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中文名称 英文名称 CAS号 化学式 结构式图片
—— 2,2-dimethyl-1-[(4S)-4-(3-phenyl-1,2,4-oxadiazol-5-yl)-8-oxa-2-azaspiro[4.5]decan-2-yl]butan-1-one —— C22H29N3O3
2,2-dimethyl-1-[(4S)-4-(3-phenyl-1,2,4-oxadiazol-5-yl)-8-oxa-2-azaspiro[4.5]decan-2-yl]butan-1-one
—— (4R)-N,N-diethyl-4-(3-phenyl-1,2,4-oxadiazol-5-yl)-8-oxa-2-azaspiro[4.5]decane-2-carboxamide —— C21H28N4O3
(4R)-N,N-diethyl-4-(3-phenyl-1,2,4-oxadiazol-5-yl)-8-oxa-2-azaspiro[4.5]decane-2-carboxamide
—— (4S)-N,N-diethyl-4-(3-phenyl-1,2,4-oxadiazol-5-yl)-8-oxa-2-azaspiro[4.5]decane-2-carboxamide —— C21H28N4O3
(4S)-N,N-diethyl-4-(3-phenyl-1,2,4-oxadiazol-5-yl)-8-oxa-2-azaspiro[4.5]decane-2-carboxamide
—— (Z)-N-[[1-(4-methoxyphenyl)pyrazol-3-yl]methyl]-3-(1-methylpyrazol-4-yl)prop-2-enamide —— C18H19N5O2
(Z)-N-[[1-(4-methoxyphenyl)pyrazol-3-yl]methyl]-3-(1-methylpyrazol-4-yl)prop-2-enamide
—— cyclohexyl-[(4R)-4-(3-phenyl-1,2,4-oxadiazol-5-yl)-8-oxa-2-azaspiro[4.5]decan-2-yl]methanone —— C23H29N3O3
cyclohexyl-[(4R)-4-(3-phenyl-1,2,4-oxadiazol-5-yl)-8-oxa-2-azaspiro[4.5]decan-2-yl]methanone
—— 3-(4-chlorophenyl)-5-[[(4R)-4-methyl-6,7-dihydro-4H-thieno[3,2-c]pyridin-5-yl]methyl]-1,2,4-oxadiazole —— C17H16ClN3OS
3-(4-chlorophenyl)-5-[[(4R)-4-methyl-6,7-dihydro-4H-thieno[3,2-c]pyridin-5-yl]methyl]-1,2,4-oxadiazole
—— (Z)-N-[3-fluoro-4-(1,2,4-triazol-1-yl)phenyl]-3-(5-methylfuran-2-yl)prop-2-enamide —— C16H13FN4O2
(Z)-N-[3-fluoro-4-(1,2,4-triazol-1-yl)phenyl]-3-(5-methylfuran-2-yl)prop-2-enamide
—— (4S)-N-(2-methylpropyl)-4-(3-phenyl-1,2,4-oxadiazol-5-yl)-8-oxa-2-azaspiro[4.5]decane-2-carboxamide —— C21H28N4O3
(4S)-N-(2-methylpropyl)-4-(3-phenyl-1,2,4-oxadiazol-5-yl)-8-oxa-2-azaspiro[4.5]decane-2-carboxamide
—— 2-cyclopentyl-1-[(4S)-4-(3-phenyl-1,2,4-oxadiazol-5-yl)-8-oxa-2-azaspiro[4.5]decan-2-yl]ethanone —— C23H29N3O3
2-cyclopentyl-1-[(4S)-4-(3-phenyl-1,2,4-oxadiazol-5-yl)-8-oxa-2-azaspiro[4.5]decan-2-yl]ethanone
—— (Z)-3-(2-methyl-1,3-thiazol-4-yl)-N-[(1R)-1-(5-methylthiophen-2-yl)ethyl]prop-2-enamide —— C14H16N2OS2
(Z)-3-(2-methyl-1,3-thiazol-4-yl)-N-[(1R)-1-(5-methylthiophen-2-yl)ethyl]prop-2-enamide
—— [(4R)-4-(3-phenyl-1,2,4-oxadiazol-5-yl)-8-oxa-2-azaspiro[4.5]decan-2-yl]-pyridin-2-ylmethanone —— C22H22N4O3
[(4R)-4-(3-phenyl-1,2,4-oxadiazol-5-yl)-8-oxa-2-azaspiro[4.5]decan-2-yl]-pyridin-2-ylmethanone
—— 3,3-dimethyl-1-[(4S)-4-(3-phenyl-1,2,4-oxadiazol-5-yl)-8-oxa-2-azaspiro[4.5]decan-2-yl]butan-1-one —— C22H29N3O3
3,3-dimethyl-1-[(4S)-4-(3-phenyl-1,2,4-oxadiazol-5-yl)-8-oxa-2-azaspiro[4.5]decan-2-yl]butan-1-one
