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二氮杂卓

中文名称 英文名称 CAS号 化学式 结构式图片
—— (2R)-1-[4-[(5-tert-butyl-1,3-oxazol-2-yl)methyl]-1,4-diazepan-1-yl]-2-(5-methylpyrazol-1-yl)propan-1-one —— C20H31N5O2
(2R)-1-[4-[(5-tert-butyl-1,3-oxazol-2-yl)methyl]-1,4-diazepan-1-yl]-2-(5-methylpyrazol-1-yl)propan-1-one
—— (2S)-1-[4-[(5-tert-butyl-1,3-oxazol-2-yl)methyl]-1,4-diazepan-1-yl]-2-(5-methylpyrazol-1-yl)propan-1-one —— C20H31N5O2
(2S)-1-[4-[(5-tert-butyl-1,3-oxazol-2-yl)methyl]-1,4-diazepan-1-yl]-2-(5-methylpyrazol-1-yl)propan-1-one
—— 5-Tert-butyl-2-[[4-(2-methoxyethylsulfonyl)-1,4-diazepan-1-yl]methyl]-1,3-oxazole —— C16H29N3O4S
5-Tert-butyl-2-[[4-(2-methoxyethylsulfonyl)-1,4-diazepan-1-yl]methyl]-1,3-oxazole
—— (2S)-1-[4-[(5-tert-butyl-1,3-oxazol-2-yl)methyl]-1,4-diazepan-1-yl]-3-(4-chloropyrazol-1-yl)-2-methylpropan-1-one —— C20H30ClN5O2
(2S)-1-[4-[(5-tert-butyl-1,3-oxazol-2-yl)methyl]-1,4-diazepan-1-yl]-3-(4-chloropyrazol-1-yl)-2-methylpropan-1-one
—— [4-[(5-Tert-butyl-1,3-oxazol-2-yl)methyl]-1,4-diazepan-1-yl]-cyclopropylmethanone —— C17H27N3O2
[4-[(5-Tert-butyl-1,3-oxazol-2-yl)methyl]-1,4-diazepan-1-yl]-cyclopropylmethanone
—— (2R)-1-[4-[(5-tert-butyl-1,3-oxazol-2-yl)methyl]-1,4-diazepan-1-yl]-2-[4-chloro-5-methyl-3-(trifluoromethyl)pyrazol-1-yl]propan-1-one —— C21H29ClF3N5O2
(2R)-1-[4-[(5-tert-butyl-1,3-oxazol-2-yl)methyl]-1,4-diazepan-1-yl]-2-[4-chloro-5-methyl-3-(trifluoromethyl)pyrazol-1-yl]propan-1-one
—— [4-(cyclopropylmethyl)-1,4-diazepan-1-yl]-[(1S,2R)-2-phenylcyclopropyl]methanone —— C19H26N2O
[4-(cyclopropylmethyl)-1,4-diazepan-1-yl]-[(1S,2R)-2-phenylcyclopropyl]methanone
—— 1-(Azepan-1-yl)-5-[4-[(5-tert-butyl-1,3-oxazol-2-yl)methyl]-1,4-diazepan-1-yl]pentane-1,5-dione —— C24H40N4O3
1-(Azepan-1-yl)-5-[4-[(5-tert-butyl-1,3-oxazol-2-yl)methyl]-1,4-diazepan-1-yl]pentane-1,5-dione
—— 5-Tert-butyl-2-[[4-(1,5-dimethylpyrazol-4-yl)sulfonyl-1,4-diazepan-1-yl]methyl]-1,3-oxazole —— C18H29N5O3S
5-Tert-butyl-2-[[4-(1,5-dimethylpyrazol-4-yl)sulfonyl-1,4-diazepan-1-yl]methyl]-1,3-oxazole
—— 1-[4-[(5-Tert-butyl-1,3-oxazol-2-yl)methyl]-1,4-diazepan-1-yl]-3-(2-fluorophenyl)propan-1-one —— C22H30FN3O2
1-[4-[(5-Tert-butyl-1,3-oxazol-2-yl)methyl]-1,4-diazepan-1-yl]-3-(2-fluorophenyl)propan-1-one
—— 2-(4-Bromo-3,5-dimethylpyrazol-1-yl)-1-[4-[(5-tert-butyl-1,3-oxazol-2-yl)methyl]-1,4-diazepan-1-yl]ethanone —— C20H30BrN5O2
2-(4-Bromo-3,5-dimethylpyrazol-1-yl)-1-[4-[(5-tert-butyl-1,3-oxazol-2-yl)methyl]-1,4-diazepan-1-yl]ethanone
—— [4-(cyclopropylmethyl)-1,4-diazepan-1-yl]-[(2S)-oxolan-2-yl]methanone —— C14H24N2O2
