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—— (S)-2-(tert-butoxy)-2-(2-((3,3-dimethylbutyl)carbamoyl)-7-(4,4-dimethylpiperidin-1-yl)-5-methylpyrazolo[1,5-a]pyrimidin-6-yl)acetic acid 1423742-64-6 C27H43N5O4
(S)-2-(tert-butoxy)-2-(2-((3,3-dimethylbutyl)carbamoyl)-7-(4,4-dimethylpiperidin-1-yl)-5-methylpyrazolo[1,5-a]pyrimidin-6-yl)acetic acid
—— ethyl 6-((S)-1-(tert-butoxy)-2-ethoxy-2-oxoethyl)-7-(5-chloro-3,4-dihydro-2H-benzo[b][1,4]oxazin-6-yl)-5-methylpyrazolo[1,5-a]pyrimidine-2-carboxylate 1423742-77-1 C26H31ClN4O6
ethyl 6-((S)-1-(tert-butoxy)-2-ethoxy-2-oxoethyl)-7-(5-chloro-3,4-dihydro-2H-benzo[b][1,4]oxazin-6-yl)-5-methylpyrazolo[1,5-a]pyrimidine-2-carboxylate
—— (2S)-2-(tert-butoxy)-2-(7-(5-chloro-3,4-dihydro-2H-benzo[b][1,4]oxazin-6-yl)-2-((4-fluoro-3-methylbenzyl)carbamoyl)-5-methylpyrazolo[1,5-a]pyrimidin-6-yl)acetic acid 1423742-53-3 C30H31ClFN5O5
(2S)-2-(tert-butoxy)-2-(7-(5-chloro-3,4-dihydro-2H-benzo[b][1,4]oxazin-6-yl)-2-((4-fluoro-3-methylbenzyl)carbamoyl)-5-methylpyrazolo[1,5-a]pyrimidin-6-yl)acetic acid
—— (2S)-2-(tert-butoxy)-2-(7-(7-fluoro-3,4-dihydro-2H-benzo[b][1,4]oxazin-6-yl)-2-((4-fluoro-3-methylbenzyl)carbamoyl)-5-methylpyrazolo[1,5-a]pyrimidin-6-yl)acetic acid 1423742-57-7 C30H31F2N5O5
(2S)-2-(tert-butoxy)-2-(7-(7-fluoro-3,4-dihydro-2H-benzo[b][1,4]oxazin-6-yl)-2-((4-fluoro-3-methylbenzyl)carbamoyl)-5-methylpyrazolo[1,5-a]pyrimidin-6-yl)acetic acid
—— 6-((S)-1-(tert-butoxy)-2-ethoxy-2-oxoethyl)-7-(7-fluoro-3,4-dihydro-2H-benzo[b][1,4]oxazin-6-yl)-5-methylpyrazolo[1,5-a]pyrimidine-2-carboxylic acid 1423742-80-6 C24H27FN4O6
6-((S)-1-(tert-butoxy)-2-ethoxy-2-oxoethyl)-7-(7-fluoro-3,4-dihydro-2H-benzo[b][1,4]oxazin-6-yl)-5-methylpyrazolo[1,5-a]pyrimidine-2-carboxylic acid
—— (S,E)-ethyl 6-(1-(tert-butoxy)-2-ethoxy-2-oxoethyl)-5-methyl-7-(4-methylpent-1-en-1-yl)pyrazolo[1,5-a]pyrimidine-2-carboxylate 1423742-83-9 C24H35N3O5
(S,E)-ethyl 6-(1-(tert-butoxy)-2-ethoxy-2-oxoethyl)-5-methyl-7-(4-methylpent-1-en-1-yl)pyrazolo[1,5-a]pyrimidine-2-carboxylate
—— ethyl 6-((S)-1-(tert-butoxy)-2-ethoxy-2-oxoethyl)-7-(7-fluoro-3,4-dihydro-2H-benzo[b][1,4]oxazin-6-yl)-5-methylpyrazolo[1,5-a]pyrimidine-2-carboxylate 1423742-79-3 C26H31FN4O6
ethyl 6-((S)-1-(tert-butoxy)-2-ethoxy-2-oxoethyl)-7-(7-fluoro-3,4-dihydro-2H-benzo[b][1,4]oxazin-6-yl)-5-methylpyrazolo[1,5-a]pyrimidine-2-carboxylate
—— (S,E)-6-(1-(tert-butoxy)-2-ethoxy-2-oxoethyl)-5-methyl-7-(4-methylpent-1-en-1-yl)pyrazolo[1,5-a]pyrimidine-2-carboxylic acid 1423742-84-0 C22H31N3O5
(S,E)-6-(1-(tert-butoxy)-2-ethoxy-2-oxoethyl)-5-methyl-7-(4-methylpent-1-en-1-yl)pyrazolo[1,5-a]pyrimidine-2-carboxylic acid
