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中文名称 英文名称 CAS号 化学式 结构式图片
—— (Z)-3-[1-[(4-bromophenyl)methyl]-3-phenylpyrazol-4-yl]-2-cyano-N-(pyridin-2-ylmethyl)prop-2-enamide —— C26H20BrN5O
(Z)-3-[1-[(4-bromophenyl)methyl]-3-phenylpyrazol-4-yl]-2-cyano-N-(pyridin-2-ylmethyl)prop-2-enamide
—— N-[(1S)-1-(2,4-difluorophenyl)ethyl]-1-phenyltetrazol-5-amine —— C15H13F2N5
N-[(1S)-1-(2,4-difluorophenyl)ethyl]-1-phenyltetrazol-5-amine
—— (Z)-3-[1-benzyl-3-(4-methoxyphenyl)pyrazol-4-yl]-2-(4-chlorophenyl)sulfonylprop-2-enenitrile —— C26H20ClN3O3S
(Z)-3-[1-benzyl-3-(4-methoxyphenyl)pyrazol-4-yl]-2-(4-chlorophenyl)sulfonylprop-2-enenitrile
—— 1-[(1R)-1-[(2S)-oxolan-2-yl]ethyl]-3-[(3-pentan-3-yl-1,2-oxazol-5-yl)methyl]urea —— C16H27N3O3
1-[(1R)-1-[(2S)-oxolan-2-yl]ethyl]-3-[(3-pentan-3-yl-1,2-oxazol-5-yl)methyl]urea
—— (Z)-2-cyano-3-[5-(3,4-dimethoxyphenyl)-1H-pyrazol-4-yl]prop-2-enamide —— C15H14N4O3
(Z)-2-cyano-3-[5-(3,4-dimethoxyphenyl)-1H-pyrazol-4-yl]prop-2-enamide
—— [(2R)-1-(2-methyl-1H-indol-3-yl)-1-oxopropan-2-yl] 2-(tetrazol-1-yl)benzoate —— C20H17N5O3
[(2R)-1-(2-methyl-1H-indol-3-yl)-1-oxopropan-2-yl] 2-(tetrazol-1-yl)benzoate
—— (Z)-2-cyano-3-[5-(4-ethylphenyl)-1H-pyrazol-4-yl]prop-2-enamide —— C15H14N4O
(Z)-2-cyano-3-[5-(4-ethylphenyl)-1H-pyrazol-4-yl]prop-2-enamide
—— Methyl 6-[(1-phenyltetrazol-5-yl)amino]hexanoate —— C14H19N5O2
Methyl 6-[(1-phenyltetrazol-5-yl)amino]hexanoate
—— (Z)-2-cyano-3-[5-(4-ethylphenyl)-1H-pyrazol-4-yl]-N-(thiophen-2-ylmethyl)prop-2-enamide —— C20H18N4OS
(Z)-2-cyano-3-[5-(4-ethylphenyl)-1H-pyrazol-4-yl]-N-(thiophen-2-ylmethyl)prop-2-enamide
—— (Z)-2-cyano-3-[5-(4-fluorophenyl)-1H-pyrazol-4-yl]-N-(pyridin-4-ylmethyl)prop-2-enamide —— C19H14FN5O
(Z)-2-cyano-3-[5-(4-fluorophenyl)-1H-pyrazol-4-yl]-N-(pyridin-4-ylmethyl)prop-2-enamide
—— (Z)-2-cyano-3-[5-(4-methylphenyl)-1H-pyrazol-4-yl]-N-(1,3-thiazol-2-yl)prop-2-enamide —— C17H13N5OS
(Z)-2-cyano-3-[5-(4-methylphenyl)-1H-pyrazol-4-yl]-N-(1,3-thiazol-2-yl)prop-2-enamide
—— 1-[(1S)-1-[(2R)-oxolan-2-yl]ethyl]-3-[(3-pentan-3-yl-1,2-oxazol-5-yl)methyl]urea —— C16H27N3O3
1-[(1S)-1-[(2R)-oxolan-2-yl]ethyl]-3-[(3-pentan-3-yl-1,2-oxazol-5-yl)methyl]urea
—— 1-[(1R)-1-(3-imidazol-1-ylphenyl)ethyl]-3-[(1R)-1-pyridin-2-ylethyl]urea —— C19H21N5O
1-[(1R)-1-(3-imidazol-1-ylphenyl)ethyl]-3-[(1R)-1-pyridin-2-ylethyl]urea
