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中文名称 英文名称 CAS号 化学式 结构式图片
—— N-[[2-[(3R)-1-(1-ethylpyrazol-4-yl)sulfonylpiperidin-3-yl]-1,3-thiazol-4-yl]methyl]acetamide —— C16H23N5O3S2
N-[[2-[(3R)-1-(1-ethylpyrazol-4-yl)sulfonylpiperidin-3-yl]-1,3-thiazol-4-yl]methyl]acetamide
—— (5E)-5-[[5-(4-chlorophenyl)-1H-pyrazol-4-yl]methylidene]-3-(4-methylphenyl)-2-sulfanylideneimidazolidin-4-one —— C20H15ClN4OS
(5E)-5-[[5-(4-chlorophenyl)-1H-pyrazol-4-yl]methylidene]-3-(4-methylphenyl)-2-sulfanylideneimidazolidin-4-one
—— N-[[2-[(3R)-1-[(2-fluorophenyl)methylsulfonyl]piperidin-3-yl]-1,3-thiazol-4-yl]methyl]acetamide —— C18H22FN3O3S2
N-[[2-[(3R)-1-[(2-fluorophenyl)methylsulfonyl]piperidin-3-yl]-1,3-thiazol-4-yl]methyl]acetamide
—— [(3R)-3-(4-chlorophenyl)sulfonylpyrrolidin-1-yl]-[3-(2-methoxyphenyl)-1H-pyrazol-5-yl]methanone —— C21H20ClN3O4S
[(3R)-3-(4-chlorophenyl)sulfonylpyrrolidin-1-yl]-[3-(2-methoxyphenyl)-1H-pyrazol-5-yl]methanone
—— [4-(3,5-dimethylphenyl)-5-sulfanylidenetetrazol-1-yl]methyl-ethyl-[(4-oxo-3H-quinazolin-2-yl)methyl]azanium —— C21H24N7OS+
[4-(3,5-dimethylphenyl)-5-sulfanylidenetetrazol-1-yl]methyl-ethyl-[(4-oxo-3H-quinazolin-2-yl)methyl]azanium
—— (5E)-5-[[5-(4-chlorophenyl)-1H-pyrazol-4-yl]methylidene]-3-(3,5-dimethylphenyl)-2-sulfanylideneimidazolidin-4-one —— C21H17ClN4OS
(5E)-5-[[5-(4-chlorophenyl)-1H-pyrazol-4-yl]methylidene]-3-(3,5-dimethylphenyl)-2-sulfanylideneimidazolidin-4-one
—— 2-[[[4-(2,6-dimethylphenyl)-5-sulfanylidenetetrazol-1-yl]methyl-ethylamino]methyl]-3H-quinazolin-4-one —— C21H23N7OS
2-[[[4-(2,6-dimethylphenyl)-5-sulfanylidenetetrazol-1-yl]methyl-ethylamino]methyl]-3H-quinazolin-4-one
—— 3-[(2Z)-2-[(4-imidazol-1-ylphenyl)methylidene]hydrazinyl]-6-methyl-4H-1,2,4-triazin-5-one —— C14H13N7O
3-[(2Z)-2-[(4-imidazol-1-ylphenyl)methylidene]hydrazinyl]-6-methyl-4H-1,2,4-triazin-5-one
—— 3-[(2Z)-2-[[1-benzyl-3-(3-methoxyphenyl)pyrazol-4-yl]methylidene]hydrazinyl]-6-methyl-4H-1,2,4-triazin-5-one —— C22H21N7O2
3-[(2Z)-2-[[1-benzyl-3-(3-methoxyphenyl)pyrazol-4-yl]methylidene]hydrazinyl]-6-methyl-4H-1,2,4-triazin-5-one
—— N-(4-ethoxy-3-methoxyphenyl)-2-[1-(4-methoxyphenyl)imidazol-2-yl]sulfanylacetamide —— C21H23N3O4S
N-(4-ethoxy-3-methoxyphenyl)-2-[1-(4-methoxyphenyl)imidazol-2-yl]sulfanylacetamide
—— N-(4-ethoxy-3-methoxyphenyl)-2-[1-(3-fluorophenyl)imidazol-2-yl]sulfanylacetamide —— C20H20FN3O3S
N-(4-ethoxy-3-methoxyphenyl)-2-[1-(3-fluorophenyl)imidazol-2-yl]sulfanylacetamide
—— 2-[1-(2,3-dimethylphenyl)imidazol-2-yl]sulfanyl-N-(4-ethoxy-3-methoxyphenyl)acetamide —— C22H25N3O3S
2-[1-(2,3-dimethylphenyl)imidazol-2-yl]sulfanyl-N-(4-ethoxy-3-methoxyphenyl)acetamide