—— (2S)-2-(tert-butoxy)-2-(7-(5-chloro-3,4-dihydro-2H-benzo[b][1,4]oxazin-6-yl)-2-((3,3-dimethylbutyl)carbamoyl)-5-methylpyrazolo[1,5-a]pyrimidin-6-yl)acetic acid 1423742-56-6 C28H36ClN5O5
(2S)-2-(tert-butoxy)-2-(7-(5-chloro-3,4-dihydro-2H-benzo[b][1,4]oxazin-6-yl)-2-((3,3-dimethylbutyl)carbamoyl)-5-methylpyrazolo[1,5-a]pyrimidin-6-yl)acetic acid
—— trans-2-trifluoromethylcyclohexane-1-carboxylic acid 161274-54-0 C8H11F3O2
trans-2-trifluoromethylcyclohexane-1-carboxylic acid
—— (2S)-2-(tert-butoxy)-2-(2-((3,3-dimethylbutyl)carbamoyl)-7-(8-fluoro-5-methylchroman-6-yl)-5-methylpyrazolo[1,5-a]pyrimidin-6-yl)acetic acid 1423741-70-1 C30H39FN4O5
(2S)-2-(tert-butoxy)-2-(2-((3,3-dimethylbutyl)carbamoyl)-7-(8-fluoro-5-methylchroman-6-yl)-5-methylpyrazolo[1,5-a]pyrimidin-6-yl)acetic acid
—— (2S)-2-(tert-butoxy)-2-(2-((cyclohexylmethyl)carbamoyl)-7-(8-fluoro-5-methylchroman-6-yl)-5-methylpyrazolo[1,5-a]pyrimidin-6-yl)acetic acid 1423741-22-3 C31H39FN4O5
(2S)-2-(tert-butoxy)-2-(2-((cyclohexylmethyl)carbamoyl)-7-(8-fluoro-5-methylchroman-6-yl)-5-methylpyrazolo[1,5-a]pyrimidin-6-yl)acetic acid
—— (2S)-2-(tert-butoxy)-2-(7-(8-fluoro-5-methylchroman-6-yl)-2-(isopentylcarbamoyl)-5-methylpyrazolo[1,5-a]pyrimidin-6-yl)acetic acid 1423741-57-4 C29H37FN4O5
(2S)-2-(tert-butoxy)-2-(7-(8-fluoro-5-methylchroman-6-yl)-2-(isopentylcarbamoyl)-5-methylpyrazolo[1,5-a]pyrimidin-6-yl)acetic acid
—— (2S)-2-(tert-butoxy)-2-(7-(8-fluoro-5-methylchroman-6-yl)-5-methyl-2-((2-morpholinoethyl)carbamoyl)pyrazolo[1,5-a]pyrimidin-6-yl)acetic acid 1423741-96-1 C30H38FN5O6
(2S)-2-(tert-butoxy)-2-(7-(8-fluoro-5-methylchroman-6-yl)-5-methyl-2-((2-morpholinoethyl)carbamoyl)pyrazolo[1,5-a]pyrimidin-6-yl)acetic acid
—— (2S)-2-(tert-butoxy)-2-(7-(8-fluoro-5-methylchroman-6-yl)-5-methyl-2-(((tetrahydro-2H-pyran-4-yl)methyl)carbamoyl)pyrazolo[1,5-a]pyrimidin-6-yl)acetic acid 1423742-09-9 C30H37FN4O6
(2S)-2-(tert-butoxy)-2-(7-(8-fluoro-5-methylchroman-6-yl)-5-methyl-2-(((tetrahydro-2H-pyran-4-yl)methyl)carbamoyl)pyrazolo[1,5-a]pyrimidin-6-yl)acetic acid
—— (2S)-2-(tert-butoxy)-2-(7-(8-fluoro-5-methylchroman-6-yl)-5-methyl-2-((2-(tetrahydro-2H-pyran-4-yl)ethyl)carbamoyl)pyrazolo[1,5-a]pyrimidin-6-yl)acetic acid 1423742-38-4 C31H39FN4O6
(2S)-2-(tert-butoxy)-2-(7-(8-fluoro-5-methylchroman-6-yl)-5-methyl-2-((2-(tetrahydro-2H-pyran-4-yl)ethyl)carbamoyl)pyrazolo[1,5-a]pyrimidin-6-yl)acetic acid
—— (2S)-2-(tert-butoxy)-2-(2-((2-cyclohexylethyl)carbamoyl)-7-(8-fluoro-5-methylchroman-6-yl)-5-methylpyrazolo[1,5-a]pyrimidin-6-yl)acetic acid 1423742-37-3 C32H41FN4O5
(2S)-2-(tert-butoxy)-2-(2-((2-cyclohexylethyl)carbamoyl)-7-(8-fluoro-5-methylchroman-6-yl)-5-methylpyrazolo[1,5-a]pyrimidin-6-yl)acetic acid