[4-(cyclopropylmethyl)-1,4-diazepan-1-yl]-[(2S)-oxolan-2-yl]methanone
—— 1-[4-[(5-Tert-butyl-1,3-oxazol-2-yl)methyl]-1,4-diazepan-1-yl]-3-(4-fluorophenyl)propan-1-one —— C22H30FN3O2
1-[4-[(5-Tert-butyl-1,3-oxazol-2-yl)methyl]-1,4-diazepan-1-yl]-3-(4-fluorophenyl)propan-1-one
—— 1-[4-[(5-Tert-butyl-1,3-oxazol-2-yl)methyl]-1,4-diazepan-1-yl]-3-(1-ethyl-3-methylpyrazol-4-yl)propan-1-one —— C22H35N5O2
1-[4-[(5-Tert-butyl-1,3-oxazol-2-yl)methyl]-1,4-diazepan-1-yl]-3-(1-ethyl-3-methylpyrazol-4-yl)propan-1-one
—— (2R)-1-[4-[(5-tert-butyl-1,3-oxazol-2-yl)methyl]-1,4-diazepan-1-yl]-2-[3-(trifluoromethyl)pyrazol-1-yl]propan-1-one —— C20H28F3N5O2
(2R)-1-[4-[(5-tert-butyl-1,3-oxazol-2-yl)methyl]-1,4-diazepan-1-yl]-2-[3-(trifluoromethyl)pyrazol-1-yl]propan-1-one
—— Cyclohexyl-[4-(cyclopropylmethyl)-1,4-diazepan-1-yl]methanone —— C16H28N2O
Cyclohexyl-[4-(cyclopropylmethyl)-1,4-diazepan-1-yl]methanone
—— (2S)-1-[4-(cyclopropylmethyl)-1,4-diazepan-1-yl]-2-ethylhexan-1-one —— C17H32N2O
(2S)-1-[4-(cyclopropylmethyl)-1,4-diazepan-1-yl]-2-ethylhexan-1-one
—— (2R)-1-[4-[(5-tert-butyl-1,3-oxazol-2-yl)methyl]-1,4-diazepan-1-yl]-3-(4-chloropyrazol-1-yl)-2-methylpropan-1-one —— C20H30ClN5O2
(2R)-1-[4-[(5-tert-butyl-1,3-oxazol-2-yl)methyl]-1,4-diazepan-1-yl]-3-(4-chloropyrazol-1-yl)-2-methylpropan-1-one
—— 1-[4-(Cyclopropylmethyl)-1,4-diazepan-1-yl]-4-phenylbutan-1-one —— C19H28N2O
1-[4-(Cyclopropylmethyl)-1,4-diazepan-1-yl]-4-phenylbutan-1-one
—— [4-(cyclopropylmethyl)-1,4-diazepan-1-yl]-[(1S,2S)-2-phenylcyclopropyl]methanone —— C19H26N2O
[4-(cyclopropylmethyl)-1,4-diazepan-1-yl]-[(1S,2S)-2-phenylcyclopropyl]methanone
—— 1-[4-[(5-Tert-butyl-1,3-oxazol-2-yl)methyl]-1,4-diazepan-1-yl]-3-(1,5-dimethylpyrazol-4-yl)propan-1-one —— C21H33N5O2
1-[4-[(5-Tert-butyl-1,3-oxazol-2-yl)methyl]-1,4-diazepan-1-yl]-3-(1,5-dimethylpyrazol-4-yl)propan-1-one
—— [4-(cyclopropylmethyl)-1,4-diazepan-1-yl]-[(1R,2R)-2-methylcyclopropyl]methanone —— C14H24N2O
[4-(cyclopropylmethyl)-1,4-diazepan-1-yl]-[(1R,2R)-2-methylcyclopropyl]methanone
—— 3-(4-Bromopyrazol-1-yl)-1-[4-[(5-tert-butyl-1,3-oxazol-2-yl)methyl]-1,4-diazepan-1-yl]propan-1-one —— C19H28BrN5O2
3-(4-Bromopyrazol-1-yl)-1-[4-[(5-tert-butyl-1,3-oxazol-2-yl)methyl]-1,4-diazepan-1-yl]propan-1-one
—— Cyclopropyl-[4-(cyclopropylmethyl)-1,4-diazepan-1-yl]methanone —— C13H22N2O
Cyclopropyl-[4-(cyclopropylmethyl)-1,4-diazepan-1-yl]methanone
—— (2R)-2-[4-bromo-5-methyl-3-(trifluoromethyl)pyrazol-1-yl]-1-[4-[(5-tert-butyl-1,3-oxazol-2-yl)methyl]-1,4-diazepan-1-yl]propan-1-one —— C21H29BrF3N5O2