—— (Z)-3-(2-methyl-1,3-thiazol-4-yl)-N-[3-(3-oxo-[1,2,4]triazolo[4,3-a]pyridin-2-yl)propyl]prop-2-enamide —— C16H17N5O2S
(Z)-3-(2-methyl-1,3-thiazol-4-yl)-N-[3-(3-oxo-[1,2,4]triazolo[4,3-a]pyridin-2-yl)propyl]prop-2-enamide
—— 3,3-dimethyl-1-[(4R)-4-(3-phenyl-1,2,4-oxadiazol-5-yl)-8-oxa-2-azaspiro[4.5]decan-2-yl]butan-1-one —— C22H29N3O3
3,3-dimethyl-1-[(4R)-4-(3-phenyl-1,2,4-oxadiazol-5-yl)-8-oxa-2-azaspiro[4.5]decan-2-yl]butan-1-one
—— (4R)-N-(3-methylbutyl)-4-(3-phenyl-1,2,4-oxadiazol-5-yl)-8-oxa-2-azaspiro[4.5]decane-2-carboxamide —— C22H30N4O3
(4R)-N-(3-methylbutyl)-4-(3-phenyl-1,2,4-oxadiazol-5-yl)-8-oxa-2-azaspiro[4.5]decane-2-carboxamide
—— (4S)-N-(3-methylbutyl)-4-(3-phenyl-1,2,4-oxadiazol-5-yl)-8-oxa-2-azaspiro[4.5]decane-2-carboxamide —— C22H30N4O3
(4S)-N-(3-methylbutyl)-4-(3-phenyl-1,2,4-oxadiazol-5-yl)-8-oxa-2-azaspiro[4.5]decane-2-carboxamide
—— (Z)-N-[(4S)-1-tert-butyl-4,5,6,7-tetrahydroindazol-4-yl]-3-(2-methyl-1,3-thiazol-4-yl)prop-2-enamide —— C18H24N4OS
(Z)-N-[(4S)-1-tert-butyl-4,5,6,7-tetrahydroindazol-4-yl]-3-(2-methyl-1,3-thiazol-4-yl)prop-2-enamide
—— (Z)-N-[2-(3-oxo-[1,2,4]triazolo[4,3-a]pyridin-2-yl)ethyl]-3-thiophen-3-ylprop-2-enamide —— C15H14N4O2S
(Z)-N-[2-(3-oxo-[1,2,4]triazolo[4,3-a]pyridin-2-yl)ethyl]-3-thiophen-3-ylprop-2-enamide
—— 2,2-dimethyl-1-[(4R)-4-(3-phenyl-1,2,4-oxadiazol-5-yl)-8-oxa-2-azaspiro[4.5]decan-2-yl]butan-1-one —— C22H29N3O3
2,2-dimethyl-1-[(4R)-4-(3-phenyl-1,2,4-oxadiazol-5-yl)-8-oxa-2-azaspiro[4.5]decan-2-yl]butan-1-one
—— (Z)-N-[(4R)-1-tert-butyl-4,5,6,7-tetrahydroindazol-4-yl]-3-(2-methyl-1,3-thiazol-4-yl)prop-2-enamide —— C18H24N4OS
(Z)-N-[(4R)-1-tert-butyl-4,5,6,7-tetrahydroindazol-4-yl]-3-(2-methyl-1,3-thiazol-4-yl)prop-2-enamide
—— (Z)-3-(2-methyl-1,3-thiazol-4-yl)-N-[(1S)-1-(5-methylthiophen-2-yl)ethyl]prop-2-enamide —— C14H16N2OS2
(Z)-3-(2-methyl-1,3-thiazol-4-yl)-N-[(1S)-1-(5-methylthiophen-2-yl)ethyl]prop-2-enamide
—— (Z)-N-[4-(4,5-dimethyl-1,3-oxazol-2-yl)phenyl]-3-pyridin-3-ylprop-2-enamide —— C19H17N3O2
(Z)-N-[4-(4,5-dimethyl-1,3-oxazol-2-yl)phenyl]-3-pyridin-3-ylprop-2-enamide
—— (Z)-N-methyl-N-[(2-methylfuran-3-yl)methyl]-3-(1-phenylpyrazol-4-yl)prop-2-enamide —— C19H19N3O2
(Z)-N-methyl-N-[(2-methylfuran-3-yl)methyl]-3-(1-phenylpyrazol-4-yl)prop-2-enamide
—— (Z)-N-[3-fluoro-4-(1,2,4-triazol-1-yl)phenyl]-3-thiophen-3-ylprop-2-enamide —— C15H11FN4OS
(Z)-N-[3-fluoro-4-(1,2,4-triazol-1-yl)phenyl]-3-thiophen-3-ylprop-2-enamide
—— (Z)-3-(1-methylpyrazol-4-yl)-N-(2-methylsulfonylethyl)prop-2-enamide —— C10H15N3O3S
(Z)-3-(1-methylpyrazol-4-yl)-N-(2-methylsulfonylethyl)prop-2-enamide