—— 1-[(S)-cyclopropyl-(4-methyl-1,3-thiazol-2-yl)methyl]-3-[(1R)-1-(4-fluorophenyl)ethyl]urea —— C17H20FN3OS
1-[(S)-cyclopropyl-(4-methyl-1,3-thiazol-2-yl)methyl]-3-[(1R)-1-(4-fluorophenyl)ethyl]urea
—— 1-[(1S)-1-(2-ethyl-4-methyl-1,3-thiazol-5-yl)ethyl]-3-[(2-methoxypyridin-4-yl)methyl]-1-methylurea —— C17H24N4O2S
1-[(1S)-1-(2-ethyl-4-methyl-1,3-thiazol-5-yl)ethyl]-3-[(2-methoxypyridin-4-yl)methyl]-1-methylurea
—— 5-chloro-1-methyl-N-[(2R)-2-methyl-3-(2-methyl-1,3-dioxolan-2-yl)propyl]-3-propan-2-ylpyrazole-4-carboxamide —— C16H26ClN3O3
5-chloro-1-methyl-N-[(2R)-2-methyl-3-(2-methyl-1,3-dioxolan-2-yl)propyl]-3-propan-2-ylpyrazole-4-carboxamide
—— 1-[(S)-cyclopropyl-(4-methyl-1,3-thiazol-2-yl)methyl]-3-[(1S)-1-(4-fluorophenyl)ethyl]urea —— C17H20FN3OS
1-[(S)-cyclopropyl-(4-methyl-1,3-thiazol-2-yl)methyl]-3-[(1S)-1-(4-fluorophenyl)ethyl]urea
—— 1-[(1S)-1-(3,4-difluorophenyl)ethyl]-3-[(4,5-dimethyl-1,3-thiazol-2-yl)methyl]urea —— C15H17F2N3OS
1-[(1S)-1-(3,4-difluorophenyl)ethyl]-3-[(4,5-dimethyl-1,3-thiazol-2-yl)methyl]urea
—— 1-[(1S)-1-(3-imidazol-1-ylphenyl)ethyl]-3-[(1R)-1-pyridin-2-ylethyl]urea —— C19H21N5O
1-[(1S)-1-(3-imidazol-1-ylphenyl)ethyl]-3-[(1R)-1-pyridin-2-ylethyl]urea
—— 1-(benzimidazol-1-yl)-3-[(1S)-1-(4-pyrazol-1-ylphenyl)ethyl]urea —— C19H18N6O
1-(benzimidazol-1-yl)-3-[(1S)-1-(4-pyrazol-1-ylphenyl)ethyl]urea
—— 1-[(1R)-1-(3-imidazol-1-ylphenyl)ethyl]-3-[(1S)-1-pyridin-2-ylethyl]urea —— C19H21N5O
1-[(1R)-1-(3-imidazol-1-ylphenyl)ethyl]-3-[(1S)-1-pyridin-2-ylethyl]urea
—— 1-[(1S)-1-(3-imidazol-1-ylphenyl)ethyl]-3-[(1S)-1-pyridin-2-ylethyl]urea —— C19H21N5O
1-[(1S)-1-(3-imidazol-1-ylphenyl)ethyl]-3-[(1S)-1-pyridin-2-ylethyl]urea
—— N-[(2R)-2-(2,5-dimethylfuran-3-yl)-2-hydroxypropyl]-1-phenylpyrazole-4-carboxamide —— C19H21N3O3
N-[(2R)-2-(2,5-dimethylfuran-3-yl)-2-hydroxypropyl]-1-phenylpyrazole-4-carboxamide
—— 1-[(1R)-1-(2-ethyl-4-methyl-1,3-thiazol-5-yl)ethyl]-3-[(2-methoxypyridin-4-yl)methyl]-1-methylurea —— C17H24N4O2S
1-[(1R)-1-(2-ethyl-4-methyl-1,3-thiazol-5-yl)ethyl]-3-[(2-methoxypyridin-4-yl)methyl]-1-methylurea
—— N-[(2S)-2-hydroxy-2-(1-methylpyrazol-4-yl)propyl]-5-(4-methylphenyl)-1,3-oxazole-4-carboxamide —— C18H20N4O3
N-[(2S)-2-hydroxy-2-(1-methylpyrazol-4-yl)propyl]-5-(4-methylphenyl)-1,3-oxazole-4-carboxamide
—— 1-(benzimidazol-1-yl)-3-[(1S)-1-(3-imidazol-1-ylphenyl)ethyl]urea —— C19H18N6O
