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中文名称 英文名称 CAS号 化学式 结构式图片
—— 5-amino-1-(3,4-difluorophenyl)-N-(2-((ethyl)(phenylcarbonyl)aminomethyl)-3,3,3-trifluoro-2-hydroxypropyl)-1H-pyrazole-4-carboxamide 1034141-43-9 C23H22F5N5O3
5-amino-1-(3,4-difluorophenyl)-N-(2-((ethyl)(phenylcarbonyl)aminomethyl)-3,3,3-trifluoro-2-hydroxypropyl)-1H-pyrazole-4-carboxamide
—— 3-(6-bromo-3-{2,2,2-trifluoro-1-[1-(4-fluorophenyl)-1H-indazol-5-yl]-1-hydroxyethyl}indol-1-yl)propane-1,2-diol 1032648-82-0 C26H20BrF4N3O3
3-(6-bromo-3-{2,2,2-trifluoro-1-[1-(4-fluorophenyl)-1H-indazol-5-yl]-1-hydroxyethyl}indol-1-yl)propane-1,2-diol
—— 3-{2,2,2-trifluoro-1-[1-(4-fluorophenyl)-1H-indazol-5-yl]-1-hydroxyethyl}pyrrolo[2,3-b]pyridine-1-sulfonic acid dimethylamide 1032648-13-7 C24H19F4N5O3S
3-{2,2,2-trifluoro-1-[1-(4-fluorophenyl)-1H-indazol-5-yl]-1-hydroxyethyl}pyrrolo[2,3-b]pyridine-1-sulfonic acid dimethylamide
—— (2R,6R)-6-(aminomethyl)-4-{(1R)-1-[1-benzyl-4-(3-fluorophenyl)-1H-imidazol-2-yl]-2,2-dimethylpropyl}-2-methylmorpholin-3-one 1039747-03-9 C27H33FN4O2
(2R,6R)-6-(aminomethyl)-4-{(1R)-1-[1-benzyl-4-(3-fluorophenyl)-1H-imidazol-2-yl]-2,2-dimethylpropyl}-2-methylmorpholin-3-one
—— 3-(4-chloro-7-{2,2,2-trifluoro-1-[1-(4-fluorophenyl)-1H-indazol-5-yl]-1-hydroxyethyl}pyrrolo[3,2-d]pyrimidin-5-yl)propane-1,2-diol 1032648-86-4 C24H18ClF4N5O3
3-(4-chloro-7-{2,2,2-trifluoro-1-[1-(4-fluorophenyl)-1H-indazol-5-yl]-1-hydroxyethyl}pyrrolo[3,2-d]pyrimidin-5-yl)propane-1,2-diol
—— 1-[4-chloro-5-(2-hydroxyethyl)-5H-pyrrolo[3,2-d]pyrimidin-7-yl]-2,2,2-trifluoro-1-[1-(4-fluorophenyl)-1H-indazol-5-yl]ethanol 1032648-85-3 C23H16ClF4N5O2
1-[4-chloro-5-(2-hydroxyethyl)-5H-pyrrolo[3,2-d]pyrimidin-7-yl]-2,2,2-trifluoro-1-[1-(4-fluorophenyl)-1H-indazol-5-yl]ethanol
—— {3-[7-(2-methyl-2H-tetrazol-5-yl)imidazo[1,2-a]pyridin-3-yl]-phenyl}[1,3,4]thiadiazol-2-yl-amine 1036761-80-4 C17H13N9S
{3-[7-(2-methyl-2H-tetrazol-5-yl)imidazo[1,2-a]pyridin-3-yl]-phenyl}[1,3,4]thiadiazol-2-yl-amine
—— 1-(7-chloro-1H-pyrrolo[2,3-c]pyridin-3-yl)-2,2,2-trifluoro-1-[1-(4-fluorophenyl)-1H-indazol-5-yl]ethanol 1032648-07-9 C22H13ClF4N4O
1-(7-chloro-1H-pyrrolo[2,3-c]pyridin-3-yl)-2,2,2-trifluoro-1-[1-(4-fluorophenyl)-1H-indazol-5-yl]ethanol
