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中文名称 英文名称 CAS号 化学式 结构式图片
—— 1-[(1S,3S)-3-ethoxyspiro[3.4]octan-1-yl]-3-[(4R)-1-methyl-4,5,6,7-tetrahydroindazol-4-yl]urea —— C19H30N4O2
1-[(1S,3S)-3-ethoxyspiro[3.4]octan-1-yl]-3-[(4R)-1-methyl-4,5,6,7-tetrahydroindazol-4-yl]urea
—— N-[(3R)-1-benzylpyrrolidin-1-ium-3-yl]-1-phenyltetrazol-5-amine —— C18H21N6+
N-[(3R)-1-benzylpyrrolidin-1-ium-3-yl]-1-phenyltetrazol-5-amine
—— (2S)-N-[2-(2-methyl-1,3-thiazol-4-yl)ethyl]-2-propan-2-ylthiomorpholine-4-carboxamide —— C14H23N3OS2
(2S)-N-[2-(2-methyl-1,3-thiazol-4-yl)ethyl]-2-propan-2-ylthiomorpholine-4-carboxamide
—— 1-[[1-(2-methylpropyl)imidazol-2-yl]methyl]-3-[(4R)-1-methyl-4,5,6,7-tetrahydroindazol-4-yl]urea —— C17H26N6O
1-[[1-(2-methylpropyl)imidazol-2-yl]methyl]-3-[(4R)-1-methyl-4,5,6,7-tetrahydroindazol-4-yl]urea
—— 1-[(1R,3R)-3-ethoxyspiro[3.4]octan-1-yl]-3-[(4R)-1-methyl-4,5,6,7-tetrahydroindazol-4-yl]urea —— C19H30N4O2
1-[(1R,3R)-3-ethoxyspiro[3.4]octan-1-yl]-3-[(4R)-1-methyl-4,5,6,7-tetrahydroindazol-4-yl]urea
—— (2S)-N-[(E)-1-(4-imidazol-1-ylphenyl)ethylideneamino]-2-(2-methylphenoxy)propanamide —— C21H22N4O2
(2S)-N-[(E)-1-(4-imidazol-1-ylphenyl)ethylideneamino]-2-(2-methylphenoxy)propanamide
—— 1-[2-[(1S,2R)-2-methylcyclohexyl]oxyethyl]-3-[(1S)-1-(1-methylpyrazol-4-yl)ethyl]urea —— C16H28N4O2
1-[2-[(1S,2R)-2-methylcyclohexyl]oxyethyl]-3-[(1S)-1-(1-methylpyrazol-4-yl)ethyl]urea
—— 1-[3-[(3,4-Dichlorophenyl)methoxy]phenyl]tetrazole —— C14H10Cl2N4O
1-[3-[(3,4-Dichlorophenyl)methoxy]phenyl]tetrazole
—— 1-[(2R)-2-(2,5-dimethylfuran-3-yl)-2-hydroxypropyl]-3-[(2R)-1-(3,5-dimethylpyrazol-1-yl)propan-2-yl]urea —— C18H28N4O3
1-[(2R)-2-(2,5-dimethylfuran-3-yl)-2-hydroxypropyl]-3-[(2R)-1-(3,5-dimethylpyrazol-1-yl)propan-2-yl]urea
—— 1-[(1R,2S)-2-methylsulfanylcyclopentyl]-3-[(4-pyrazol-1-ylphenyl)methyl]urea —— C17H22N4OS
1-[(1R,2S)-2-methylsulfanylcyclopentyl]-3-[(4-pyrazol-1-ylphenyl)methyl]urea
—— (7R)-4-[5-(3-methoxyphenyl)tetrazol-2-yl]-7-methyl-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidine —— C19H18N6OS
(7R)-4-[5-(3-methoxyphenyl)tetrazol-2-yl]-7-methyl-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidine
—— (Z)-3-[5-(4-bromophenyl)-1H-pyrazol-4-yl]-2-cyano-N-(1,3-thiazol-2-yl)prop-2-enamide —— C16H10BrN5OS
(Z)-3-[5-(4-bromophenyl)-1H-pyrazol-4-yl]-2-cyano-N-(1,3-thiazol-2-yl)prop-2-enamide
—— (Z)-3-[1-benzyl-3-(4-methoxyphenyl)pyrazol-4-yl]-2-cyano-N-(1,3-thiazol-2-yl)prop-2-enamide —— C24H19N5O2S
(Z)-3-[1-benzyl-3-(4-methoxyphenyl)pyrazol-4-yl]-2-cyano-N-(1,3-thiazol-2-yl)prop-2-enamide