—— [(3S)-3-(4-chlorophenyl)sulfonylpyrrolidin-1-yl]-[3-(2-methoxyphenyl)-1H-pyrazol-5-yl]methanone —— C21H20ClN3O4S
[(3S)-3-(4-chlorophenyl)sulfonylpyrrolidin-1-yl]-[3-(2-methoxyphenyl)-1H-pyrazol-5-yl]methanone
—— 5-(2,5-dimethoxyphenyl)-N-[(2S)-2-hydroxy-2-(1-methyl-2,3-dihydroindol-5-yl)ethyl]-2-methylpyrazole-3-carboxamide —— C24H28N4O4
5-(2,5-dimethoxyphenyl)-N-[(2S)-2-hydroxy-2-(1-methyl-2,3-dihydroindol-5-yl)ethyl]-2-methylpyrazole-3-carboxamide
—— N-[(2S)-butan-2-yl]-1-[3,5-dimethyl-1-(4-methylphenyl)pyrazol-4-yl]sulfonylpiperidine-4-carboxamide —— C22H32N4O3S
N-[(2S)-butan-2-yl]-1-[3,5-dimethyl-1-(4-methylphenyl)pyrazol-4-yl]sulfonylpiperidine-4-carboxamide
—— 5-(2,5-dimethoxyphenyl)-N-[(2R)-2-hydroxy-2-(1-methyl-2,3-dihydroindol-5-yl)ethyl]-2-methylpyrazole-3-carboxamide —— C24H28N4O4
5-(2,5-dimethoxyphenyl)-N-[(2R)-2-hydroxy-2-(1-methyl-2,3-dihydroindol-5-yl)ethyl]-2-methylpyrazole-3-carboxamide
—— 3-methoxy-N-[(2S)-2-methoxy-2-thiophen-3-ylethyl]-1-methylpyrazole-4-carboxamide —— C13H17N3O3S
3-methoxy-N-[(2S)-2-methoxy-2-thiophen-3-ylethyl]-1-methylpyrazole-4-carboxamide
—— 1-[3,5-dimethyl-1-(4-methylphenyl)pyrazol-4-yl]sulfonyl-N-[[(2S)-oxolan-2-yl]methyl]piperidine-4-carboxamide —— C23H32N4O4S
1-[3,5-dimethyl-1-(4-methylphenyl)pyrazol-4-yl]sulfonyl-N-[[(2S)-oxolan-2-yl]methyl]piperidine-4-carboxamide
—— 2-(1-adamantyl)-N-[[2-(4-butylphenyl)benzotriazol-5-yl]carbamothioyl]acetamide —— C29H35N5OS
2-(1-adamantyl)-N-[[2-(4-butylphenyl)benzotriazol-5-yl]carbamothioyl]acetamide
—— 1-[1-(4-chlorophenyl)-3,5-dimethylpyrazol-4-yl]sulfonyl-N-[[(2S)-oxolan-2-yl]methyl]piperidine-4-carboxamide —— C22H29ClN4O4S
1-[1-(4-chlorophenyl)-3,5-dimethylpyrazol-4-yl]sulfonyl-N-[[(2S)-oxolan-2-yl]methyl]piperidine-4-carboxamide
—— 1-[1-(4-chlorophenyl)-3,5-dimethylpyrazol-4-yl]sulfonyl-N-[[(2R)-oxolan-2-yl]methyl]piperidine-4-carboxamide —— C22H29ClN4O4S
1-[1-(4-chlorophenyl)-3,5-dimethylpyrazol-4-yl]sulfonyl-N-[[(2R)-oxolan-2-yl]methyl]piperidine-4-carboxamide
—— N-[(2S)-butan-2-yl]-1-[1-(4-fluorophenyl)-3,5-dimethylpyrazol-4-yl]sulfonylpiperidine-4-carboxamide —— C21H29FN4O3S
N-[(2S)-butan-2-yl]-1-[1-(4-fluorophenyl)-3,5-dimethylpyrazol-4-yl]sulfonylpiperidine-4-carboxamide
—— 1-[1-(4-fluorophenyl)-3,5-dimethylpyrazol-4-yl]sulfonyl-N-[[(2R)-oxolan-2-yl]methyl]piperidine-4-carboxamide —— C22H29FN4O4S
1-[1-(4-fluorophenyl)-3,5-dimethylpyrazol-4-yl]sulfonyl-N-[[(2R)-oxolan-2-yl]methyl]piperidine-4-carboxamide
—— 1-[1-(4-fluorophenyl)-3,5-dimethylpyrazol-4-yl]sulfonyl-N-[[(2S)-oxolan-2-yl]methyl]piperidine-4-carboxamide —— C22H29FN4O4S
