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二氮杂卓

中文名称 英文名称 CAS号 化学式 结构式图片
—— (6R)-1-(2-cyclopropylacetyl)-4-[2-(1H-pyrazol-4-yl)ethyl]-1,4-diazepane-6-carboxylic acid —— C16H24N4O3
(6R)-1-(2-cyclopropylacetyl)-4-[2-(1H-pyrazol-4-yl)ethyl]-1,4-diazepane-6-carboxylic acid
—— [(6R)-4-[(2-aminopyridin-3-yl)methyl]-6-hydroxy-1,4-diazepan-1-yl]-(oxan-4-yl)methanone —— C17H26N4O3
[(6R)-4-[(2-aminopyridin-3-yl)methyl]-6-hydroxy-1,4-diazepan-1-yl]-(oxan-4-yl)methanone
—— (6R)-1-[[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl]-4-(oxan-4-yl)-1,4-diazepan-6-ol —— C15H26N4O4
(6R)-1-[[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl]-4-(oxan-4-yl)-1,4-diazepan-6-ol
—— [(6S)-4-[(2-aminopyridin-3-yl)methyl]-6-hydroxy-1,4-diazepan-1-yl]-(oxan-4-yl)methanone —— C17H26N4O3
[(6S)-4-[(2-aminopyridin-3-yl)methyl]-6-hydroxy-1,4-diazepan-1-yl]-(oxan-4-yl)methanone
—— (6R)-1-[[1-(2-hydroxyethyl)-3-methylpyrazol-4-yl]methyl]-1,4-diazepane-6-carboxylic acid —— C13H22N4O3
(6R)-1-[[1-(2-hydroxyethyl)-3-methylpyrazol-4-yl]methyl]-1,4-diazepane-6-carboxylic acid
—— (6S)-1-[[1-(2-hydroxyethyl)-3-methylpyrazol-4-yl]methyl]-1,4-diazepane-6-carboxylic acid —— C13H22N4O3
(6S)-1-[[1-(2-hydroxyethyl)-3-methylpyrazol-4-yl]methyl]-1,4-diazepane-6-carboxylic acid
—— (6S)-1-[(1-benzylimidazol-2-yl)methyl]-4-(3-hydroxypropyl)-1,4-diazepan-6-ol —— C19H28N4O2
(6S)-1-[(1-benzylimidazol-2-yl)methyl]-4-(3-hydroxypropyl)-1,4-diazepan-6-ol
—— (6S)-1-[(E)-but-2-enyl]-4-[1-(methoxymethyl)cyclobutanecarbonyl]-1,4-diazepane-6-carboxylic acid —— C17H28N2O4
(6S)-1-[(E)-but-2-enyl]-4-[1-(methoxymethyl)cyclobutanecarbonyl]-1,4-diazepane-6-carboxylic acid
—— (6S)-1-[(2,4-dimethylpyrazol-3-yl)methyl]-4-(2-ethoxyethyl)-1,4-diazepan-6-ol —— C15H28N4O2
(6S)-1-[(2,4-dimethylpyrazol-3-yl)methyl]-4-(2-ethoxyethyl)-1,4-diazepan-6-ol
—— (6R)-1-[(E)-but-2-enyl]-4-[1-(methoxymethyl)cyclobutanecarbonyl]-1,4-diazepane-6-carboxylic acid —— C17H28N2O4
(6R)-1-[(E)-but-2-enyl]-4-[1-(methoxymethyl)cyclobutanecarbonyl]-1,4-diazepane-6-carboxylic acid
—— (6R)-1-(furan-2-ylmethyl)-4-(2-methoxyethylcarbamoyl)-1,4-diazepane-6-carboxylic acid —— C15H23N3O5
(6R)-1-(furan-2-ylmethyl)-4-(2-methoxyethylcarbamoyl)-1,4-diazepane-6-carboxylic acid
—— (6S)-1-(furan-2-ylmethyl)-4-(2-methoxyethylcarbamoyl)-1,4-diazepane-6-carboxylic acid —— C15H23N3O5
(6S)-1-(furan-2-ylmethyl)-4-(2-methoxyethylcarbamoyl)-1,4-diazepane-6-carboxylic acid
—— (6S)-1-(2-methoxyethylcarbamoyl)-4-(2H-triazol-4-ylmethyl)-1,4-diazepane-6-carboxylic acid —— C13H22N6O4
