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中文名称 英文名称 CAS号 化学式 结构式图片
—— N-(5-(1,4-diazepan-1-yl)-1-methyl-1H-pyrazol-4-yl)-5-amino-2-(2,6-difluorophenyl)thiazole-4-carboxamide 1338715-44-8 C19H21F2N7OS
N-(5-(1,4-diazepan-1-yl)-1-methyl-1H-pyrazol-4-yl)-5-amino-2-(2,6-difluorophenyl)thiazole-4-carboxamide
—— 2-carbamoyloxymethyl-3-methyl-5-nitro-3<i>H</i>-imidazole-4-carbonitrile 41605-10-1 C7H7N5O4
2-carbamoyloxymethyl-3-methyl-5-nitro-3<i>H</i>-imidazole-4-carbonitrile
—— M-4-NImOH 14953-66-3 C5H7N3O3
M-4-NImOH
—— 2-(4-Fluoro-phenyl)-5-isopropyl-4-thiophen-3-yl-1H-imidazole 113399-12-5 C16H15FN2S
2-(4-Fluoro-phenyl)-5-isopropyl-4-thiophen-3-yl-1H-imidazole
—— 1-Methyl-2-hydroxymethyl-4-nitro-5-methylsulfonylimidazol 41605-00-9 C6H9N3O5S
1-Methyl-2-hydroxymethyl-4-nitro-5-methylsulfonylimidazol
—— 5-(3-chloro-4-methoxyphenyl)-1-(3,4,5-trimethoxyphenyl)-1H-tetrazole 1352545-25-5 C17H17ClN4O4
5-(3-chloro-4-methoxyphenyl)-1-(3,4,5-trimethoxyphenyl)-1H-tetrazole
—— 3-(Piperidinopropoxy)-1-(alpha,alpha,alpha-trifluoro-m-tolyl)-1H-indazole 26660-66-2 C22H24F3N3O
3-(Piperidinopropoxy)-1-(alpha,alpha,alpha-trifluoro-m-tolyl)-1H-indazole
—— 5-amino-N-(5-((2R,4R,5S,6R)-4-amino-5-hydroxy-5,6-dimethyltetrahydro-2H-pyran-2-yl)-1-methyl-1H-pyrazol-4-yl)-2-(2,6-difluorophenyl)thiazole-4-carboxamide 1586041-82-8 C21H24F2N6O3S
5-amino-N-(5-((2R,4R,5S,6R)-4-amino-5-hydroxy-5,6-dimethyltetrahydro-2H-pyran-2-yl)-1-methyl-1H-pyrazol-4-yl)-2-(2,6-difluorophenyl)thiazole-4-carboxamide
—— 5-amino-2-(2,6-difluorophenyl)-N-[5-(3,4-dihydro-2H-pyran-6-yl)-1-methyl-pyrazol-4-yl]thiazole-4-carboxamide 1586039-48-6 C19H17F2N5O2S
5-amino-2-(2,6-difluorophenyl)-N-[5-(3,4-dihydro-2H-pyran-6-yl)-1-methyl-pyrazol-4-yl]thiazole-4-carboxamide
—— 5-amino-N-(5-((4S,5R)-4-amino-5-hydroxyazepan-1-yl)-1-methyl-1H-pyrazol-4-yl)-2-(2,6-difluorophenyl)thiazole-4-carboxamide 1428571-51-0 C20H23F2N7O2S
5-amino-N-(5-((4S,5R)-4-amino-5-hydroxyazepan-1-yl)-1-methyl-1H-pyrazol-4-yl)-2-(2,6-difluorophenyl)thiazole-4-carboxamide
—— 1-methyl-4-(naphthalen-2-yl)-5-(3,4,5-trimethoxyphenyl)-1H-imidazole 1111266-65-9 C23H22N2O3
1-methyl-4-(naphthalen-2-yl)-5-(3,4,5-trimethoxyphenyl)-1H-imidazole
—— 7-methoxy-3-(4-methoxyphenyl)-1H-benzofuro[3,2-c]pyrazole 1341184-96-0 C17H14N2O3
