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二氮杂卓

中文名称 英文名称 CAS号 化学式 结构式图片
—— (3R)-4-benzyl-3-ethyl-1-[2-(2-methyl-6-oxo-1H-pyrimidin-5-yl)acetyl]-1,4-diazepan-5-one —— C21H26N4O3
(3R)-4-benzyl-3-ethyl-1-[2-(2-methyl-6-oxo-1H-pyrimidin-5-yl)acetyl]-1,4-diazepan-5-one
—— (3R)-4-[(4-fluorophenyl)methyl]-1-(6-oxo-4,5-dihydro-1H-pyridazine-3-carbonyl)-3-propan-2-yl-1,4-diazepan-5-one —— C20H25FN4O3
(3R)-4-[(4-fluorophenyl)methyl]-1-(6-oxo-4,5-dihydro-1H-pyridazine-3-carbonyl)-3-propan-2-yl-1,4-diazepan-5-one
—— (3S)-4-benzyl-3-ethyl-1-(1,3-thiazol-4-ylmethyl)-1,4-diazepan-5-one —— C18H23N3OS
(3S)-4-benzyl-3-ethyl-1-(1,3-thiazol-4-ylmethyl)-1,4-diazepan-5-one
—— (3S)-4-[(4-fluorophenyl)methyl]-3-propan-2-yl-1-[2-(tetrazol-2-yl)acetyl]-1,4-diazepan-5-one —— C18H23FN6O2
(3S)-4-[(4-fluorophenyl)methyl]-3-propan-2-yl-1-[2-(tetrazol-2-yl)acetyl]-1,4-diazepan-5-one
—— (3R)-4-benzyl-3-ethyl-1-[2-(1,2,4-triazol-1-yl)acetyl]-1,4-diazepan-5-one —— C18H23N5O2
(3R)-4-benzyl-3-ethyl-1-[2-(1,2,4-triazol-1-yl)acetyl]-1,4-diazepan-5-one
—— (3R)-4-benzyl-3-ethyl-1-(1,3-thiazol-4-ylmethyl)-1,4-diazepan-5-one —— C18H23N3OS
(3R)-4-benzyl-3-ethyl-1-(1,3-thiazol-4-ylmethyl)-1,4-diazepan-5-one
—— (3S)-4-(cyclopropylmethyl)-3-propan-2-yl-1-[2-(tetrazol-1-yl)acetyl]-1,4-diazepan-5-one —— C15H24N6O2
(3S)-4-(cyclopropylmethyl)-3-propan-2-yl-1-[2-(tetrazol-1-yl)acetyl]-1,4-diazepan-5-one
—— (3S)-N-cyclohexyl-4-(cyclopropylmethyl)-5-oxo-3-propan-2-yl-1,4-diazepane-1-carboxamide —— C19H33N3O2
(3S)-N-cyclohexyl-4-(cyclopropylmethyl)-5-oxo-3-propan-2-yl-1,4-diazepane-1-carboxamide
—— (3R)-N-cyclohexyl-4-(cyclopropylmethyl)-5-oxo-3-propan-2-yl-1,4-diazepane-1-carboxamide —— C19H33N3O2
(3R)-N-cyclohexyl-4-(cyclopropylmethyl)-5-oxo-3-propan-2-yl-1,4-diazepane-1-carboxamide
—— (3R)-4-benzyl-3-ethyl-1-[(2-ethylpyrimidin-5-yl)methyl]-1,4-diazepan-5-one —— C21H28N4O
(3R)-4-benzyl-3-ethyl-1-[(2-ethylpyrimidin-5-yl)methyl]-1,4-diazepan-5-one
—— (3S)-4-benzyl-3-ethyl-1-(oxan-4-yl)-1,4-diazepan-5-one —— C19H28N2O2
(3S)-4-benzyl-3-ethyl-1-(oxan-4-yl)-1,4-diazepan-5-one
—— (3S)-4-[(4-fluorophenyl)methyl]-1-[2-(3-methyl-1,2-oxazol-5-yl)acetyl]-3-propan-2-yl-1,4-diazepan-5-one —— C21H26FN3O3
(3S)-4-[(4-fluorophenyl)methyl]-1-[2-(3-methyl-1,2-oxazol-5-yl)acetyl]-3-propan-2-yl-1,4-diazepan-5-one
—— (3R)-4-(cyclopropylmethyl)-3-propan-2-yl-1-[2-(tetrazol-1-yl)acetyl]-1,4-diazepan-5-one —— C15H24N6O2