1-[1-(4-fluorophenyl)-3,5-dimethylpyrazol-4-yl]sulfonyl-N-[[(2S)-oxolan-2-yl]methyl]piperidine-4-carboxamide
—— N-[(2R)-butan-2-yl]-1-[3,5-dimethyl-1-(4-methylphenyl)pyrazol-4-yl]sulfonylpiperidine-4-carboxamide —— C22H32N4O3S
N-[(2R)-butan-2-yl]-1-[3,5-dimethyl-1-(4-methylphenyl)pyrazol-4-yl]sulfonylpiperidine-4-carboxamide
—— N-[(2R)-butan-2-yl]-1-[1-(4-fluorophenyl)-3,5-dimethylpyrazol-4-yl]sulfonylpiperidine-4-carboxamide —— C21H29FN4O3S
N-[(2R)-butan-2-yl]-1-[1-(4-fluorophenyl)-3,5-dimethylpyrazol-4-yl]sulfonylpiperidine-4-carboxamide
—— 1-[3,5-dimethyl-1-(4-methylphenyl)pyrazol-4-yl]sulfonyl-N-[[(2R)-oxolan-2-yl]methyl]piperidine-4-carboxamide —— C23H32N4O4S
1-[3,5-dimethyl-1-(4-methylphenyl)pyrazol-4-yl]sulfonyl-N-[[(2R)-oxolan-2-yl]methyl]piperidine-4-carboxamide
—— 3-methoxy-N-[(2R)-2-methoxy-2-thiophen-3-ylethyl]-1-methylpyrazole-4-carboxamide —— C13H17N3O3S
3-methoxy-N-[(2R)-2-methoxy-2-thiophen-3-ylethyl]-1-methylpyrazole-4-carboxamide
—— 1-phenyl-N-[(1R)-1,2,3,4-tetrahydronaphthalen-1-yl]pyrazolo[3,4-d]pyrimidin-4-amine —— C21H19N5
1-phenyl-N-[(1R)-1,2,3,4-tetrahydronaphthalen-1-yl]pyrazolo[3,4-d]pyrimidin-4-amine
—— 4-amino-N-[(3S)-1,1-dioxothiolan-3-yl]-3-(3-morpholin-4-ylpropyl)-2-sulfanylidene-1,3-thiazole-5-carboxamide —— C15H24N4O4S3
4-amino-N-[(3S)-1,1-dioxothiolan-3-yl]-3-(3-morpholin-4-ylpropyl)-2-sulfanylidene-1,3-thiazole-5-carboxamide
—— 1-phenyl-N-[(1S)-1,2,3,4-tetrahydronaphthalen-1-yl]pyrazolo[3,4-d]pyrimidin-4-amine —— C21H19N5
1-phenyl-N-[(1S)-1,2,3,4-tetrahydronaphthalen-1-yl]pyrazolo[3,4-d]pyrimidin-4-amine
—— 2-[(1R,2R)-2-phenylcyclopropyl]-5-piperidin-1-yl-1,3-oxazole-4-carbonitrile —— C18H19N3O
2-[(1R,2R)-2-phenylcyclopropyl]-5-piperidin-1-yl-1,3-oxazole-4-carbonitrile
—— 5-[[(2S)-2-(4-tert-butylphenyl)-2-(dimethylamino)ethyl]amino]-2-phenyl-1,3-oxazole-4-carbonitrile —— C24H28N4O
5-[[(2S)-2-(4-tert-butylphenyl)-2-(dimethylamino)ethyl]amino]-2-phenyl-1,3-oxazole-4-carbonitrile
—— 4-amino-N-[(3R)-1,1-dioxothiolan-3-yl]-3-(3-morpholin-4-ylpropyl)-2-sulfanylidene-1,3-thiazole-5-carboxamide —— C15H24N4O4S3
4-amino-N-[(3R)-1,1-dioxothiolan-3-yl]-3-(3-morpholin-4-ylpropyl)-2-sulfanylidene-1,3-thiazole-5-carboxamide
—— 2-(3-fluorophenyl)-5-[[(2S)-2-morpholin-4-yl-2-thiophen-2-ylethyl]amino]-1,3-oxazole-4-carbonitrile —— C20H19FN4O2S
2-(3-fluorophenyl)-5-[[(2S)-2-morpholin-4-yl-2-thiophen-2-ylethyl]amino]-1,3-oxazole-4-carbonitrile
—— 2-(4-chlorophenyl)-5-[(3R)-3-hydroxypiperidin-1-yl]-1,3-oxazole-4-carbonitrile —— C15H14ClN3O2
2-(4-chlorophenyl)-5-[(3R)-3-hydroxypiperidin-1-yl]-1,3-oxazole-4-carbonitrile