7-methoxy-3-(4-methoxyphenyl)-1H-benzofuro[3,2-c]pyrazole
—— 5-amino-N-(5-(5-amino-3-methoxyazepan-1-yl)-1-methyl-1H-pyrazol-4-yl)-2-(2,6-difluorophenyl)thiazole-4-carboxamide 1428570-65-3 C21H25F2N7O2S
5-amino-N-(5-(5-amino-3-methoxyazepan-1-yl)-1-methyl-1H-pyrazol-4-yl)-2-(2,6-difluorophenyl)thiazole-4-carboxamide
—— (S)-5-amino-N-(5-(4-aminoazepan-1-yl)-1-methyl-1H-pyrazol-4-yl)-2-(2,6-difluorophenyl)thiazole-4-carboxamide 1338715-19-7 C20H23F2N7OS
(S)-5-amino-N-(5-(4-aminoazepan-1-yl)-1-methyl-1H-pyrazol-4-yl)-2-(2,6-difluorophenyl)thiazole-4-carboxamide
—— R-5-amino-N-(5-(4-aminoazepan-1-yl)-1-methyl-1H-pyrazol-4-yl)-2-(2,6-difluorophenyl)thiazole-4-carboxamide 1338715-21-1 C20H23F2N7OS
R-5-amino-N-(5-(4-aminoazepan-1-yl)-1-methyl-1H-pyrazol-4-yl)-2-(2,6-difluorophenyl)thiazole-4-carboxamide
—— 1-Methyl-2-acetoxymethyl-4-nitroimidazol 41604-87-9 C7H9N3O4
1-Methyl-2-acetoxymethyl-4-nitroimidazol
—— 5-amino-2-(2,6-difluorophenyl)-N-(1-methyl-5-(4-((methylamino)methyl)piperidin-1-yl)-1H-pyrazol-4-yl)thiazole-4-carboxamide 1428569-43-0 C21H25F2N7OS
5-amino-2-(2,6-difluorophenyl)-N-(1-methyl-5-(4-((methylamino)methyl)piperidin-1-yl)-1H-pyrazol-4-yl)thiazole-4-carboxamide
—— tert-butyl {(3S)-1-[5-({[5-[(tert-butoxycarbonyl)amino]-2-(2,6-difluorophenyl)-1,3-thiazol-4-yl]carbonyl}amino)-2,3-dihydrofuro[2,3-b]pyridin-4-yl]piperidin-3-yl}carbamate 1620011-30-4 C32H38F2N6O6S
tert-butyl {(3S)-1-[5-({[5-[(tert-butoxycarbonyl)amino]-2-(2,6-difluorophenyl)-1,3-thiazol-4-yl]carbonyl}amino)-2,3-dihydrofuro[2,3-b]pyridin-4-yl]piperidin-3-yl}carbamate
—— (S)-5-amino-N-(4-(3-aminopiperidin-1-yl)pyridin-3-yl)-2-(2,6-difluorophenyl)thiazole-4-carboxamide 1187055-13-5 C20H20F2N6OS
(S)-5-amino-N-(4-(3-aminopiperidin-1-yl)pyridin-3-yl)-2-(2,6-difluorophenyl)thiazole-4-carboxamide
—— 5-amino-N-{4-[(3S)-3-aminopiperidin-1-yl]-2,3-dihydrofuro[2,3-b]pyridin-5-yl}-2-(2,6-difluorophenyl)-1,3-thiazole-4-carboxamide 1620011-24-6 C22H22F2N6O2S
5-amino-N-{4-[(3S)-3-aminopiperidin-1-yl]-2,3-dihydrofuro[2,3-b]pyridin-5-yl}-2-(2,6-difluorophenyl)-1,3-thiazole-4-carboxamide
—— 5-amino-N-{4-[(3S,5R)-3-amino-5-(trifluoromethyl)piperidin-1-yl]-2,3-dihydrofuro[2,3-b]pyridin-5-yl}-2-(2,6-difluorophenyl)-1,3-thiazole-4-carboxamide 1620012-49-8 C23H21F5N6O2S