(3R)-4-(cyclopropylmethyl)-3-propan-2-yl-1-[2-(tetrazol-1-yl)acetyl]-1,4-diazepan-5-one
—— (3S)-4-benzyl-3-ethyl-1-[(2-ethylpyrimidin-5-yl)methyl]-1,4-diazepan-5-one —— C21H28N4O
(3S)-4-benzyl-3-ethyl-1-[(2-ethylpyrimidin-5-yl)methyl]-1,4-diazepan-5-one
—— (2R)-1-(cyclopropylmethyl)-2-propan-2-yl-4-[(1-propylimidazol-2-yl)methyl]-1,4-diazepane —— C19H34N4
(2R)-1-(cyclopropylmethyl)-2-propan-2-yl-4-[(1-propylimidazol-2-yl)methyl]-1,4-diazepane
—— (2R)-1-(cyclopropylmethyl)-4-(1H-imidazol-5-ylmethyl)-2-propan-2-yl-1,4-diazepane —— C16H28N4
(2R)-1-(cyclopropylmethyl)-4-(1H-imidazol-5-ylmethyl)-2-propan-2-yl-1,4-diazepane
—— (3R)-4-benzyl-3-ethyl-1-(oxan-4-yl)-1,4-diazepan-5-one —— C19H28N2O2
(3R)-4-benzyl-3-ethyl-1-(oxan-4-yl)-1,4-diazepan-5-one
—— (3R)-4-[(4-fluorophenyl)methyl]-1-[2-(3-methyl-1,2-oxazol-5-yl)acetyl]-3-propan-2-yl-1,4-diazepan-5-one —— C21H26FN3O3
(3R)-4-[(4-fluorophenyl)methyl]-1-[2-(3-methyl-1,2-oxazol-5-yl)acetyl]-3-propan-2-yl-1,4-diazepan-5-one
—— (2S)-1-(cyclopropylmethyl)-4-(1H-imidazol-5-ylmethyl)-2-propan-2-yl-1,4-diazepane —— C16H28N4
(2S)-1-(cyclopropylmethyl)-4-(1H-imidazol-5-ylmethyl)-2-propan-2-yl-1,4-diazepane
—— (3S)-4-(cyclopropylmethyl)-1-[(5-methoxy-4-oxopyran-2-yl)methyl]-3-propan-2-yl-1,4-diazepan-5-one —— C19H28N2O4
(3S)-4-(cyclopropylmethyl)-1-[(5-methoxy-4-oxopyran-2-yl)methyl]-3-propan-2-yl-1,4-diazepan-5-one
—— (3R)-4-[(4-fluorophenyl)methyl]-3-propan-2-yl-1-(2-pyridin-2-ylethyl)-1,4-diazepan-5-one —— C22H28FN3O
(3R)-4-[(4-fluorophenyl)methyl]-3-propan-2-yl-1-(2-pyridin-2-ylethyl)-1,4-diazepan-5-one
—— (3R)-1-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-4-[(4-fluorophenyl)methyl]-3-propan-2-yl-1,4-diazepan-5-one —— C21H29FN4O
(3R)-1-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-4-[(4-fluorophenyl)methyl]-3-propan-2-yl-1,4-diazepan-5-one
—— (3R)-4-benzyl-3-ethyl-1-[(1-methylimidazol-2-yl)methyl]-1,4-diazepan-5-one —— C19H26N4O
(3R)-4-benzyl-3-ethyl-1-[(1-methylimidazol-2-yl)methyl]-1,4-diazepan-5-one
—— (3R)-4-[(4-fluorophenyl)methyl]-3-propan-2-yl-1-(3-pyrazol-1-ylpropyl)-1,4-diazepan-5-one —— C21H29FN4O
(3R)-4-[(4-fluorophenyl)methyl]-3-propan-2-yl-1-(3-pyrazol-1-ylpropyl)-1,4-diazepan-5-one
—— (3R)-4-[(4-fluorophenyl)methyl]-1-(3-fluoropropyl)-3-propan-2-yl-1,4-diazepan-5-one —— C18H26F2N2O
(3R)-4-[(4-fluorophenyl)methyl]-1-(3-fluoropropyl)-3-propan-2-yl-1,4-diazepan-5-one