1-(benzimidazol-1-yl)-3-[(1S)-1-(3-imidazol-1-ylphenyl)ethyl]urea
—— 1-[(1R)-1-(3,4-difluorophenyl)ethyl]-3-[(4,5-dimethyl-1,3-thiazol-2-yl)methyl]urea —— C15H17F2N3OS
1-[(1R)-1-(3,4-difluorophenyl)ethyl]-3-[(4,5-dimethyl-1,3-thiazol-2-yl)methyl]urea
—— N-[(2-fluorophenyl)methyl]-3-methyl-1-phenylthieno[2,3-c]pyrazole-5-carboxamide —— C20H16FN3OS
N-[(2-fluorophenyl)methyl]-3-methyl-1-phenylthieno[2,3-c]pyrazole-5-carboxamide
—— 1-[(R)-cyclopropyl-(4-methyl-1,3-thiazol-2-yl)methyl]-3-[(1S)-1-(4-fluorophenyl)ethyl]urea —— C17H20FN3OS
1-[(R)-cyclopropyl-(4-methyl-1,3-thiazol-2-yl)methyl]-3-[(1S)-1-(4-fluorophenyl)ethyl]urea
—— N-[(2S)-2-(2,5-dimethylfuran-3-yl)-2-hydroxypropyl]-1-phenylpyrazole-4-carboxamide —— C19H21N3O3
N-[(2S)-2-(2,5-dimethylfuran-3-yl)-2-hydroxypropyl]-1-phenylpyrazole-4-carboxamide
—— N-[(2R)-2-hydroxy-2-thiophen-2-ylpropyl]-5-(4-methylphenyl)-1,3-oxazole-4-carboxamide —— C18H18N2O3S
N-[(2R)-2-hydroxy-2-thiophen-2-ylpropyl]-5-(4-methylphenyl)-1,3-oxazole-4-carboxamide
—— 1-(benzimidazol-1-yl)-3-[(1R)-1-(4-pyrazol-1-ylphenyl)ethyl]urea —— C19H18N6O
1-(benzimidazol-1-yl)-3-[(1R)-1-(4-pyrazol-1-ylphenyl)ethyl]urea
—— N-[(2R)-2-hydroxy-2-(1-methylpyrazol-4-yl)propyl]-5-(4-methylphenyl)-1,3-oxazole-4-carboxamide —— C18H20N4O3
N-[(2R)-2-hydroxy-2-(1-methylpyrazol-4-yl)propyl]-5-(4-methylphenyl)-1,3-oxazole-4-carboxamide
—— 1-[(R)-cyclopropyl-(4-methyl-1,3-thiazol-2-yl)methyl]-3-[(1R)-1-(4-fluorophenyl)ethyl]urea —— C17H20FN3OS
1-[(R)-cyclopropyl-(4-methyl-1,3-thiazol-2-yl)methyl]-3-[(1R)-1-(4-fluorophenyl)ethyl]urea
—— N-[(2R)-2-hydroxy-2-thiophen-3-ylpropyl]-5-(4-methylphenyl)-1,3-oxazole-4-carboxamide —— C18H18N2O3S
N-[(2R)-2-hydroxy-2-thiophen-3-ylpropyl]-5-(4-methylphenyl)-1,3-oxazole-4-carboxamide
—— 5-chloro-1-methyl-N-[(2S)-2-methyl-3-(2-methyl-1,3-dioxolan-2-yl)propyl]-3-propan-2-ylpyrazole-4-carboxamide —— C16H26ClN3O3
5-chloro-1-methyl-N-[(2S)-2-methyl-3-(2-methyl-1,3-dioxolan-2-yl)propyl]-3-propan-2-ylpyrazole-4-carboxamide
—— 1-(benzimidazol-1-yl)-3-[(1R)-1-(3-imidazol-1-ylphenyl)ethyl]urea —— C19H18N6O
1-(benzimidazol-1-yl)-3-[(1R)-1-(3-imidazol-1-ylphenyl)ethyl]urea
—— (1S)-1-[3-fluoro-4-(4-methylpyrazol-1-yl)phenyl]-N-[(1S)-1-(5-methyl-1,3,4-oxadiazol-2-yl)ethyl]ethanamine —— C17H20FN5O
(1S)-1-[3-fluoro-4-(4-methylpyrazol-1-yl)phenyl]-N-[(1S)-1-(5-methyl-1,3,4-oxadiazol-2-yl)ethyl]ethanamine