(6S)-1-(2-methoxyethylcarbamoyl)-4-(2H-triazol-4-ylmethyl)-1,4-diazepane-6-carboxylic acid
—— (6R)-1-(2-methoxyethylcarbamoyl)-4-(2H-triazol-4-ylmethyl)-1,4-diazepane-6-carboxylic acid —— C13H22N6O4
(6R)-1-(2-methoxyethylcarbamoyl)-4-(2H-triazol-4-ylmethyl)-1,4-diazepane-6-carboxylic acid
—— 1-[(6S)-4-acetyl-6-hydroxy-1,4-diazepan-1-yl]-3-(3-fluorophenyl)propan-1-one —— C16H21FN2O3
1-[(6S)-4-acetyl-6-hydroxy-1,4-diazepan-1-yl]-3-(3-fluorophenyl)propan-1-one
—— (6R)-1-(cyclopent-3-ene-1-carbonyl)-4-methylsulfonyl-1,4-diazepane-6-carboxylic acid —— C13H20N2O5S
(6R)-1-(cyclopent-3-ene-1-carbonyl)-4-methylsulfonyl-1,4-diazepane-6-carboxylic acid
—— (6S)-1-(cyclopent-3-ene-1-carbonyl)-4-methylsulfonyl-1,4-diazepane-6-carboxylic acid —— C13H20N2O5S
(6S)-1-(cyclopent-3-ene-1-carbonyl)-4-methylsulfonyl-1,4-diazepane-6-carboxylic acid
—— 1-[(6R)-4-acetyl-6-hydroxy-1,4-diazepan-1-yl]-3-(3-fluorophenyl)propan-1-one —— C16H21FN2O3
1-[(6R)-4-acetyl-6-hydroxy-1,4-diazepan-1-yl]-3-(3-fluorophenyl)propan-1-one
—— 4-[(6R)-4-[(4-chloro-5-methyl-1H-pyrazol-3-yl)methyl]-6-hydroxy-1,4-diazepan-1-yl]-4-oxobutanoic acid —— C14H21ClN4O4
4-[(6R)-4-[(4-chloro-5-methyl-1H-pyrazol-3-yl)methyl]-6-hydroxy-1,4-diazepan-1-yl]-4-oxobutanoic acid
—— 1-[(6R)-4-cyclopentyl-6-hydroxy-1,4-diazepan-1-yl]-2-(5-methyltetrazol-1-yl)ethanone —— C14H24N6O2
1-[(6R)-4-cyclopentyl-6-hydroxy-1,4-diazepan-1-yl]-2-(5-methyltetrazol-1-yl)ethanone
—— 1-[(6S)-4-cyclopentyl-6-hydroxy-1,4-diazepan-1-yl]-2-(5-methyltetrazol-1-yl)ethanone —— C14H24N6O2
1-[(6S)-4-cyclopentyl-6-hydroxy-1,4-diazepan-1-yl]-2-(5-methyltetrazol-1-yl)ethanone
—— 2-methoxy-1-[4-[(3R)-3-(5-methylfuran-2-yl)butyl]-1,4-diazepan-1-yl]ethanone —— C17H28N2O3
2-methoxy-1-[4-[(3R)-3-(5-methylfuran-2-yl)butyl]-1,4-diazepan-1-yl]ethanone
—— (6R)-1-(oxan-4-yl)-4-[2-(1,2,4-triazol-1-yl)acetyl]-1,4-diazepane-6-carboxylic acid —— C15H23N5O4
(6R)-1-(oxan-4-yl)-4-[2-(1,2,4-triazol-1-yl)acetyl]-1,4-diazepane-6-carboxylic acid
—— 2-methoxy-1-[4-[(3S)-3-(5-methylfuran-2-yl)butyl]-1,4-diazepan-1-yl]ethanone —— C17H28N2O3
2-methoxy-1-[4-[(3S)-3-(5-methylfuran-2-yl)butyl]-1,4-diazepan-1-yl]ethanone
—— 1-[(6S)-6-hydroxy-4-[[5-(hydroxymethyl)furan-2-yl]methyl]-1,4-diazepan-1-yl]-2-(triazol-2-yl)ethanone —— C15H21N5O4
1-[(6S)-6-hydroxy-4-[[5-(hydroxymethyl)furan-2-yl]methyl]-1,4-diazepan-1-yl]-2-(triazol-2-yl)ethanone
—— (6S)-1-(furan-2-ylmethylcarbamoyl)-4-(2H-triazol-4-ylmethyl)-1,4-diazepane-6-carboxylic acid —— C15H20N6O4
(6S)-1-(furan-2-ylmethylcarbamoyl)-4-(2H-triazol-4-ylmethyl)-1,4-diazepane-6-carboxylic acid