—— (3S)-4-[(4-fluorophenyl)methyl]-1-(3-fluoropropyl)-3-propan-2-yl-1,4-diazepan-5-one —— C18H26F2N2O
(3S)-4-[(4-fluorophenyl)methyl]-1-(3-fluoropropyl)-3-propan-2-yl-1,4-diazepan-5-one
—— (3S)-4-[(4-fluorophenyl)methyl]-3-propan-2-yl-1-(2-pyridin-2-ylethyl)-1,4-diazepan-5-one —— C22H28FN3O
(3S)-4-[(4-fluorophenyl)methyl]-3-propan-2-yl-1-(2-pyridin-2-ylethyl)-1,4-diazepan-5-one
—— (3S)-4-benzyl-3-ethyl-1-[(1-methylimidazol-2-yl)methyl]-1,4-diazepan-5-one —— C19H26N4O
(3S)-4-benzyl-3-ethyl-1-[(1-methylimidazol-2-yl)methyl]-1,4-diazepan-5-one
—— (3S)-4-[(4-fluorophenyl)methyl]-3-propan-2-yl-1-(3-pyrazol-1-ylpropyl)-1,4-diazepan-5-one —— C21H29FN4O
(3S)-4-[(4-fluorophenyl)methyl]-3-propan-2-yl-1-(3-pyrazol-1-ylpropyl)-1,4-diazepan-5-one
—— (3S)-4-(cyclopropylmethyl)-1-[(1-methylpyrazol-4-yl)methyl]-3-propan-2-yl-1,4-diazepan-5-one —— C17H28N4O
(3S)-4-(cyclopropylmethyl)-1-[(1-methylpyrazol-4-yl)methyl]-3-propan-2-yl-1,4-diazepan-5-one
—— (3S)-1-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-4-[(4-fluorophenyl)methyl]-3-propan-2-yl-1,4-diazepan-5-one —— C21H29FN4O
(3S)-1-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-4-[(4-fluorophenyl)methyl]-3-propan-2-yl-1,4-diazepan-5-one
—— (3S)-4-benzyl-3-ethyl-1-[(2-propan-2-ylpyrimidin-4-yl)methyl]-1,4-diazepan-5-one —— C22H30N4O
(3S)-4-benzyl-3-ethyl-1-[(2-propan-2-ylpyrimidin-4-yl)methyl]-1,4-diazepan-5-one
—— (3R)-4-(cyclopropylmethyl)-1-[(1-methylpyrazol-4-yl)methyl]-3-propan-2-yl-1,4-diazepan-5-one —— C17H28N4O
(3R)-4-(cyclopropylmethyl)-1-[(1-methylpyrazol-4-yl)methyl]-3-propan-2-yl-1,4-diazepan-5-one
—— (3S)-4-benzyl-3-ethyl-1-(2-pyridin-2-ylethyl)-1,4-diazepan-5-one —— C21H27N3O
(3S)-4-benzyl-3-ethyl-1-(2-pyridin-2-ylethyl)-1,4-diazepan-5-one
—— (3R)-4-benzyl-3-ethyl-1-[(2-propan-2-ylpyrimidin-4-yl)methyl]-1,4-diazepan-5-one —— C22H30N4O
(3R)-4-benzyl-3-ethyl-1-[(2-propan-2-ylpyrimidin-4-yl)methyl]-1,4-diazepan-5-one
—— (3S)-4-[(4-fluorophenyl)methyl]-1-[(5-methyl-1,3,4-thiadiazol-2-yl)methyl]-3-propan-2-yl-1,4-diazepan-5-one —— C19H25FN4OS
(3S)-4-[(4-fluorophenyl)methyl]-1-[(5-methyl-1,3,4-thiadiazol-2-yl)methyl]-3-propan-2-yl-1,4-diazepan-5-one
—— (3R)-4-benzyl-3-ethyl-1-[2-(2-oxopyridin-1-yl)acetyl]-1,4-diazepan-5-one —— C21H25N3O3
(3R)-4-benzyl-3-ethyl-1-[2-(2-oxopyridin-1-yl)acetyl]-1,4-diazepan-5-one