5-amino-N-{4-[(3S,5R)-3-amino-5-(trifluoromethyl)piperidin-1-yl]-2,3-dihydrofuro[2,3-b]pyridin-5-yl}-2-(2,6-difluorophenyl)-1,3-thiazole-4-carboxamide
—— 5-amino-2-(2,6-difluorophenyl)-N-(1-methyl-5-tetrahydropyran-2-yl-pyrazol-4-yl)thiazole-4-carboxamide 1586039-50-0 C19H19F2N5O2S
5-amino-2-(2,6-difluorophenyl)-N-(1-methyl-5-tetrahydropyran-2-yl-pyrazol-4-yl)thiazole-4-carboxamide
—— 2-(4-Fluoro-phenyl)-5-propyl-4-thiophen-3-yl-1H-imidazole 113399-11-4 C16H15FN2S
2-(4-Fluoro-phenyl)-5-propyl-4-thiophen-3-yl-1H-imidazole
—— 5-amino-2-(2,6-difluorophenyl)-N-(5-morpholinoisothiazol-4-yl)thiazole-4-carboxamide 1422394-36-2 C17H15F2N5O2S2
5-amino-2-(2,6-difluorophenyl)-N-(5-morpholinoisothiazol-4-yl)thiazole-4-carboxamide
—— 5-Cyclohexyl-2-(4-fluoro-phenyl)-4-thiophen-3-yl-1H-imidazole 113399-18-1 C19H19FN2S
5-Cyclohexyl-2-(4-fluoro-phenyl)-4-thiophen-3-yl-1H-imidazole
—— tert-butyl 2-(2,6-difluorophenyl)-4-(5-(2-ethoxytetrahydro-2H-pyran-2-yl)-1-methyl-1H-pyrazol-4-ylcarbamoyl)thiazol-5-ylcarbamate 1586046-34-5 C26H31F2N5O5S
tert-butyl 2-(2,6-difluorophenyl)-4-(5-(2-ethoxytetrahydro-2H-pyran-2-yl)-1-methyl-1H-pyrazol-4-ylcarbamoyl)thiazol-5-ylcarbamate
—— 5-amino-N-(5-((1S,4S,5S)-4-amino-8-oxabicyclo[3.2.1]octan-1-yl)-1-methyl-1H-pyrazol-4-yl)-2-(2,6-difluorophenyl)thiazole-4-carboxamide 1586039-62-4 C21H22F2N6O2S
5-amino-N-(5-((1S,4S,5S)-4-amino-8-oxabicyclo[3.2.1]octan-1-yl)-1-methyl-1H-pyrazol-4-yl)-2-(2,6-difluorophenyl)thiazole-4-carboxamide
—— 5-amino-N-(5-(4-amino-3-fluoroazepan-1-yl)-1-methyl-1H-pyrazol-4-yl)-2-(2,6-difluorophenyl)thiazole-4-carboxamide 1428573-61-8 C20H22F3N7OS
5-amino-N-(5-(4-amino-3-fluoroazepan-1-yl)-1-methyl-1H-pyrazol-4-yl)-2-(2,6-difluorophenyl)thiazole-4-carboxamide
—— 2-(4-fluorophenyl)-5-(3-thienyl)oxazole 113398-97-3 C13H8FNOS
2-(4-fluorophenyl)-5-(3-thienyl)oxazole
—— 5-Butyl-2-(4-fluoro-phenyl)-4-thiophen-3-yl-1H-imidazole 113399-13-6 C17H17FN2S
5-Butyl-2-(4-fluoro-phenyl)-4-thiophen-3-yl-1H-imidazole
—— 5-amino-N-(5-(4-aminoazepan-1-yl)-1-ethyl-1H-pyrazol-4-yl)-2-(2,6-difluorophenyl)thiazole-4-carboxamide 1338716-13-4 C21H25F2N7OS
5-amino-N-(5-(4-aminoazepan-1-yl)-1-ethyl-1H-pyrazol-4-yl)-2-(2,6-difluorophenyl)thiazole-4-carboxamide