—— 5-(2-chlorophenyl)-12-[(2S)-oxolane-2-carbonyl]-2,6,7,12-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one —— C20H19ClN4O3
5-(2-chlorophenyl)-12-[(2S)-oxolane-2-carbonyl]-2,6,7,12-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one
—— 5-(2-chlorophenyl)-12-[(2R)-2-methylbutanoyl]-2,6,7,12-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one —— C20H21ClN4O2
5-(2-chlorophenyl)-12-[(2R)-2-methylbutanoyl]-2,6,7,12-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one
—— 5-(2-chlorophenyl)-12-[(2S)-2-methylbutanoyl]-2,6,7,12-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one —— C20H21ClN4O2
5-(2-chlorophenyl)-12-[(2S)-2-methylbutanoyl]-2,6,7,12-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one
—— N-[(3R)-1-(5-phenyl-1H-pyrazol-3-yl)pyrrolidin-3-yl]-1,3-benzodioxole-5-carboxamide —— C21H20N4O3
N-[(3R)-1-(5-phenyl-1H-pyrazol-3-yl)pyrrolidin-3-yl]-1,3-benzodioxole-5-carboxamide
—— (Z)-N-[(4R)-1-tert-butyl-4,5,6,7-tetrahydroindazol-4-yl]-3-(1-methylpyrazol-4-yl)prop-2-enamide —— C18H25N5O
(Z)-N-[(4R)-1-tert-butyl-4,5,6,7-tetrahydroindazol-4-yl]-3-(1-methylpyrazol-4-yl)prop-2-enamide
—— (Z)-N-[(4S)-1-tert-butyl-4,5,6,7-tetrahydroindazol-4-yl]-3-(1-methylpyrazol-4-yl)prop-2-enamide —— C18H25N5O
(Z)-N-[(4S)-1-tert-butyl-4,5,6,7-tetrahydroindazol-4-yl]-3-(1-methylpyrazol-4-yl)prop-2-enamide
—— (Z)-N-[(3S)-1,1-dioxothiolan-3-yl]-3-(1-phenylpyrazol-4-yl)-N-prop-2-enylprop-2-enamide —— C19H21N3O3S
(Z)-N-[(3S)-1,1-dioxothiolan-3-yl]-3-(1-phenylpyrazol-4-yl)-N-prop-2-enylprop-2-enamide
—— 5-(2-chlorophenyl)-12-[(2R)-oxolane-2-carbonyl]-2,6,7,12-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one —— C20H19ClN4O3
5-(2-chlorophenyl)-12-[(2R)-oxolane-2-carbonyl]-2,6,7,12-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one
—— (Z)-N-(2-methoxyethyl)-3-(1-phenylpyrazol-4-yl)-N-(pyridin-2-ylmethyl)prop-2-enamide —— C21H22N4O2
(Z)-N-(2-methoxyethyl)-3-(1-phenylpyrazol-4-yl)-N-(pyridin-2-ylmethyl)prop-2-enamide
—— (Z)-N-[(3R)-1,1-dioxothiolan-3-yl]-3-(1-phenylpyrazol-4-yl)-N-prop-2-enylprop-2-enamide —— C19H21N3O3S
(Z)-N-[(3R)-1,1-dioxothiolan-3-yl]-3-(1-phenylpyrazol-4-yl)-N-prop-2-enylprop-2-enamide
—— (Z)-N-[3-[3-(3-fluorophenyl)-1H-pyrazol-5-yl]propyl]-N-methyl-3-(1-methylpyrazol-4-yl)prop-2-enamide —— C20H22FN5O
(Z)-N-[3-[3-(3-fluorophenyl)-1H-pyrazol-5-yl]propyl]-N-methyl-3-(1-methylpyrazol-4-yl)prop-2-enamide
—— (Z)-N-(3-methylsulfonylpropyl)-3-(1-phenylpyrazol-4-yl)prop-2-enamide —— C16H19N3O3S
(Z)-N-(3-methylsulfonylpropyl)-3-(1-phenylpyrazol-4-yl)prop-2-enamide