(2R)-2-[4-bromo-5-methyl-3-(trifluoromethyl)pyrazol-1-yl]-1-[4-[(5-tert-butyl-1,3-oxazol-2-yl)methyl]-1,4-diazepan-1-yl]propan-1-one
—— 1-[4-(Cyclopropylmethyl)-1,4-diazepan-1-yl]-3-methylbutan-1-one —— C14H26N2O
1-[4-(Cyclopropylmethyl)-1,4-diazepan-1-yl]-3-methylbutan-1-one
—— 3-Cyclopentyl-1-[4-(cyclopropylmethyl)-1,4-diazepan-1-yl]propan-1-one —— C17H30N2O
3-Cyclopentyl-1-[4-(cyclopropylmethyl)-1,4-diazepan-1-yl]propan-1-one
—— (2S)-1-[4-[(5-tert-butyl-1,3-oxazol-2-yl)methyl]-1,4-diazepan-1-yl]-2-[4-chloro-5-methyl-3-(trifluoromethyl)pyrazol-1-yl]propan-1-one —— C21H29ClF3N5O2
(2S)-1-[4-[(5-tert-butyl-1,3-oxazol-2-yl)methyl]-1,4-diazepan-1-yl]-2-[4-chloro-5-methyl-3-(trifluoromethyl)pyrazol-1-yl]propan-1-one
—— (E)-1-[4-[(5-tert-butyl-1,3-oxazol-2-yl)methyl]-1,4-diazepan-1-yl]-3-thiophen-2-ylprop-2-en-1-one —— C20H27N3O2S
(E)-1-[4-[(5-tert-butyl-1,3-oxazol-2-yl)methyl]-1,4-diazepan-1-yl]-3-thiophen-2-ylprop-2-en-1-one
—— 1-[4-[(5-Tert-butyl-1,3-oxazol-2-yl)methyl]-1,4-diazepan-1-yl]-3-cyclopentylpropan-1-one —— C21H35N3O2
1-[4-[(5-Tert-butyl-1,3-oxazol-2-yl)methyl]-1,4-diazepan-1-yl]-3-cyclopentylpropan-1-one
—— (2S)-1-[4-[(5-tert-butyl-1,3-oxazol-2-yl)methyl]-1,4-diazepan-1-yl]-2-[3-(trifluoromethyl)pyrazol-1-yl]propan-1-one —— C20H28F3N5O2
(2S)-1-[4-[(5-tert-butyl-1,3-oxazol-2-yl)methyl]-1,4-diazepan-1-yl]-2-[3-(trifluoromethyl)pyrazol-1-yl]propan-1-one
—— [(3R,4aS,8aR)-2,3,4a,8a-tetrahydro-1,4-benzodioxin-3-yl]-[4-(cyclopropylmethyl)-1,4-diazepan-1-yl]methanone —— C18H26N2O3
[(3R,4aS,8aR)-2,3,4a,8a-tetrahydro-1,4-benzodioxin-3-yl]-[4-(cyclopropylmethyl)-1,4-diazepan-1-yl]methanone
—— 1-[4-(Cyclopropylmethyl)-1,4-diazepan-1-yl]pentan-1-one —— C14H26N2O
1-[4-(Cyclopropylmethyl)-1,4-diazepan-1-yl]pentan-1-one
—— 1-[4-(Cyclopropylmethyl)-1,4-diazepan-1-yl]-2-ethylbutan-1-one —— C15H28N2O
1-[4-(Cyclopropylmethyl)-1,4-diazepan-1-yl]-2-ethylbutan-1-one
—— (2S)-2-[4-bromo-5-methyl-3-(trifluoromethyl)pyrazol-1-yl]-1-[4-[(5-tert-butyl-1,3-oxazol-2-yl)methyl]-1,4-diazepan-1-yl]propan-1-one —— C21H29BrF3N5O2
(2S)-2-[4-bromo-5-methyl-3-(trifluoromethyl)pyrazol-1-yl]-1-[4-[(5-tert-butyl-1,3-oxazol-2-yl)methyl]-1,4-diazepan-1-yl]propan-1-one
—— (2R)-1-[4-(cyclopropylmethyl)-1,4-diazepan-1-yl]-2-methylbutan-1-one —— C14H26N2O
(2R)-1-[4-(cyclopropylmethyl)-1,4-diazepan-1-yl]-2-methylbutan-1-one
—— 3-Cyclohexyl-1-[4-(cyclopropylmethyl)-1,4-diazepan-1-yl]propan-1-one —— C18H32N2O
3-Cyclohexyl-1-[4-(cyclopropylmethyl)-1,4-diazepan-1-yl]propan-1-one