—— 2-hydroxy-1-[(6S)-6-hydroxy-4-[[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl]-1,4-diazepan-1-yl]ethanone —— C13H22N4O5
2-hydroxy-1-[(6S)-6-hydroxy-4-[[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl]-1,4-diazepan-1-yl]ethanone
—— 1-[(6R)-6-hydroxy-4-(3-hydroxypropyl)-1,4-diazepan-1-yl]-2-(4-methylpyrazol-1-yl)ethanone —— C14H24N4O3
1-[(6R)-6-hydroxy-4-(3-hydroxypropyl)-1,4-diazepan-1-yl]-2-(4-methylpyrazol-1-yl)ethanone
—— 2-hydroxy-1-[(6R)-6-hydroxy-4-[[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl]-1,4-diazepan-1-yl]ethanone —— C13H22N4O5
2-hydroxy-1-[(6R)-6-hydroxy-4-[[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl]-1,4-diazepan-1-yl]ethanone
—— 1-[(6S)-6-hydroxy-4-(3-hydroxypropyl)-1,4-diazepan-1-yl]-2-(4-methylpyrazol-1-yl)ethanone —— C14H24N4O3
1-[(6S)-6-hydroxy-4-(3-hydroxypropyl)-1,4-diazepan-1-yl]-2-(4-methylpyrazol-1-yl)ethanone
—— 1-[(6R)-6-hydroxy-4-[[5-(hydroxymethyl)furan-2-yl]methyl]-1,4-diazepan-1-yl]-2-(triazol-2-yl)ethanone —— C15H21N5O4
1-[(6R)-6-hydroxy-4-[[5-(hydroxymethyl)furan-2-yl]methyl]-1,4-diazepan-1-yl]-2-(triazol-2-yl)ethanone
—— (6R)-1-(furan-2-ylmethylcarbamoyl)-4-(2H-triazol-4-ylmethyl)-1,4-diazepane-6-carboxylic acid —— C15H20N6O4
(6R)-1-(furan-2-ylmethylcarbamoyl)-4-(2H-triazol-4-ylmethyl)-1,4-diazepane-6-carboxylic acid
—— 2-[(6R)-6-hydroxy-4-[[3-(2-methoxyethyl)imidazol-4-yl]methyl]-1,4-diazepan-1-yl]propane-1,3-diol —— C15H28N4O4
2-[(6R)-6-hydroxy-4-[[3-(2-methoxyethyl)imidazol-4-yl]methyl]-1,4-diazepan-1-yl]propane-1,3-diol
—— 1-[(6S)-6-hydroxy-4-[[5-(1H-pyrazol-5-yl)furan-2-yl]methyl]-1,4-diazepan-1-yl]-3-methylbut-2-en-1-one —— C18H24N4O3
1-[(6S)-6-hydroxy-4-[[5-(1H-pyrazol-5-yl)furan-2-yl]methyl]-1,4-diazepan-1-yl]-3-methylbut-2-en-1-one
—— 2-ethyl-1-[(6R)-6-hydroxy-4-[(5-methyl-1H-1,2,4-triazol-3-yl)methyl]-1,4-diazepan-1-yl]butan-1-one —— C15H27N5O2
2-ethyl-1-[(6R)-6-hydroxy-4-[(5-methyl-1H-1,2,4-triazol-3-yl)methyl]-1,4-diazepan-1-yl]butan-1-one
—— 2-ethyl-1-[(6S)-6-hydroxy-4-[(5-methyl-1H-1,2,4-triazol-3-yl)methyl]-1,4-diazepan-1-yl]butan-1-one —— C15H27N5O2
2-ethyl-1-[(6S)-6-hydroxy-4-[(5-methyl-1H-1,2,4-triazol-3-yl)methyl]-1,4-diazepan-1-yl]butan-1-one
—— 1-[(6R)-6-hydroxy-4-[[5-(1H-pyrazol-5-yl)furan-2-yl]methyl]-1,4-diazepan-1-yl]-3-methylbut-2-en-1-one —— C18H24N4O3
1-[(6R)-6-hydroxy-4-[[5-(1H-pyrazol-5-yl)furan-2-yl]methyl]-1,4-diazepan-1-yl]-3-methylbut-2-en-1-one
—— 5-[3-[(6R)-6-hydroxy-1,4-diazepan-1-yl]-3-oxopropyl]-1,2-oxazol-3-one —— C11H17N3O4