—— N-[(3S)-1-(5-phenyl-1H-pyrazol-3-yl)pyrrolidin-3-yl]-1,3-benzodioxole-5-carboxamide —— C21H20N4O3
N-[(3S)-1-(5-phenyl-1H-pyrazol-3-yl)pyrrolidin-3-yl]-1,3-benzodioxole-5-carboxamide
—— (Z)-N-[(1R)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]-3-(1,3-thiazol-2-yl)prop-2-enamide —— C18H17FN4OS
(Z)-N-[(1R)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]-3-(1,3-thiazol-2-yl)prop-2-enamide
—— (Z)-3-(2-phenyltriazol-4-yl)-N-(1-propan-2-ylpiperidin-4-yl)prop-2-enamide —— C19H25N5O
(Z)-3-(2-phenyltriazol-4-yl)-N-(1-propan-2-ylpiperidin-4-yl)prop-2-enamide
—— (Z)-2-(4-methylphenyl)-N-[(1S)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]ethenesulfonamide —— C19H20N4O2S
(Z)-2-(4-methylphenyl)-N-[(1S)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]ethenesulfonamide
—— (Z)-3-(2-methyl-1,3-thiazol-4-yl)-N-[[3-(2-oxo-1,3-oxazolidin-3-yl)phenyl]methyl]prop-2-enamide —— C17H17N3O3S
(Z)-3-(2-methyl-1,3-thiazol-4-yl)-N-[[3-(2-oxo-1,3-oxazolidin-3-yl)phenyl]methyl]prop-2-enamide
—— (Z)-3-(2-methyl-1,3-thiazol-4-yl)-N-[[3-(1,2,4-triazol-1-ylmethyl)phenyl]methyl]prop-2-enamide —— C17H17N5OS
(Z)-3-(2-methyl-1,3-thiazol-4-yl)-N-[[3-(1,2,4-triazol-1-ylmethyl)phenyl]methyl]prop-2-enamide
—— (Z)-N-[2-(3-oxo-[1,2,4]triazolo[4,3-a]pyridin-2-yl)ethyl]-3-(1-phenylpyrazol-4-yl)prop-2-enamide —— C20H18N6O2
(Z)-N-[2-(3-oxo-[1,2,4]triazolo[4,3-a]pyridin-2-yl)ethyl]-3-(1-phenylpyrazol-4-yl)prop-2-enamide
—— (Z)-N-[(1S)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]-3-(1,3-thiazol-2-yl)prop-2-enamide —— C18H17FN4OS
(Z)-N-[(1S)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]-3-(1,3-thiazol-2-yl)prop-2-enamide
—— (Z)-3-(1-phenylpyrazol-4-yl)-N-[[2-(1,2,4-triazol-1-yl)pyridin-3-yl]methyl]prop-2-enamide —— C20H17N7O
(Z)-3-(1-phenylpyrazol-4-yl)-N-[[2-(1,2,4-triazol-1-yl)pyridin-3-yl]methyl]prop-2-enamide
—— (Z)-N-(3-ethoxypropyl)-3-(2-phenyltriazol-4-yl)prop-2-enamide —— C16H20N4O2
(Z)-N-(3-ethoxypropyl)-3-(2-phenyltriazol-4-yl)prop-2-enamide
—— (Z)-3-(3,5-dimethyl-1-phenylpyrazol-4-yl)-1-(1,3-dimethylpyrazol-4-yl)prop-2-en-1-one —— C19H20N4O
(Z)-3-(3,5-dimethyl-1-phenylpyrazol-4-yl)-1-(1,3-dimethylpyrazol-4-yl)prop-2-en-1-one
—— (Z)-2-(4-methylphenyl)-N-[(1R)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]ethenesulfonamide —— C19H20N4O2S
(Z)-2-(4-methylphenyl)-N-[(1R)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]ethenesulfonamide
—— (Z)-1-(5-methyl-2-phenyl-1H-imidazol-4-yl)-3-(thiadiazol-4-yl)prop-2-en-1-one —— C15H12N4OS
(Z)-1-(5-methyl-2-phenyl-1H-imidazol-4-yl)-3-(thiadiazol-4-yl)prop-2-en-1-one