—— tert-butyl 2-(2,6-difluorophenyl)-4-(5-(4-hydroxy-5-(2,2,2-trifluoroacetamido)azepan-1-yl)-1-methyl-1H-pyrazol-4-ylcarbamoyl)thiazol-5-ylcarbamate 1428576-67-3 C27H30F5N7O5S
tert-butyl 2-(2,6-difluorophenyl)-4-(5-(4-hydroxy-5-(2,2,2-trifluoroacetamido)azepan-1-yl)-1-methyl-1H-pyrazol-4-ylcarbamoyl)thiazol-5-ylcarbamate
—— tert-butyl N-[6-[4-[[5-(tert-butoxycarbonylamino)-2-(2,6-difluorophenyl)thiazole-4-carbonyl]amino]-2-methyl-pyrazol-3-yl]oxepan-3-yl]carbamate 1586043-89-1 C30H38F2N6O6S
tert-butyl N-[6-[4-[[5-(tert-butoxycarbonylamino)-2-(2,6-difluorophenyl)thiazole-4-carbonyl]amino]-2-methyl-pyrazol-3-yl]oxepan-3-yl]carbamate
—— tert-butyl 4-(5-chloro-1-methyl-1H-pyrazol-4-ylcarbamoyl)-2-(2,6-difluorophenyl)thiazol-5-ylcarbamate 1586042-47-8 C19H18ClF2N5O3S
tert-butyl 4-(5-chloro-1-methyl-1H-pyrazol-4-ylcarbamoyl)-2-(2,6-difluorophenyl)thiazol-5-ylcarbamate
—— 2-(4-Fluoro-phenyl)-5-methyl-4-thiophen-3-yl-1H-imidazole 113399-08-9 C14H11FN2S
2-(4-Fluoro-phenyl)-5-methyl-4-thiophen-3-yl-1H-imidazole
—— 5-amino-N-(5-((4S,5R)-4-amino-5-fluoroazepan-1-yl)-1-methyl-1H-pyrazol-4-yl)-2-(2,6-difluorophenyl)thiazole-4-carboxamide 1428569-93-0 C20H22F3N7OS
5-amino-N-(5-((4S,5R)-4-amino-5-fluoroazepan-1-yl)-1-methyl-1H-pyrazol-4-yl)-2-(2,6-difluorophenyl)thiazole-4-carboxamide
—— 5-amino-2-(2,6-difluorophenyl)-N-[5-(2-methoxytetrahydropyran-2-yl)-1-methyl-pyrazol-4-yl]thiazole-4-carboxamide 1586039-49-7 C20H21F2N5O3S
5-amino-2-(2,6-difluorophenyl)-N-[5-(2-methoxytetrahydropyran-2-yl)-1-methyl-pyrazol-4-yl]thiazole-4-carboxamide
—— tert-butyl (1-(4-(5-amino-2-(2,6-difluorophenyl)thiazole-4-carboxamido)isothiazol-5-yl)piperidin-3-yl)carbamate 1422394-44-2 C23H26F2N6O3S2
tert-butyl (1-(4-(5-amino-2-(2,6-difluorophenyl)thiazole-4-carboxamido)isothiazol-5-yl)piperidin-3-yl)carbamate
—— 5-amino-2-(2,6-difluorophenyl)-N-[5-(3,6-dihydro-2H-pyran-4-yl)-1-methyl-pyrazol-4-yl]thiazole-4-carboxamide 1586039-47-5 C19H17F2N5O2S
5-amino-2-(2,6-difluorophenyl)-N-[5-(3,6-dihydro-2H-pyran-4-yl)-1-methyl-pyrazol-4-yl]thiazole-4-carboxamide
—— N-(5-((2S,5R,6S)-5-amino-6-fluorooxepan-2-yl)-1-methyl-1H-pyrazol-4-yl)-2-(2,6-difluorophenyl)thiazole-4-carboxamide 1586041-58-8 C20H20F3N5O2S
N-(5-((2S,5R,6S)-5-amino-6-fluorooxepan-2-yl)-1-methyl-1H-pyrazol-4-yl)-2-(2,6-difluorophenyl)thiazole-4-carboxamide