—— N5,N5-Dibenzyl-3-(2,4-difluorophenyl)-3,4-diazatricyclo[5.2.1.02,6]deca-2(6),4-dien-5-amine 1024003-70-0 C28H25F2N3
N5,N5-Dibenzyl-3-(2,4-difluorophenyl)-3,4-diazatricyclo[5.2.1.02,6]deca-2(6),4-dien-5-amine
—— 3-(2,4-difluorophenyl)-5-[(E)-3,3-dimethyl-1-butenyl]-3,4-diazatricyclo[5.2.1.0(2,6)]deca-2(6),4-diene 1024003-91-5 C20H22F2N2
3-(2,4-difluorophenyl)-5-[(E)-3,3-dimethyl-1-butenyl]-3,4-diazatricyclo[5.2.1.0(2,6)]deca-2(6),4-diene
—— 3-(2,4-difluorophenyl)-5-(1-fluro-3,3-dimethylbutyl)-3,4-diazatricyclo[5.2.1.0(2,6)]deca-2(6),4-diene 1024003-74-4 C20H23F3N2
3-(2,4-difluorophenyl)-5-(1-fluro-3,3-dimethylbutyl)-3,4-diazatricyclo[5.2.1.0(2,6)]deca-2(6),4-diene
—— 6-(3-Amino-4-methylphenyl)-3-(3,4,5-trimethoxyphenyl)-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazole 1022918-45-1 C19H19N5O3S
6-(3-Amino-4-methylphenyl)-3-(3,4,5-trimethoxyphenyl)-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazole
—— ethyl 2-[5-chloro-2-[[2-(2,4-difluorophenoxy)-2-methylpropanoyl]amino]thiazol-4-yl]acetate 1052720-28-1 C17H17ClF2N2O4S
ethyl 2-[5-chloro-2-[[2-(2,4-difluorophenoxy)-2-methylpropanoyl]amino]thiazol-4-yl]acetate
—— 3-(2,4-Difluorophenyl)-5-(3,3-dimethylbutyl)-3,4-diazatricyclo[5.2.1.02,6]deca-2(6),4-diene 1024003-92-6 C20H24F2N2
3-(2,4-Difluorophenyl)-5-(3,3-dimethylbutyl)-3,4-diazatricyclo[5.2.1.02,6]deca-2(6),4-diene
—— 5-(tert-Butyl)-2-[5-(2,4-difluorophenyl)-4,5-diazatricyclo[5.2.1.02,6]deca-2(6),3-dien-3yl]-1,3-oxazole 1024004-14-5 C21H21F2N3O
5-(tert-Butyl)-2-[5-(2,4-difluorophenyl)-4,5-diazatricyclo[5.2.1.02,6]deca-2(6),3-dien-3yl]-1,3-oxazole
—— 2-(4-chloro-phenyl)-4-methyl-thiazole-5-carboxylic acid 3,4-dichloro-benzylamide 1048364-19-7 C18H13Cl3N2OS
2-(4-chloro-phenyl)-4-methyl-thiazole-5-carboxylic acid 3,4-dichloro-benzylamide
—— 2-(tert-Butyl)-5-[5-(2,4-difluorophenyl)-4,5-diazatricyclo[5.2.1.02,6]deca-2(6),3-dien-3yl]-1,3,4-thiadiazole 1024003-83-5 C20H20F2N4S
2-(tert-Butyl)-5-[5-(2,4-difluorophenyl)-4,5-diazatricyclo[5.2.1.02,6]deca-2(6),3-dien-3yl]-1,3,4-thiadiazole
—— 1-({4-[5-methyl-3-(trifluoromethyl)-4,5,6,7-tetrahydro-1H-pyrazolo[4,3-c]pyridin-1-yl]phenyl}methyl)-2-pyrrolidinone 1022930-55-7 C19H21F3N4O
1-({4-[5-methyl-3-(trifluoromethyl)-4,5,6,7-tetrahydro-1H-pyrazolo[4,3-c]pyridin-1-yl]phenyl}methyl)-2-pyrrolidinone