5-[3-[(6R)-6-hydroxy-1,4-diazepan-1-yl]-3-oxopropyl]-1,2-oxazol-3-one
—— 5-[3-[(6S)-6-hydroxy-1,4-diazepan-1-yl]-3-oxopropyl]-1,2-oxazol-3-one —— C11H17N3O4
5-[3-[(6S)-6-hydroxy-1,4-diazepan-1-yl]-3-oxopropyl]-1,2-oxazol-3-one
—— (6R)-1-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-4-(2-pyrrolidin-1-ylethyl)-1,4-diazepane-6-carboxylic acid —— C18H31N5O2
(6R)-1-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-4-(2-pyrrolidin-1-ylethyl)-1,4-diazepane-6-carboxylic acid
—— 1-[(6R)-6-hydroxy-4-[(3-pyridin-4-yl-1,2,4-oxadiazol-5-yl)methyl]-1,4-diazepan-1-yl]ethanone —— C15H19N5O3
1-[(6R)-6-hydroxy-4-[(3-pyridin-4-yl-1,2,4-oxadiazol-5-yl)methyl]-1,4-diazepan-1-yl]ethanone
—— 1-[(6S)-6-hydroxy-4-[(3-pyridin-4-yl-1,2,4-oxadiazol-5-yl)methyl]-1,4-diazepan-1-yl]ethanone —— C15H19N5O3
1-[(6S)-6-hydroxy-4-[(3-pyridin-4-yl-1,2,4-oxadiazol-5-yl)methyl]-1,4-diazepan-1-yl]ethanone
—— [(2S)-oxolan-2-yl]-[4-[(2-propan-2-yl-1,3-oxazol-4-yl)methyl]-1,4-diazepan-1-yl]methanone —— C17H27N3O3
[(2S)-oxolan-2-yl]-[4-[(2-propan-2-yl-1,3-oxazol-4-yl)methyl]-1,4-diazepan-1-yl]methanone
—— [(2R)-oxolan-2-yl]-[4-[(2-propan-2-yl-1,3-oxazol-4-yl)methyl]-1,4-diazepan-1-yl]methanone —— C17H27N3O3
[(2R)-oxolan-2-yl]-[4-[(2-propan-2-yl-1,3-oxazol-4-yl)methyl]-1,4-diazepan-1-yl]methanone
—— [(6R)-6-hydroxy-4-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]-1,4-diazepan-1-yl]-[1-(methoxymethyl)cyclopropyl]methanone —— C15H24N4O4
[(6R)-6-hydroxy-4-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]-1,4-diazepan-1-yl]-[1-(methoxymethyl)cyclopropyl]methanone
—— [(6S)-6-hydroxy-4-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]-1,4-diazepan-1-yl]-[1-(methoxymethyl)cyclopropyl]methanone —— C15H24N4O4
[(6S)-6-hydroxy-4-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]-1,4-diazepan-1-yl]-[1-(methoxymethyl)cyclopropyl]methanone
—— (6R)-1-(4-methoxypiperidin-1-yl)sulfonyl-1,4-diazepane-6-carboxylic acid —— C12H23N3O5S
(6R)-1-(4-methoxypiperidin-1-yl)sulfonyl-1,4-diazepane-6-carboxylic acid
—— (6S)-1-(4-methoxypiperidin-1-yl)sulfonyl-1,4-diazepane-6-carboxylic acid —— C12H23N3O5S
(6S)-1-(4-methoxypiperidin-1-yl)sulfonyl-1,4-diazepane-6-carboxylic acid
—— [4-[(4-chloro-5-methyl-1H-pyrazol-3-yl)methyl]-1,4-diazepan-1-yl]-[(2S)-oxolan-2-yl]methanone —— C15H23ClN4O2
[4-[(4-chloro-5-methyl-1H-pyrazol-3-yl)methyl]-1,4-diazepan-1-yl]-[(2S)-oxolan-2-yl]methanone
—— 1-[(6R)-4-cyclopentyl-6-hydroxy-1,4-diazepan-1-yl]-2-thiophen-2-ylethanone —— C16H24N2O2S
1-[(6R)-4-cyclopentyl-6-hydroxy-1,4-diazepan-1-yl]-2-thiophen-2-ylethanone