—— (3R)-4-benzyl-3-ethyl-1-(2-pyridin-2-ylethyl)-1,4-diazepan-5-one —— C21H27N3O
(3R)-4-benzyl-3-ethyl-1-(2-pyridin-2-ylethyl)-1,4-diazepan-5-one
—— 5-[[(3S)-4-benzyl-3-ethyl-5-oxo-1,4-diazepan-1-yl]methyl]-6-methyl-1H-pyrimidine-2,4-dione —— C20H26N4O3
5-[[(3S)-4-benzyl-3-ethyl-5-oxo-1,4-diazepan-1-yl]methyl]-6-methyl-1H-pyrimidine-2,4-dione
—— 5-[[(3R)-4-benzyl-3-ethyl-5-oxo-1,4-diazepan-1-yl]methyl]-6-methyl-1H-pyrimidine-2,4-dione —— C20H26N4O3
5-[[(3R)-4-benzyl-3-ethyl-5-oxo-1,4-diazepan-1-yl]methyl]-6-methyl-1H-pyrimidine-2,4-dione
—— (3R)-4-benzyl-3-ethyl-1-(2-ethylsulfanylethyl)-1,4-diazepan-5-one —— C18H28N2OS
(3R)-4-benzyl-3-ethyl-1-(2-ethylsulfanylethyl)-1,4-diazepan-5-one
—— (3S)-4-benzyl-3-ethyl-1-[2-(2-oxopyridin-1-yl)acetyl]-1,4-diazepan-5-one —— C21H25N3O3
(3S)-4-benzyl-3-ethyl-1-[2-(2-oxopyridin-1-yl)acetyl]-1,4-diazepan-5-one
—— 1-[2-[(3R)-4-(cyclopropylmethyl)-3-propan-2-yl-1,4-diazepan-1-yl]-2-oxoethyl]pyrimidin-2-one —— C18H28N4O2
1-[2-[(3R)-4-(cyclopropylmethyl)-3-propan-2-yl-1,4-diazepan-1-yl]-2-oxoethyl]pyrimidin-2-one
—— 1-[3-[(3S)-4-(cyclopropylmethyl)-3-propan-2-yl-1,4-diazepan-1-yl]-3-oxopropyl]pyrimidine-2,4-dione —— C19H30N4O3
1-[3-[(3S)-4-(cyclopropylmethyl)-3-propan-2-yl-1,4-diazepan-1-yl]-3-oxopropyl]pyrimidine-2,4-dione
—— (3S)-4-benzyl-3-ethyl-1-[[3-(2-methoxyethyl)imidazol-4-yl]methyl]-1,4-diazepan-5-one —— C21H30N4O2
(3S)-4-benzyl-3-ethyl-1-[[3-(2-methoxyethyl)imidazol-4-yl]methyl]-1,4-diazepan-5-one
—— 1-[2-[(3S)-4-(cyclopropylmethyl)-3-propan-2-yl-1,4-diazepan-1-yl]-2-oxoethyl]pyrimidin-2-one —— C18H28N4O2
1-[2-[(3S)-4-(cyclopropylmethyl)-3-propan-2-yl-1,4-diazepan-1-yl]-2-oxoethyl]pyrimidin-2-one
—— (3S)-4-[(4-fluorophenyl)methyl]-3-propan-2-yl-1-[2-(1,2,4-triazol-1-yl)acetyl]-1,4-diazepan-5-one —— C19H24FN5O2
(3S)-4-[(4-fluorophenyl)methyl]-3-propan-2-yl-1-[2-(1,2,4-triazol-1-yl)acetyl]-1,4-diazepan-5-one
—— (3R)-4-[(4-fluorophenyl)methyl]-3-propan-2-yl-1-[2-(1,2,4-triazol-1-yl)acetyl]-1,4-diazepan-5-one —— C19H24FN5O2
(3R)-4-[(4-fluorophenyl)methyl]-3-propan-2-yl-1-[2-(1,2,4-triazol-1-yl)acetyl]-1,4-diazepan-5-one
—— (3S)-4-benzyl-1-(3-ethoxypropanoyl)-3-ethyl-1,4-diazepan-5-one —— C19H28N2O3
(3S)-4-benzyl-1-(3-ethoxypropanoyl)-3-ethyl-1,4-diazepan-5-one
—— (3S)-4-benzyl-3-ethyl-1-[4-(1,2,4-triazol-1-yl)butanoyl]-1,4-diazepan-5-one —— C20H27N5O2
(3S)-4-benzyl-3-ethyl-1-[4-(1,2,4-triazol-1-yl)butanoyl]-1,4-diazepan-5-one