3-propan-2-yl-1,4-diazepan-5-one —— C18H26N4O3
(3S)-4-(cyclopropylmethyl)-1-[2-(2-oxopyrimidin-1-yl)acetyl]-3-propan-2-yl-1,4-diazepan-5-one
—— (3S)-4-(cyclopropylmethyl)-3-propan-2-yl-1-[4-(1,2,4-triazol-1-yl)butanoyl]-1,4-diazepan-5-one —— C18H29N5O2
(3S)-4-(cyclopropylmethyl)-3-propan-2-yl-1-[4-(1,2,4-triazol-1-yl)butanoyl]-1,4-diazepan-5-one
—— (3S)-4-[(4-fluorophenyl)methyl]-1-[2-(4-methylpyrazol-1-yl)acetyl]-3-propan-2-yl-1,4-diazepan-5-one —— C21H27FN4O2
(3S)-4-[(4-fluorophenyl)methyl]-1-[2-(4-methylpyrazol-1-yl)acetyl]-3-propan-2-yl-1,4-diazepan-5-one
—— (3R)-4-[(4-fluorophenyl)methyl]-1-[2-(4-methylpyrazol-1-yl)acetyl]-3-propan-2-yl-1,4-diazepan-5-one —— C21H27FN4O2
(3R)-4-[(4-fluorophenyl)methyl]-1-[2-(4-methylpyrazol-1-yl)acetyl]-3-propan-2-yl-1,4-diazepan-5-one
—— (3R)-4-[(4-fluorophenyl)methyl]-3-propan-2-yl-1-[3-(1,2,4-triazol-4-yl)propanoyl]-1,4-diazepan-5-one —— C20H26FN5O2
(3R)-4-[(4-fluorophenyl)methyl]-3-propan-2-yl-1-[3-(1,2,4-triazol-4-yl)propanoyl]-1,4-diazepan-5-one
—— (3S)-4-[(4-fluorophenyl)methyl]-3-propan-2-yl-1-[3-(1,2,4-triazol-4-yl)propanoyl]-1,4-diazepan-5-one —— C20H26FN5O2
(3S)-4-[(4-fluorophenyl)methyl]-3-propan-2-yl-1-[3-(1,2,4-triazol-4-yl)propanoyl]-1,4-diazepan-5-one
—— (3S)-4-[(4-fluorophenyl)methyl]-1-[2-(2-hydroxyethoxy)ethyl]-3-propan-2-yl-1,4-diazepan-5-one —— C19H29FN2O3
(3S)-4-[(4-fluorophenyl)methyl]-1-[2-(2-hydroxyethoxy)ethyl]-3-propan-2-yl-1,4-diazepan-5-one
—— (3R)-4-[(4-fluorophenyl)methyl]-1-[2-(2-hydroxyethoxy)ethyl]-3-propan-2-yl-1,4-diazepan-5-one —— C19H29FN2O3
(3R)-4-[(4-fluorophenyl)methyl]-1-[2-(2-hydroxyethoxy)ethyl]-3-propan-2-yl-1,4-diazepan-5-one
—— (3S)-1-(3-ethoxypropanoyl)-4-[(4-fluorophenyl)methyl]-3-propan-2-yl-1,4-diazepan-5-one —— C20H29FN2O3
(3S)-1-(3-ethoxypropanoyl)-4-[(4-fluorophenyl)methyl]-3-propan-2-yl-1,4-diazepan-5-one
—— (3R)-1-(3-ethoxypropanoyl)-4-[(4-fluorophenyl)methyl]-3-propan-2-yl-1,4-diazepan-5-one —— C20H29FN2O3
(3R)-1-(3-ethoxypropanoyl)-4-[(4-fluorophenyl)methyl]-3-propan-2-yl-1,4-diazepan-5-one
—— (3S)-4-benzyl-3-ethyl-1-(2-imidazol-1-ylacetyl)-1,4-diazepan-5-one —— C19H24N4O2
(3S)-4-benzyl-3-ethyl-1-(2-imidazol-1-ylacetyl)-1,4-diazepan-5-one
—— (3R)-4-benzyl-3-ethyl-1-(2-imidazol-1-ylacetyl)-1,4-diazepan-5-one —— C19H24N4O2
(3R)-4-benzyl-3-ethyl-1-(2-imidazol-1-ylacetyl)-1,4-diazepan-5-one
—— (3R)-4-(cyclopropylmethyl)-1-[4-(2-methylimidazol-1-yl)butanoyl]-3-propan-2-yl-1,4-diazepan-5-one —— C20H32N4O2
(3R)-4-(cyclopropylmethyl)-1-[4-(2-methylimidazol-1-yl)butanoyl]-3-propan-2-yl-1,4-diazepan-5-one
—— (3R)-4-[(4-fluorophenyl)methyl]-3-propan-2-yl-1-(2-propan-2-ylsulfanylacetyl)-1,4-diazepan-5-one —— C20H29FN2O2S
(3R)-4-[(4-fluorophenyl)methyl]-3-propan-2-yl-1-(2-propan-2-ylsulfanylacetyl)-1,4-diazepan-5-one
—— (3S)-4-[(4-fluorophenyl)methyl]-3-propan-2-yl-1-(2-propan-2-ylsulfanylacetyl)-1,4-diazepan-5-one —— C20H29FN2O2S
(3S)-4-[(4-fluorophenyl)methyl]-3-propan-2-yl-1-(2-propan-2-ylsulfanylacetyl)-1,4-diazepan-5-one
—— (3S)-4-[(4-fluorophenyl)methyl]-1-(3-imidazol-1-ylpropanoyl)-3-propan-2-yl-1,4-diazepan-5-one —— C21H27FN4O2
(3S)-4-[(4-fluorophenyl)methyl]-1-(3-imidazol-1-ylpropanoyl)-3-propan-2-yl-1,4-diazepan-5-one
—— (3R)-1-(6-aminohexanoyl)-4-[(4-fluorophenyl)methyl]-3-propan-2-yl-1,4-diazepan-5-one —— C21H32FN3O2
(3R)-1-(6-aminohexanoyl)-4-[(4-fluorophenyl)methyl]-3-propan-2-yl-1,4-diazepan-5-one
—— (3R)-4-[(4-fluorophenyl)methyl]-1-(3-imidazol-1-ylpropanoyl)-3-propan-2-yl-1,4-diazepan-5-one —— C21H27FN4O2
(3R)-4-[(4-fluorophenyl)methyl]-1-(3-imidazol-1-ylpropanoyl)-3-propan-2-yl-1,4-diazepan-5-one
—— [(2R)-oxolan-2-yl]-[4-(5,6,7,8-tetrahydro-4H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl)-1,4-diazepan-1-yl]methanone —— C18H29N5O2
[(2R)-oxolan-2-yl]-[4-(5,6,7,8-tetrahydro-4H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl)-1,4-diazepan-1-yl]methanone