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二氮杂卓

中文名称 英文名称 CAS号 化学式 结构式图片
—— 1-[4-[(2-Tert-butyl-1,3-thiazol-4-yl)methyl]-1,4-diazepan-1-yl]propan-1-one —— C16H27N3OS
1-[4-[(2-Tert-butyl-1,3-thiazol-4-yl)methyl]-1,4-diazepan-1-yl]propan-1-one
—— tert-butyl 4-[(2S)-3-(4-bromo-3,5-dimethylpyrazol-1-yl)-2-methylpropanoyl]-1,4-diazepane-1-carboxylate —— C19H31BrN4O3
tert-butyl 4-[(2S)-3-(4-bromo-3,5-dimethylpyrazol-1-yl)-2-methylpropanoyl]-1,4-diazepane-1-carboxylate
—— 1-[4-[(2-Tert-butyl-1,3-thiazol-4-yl)methyl]-1,4-diazepan-1-yl]-3-(4-methylphenyl)propan-1-one —— C23H33N3OS
1-[4-[(2-Tert-butyl-1,3-thiazol-4-yl)methyl]-1,4-diazepan-1-yl]-3-(4-methylphenyl)propan-1-one
—— [4-[(2-tert-butyl-1,3-thiazol-4-yl)methyl]-1,4-diazepan-1-yl]-[(1R,2S)-2-phenylcyclopropyl]methanone —— C23H31N3OS
[4-[(2-tert-butyl-1,3-thiazol-4-yl)methyl]-1,4-diazepan-1-yl]-[(1R,2S)-2-phenylcyclopropyl]methanone
—— [4-[(2-Tert-butyl-1,3-thiazol-4-yl)methyl]-1,4-diazepan-1-yl]-cyclopropylmethanone —— C17H27N3OS
[4-[(2-Tert-butyl-1,3-thiazol-4-yl)methyl]-1,4-diazepan-1-yl]-cyclopropylmethanone
—— Tert-butyl 4-(1,5-dimethylpyrazol-4-yl)sulfonyl-1,4-diazepane-1-carboxylate —— C15H26N4O4S
Tert-butyl 4-(1,5-dimethylpyrazol-4-yl)sulfonyl-1,4-diazepane-1-carboxylate
—— Tert-butyl 4-[3-(1,5-dimethylpyrazol-4-yl)propanoyl]-1,4-diazepane-1-carboxylate —— C18H30N4O3
Tert-butyl 4-[3-(1,5-dimethylpyrazol-4-yl)propanoyl]-1,4-diazepane-1-carboxylate
—— (2S)-1-[4-[(2-tert-butyl-1,3-thiazol-4-yl)methyl]-1,4-diazepan-1-yl]-2-ethylhexan-1-one —— C21H37N3OS
(2S)-1-[4-[(2-tert-butyl-1,3-thiazol-4-yl)methyl]-1,4-diazepan-1-yl]-2-ethylhexan-1-one
—— (E)-1-[4-[(2-tert-butyl-1,3-thiazol-4-yl)methyl]-1,4-diazepan-1-yl]-3-(5-methylfuran-2-yl)prop-2-en-1-one —— C21H29N3O2S
(E)-1-[4-[(2-tert-butyl-1,3-thiazol-4-yl)methyl]-1,4-diazepan-1-yl]-3-(5-methylfuran-2-yl)prop-2-en-1-one
—— 2-Tert-butyl-4-[(4-propan-2-ylsulfonyl-1,4-diazepan-1-yl)methyl]-1,3-thiazole —— C16H29N3O2S2
2-Tert-butyl-4-[(4-propan-2-ylsulfonyl-1,4-diazepan-1-yl)methyl]-1,3-thiazole
—— 1-[4-[(2-Tert-butyl-1,3-thiazol-4-yl)methyl]-1,4-diazepan-1-yl]-3-cyclohexylpropan-1-one —— C22H37N3OS
1-[4-[(2-Tert-butyl-1,3-thiazol-4-yl)methyl]-1,4-diazepan-1-yl]-3-cyclohexylpropan-1-one
—— [4-[(2-tert-butyl-1,3-thiazol-4-yl)methyl]-1,4-diazepan-1-yl]-[(2R)-oxolan-2-yl]methanone —— C18H29N3O2S
[4-[(2-tert-butyl-1,3-thiazol-4-yl)methyl]-1,4-diazepan-1-yl]-[(2R)-oxolan-2-yl]methanone
—— [4-[(2-tert-butyl-1,3-thiazol-4-yl)methyl]-1,4-diazepan-1-yl]-[(1R,2S)-2-methylcyclopropyl]methanone —— C18H29N3OS