—— N,N'-(Pyridine-2,6-diylbis(methylene))bis(5-p-tolyl-1H-pyrazol-3-amine) 1028363-55-4 C27H27N7
N,N'-(Pyridine-2,6-diylbis(methylene))bis(5-p-tolyl-1H-pyrazol-3-amine)
—— N-(5-(thiophen-2-yl)-1H-pyrazol-3-yl)-N'-(5-p-tolyl-1H-pyrazol-3-yl)ethane-1,2-diamine 1028363-12-3 C19H20N6S
N-(5-(thiophen-2-yl)-1H-pyrazol-3-yl)-N'-(5-p-tolyl-1H-pyrazol-3-yl)ethane-1,2-diamine
—— N5-(3,3-Dimethyl-2-oxobutyl)-3-(2,4-difluorophenyl)-3,4-diazatricyclo[5.2.1.02,6]deca-2(6),4-dien-5-carboxamide 1024003-97-1 C21H23F2N3O2
N5-(3,3-Dimethyl-2-oxobutyl)-3-(2,4-difluorophenyl)-3,4-diazatricyclo[5.2.1.02,6]deca-2(6),4-dien-5-carboxamide
—— 1-[5-(2,4-diflurophenyl)-4,5-diazatricyclo[5.2.1.0(2,6)]deca-2(6),3-dien-3-yl]-3,3,-dimethyl-1-butanol 1024003-64-2 C20H24F2N2O
1-[5-(2,4-diflurophenyl)-4,5-diazatricyclo[5.2.1.0(2,6)]deca-2(6),3-dien-3-yl]-3,3,-dimethyl-1-butanol
—— 1-({4-[3-(trifluoromethyl)-4,5,6,7-tetrahydro-1H-pyrazolo[4,3-c]pyridin-1-yl]phenyl}methyl)-2-pyrrolidinone 1022930-67-1 C18H19F3N4O
1-({4-[3-(trifluoromethyl)-4,5,6,7-tetrahydro-1H-pyrazolo[4,3-c]pyridin-1-yl]phenyl}methyl)-2-pyrrolidinone
—— 2-[5-(2,4-Difluorophenyl)-4,5-diazatricyclo[5.2.1.02,6]deca-2(6),3-dien-3yl]-4-phenyl-1,3-thiazole 1024004-39-4 C23H17F2N3S
2-[5-(2,4-Difluorophenyl)-4,5-diazatricyclo[5.2.1.02,6]deca-2(6),3-dien-3yl]-4-phenyl-1,3-thiazole
—— N-(tetrahydro-2-furanylmethyl)-4-[3-(trifluoromethyl)-6,7-dihydropyrano[4,3-c]pyrazol-1(4H)-yl]benzenesulfonamide 1022931-04-9 C18H20F3N3O4S
N-(tetrahydro-2-furanylmethyl)-4-[3-(trifluoromethyl)-6,7-dihydropyrano[4,3-c]pyrazol-1(4H)-yl]benzenesulfonamide
—— 4-(2-phenylethyl)-1H-imidazol-2-amine 1033822-52-4 C11H13N3
4-(2-phenylethyl)-1H-imidazol-2-amine
—— 1-({2-fluoro-4-[3-(trifluoromethyl)-4,5,6,7-tetrahydro-1H-pyrazolo[3,4-c]pyridin-1-yl]phenyl}methyl)-2-pyrrolidinone hydrochloride 1022931-13-0 C18H18F4N4O*ClH
1-({2-fluoro-4-[3-(trifluoromethyl)-4,5,6,7-tetrahydro-1H-pyrazolo[3,4-c]pyridin-1-yl]phenyl}methyl)-2-pyrrolidinone hydrochloride
—— N-({4-[3-(trifluoromethyl)-4,7-dihydropyrano[3,4-c]pyrazol-1(5H)-yl]phenyl}methyl)methanesulfonamide 1022930-90-0 C15H16F3N3O3S
N-({4-[3-(trifluoromethyl)-4,7-dihydropyrano[3,4-c]pyrazol-1(5H)-yl]phenyl}methyl)methanesulfonamide