—— (Z)-2-cyano-3-[3-(3,4-dimethoxyphenyl)-1-[(4-fluorophenyl)methyl]pyrazol-4-yl]-N-(furan-2-ylmethyl)prop-2-enamide —— C27H23FN4O4
(Z)-2-cyano-3-[3-(3,4-dimethoxyphenyl)-1-[(4-fluorophenyl)methyl]pyrazol-4-yl]-N-(furan-2-ylmethyl)prop-2-enamide
—— (2R)-2-(2,4-difluorophenoxy)-N-[(E)-1-(4-imidazol-1-ylphenyl)ethylideneamino]propanamide —— C20H18F2N4O2
(2R)-2-(2,4-difluorophenoxy)-N-[(E)-1-(4-imidazol-1-ylphenyl)ethylideneamino]propanamide
—— N-[[3-(4-chlorophenyl)-1-phenylpyrazol-4-yl]methyl]-N-methylcyclopropanecarboxamide —— C21H20ClN3O
N-[[3-(4-chlorophenyl)-1-phenylpyrazol-4-yl]methyl]-N-methylcyclopropanecarboxamide
—— (Z)-2-cyano-3-[5-(4-methoxyphenyl)-1H-pyrazol-4-yl]-N-(4-propan-2-ylphenyl)prop-2-enamide —— C23H22N4O2
(Z)-2-cyano-3-[5-(4-methoxyphenyl)-1H-pyrazol-4-yl]-N-(4-propan-2-ylphenyl)prop-2-enamide
—— N-[[3-(4-chlorophenyl)-1-phenylpyrazol-4-yl]methyl]-N-methylpyridine-2-carboxamide —— C23H19ClN4O
N-[[3-(4-chlorophenyl)-1-phenylpyrazol-4-yl]methyl]-N-methylpyridine-2-carboxamide
—— (5E)-2-imino-5-[[3-(2-methylpropyl)-1-phenylpyrazol-4-yl]methylidene]-3-(4-pyrrol-1-yl-1,2,5-oxadiazol-3-yl)-1,3-thiazolidin-4-one —— C23H21N7O2S
(5E)-2-imino-5-[[3-(2-methylpropyl)-1-phenylpyrazol-4-yl]methylidene]-3-(4-pyrrol-1-yl-1,2,5-oxadiazol-3-yl)-1,3-thiazolidin-4-one
—— (2R)-2-hydroxy-N-[(E)-1-(4-imidazol-1-ylphenyl)ethylideneamino]-2-phenylacetamide —— C19H18N4O2
(2R)-2-hydroxy-N-[(E)-1-(4-imidazol-1-ylphenyl)ethylideneamino]-2-phenylacetamide
—— 1-[(S)-cyclopropyl-(5-methyl-1,3-thiazol-2-yl)methyl]-3-[(2-methylpyrimidin-4-yl)methyl]urea —— C15H19N5OS
1-[(S)-cyclopropyl-(5-methyl-1,3-thiazol-2-yl)methyl]-3-[(2-methylpyrimidin-4-yl)methyl]urea
—— (Z)-2-cyano-N-[2-(3,4-dimethoxyphenyl)ethyl]-3-(3,5-dimethyl-1-phenylpyrazol-4-yl)prop-2-enamide —— C25H26N4O3
(Z)-2-cyano-N-[2-(3,4-dimethoxyphenyl)ethyl]-3-(3,5-dimethyl-1-phenylpyrazol-4-yl)prop-2-enamide
—— (2R)-2-(2-chloro-5-methylphenoxy)-N-[(E)-1-(4-imidazol-1-ylphenyl)ethylideneamino]propanamide —— C21H21ClN4O2
(2R)-2-(2-chloro-5-methylphenoxy)-N-[(E)-1-(4-imidazol-1-ylphenyl)ethylideneamino]propanamide
—— (Z)-N-[(4-chlorophenyl)methyl]-2-cyano-3-[5-(4-ethylphenyl)-1H-pyrazol-4-yl]prop-2-enamide —— C22H19ClN4O
(Z)-N-[(4-chlorophenyl)methyl]-2-cyano-3-[5-(4-ethylphenyl)-1H-pyrazol-4-yl]prop-2-enamide
—— [2-[(1-Cyanocyclohexyl)amino]-2-oxoethyl] 3-(tetrazol-1-yl)benzoate —— C17H18N6O3
[2-[(1-Cyanocyclohexyl)amino]-2-oxoethyl] 3-(tetrazol-1-yl)benzoate
—— (2S)-2-(2,4-difluorophenoxy)-N-[(E)-1-(4-imidazol-1-ylphenyl)ethylideneamino]propanamide —— C20H18F2N4O2