—— (3S)-N-[4-(3-ethyl-1,2,4-oxadiazol-5-yl)phenyl]-2,3-dihydro-1,4-benzodioxine-3-carboxamide —— C19H17N3O4
(3S)-N-[4-(3-ethyl-1,2,4-oxadiazol-5-yl)phenyl]-2,3-dihydro-1,4-benzodioxine-3-carboxamide
—— 5-[[(2S)-2-(4-tert-butylphenyl)-2-(diethylamino)ethyl]amino]-2-phenyl-1,3-oxazole-4-carbonitrile —— C26H32N4O
5-[[(2S)-2-(4-tert-butylphenyl)-2-(diethylamino)ethyl]amino]-2-phenyl-1,3-oxazole-4-carbonitrile
—— 2-(3-fluorophenyl)-5-[(3R)-3-methylpiperidin-1-yl]-1,3-oxazole-4-carbonitrile —— C16H16FN3O
2-(3-fluorophenyl)-5-[(3R)-3-methylpiperidin-1-yl]-1,3-oxazole-4-carbonitrile
—— 5-[(3R)-3-hydroxypiperidin-1-yl]-2-thiophen-2-yl-1,3-oxazole-4-carbonitrile —— C13H13N3O2S
5-[(3R)-3-hydroxypiperidin-1-yl]-2-thiophen-2-yl-1,3-oxazole-4-carbonitrile
—— N'-[2-[1-(3-fluorophenyl)imidazol-2-yl]sulfanylacetyl]benzohydrazide —— C18H15FN4O2S
N'-[2-[1-(3-fluorophenyl)imidazol-2-yl]sulfanylacetyl]benzohydrazide
—— 5-[(3S)-3-hydroxypiperidin-1-yl]-2-phenyl-1,3-oxazole-4-carbonitrile —— C15H15N3O2
5-[(3S)-3-hydroxypiperidin-1-yl]-2-phenyl-1,3-oxazole-4-carbonitrile
—— 2-[(1S,2S)-2-phenylcyclopropyl]-5-(3-propan-2-yloxypropylamino)-1,3-oxazole-4-carbonitrile —— C19H23N3O2
2-[(1S,2S)-2-phenylcyclopropyl]-5-(3-propan-2-yloxypropylamino)-1,3-oxazole-4-carbonitrile
—— 2-(3-methoxyphenyl)-5-[[(2S)-2-morpholin-4-ylpropyl]amino]-1,3-oxazole-4-carbonitrile —— C18H22N4O3
2-(3-methoxyphenyl)-5-[[(2S)-2-morpholin-4-ylpropyl]amino]-1,3-oxazole-4-carbonitrile
—— 5-[[(2S)-2-(dimethylamino)-2-thiophen-2-ylethyl]amino]-2-(3-fluorophenyl)-1,3-oxazole-4-carbonitrile —— C18H17FN4OS
5-[[(2S)-2-(dimethylamino)-2-thiophen-2-ylethyl]amino]-2-(3-fluorophenyl)-1,3-oxazole-4-carbonitrile
—— 2-(3-methoxyphenyl)-5-[[(2R)-2-morpholin-4-ylpropyl]amino]-1,3-oxazole-4-carbonitrile —— C18H22N4O3
2-(3-methoxyphenyl)-5-[[(2R)-2-morpholin-4-ylpropyl]amino]-1,3-oxazole-4-carbonitrile
—— 2-[(1S,2S)-2-phenylcyclopropyl]-5-(2-thiophen-2-ylethylamino)-1,3-oxazole-4-carbonitrile —— C19H17N3OS
2-[(1S,2S)-2-phenylcyclopropyl]-5-(2-thiophen-2-ylethylamino)-1,3-oxazole-4-carbonitrile
—— (3S)-N-[2-(3-propan-2-yl-1,2,4-oxadiazol-5-yl)phenyl]-2,3-dihydro-1,4-benzodioxine-3-carboxamide —— C20H19N3O4
(3S)-N-[2-(3-propan-2-yl-1,2,4-oxadiazol-5-yl)phenyl]-2,3-dihydro-1,4-benzodioxine-3-carboxamide
—— 2-[(1R,2R)-2-phenylcyclopropyl]-5-(2-piperidin-1-ylethylamino)-1,3-oxazole-4-carbonitrile —— C20H24N4O
2-[(1R,2R)-2-phenylcyclopropyl]-5-(2-piperidin-1-ylethylamino)-1,3-oxazole-4-carbonitrile
—— 5-[(3S,5S)-3,5-dimethylpiperidin-1-yl]sulfonyl-2-phenyl-1,3-oxazole-4-carbonitrile —— C17H19N3O3S
5-[(3S,5S)-3,5-dimethylpiperidin-1-yl]sulfonyl-2-phenyl-1,3-oxazole-4-carbonitrile