—— 3-(4-Bromo-3,5-dimethylpyrazol-1-yl)-1-[4-[(5-tert-butyl-1,3-oxazol-2-yl)methyl]-1,4-diazepan-1-yl]propan-1-one —— C21H32BrN5O2
3-(4-Bromo-3,5-dimethylpyrazol-1-yl)-1-[4-[(5-tert-butyl-1,3-oxazol-2-yl)methyl]-1,4-diazepan-1-yl]propan-1-one
—— (2S)-3-(4-bromo-3,5-dimethylpyrazol-1-yl)-1-[4-[(5-tert-butyl-1,3-oxazol-2-yl)methyl]-1,4-diazepan-1-yl]-2-methylpropan-1-one —— C22H34BrN5O2
(2S)-3-(4-bromo-3,5-dimethylpyrazol-1-yl)-1-[4-[(5-tert-butyl-1,3-oxazol-2-yl)methyl]-1,4-diazepan-1-yl]-2-methylpropan-1-one
—— [(3R,4aS,8aR)-2,3,4a,8a-tetrahydro-1,4-benzodioxin-3-yl]-[4-[(5-tert-butyl-1,3-oxazol-2-yl)methyl]-1,4-diazepan-1-yl]methanone —— C22H31N3O4
[(3R,4aS,8aR)-2,3,4a,8a-tetrahydro-1,4-benzodioxin-3-yl]-[4-[(5-tert-butyl-1,3-oxazol-2-yl)methyl]-1,4-diazepan-1-yl]methanone
—— [4-(cyclopropylmethyl)-1,4-diazepan-1-yl]-[(1S,2R)-2-methylcyclopropyl]methanone —— C14H24N2O
[4-(cyclopropylmethyl)-1,4-diazepan-1-yl]-[(1S,2R)-2-methylcyclopropyl]methanone
—— [4-(cyclopropylmethyl)-1,4-diazepan-1-yl]-[(2R)-oxolan-2-yl]methanone —— C14H24N2O2
[4-(cyclopropylmethyl)-1,4-diazepan-1-yl]-[(2R)-oxolan-2-yl]methanone
—— (2S)-1-[4-[(5-tert-butyl-1,3-oxazol-2-yl)methyl]-1,4-diazepan-1-yl]-2-ethylhexan-1-one —— C21H37N3O2
(2S)-1-[4-[(5-tert-butyl-1,3-oxazol-2-yl)methyl]-1,4-diazepan-1-yl]-2-ethylhexan-1-one
—— Cyclobutyl-[4-(cyclopropylmethyl)-1,4-diazepan-1-yl]methanone —— C14H24N2O
Cyclobutyl-[4-(cyclopropylmethyl)-1,4-diazepan-1-yl]methanone
—— 1-[4-[(5-Tert-butyl-1,3-oxazol-2-yl)methyl]-1,4-diazepan-1-yl]-2-(3,5-dimethylpyrazol-1-yl)ethanone —— C20H31N5O2
1-[4-[(5-Tert-butyl-1,3-oxazol-2-yl)methyl]-1,4-diazepan-1-yl]-2-(3,5-dimethylpyrazol-1-yl)ethanone
—— [4-(cyclopropylmethyl)-1,4-diazepan-1-yl]-[(1S,2S)-2-methylcyclopropyl]methanone —— C14H24N2O
[4-(cyclopropylmethyl)-1,4-diazepan-1-yl]-[(1S,2S)-2-methylcyclopropyl]methanone
—— 1-[4-(Cyclopropylmethyl)-1,4-diazepan-1-yl]butan-1-one —— C13H24N2O
1-[4-(Cyclopropylmethyl)-1,4-diazepan-1-yl]butan-1-one
—— 1-(Cyclopropylmethyl)-4-propan-2-ylsulfonyl-1,4-diazepane —— C12H24N2O2S
1-(Cyclopropylmethyl)-4-propan-2-ylsulfonyl-1,4-diazepane
—— (2R)-3-(4-bromo-3,5-dimethylpyrazol-1-yl)-1-[4-[(5-tert-butyl-1,3-oxazol-2-yl)methyl]-1,4-diazepan-1-yl]-2-methylpropan-1-one —— C22H34BrN5O2
(2R)-3-(4-bromo-3,5-dimethylpyrazol-1-yl)-1-[4-[(5-tert-butyl-1,3-oxazol-2-yl)methyl]-1,4-diazepan-1-yl]-2-methylpropan-1-one
—— (2S)-1-[4-(cyclopropylmethyl)-1,4-diazepan-1-yl]-2-methylbutan-1-one —— C14H26N2O
(2S)-1-[4-(cyclopropylmethyl)-1,4-diazepan-1-yl]-2-methylbutan-1-one