—— 4-chloro-6-(2-pyrazol-1-yl-benzylamino)-2H-phthalazin-1-one 1028336-77-7 C18H14ClN5O
4-chloro-6-(2-pyrazol-1-yl-benzylamino)-2H-phthalazin-1-one
—— 2-chloro-4-formylimidazole 944900-99-6 C4H3ClN2O
2-chloro-4-formylimidazole
—— 2-(6-chloro-2-(4-(3-hydroxypropoxy)phenyl)imidazol[1,2-a]pyridin-3-yl)-N,N-diethylacetamide 1009080-40-3 C22H26ClN3O3
2-(6-chloro-2-(4-(3-hydroxypropoxy)phenyl)imidazol[1,2-a]pyridin-3-yl)-N,N-diethylacetamide
—— 7-phenyl-1-(2-phenyl-2H-tetrazol-5-yl)-heptan-1-one 1042153-47-8 C20H22N4O
7-phenyl-1-(2-phenyl-2H-tetrazol-5-yl)-heptan-1-one
—— N-adamantan-2-yl-4-[3-(4-chloro-phenyl)-[1,2,4]oxadiazol-5-yl]-3,3-dimethyl-butyramide 1034144-09-6 C24H30ClN3O2
N-adamantan-2-yl-4-[3-(4-chloro-phenyl)-[1,2,4]oxadiazol-5-yl]-3,3-dimethyl-butyramide
—— 2-(6-chloro-2-(4-(3-[18F]fluoropropoxy)phenyl)imidazo[1,2-a]pyridin-3-yl)-N,N-diethylacetamide 1009080-75-4 C22H25ClFN3O2
2-(6-chloro-2-(4-(3-[18F]fluoropropoxy)phenyl)imidazo[1,2-a]pyridin-3-yl)-N,N-diethylacetamide
—— 4-chloro-6-(3-pyrazol-1-yl-benzylamino)-2H-phthalazin-1-one 1028336-78-8 C18H14ClN5O
4-chloro-6-(3-pyrazol-1-yl-benzylamino)-2H-phthalazin-1-one
—— Cuprous Imidazolide 945662-18-0 C3H3N2*Cu
Cuprous Imidazolide
—— 3-[[(2,4-dichlorophenyl)carbonyl]-(1-methylethyl)amino]-5-(4-imidazo[2,1-b][1,3]thiazol-6-ylphenyl)-2-thiophenecarboxylic acid 1019337-35-9 C26H19Cl2N3O3S2
3-[[(2,4-dichlorophenyl)carbonyl]-(1-methylethyl)amino]-5-(4-imidazo[2,1-b][1,3]thiazol-6-ylphenyl)-2-thiophenecarboxylic acid
—— 2-(3-hydroxyphenylamino)-9-(2-methoxyphenyl)-8-oxo-8,9-dihydro-7H-purine-6-carboxamide 1022155-71-0 C19H16N6O4
2-(3-hydroxyphenylamino)-9-(2-methoxyphenyl)-8-oxo-8,9-dihydro-7H-purine-6-carboxamide
—— (2S)-ethoxy-3-{4-[2-(5-methyl-2-phenyl-oxazol-4-yl)-ethoxy]-phenyl}-propanoic acid 1048667-76-0 C23H25NO5
(2S)-ethoxy-3-{4-[2-(5-methyl-2-phenyl-oxazol-4-yl)-ethoxy]-phenyl}-propanoic acid
—— 3-{[(4-chloro-2-fluorophenyl)carbonyl]-[1-methyl-2-(methyloxy)ethyl]amino}-5-(4-pyrazolo[1,5-a]pyrimidin-2-ylphenyl)-2-thiophenecarboxylic acid 1019337-60-0 C28H22ClFN4O4S
3-{[(4-chloro-2-fluorophenyl)carbonyl]-[1-methyl-2-(methyloxy)ethyl]amino}-5-(4-pyrazolo[1,5-a]pyrimidin-2-ylphenyl)-2-thiophenecarboxylic acid