—— 2-[1-(4-fluorophenyl)pyrazol-3-yl]-N-[(2S)-2-hydroxy-2-thiophen-3-ylethyl]acetamide —— C17H16FN3O2S
2-[1-(4-fluorophenyl)pyrazol-3-yl]-N-[(2S)-2-hydroxy-2-thiophen-3-ylethyl]acetamide
—— N-[(2S)-2-hydroxy-2-thiophen-2-ylpropyl]-5-(4-methylphenyl)-1,3-oxazole-4-carboxamide —— C18H18N2O3S
N-[(2S)-2-hydroxy-2-thiophen-2-ylpropyl]-5-(4-methylphenyl)-1,3-oxazole-4-carboxamide
—— 2-[1-(difluoromethyl)-3,5-dimethylpyrazol-4-yl]-N-[(2R,3R)-2-hydroxy-2,3-dimethylpentyl]acetamide —— C15H25F2N3O2
2-[1-(difluoromethyl)-3,5-dimethylpyrazol-4-yl]-N-[(2R,3R)-2-hydroxy-2,3-dimethylpentyl]acetamide
—— (1R)-1-[3-fluoro-4-(4-methylpyrazol-1-yl)phenyl]-N-[(1S)-1-(5-methyl-1,3,4-oxadiazol-2-yl)ethyl]ethanamine —— C17H20FN5O
(1R)-1-[3-fluoro-4-(4-methylpyrazol-1-yl)phenyl]-N-[(1S)-1-(5-methyl-1,3,4-oxadiazol-2-yl)ethyl]ethanamine
—— 2-[1-(4-fluorophenyl)pyrazol-3-yl]-N-[(2R)-2-hydroxy-2-thiophen-3-ylethyl]acetamide —— C17H16FN3O2S
2-[1-(4-fluorophenyl)pyrazol-3-yl]-N-[(2R)-2-hydroxy-2-thiophen-3-ylethyl]acetamide
—— (1R)-1-[3-fluoro-4-(4-methylpyrazol-1-yl)phenyl]-N-[(1R)-1-(5-methyl-1,3,4-oxadiazol-2-yl)ethyl]ethanamine —— C17H20FN5O
(1R)-1-[3-fluoro-4-(4-methylpyrazol-1-yl)phenyl]-N-[(1R)-1-(5-methyl-1,3,4-oxadiazol-2-yl)ethyl]ethanamine
—— 7-[[(1R)-1-(1-phenyltetrazol-5-yl)ethyl]amino]-3,4-dihydro-1H-quinolin-2-one —— C18H18N6O
7-[[(1R)-1-(1-phenyltetrazol-5-yl)ethyl]amino]-3,4-dihydro-1H-quinolin-2-one
—— (1S)-1-[3-fluoro-4-(4-methylpyrazol-1-yl)phenyl]-N-[(1R)-1-(5-methyl-1,3,4-oxadiazol-2-yl)ethyl]ethanamine —— C17H20FN5O
(1S)-1-[3-fluoro-4-(4-methylpyrazol-1-yl)phenyl]-N-[(1R)-1-(5-methyl-1,3,4-oxadiazol-2-yl)ethyl]ethanamine
—— 2-[1-(difluoromethyl)-3,5-dimethylpyrazol-4-yl]-N-[(2S,3S)-2-hydroxy-2,3-dimethylpentyl]acetamide —— C15H25F2N3O2
2-[1-(difluoromethyl)-3,5-dimethylpyrazol-4-yl]-N-[(2S,3S)-2-hydroxy-2,3-dimethylpentyl]acetamide
—— 7-[[(1S)-1-(1-phenyltetrazol-5-yl)ethyl]amino]-3,4-dihydro-1H-quinolin-2-one —— C18H18N6O
7-[[(1S)-1-(1-phenyltetrazol-5-yl)ethyl]amino]-3,4-dihydro-1H-quinolin-2-one
—— 5-[[(1R)-1-(5-phenyl-1,3-oxazol-2-yl)ethyl]amino]-3H-1,3-benzoxazol-2-one —— C18H15N3O3
5-[[(1R)-1-(5-phenyl-1,3-oxazol-2-yl)ethyl]amino]-3H-1,3-benzoxazol-2-one
—— 3-fluoro-4-methoxy-N-[(1R)-1-(1-phenyltetrazol-5-yl)ethyl]aniline —— C16H16FN5O
3-fluoro-4-methoxy-N-[(1R)-1-(1-phenyltetrazol-5-yl)ethyl]aniline