(2S)-2-(2,4-difluorophenoxy)-N-[(E)-1-(4-imidazol-1-ylphenyl)ethylideneamino]propanamide
—— (2S)-2-hydroxy-N-[(E)-1-(4-imidazol-1-ylphenyl)ethylideneamino]-2-phenylacetamide —— C19H18N4O2
(2S)-2-hydroxy-N-[(E)-1-(4-imidazol-1-ylphenyl)ethylideneamino]-2-phenylacetamide
—— (2R)-2-(4-chloro-3,5-dimethylphenoxy)-N-[(E)-1-(4-imidazol-1-ylphenyl)ethylideneamino]propanamide —— C22H23ClN4O2
(2R)-2-(4-chloro-3,5-dimethylphenoxy)-N-[(E)-1-(4-imidazol-1-ylphenyl)ethylideneamino]propanamide
—— (2R)-N-[(E)-1-(4-imidazol-1-ylphenyl)ethylideneamino]-2-[3-(trifluoromethyl)phenoxy]propanamide —— C21H19F3N4O2
(2R)-N-[(E)-1-(4-imidazol-1-ylphenyl)ethylideneamino]-2-[3-(trifluoromethyl)phenoxy]propanamide
—— propan-2-yl 2-[[(Z)-2-cyano-3-(1,3-diphenylpyrazol-4-yl)prop-2-enoyl]amino]thiophene-3-carboxylate —— C27H22N4O3S
propan-2-yl 2-[[(Z)-2-cyano-3-(1,3-diphenylpyrazol-4-yl)prop-2-enoyl]amino]thiophene-3-carboxylate
—— (Z)-2-cyano-3-[5-(4-ethylphenyl)-1H-pyrazol-4-yl]-N-(2,4,6-trimethylphenyl)prop-2-enamide —— C24H24N4O
(Z)-2-cyano-3-[5-(4-ethylphenyl)-1H-pyrazol-4-yl]-N-(2,4,6-trimethylphenyl)prop-2-enamide
—— (2S)-N-[(E)-1-(4-imidazol-1-ylphenyl)ethylideneamino]-2-[3-(trifluoromethyl)phenoxy]propanamide —— C21H19F3N4O2
(2S)-N-[(E)-1-(4-imidazol-1-ylphenyl)ethylideneamino]-2-[3-(trifluoromethyl)phenoxy]propanamide
—— (Z)-2-cyano-3-[1-[(2,6-dichlorophenyl)methyl]-3-phenylpyrazol-4-yl]-N-(2-phenylethyl)prop-2-enamide —— C28H22Cl2N4O
(Z)-2-cyano-3-[1-[(2,6-dichlorophenyl)methyl]-3-phenylpyrazol-4-yl]-N-(2-phenylethyl)prop-2-enamide
—— (2R)-N-[(E)-1-(4-imidazol-1-ylphenyl)ethylideneamino]-2-(2-methylphenoxy)propanamide —— C21H22N4O2
(2R)-N-[(E)-1-(4-imidazol-1-ylphenyl)ethylideneamino]-2-(2-methylphenoxy)propanamide
—— (Z)-N-(1,3-benzodioxol-5-yl)-3-(1-benzyl-3-phenylpyrazol-4-yl)-2-cyanoprop-2-enamide —— C27H20N4O3
(Z)-N-(1,3-benzodioxol-5-yl)-3-(1-benzyl-3-phenylpyrazol-4-yl)-2-cyanoprop-2-enamide
—— (2S)-2-(2-chloro-5-methylphenoxy)-N-[(E)-1-(4-imidazol-1-ylphenyl)ethylideneamino]propanamide —— C21H21ClN4O2
(2S)-2-(2-chloro-5-methylphenoxy)-N-[(E)-1-(4-imidazol-1-ylphenyl)ethylideneamino]propanamide
—— ethyl 2-[[(Z)-2-cyano-3-[5-(4-fluorophenyl)-1H-pyrazol-4-yl]prop-2-enoyl]amino]-5-propan-2-ylthiophene-3-carboxylate —— C23H21FN4O3S
ethyl 2-[[(Z)-2-cyano-3-[5-(4-fluorophenyl)-1H-pyrazol-4-yl]prop-2-enoyl]amino]-5-propan-2-ylthiophene-3-carboxylate
—— (Z)-N-(1,3-benzodioxol-5-ylmethyl)-2-cyano-3-(1,3-diphenylpyrazol-4-yl)prop-2-enamide —— C27H20N4O3
(Z)-N-(1,3-benzodioxol-5-ylmethyl)-2-cyano-3-(1,3-diphenylpyrazol-4-yl)prop-2-enamide