[4-[(2-tert-butyl-1,3-thiazol-4-yl)methyl]-1,4-diazepan-1-yl]-[(1R,2S)-2-methylcyclopropyl]methanone
—— (2R)-1-[4-[(2-tert-butyl-1,3-thiazol-4-yl)methyl]-1,4-diazepan-1-yl]-2-ethylhexan-1-one —— C21H37N3OS
(2R)-1-[4-[(2-tert-butyl-1,3-thiazol-4-yl)methyl]-1,4-diazepan-1-yl]-2-ethylhexan-1-one
—— (2S)-1-[4-[(2-tert-butyl-1,3-thiazol-4-yl)methyl]-1,4-diazepan-1-yl]-2-methylbutan-1-one —— C18H31N3OS
(2S)-1-[4-[(2-tert-butyl-1,3-thiazol-4-yl)methyl]-1,4-diazepan-1-yl]-2-methylbutan-1-one
—— 1-[4-[(2-Tert-butyl-1,3-thiazol-4-yl)methyl]-1,4-diazepan-1-yl]-3,3-dimethylbutan-1-one —— C19H33N3OS
1-[4-[(2-Tert-butyl-1,3-thiazol-4-yl)methyl]-1,4-diazepan-1-yl]-3,3-dimethylbutan-1-one
—— Tert-butyl 4-[2-(4-chloro-3,5-dimethylpyrazol-1-yl)acetyl]-1,4-diazepane-1-carboxylate —— C17H27ClN4O3
Tert-butyl 4-[2-(4-chloro-3,5-dimethylpyrazol-1-yl)acetyl]-1,4-diazepane-1-carboxylate
—— 1-[4-[(2-Tert-butyl-1,3-thiazol-4-yl)methyl]-1,4-diazepan-1-yl]-3-methylbutan-1-one —— C18H31N3OS
1-[4-[(2-Tert-butyl-1,3-thiazol-4-yl)methyl]-1,4-diazepan-1-yl]-3-methylbutan-1-one
—— [4-[(2-Tert-butyl-1,3-thiazol-4-yl)methyl]-1,4-diazepan-1-yl]-cyclobutylmethanone —— C18H29N3OS
[4-[(2-Tert-butyl-1,3-thiazol-4-yl)methyl]-1,4-diazepan-1-yl]-cyclobutylmethanone
—— 1-[4-[(2-Tert-butyl-1,3-thiazol-4-yl)methyl]-1,4-diazepan-1-yl]-3-phenylpropan-1-one —— C22H31N3OS
1-[4-[(2-Tert-butyl-1,3-thiazol-4-yl)methyl]-1,4-diazepan-1-yl]-3-phenylpropan-1-one
—— 2-Tert-butyl-4-[[4-(2-methoxyethylsulfonyl)-1,4-diazepan-1-yl]methyl]-1,3-thiazole —— C16H29N3O3S2
2-Tert-butyl-4-[[4-(2-methoxyethylsulfonyl)-1,4-diazepan-1-yl]methyl]-1,3-thiazole
—— 1-(Azepan-1-yl)-5-[4-[(2-tert-butyl-1,3-thiazol-4-yl)methyl]-1,4-diazepan-1-yl]pentane-1,5-dione —— C24H40N4O2S
1-(Azepan-1-yl)-5-[4-[(2-tert-butyl-1,3-thiazol-4-yl)methyl]-1,4-diazepan-1-yl]pentane-1,5-dione
—— 1-[4-[(2-Tert-butyl-1,3-thiazol-4-yl)methyl]-1,4-diazepan-1-yl]-2,2,2-trifluoroethanone —— C15H22F3N3OS
1-[4-[(2-Tert-butyl-1,3-thiazol-4-yl)methyl]-1,4-diazepan-1-yl]-2,2,2-trifluoroethanone
—— tert-butyl 4-[(2R)-2-[4-chloro-5-methyl-3-(trifluoromethyl)pyrazol-1-yl]propanoyl]-1,4-diazepane-1-carboxylate —— C18H26ClF3N4O3
tert-butyl 4-[(2R)-2-[4-chloro-5-methyl-3-(trifluoromethyl)pyrazol-1-yl]propanoyl]-1,4-diazepane-1-carboxylate
—— (E)-1-[4-[(2-tert-butyl-1,3-thiazol-4-yl)methyl]-1,4-diazepan-1-yl]-3-thiophen-2-ylprop-2-en-1-one —— C20H27N3OS2
(E)-1-[4-[(2-tert-butyl-1,3-thiazol-4-yl)methyl]-1,4-diazepan-1-yl]-3-thiophen-2-ylprop-2-en-1-one
—— 1-[4-[(2-Tert-butyl-1,3-thiazol-4-yl)methyl]-1,4-diazepan-1-yl]-3-(4-fluorophenyl)propan-1-one —— C22H30FN3OS