—— 3-(4-chloro-3-fluorophenyl)-N-propyl-3H-imidazo[4,5-b]pyridine-2-carboxamide 1622208-16-5 C16H14ClFN4O
3-(4-chloro-3-fluorophenyl)-N-propyl-3H-imidazo[4,5-b]pyridine-2-carboxamide
—— 2-(3-hydroxyphenylamino)-9-(2-methoxyphenyl)-9H-purine-6-carboxamide 1022155-81-2 C19H16N6O3
2-(3-hydroxyphenylamino)-9-(2-methoxyphenyl)-9H-purine-6-carboxamide
—— 3-{[(2,4-dichlorophenyl)carbonyl]-[2-(methyloxy)ethyl]amino}-5-(4-pyrazolo[1,5-a]pyrimidin-2-ylphenyl)-2-thiophenecarboxylic acid 1019337-51-9 C27H20Cl2N4O4S
3-{[(2,4-dichlorophenyl)carbonyl]-[2-(methyloxy)ethyl]amino}-5-(4-pyrazolo[1,5-a]pyrimidin-2-ylphenyl)-2-thiophenecarboxylic acid
—— 1-(4-fluorophenyl)-6-methyl-1H-indazol-4-amine 1020153-96-1 C14H12FN3
1-(4-fluorophenyl)-6-methyl-1H-indazol-4-amine
—— 3-[{[2-fluoro-4-(trifluoromethyl)phenyl]carbonyl}-(1-methylethyl)amino]-5-(4-pyrazolo[1,5-a]pyrimidin-2-ylphenyl)-2-thiophenecarboxylic acid 1019337-45-1 C28H20F4N4O3S
3-[{[2-fluoro-4-(trifluoromethyl)phenyl]carbonyl}-(1-methylethyl)amino]-5-(4-pyrazolo[1,5-a]pyrimidin-2-ylphenyl)-2-thiophenecarboxylic acid
—— 3-{[(4-chloro-2-fluorophenyl)carbonyl]-[2-(methyloxy)ethyl]amino}-5-(4-pyrazolo[1,5-a]pyrimidin-2-ylphenyl)-2-thiophenecarboxylic acid 1019337-49-5 C27H20ClFN4O4S
3-{[(4-chloro-2-fluorophenyl)carbonyl]-[2-(methyloxy)ethyl]amino}-5-(4-pyrazolo[1,5-a]pyrimidin-2-ylphenyl)-2-thiophenecarboxylic acid
—— (2S)-ethoxy-3-{4-[5-methyl-2-phenyl-oxazol-4-yl-methoxy]-phenyl}-propanoic acid 1048667-75-9 C22H23NO5
(2S)-ethoxy-3-{4-[5-methyl-2-phenyl-oxazol-4-yl-methoxy]-phenyl}-propanoic acid
—— {4-[6-(2.5-difluoro-benzylamino)-imidazo[1,2-b]pyridazin-3-yl]-phenyl}-(4-methyl-piperazin-1-yl)-methanone 1022981-52-7 C25H24F2N6O
{4-[6-(2.5-difluoro-benzylamino)-imidazo[1,2-b]pyridazin-3-yl]-phenyl}-(4-methyl-piperazin-1-yl)-methanone
—— 6-methyl-1-phenyl-1H-indazole-4-amine 913002-95-6 C14H13N3
6-methyl-1-phenyl-1H-indazole-4-amine
—— [<sup>18</sup>F]-2-methyl-4-(morpholine-4-carbonyl)-2H-pyrazole-3-carboxylic acid {2-[3-(2-fluoroethoxy)phenyl]-[1,2,4]triazolo[1,5-a]pyridin-7-yl}amide 1621268-48-1 C24H24FN7O4
[<sup>18</sup>F]-2-methyl-4-(morpholine-4-carbonyl)-2H-pyrazole-3-carboxylic acid {2-[3-(2-fluoroethoxy)phenyl]-[1,2,4]triazolo[1,5-a]pyridin-7-yl}amide