—— N'-methyl-N'-phenyl-N-(1-phenyltetrazol-5-yl)propane-1,3-diamine —— C17H20N6
N'-methyl-N'-phenyl-N-(1-phenyltetrazol-5-yl)propane-1,3-diamine
—— ethyl 2-[[(Z)-2-cyano-3-[5-(4-methoxyphenyl)-1H-pyrazol-4-yl]prop-2-enoyl]amino]thiophene-3-carboxylate —— C21H18N4O4S
ethyl 2-[[(Z)-2-cyano-3-[5-(4-methoxyphenyl)-1H-pyrazol-4-yl]prop-2-enoyl]amino]thiophene-3-carboxylate
—— N-[(1S)-1-(4-bromophenyl)propyl]-1-phenyltetrazol-5-amine —— C16H16BrN5
N-[(1S)-1-(4-bromophenyl)propyl]-1-phenyltetrazol-5-amine
—— (Z)-3-[1-benzyl-3-(4-methoxyphenyl)pyrazol-4-yl]-2-cyano-N-(3-cyano-4-ethyl-5-methylthiophen-2-yl)prop-2-enamide —— C29H25N5O2S
(Z)-3-[1-benzyl-3-(4-methoxyphenyl)pyrazol-4-yl]-2-cyano-N-(3-cyano-4-ethyl-5-methylthiophen-2-yl)prop-2-enamide
—— (Z)-2-cyano-N-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-[5-(4-methylphenyl)-1H-pyrazol-4-yl]prop-2-enamide —— C22H18N4O3
(Z)-2-cyano-N-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-[5-(4-methylphenyl)-1H-pyrazol-4-yl]prop-2-enamide
—— [(2R)-1-oxo-1-[[(1R)-1,2,3,4-tetrahydronaphthalen-1-yl]amino]propan-2-yl] 3-(tetrazol-1-yl)benzoate —— C21H21N5O3
[(2R)-1-oxo-1-[[(1R)-1,2,3,4-tetrahydronaphthalen-1-yl]amino]propan-2-yl] 3-(tetrazol-1-yl)benzoate
—— (Z)-2-cyano-3-[3-(3,4-dimethoxyphenyl)-1-[(2-fluorophenyl)methyl]pyrazol-4-yl]-N-(1,3-thiazol-2-yl)prop-2-enamide —— C25H20FN5O3S
(Z)-2-cyano-3-[3-(3,4-dimethoxyphenyl)-1-[(2-fluorophenyl)methyl]pyrazol-4-yl]-N-(1,3-thiazol-2-yl)prop-2-enamide
—— (Z)-N-(1,3-benzodioxol-5-yl)-3-[5-(4-chlorophenyl)-1H-pyrazol-4-yl]-2-cyanoprop-2-enamide —— C20H13ClN4O3
(Z)-N-(1,3-benzodioxol-5-yl)-3-[5-(4-chlorophenyl)-1H-pyrazol-4-yl]-2-cyanoprop-2-enamide
—— (Z)-3-[5-(4-chlorophenyl)-1H-pyrazol-4-yl]-2-cyano-N-[(4-methoxyphenyl)methyl]prop-2-enamide —— C21H17ClN4O2
(Z)-3-[5-(4-chlorophenyl)-1H-pyrazol-4-yl]-2-cyano-N-[(4-methoxyphenyl)methyl]prop-2-enamide
—— (Z)-3-[5-(4-bromophenyl)-1H-pyrazol-4-yl]-2-cyano-N-(2,3-dihydro-1,4-benzodioxin-6-yl)prop-2-enamide —— C21H15BrN4O3
(Z)-3-[5-(4-bromophenyl)-1H-pyrazol-4-yl]-2-cyano-N-(2,3-dihydro-1,4-benzodioxin-6-yl)prop-2-enamide
—— (Z)-3-[1-[(4-chlorophenyl)methyl]-3-(3,4-dimethoxyphenyl)pyrazol-4-yl]-2-cyano-N-(pyridin-3-ylmethyl)prop-2-enamide —— C28H24ClN5O3
(Z)-3-[1-[(4-chlorophenyl)methyl]-3-(3,4-dimethoxyphenyl)pyrazol-4-yl]-2-cyano-N-(pyridin-3-ylmethyl)prop-2-enamide
—— (Z)-3-[1-[(2-chloro-6-fluorophenyl)methyl]-3-phenylpyrazol-4-yl]-2-cyano-N-(3-cyanothiophen-2-yl)prop-2-enamide —— C25H15ClFN5OS
(Z)-3-[1-[(2-chloro-6-fluorophenyl)methyl]-3-phenylpyrazol-4-yl]-2-cyano-N-(3-cyanothiophen-2-yl)prop-2-enamide