1-[4-[(2-Tert-butyl-1,3-thiazol-4-yl)methyl]-1,4-diazepan-1-yl]-3-(4-fluorophenyl)propan-1-one
—— 1-[4-[(2-Tert-butyl-1,3-thiazol-4-yl)methyl]-1,4-diazepan-1-yl]-3-(1,3,5-trimethylpyrazol-4-yl)propan-1-one —— C22H35N5OS
1-[4-[(2-Tert-butyl-1,3-thiazol-4-yl)methyl]-1,4-diazepan-1-yl]-3-(1,3,5-trimethylpyrazol-4-yl)propan-1-one
—— [4-[(2-tert-butyl-1,3-thiazol-4-yl)methyl]-1,4-diazepan-1-yl]-[(1S,2R)-2-methylcyclopropyl]methanone —— C18H29N3OS
[4-[(2-tert-butyl-1,3-thiazol-4-yl)methyl]-1,4-diazepan-1-yl]-[(1S,2R)-2-methylcyclopropyl]methanone
—— tert-butyl 4-[(2R)-3-(4-bromo-3,5-dimethylpyrazol-1-yl)-2-methylpropanoyl]-1,4-diazepane-1-carboxylate —— C19H31BrN4O3
tert-butyl 4-[(2R)-3-(4-bromo-3,5-dimethylpyrazol-1-yl)-2-methylpropanoyl]-1,4-diazepane-1-carboxylate
—— 1-[4-[(2-Tert-butyl-1,3-thiazol-4-yl)methyl]-1,4-diazepan-1-yl]-4-phenylbutan-1-one —— C23H33N3OS
1-[4-[(2-Tert-butyl-1,3-thiazol-4-yl)methyl]-1,4-diazepan-1-yl]-4-phenylbutan-1-one
—— Tert-butyl 4-[2-(3,5-dimethylpyrazol-1-yl)acetyl]-1,4-diazepane-1-carboxylate —— C17H28N4O3
Tert-butyl 4-[2-(3,5-dimethylpyrazol-1-yl)acetyl]-1,4-diazepane-1-carboxylate
—— tert-butyl 4-[(2S)-2-[4-bromo-5-methyl-3-(trifluoromethyl)pyrazol-1-yl]propanoyl]-1,4-diazepane-1-carboxylate —— C18H26BrF3N4O3
tert-butyl 4-[(2S)-2-[4-bromo-5-methyl-3-(trifluoromethyl)pyrazol-1-yl]propanoyl]-1,4-diazepane-1-carboxylate
—— 1-[4-[(2-Tert-butyl-1,3-thiazol-4-yl)methyl]-1,4-diazepan-1-yl]-3-(2-fluorophenyl)propan-1-one —— C22H30FN3OS
1-[4-[(2-Tert-butyl-1,3-thiazol-4-yl)methyl]-1,4-diazepan-1-yl]-3-(2-fluorophenyl)propan-1-one
—— [4-[(2-tert-butyl-1,3-thiazol-4-yl)methyl]-1,4-diazepan-1-yl]-[(2S)-oxolan-2-yl]methanone —— C18H29N3O2S
[4-[(2-tert-butyl-1,3-thiazol-4-yl)methyl]-1,4-diazepan-1-yl]-[(2S)-oxolan-2-yl]methanone
—— tert-butyl 4-[(2R)-2-[4-bromo-5-methyl-3-(trifluoromethyl)pyrazol-1-yl]propanoyl]-1,4-diazepane-1-carboxylate —— C18H26BrF3N4O3
tert-butyl 4-[(2R)-2-[4-bromo-5-methyl-3-(trifluoromethyl)pyrazol-1-yl]propanoyl]-1,4-diazepane-1-carboxylate
—— [4-[(2-Tert-butyl-1,3-thiazol-4-yl)methyl]-1,4-diazepan-1-yl]-cyclohexylmethanone —— C20H33N3OS
[4-[(2-Tert-butyl-1,3-thiazol-4-yl)methyl]-1,4-diazepan-1-yl]-cyclohexylmethanone
—— [4-[(2-Tert-butyl-1,3-thiazol-4-yl)methyl]-1,4-diazepan-1-yl]-cyclopentylmethanone —— C19H31N3OS
[4-[(2-Tert-butyl-1,3-thiazol-4-yl)methyl]-1,4-diazepan-1-yl]-cyclopentylmethanone
—— 1-[4-[(2-Tert-butyl-1,3-thiazol-4-yl)methyl]-1,4-diazepan-1-yl]pentan-1-one —— C18H31N3OS
1-[4-[(2-Tert-butyl-1,3-thiazol-4-yl)methyl]-1,4-diazepan-1-yl]pentan-1-one