—— tert-butyl 2-(2,6-difluorophenyl)-4-(5-(4-fluoro-5-(2,2,2-trifluoroacetamido)azepan-1-yl)-1-methyl-1H-pyrazol-4-ylcarbamoyl)thiazol-5-ylcarbamate 1428576-48-0 C27H29F6N7O4S
tert-butyl 2-(2,6-difluorophenyl)-4-(5-(4-fluoro-5-(2,2,2-trifluoroacetamido)azepan-1-yl)-1-methyl-1H-pyrazol-4-ylcarbamoyl)thiazol-5-ylcarbamate
—— 5-amino-2-(2,6-difluorophenyl)-N-(5-(3-hydroxypiperidin-1-yl)isothiazol-4-yl)thiazole-4-carboxamide 1422394-97-5 C18H17F2N5O2S2
5-amino-2-(2,6-difluorophenyl)-N-(5-(3-hydroxypiperidin-1-yl)isothiazol-4-yl)thiazole-4-carboxamide
—— 5-amino-N-(5-((4S,5S)-4-amino-5-hydroxy-4-methylazepan-1-yl)-1-methyl-1H-pyrazol-4-yl)-2-(2,6-difluorophenyl)thiazole-4-carboxamide 1428572-47-7 C21H25F2N7O2S
5-amino-N-(5-((4S,5S)-4-amino-5-hydroxy-4-methylazepan-1-yl)-1-methyl-1H-pyrazol-4-yl)-2-(2,6-difluorophenyl)thiazole-4-carboxamide
—— tert-butyl 2-(2,6-difluorophenyl)-4-(5-(4-hydroxy-4-methylazepan-1-yl)-1-methyl-1H-pyrazol-4-ylcarbamoyl)thiazol-5-ylcarbamate 1428576-47-9 C26H32F2N6O4S
tert-butyl 2-(2,6-difluorophenyl)-4-(5-(4-hydroxy-4-methylazepan-1-yl)-1-methyl-1H-pyrazol-4-ylcarbamoyl)thiazol-5-ylcarbamate
—— tert-butyl 2-(2,6-difluorophenyl)-4-(1-ethyl-5-(4-(2,2,2-trifluoroacetamido)azepan-1-yl)-1H-pyrazol-4-ylcarbamoyl)thiazol-5-ylcarbamate 1338718-53-8 C28H32F5N7O4S
tert-butyl 2-(2,6-difluorophenyl)-4-(1-ethyl-5-(4-(2,2,2-trifluoroacetamido)azepan-1-yl)-1H-pyrazol-4-ylcarbamoyl)thiazol-5-ylcarbamate
—— N-(5-morpholinoisothiazol-4-yl)-2-phenyloxazole-4-carboxamide 1422394-59-9 C17H16N4O3S
N-(5-morpholinoisothiazol-4-yl)-2-phenyloxazole-4-carboxamide
—— N-(5-morpholinoisothiazol-4-yl)-2-(pyridin-4-yl)thiazole-4-carboxamide 1422394-48-6 C16H15N5O2S2
N-(5-morpholinoisothiazol-4-yl)-2-(pyridin-4-yl)thiazole-4-carboxamide
—— 2-morpholino-N-(5-morpholinoisothiazol-4-yl)thiazole-4-carboxamide 1422394-53-3 C15H19N5O3S2
2-morpholino-N-(5-morpholinoisothiazol-4-yl)thiazole-4-carboxamide
—— methyl 5-[(tert-butoxycarbonyl)amino]-2-(2,6-difluorophenyl)-1,3-thiazole-4-carboxylate 1620011-01-9 C16H16F2N2O4S
methyl 5-[(tert-butoxycarbonyl)amino]-2-(2,6-difluorophenyl)-1,3-thiazole-4-carboxylate
—— N-(5-morpholinoisothiazol-4-yl)-2-(piperidin-1-yl)thiazole-4-carboxamide 1422394-52-2 C16H21N5O2S2
N-(5-morpholinoisothiazol-4-yl)-2-(piperidin-1-yl)thiazole-4-carboxamide