—— [4-[(2-tert-butyl-1,3-thiazol-4-yl)methyl]-1,4-diazepan-1-yl]-[(1S,2S)-2-methylcyclopropyl]methanone —— C18H29N3OS
[4-[(2-tert-butyl-1,3-thiazol-4-yl)methyl]-1,4-diazepan-1-yl]-[(1S,2S)-2-methylcyclopropyl]methanone
—— 1-[4-[(2-Tert-butyl-1,3-thiazol-4-yl)methyl]-1,4-diazepan-1-yl]-3-cyclopentylpropan-1-one —— C21H35N3OS
1-[4-[(2-Tert-butyl-1,3-thiazol-4-yl)methyl]-1,4-diazepan-1-yl]-3-cyclopentylpropan-1-one
—— Tert-butyl 4-[3-(4-bromo-3,5-dimethylpyrazol-1-yl)propanoyl]-1,4-diazepane-1-carboxylate —— C18H29BrN4O3
Tert-butyl 4-[3-(4-bromo-3,5-dimethylpyrazol-1-yl)propanoyl]-1,4-diazepane-1-carboxylate
—— [4-[(2-tert-butyl-1,3-thiazol-4-yl)methyl]-1,4-diazepan-1-yl]-[(1S,2S)-2-phenylcyclopropyl]methanone —— C23H31N3OS
[4-[(2-tert-butyl-1,3-thiazol-4-yl)methyl]-1,4-diazepan-1-yl]-[(1S,2S)-2-phenylcyclopropyl]methanone
—— Tert-butyl 4-[2-(4-bromo-3,5-dimethylpyrazol-1-yl)acetyl]-1,4-diazepane-1-carboxylate —— C17H27BrN4O3
Tert-butyl 4-[2-(4-bromo-3,5-dimethylpyrazol-1-yl)acetyl]-1,4-diazepane-1-carboxylate
—— 1-[4-[(2-Tert-butyl-1,3-thiazol-4-yl)methyl]-1,4-diazepan-1-yl]-2-methoxyethanone —— C16H27N3O2S
1-[4-[(2-Tert-butyl-1,3-thiazol-4-yl)methyl]-1,4-diazepan-1-yl]-2-methoxyethanone
—— 2-Tert-butyl-4-[(4-propylsulfonyl-1,4-diazepan-1-yl)methyl]-1,3-thiazole —— C16H29N3O2S2
2-Tert-butyl-4-[(4-propylsulfonyl-1,4-diazepan-1-yl)methyl]-1,3-thiazole
—— 1-[4-[(2-Tert-butyl-1,3-thiazol-4-yl)methyl]-1,4-diazepan-1-yl]-2-ethylbutan-1-one —— C19H33N3OS
1-[4-[(2-Tert-butyl-1,3-thiazol-4-yl)methyl]-1,4-diazepan-1-yl]-2-ethylbutan-1-one
—— [(3S,4aS,8aR)-2,3,4a,8a-tetrahydro-1,4-benzodioxin-3-yl]-[4-[(2-tert-butyl-1,3-thiazol-4-yl)methyl]-1,4-diazepan-1-yl]methanone —— C22H31N3O3S
[(3S,4aS,8aR)-2,3,4a,8a-tetrahydro-1,4-benzodioxin-3-yl]-[4-[(2-tert-butyl-1,3-thiazol-4-yl)methyl]-1,4-diazepan-1-yl]methanone
—— 3-(4-Bromo-3,5-dimethylpyrazol-1-yl)-1-[4-[(2-tert-butyl-1,3-thiazol-4-yl)methyl]-1,4-diazepan-1-yl]propan-1-one —— C21H32BrN5OS
3-(4-Bromo-3,5-dimethylpyrazol-1-yl)-1-[4-[(2-tert-butyl-1,3-thiazol-4-yl)methyl]-1,4-diazepan-1-yl]propan-1-one
—— (2S)-1-[4-[(2-tert-butyl-1,3-thiazol-4-yl)methyl]-1,4-diazepan-1-yl]-2-[3-(trifluoromethyl)pyrazol-1-yl]propan-1-one —— C20H28F3N5OS
(2S)-1-[4-[(2-tert-butyl-1,3-thiazol-4-yl)methyl]-1,4-diazepan-1-yl]-2-[3-(trifluoromethyl)pyrazol-1-yl]propan-1-one
—— 1-[4-[(2-Tert-butyl-1,3-thiazol-4-yl)methyl]-1,4-diazepan-1-yl]-2-(3-methylpyrazol-1-yl)ethanone —— C19H29N5OS
1-[4-[(2-Tert-butyl-1,3-thiazol-4-yl)methyl]-1,4-diazepan-1-yl]-2-(3-methylpyrazol-1-yl)ethanone