—— (2S)-2-(tert-butoxy)-2-(2-((4-fluoro-2-(1H-1,2,4-triazol-1-yl)benzyl)carbamoyl)-7-(8-fluoro-5-methylchroman-6-yl)-5-methylpyrazolo[1,5-a]pyrimidin-6-yl)acetic acid 1423741-17-6 C33H33F2N7O5
(2S)-2-(tert-butoxy)-2-(2-((4-fluoro-2-(1H-1,2,4-triazol-1-yl)benzyl)carbamoyl)-7-(8-fluoro-5-methylchroman-6-yl)-5-methylpyrazolo[1,5-a]pyrimidin-6-yl)acetic acid
—— (2S)-2-(tert-butoxy)-2-(7-(8-fluoro-5-methylchroman-6-yl)-5-methyl-2-(propylcarbamoyl)pyrazolo[1,5-a]pyrimidin-6-yl)acetic acid 1423742-33-9 C27H33FN4O5
(2S)-2-(tert-butoxy)-2-(7-(8-fluoro-5-methylchroman-6-yl)-5-methyl-2-(propylcarbamoyl)pyrazolo[1,5-a]pyrimidin-6-yl)acetic acid
—— (2S)-2-(tert-butoxy)-2-(2-((4-fluoro-2-hydroxybenzyl)carbamoyl)-7-(8-fluoro-5-methylchroman-6-yl)-5-methylpyrazolo[1,4-a]pyrimidin-6yl)acetic acid 1423741-71-2 C31H32F2N4O6
(2S)-2-(tert-butoxy)-2-(2-((4-fluoro-2-hydroxybenzyl)carbamoyl)-7-(8-fluoro-5-methylchroman-6-yl)-5-methylpyrazolo[1,4-a]pyrimidin-6yl)acetic acid
—— (2S)-2-(tert-butoxy)-2-(2-((4-fluoro-3-methoxybenzyl)carbamoyl)-7-(8-fluoro-5-ethylchroman-6-yl)-5-methylpyrazolo[1,5-a]pyrimidin-6-yl)acetic acid 1423741-43-8 C32H34F2N4O6
(2S)-2-(tert-butoxy)-2-(2-((4-fluoro-3-methoxybenzyl)carbamoyl)-7-(8-fluoro-5-ethylchroman-6-yl)-5-methylpyrazolo[1,5-a]pyrimidin-6-yl)acetic acid
—— (2S)-2-(tert-butoxy)-2-(2-((4-fluoro-3-propylbenzyl)carbamoyl)-7-(8-fluoro-5-methylchroman-6-yl)-5-methylpyrazolo[1,5-a]pyrimidin-6-yl)acetic acid 1423741-31-4 C34H38F2N4O5
(2S)-2-(tert-butoxy)-2-(2-((4-fluoro-3-propylbenzyl)carbamoyl)-7-(8-fluoro-5-methylchroman-6-yl)-5-methylpyrazolo[1,5-a]pyrimidin-6-yl)acetic acid
—— (2S)-2-(tert-butoxy)-2-(2-((4-fluoro-2-(methylcarbamoyl)benzyl)carbamoyl)-7-(8-fluoro-5-methylchroman-6-yl)-5-methylpyrazolo[1,5-a]pyrimidin-6-yl)acetic acid 1423741-38-1 C33H35F2N5O6
(2S)-2-(tert-butoxy)-2-(2-((4-fluoro-2-(methylcarbamoyl)benzyl)carbamoyl)-7-(8-fluoro-5-methylchroman-6-yl)-5-methylpyrazolo[1,5-a]pyrimidin-6-yl)acetic acid
—— (2S)-2-(tert-butoxy)-2-(2-((3-ethyl-4-fluorobenzyl)carbamoyl)-7-(8-fluoro-5-methylchroman-6-yl)-5-methylpyrazolo[1,5-a]pyrimidin-6-yl)acetic acid 1423741-30-3 C33H36F2N4O5
(2S)-2-(tert-butoxy)-2-(2-((3-ethyl-4-fluorobenzyl)carbamoyl)-7-(8-fluoro-5-methylchroman-6-yl)-5-methylpyrazolo[1,5-a]pyrimidin-6-yl)acetic acid
—— (2S)-2-(tert-butoxy)-2-(2-((4-fluoro-3-methylbenzyl)carbamoyl)-7-(8-fluoro-5-methylchroman-6-yl)-5-methylpyrazolo[1,5-a]pyrimidin-6-yl)acetic acid 1423741-08-5 C32H34F2N4O5
(2S)-2-(tert-butoxy)-2-(2-((4-fluoro-3-methylbenzyl)carbamoyl)-7-(8-fluoro-5-methylchroman-6-yl)-5-methylpyrazolo[1,5-a]pyrimidin-6-yl)acetic acid
—— (2S)-2-(tert-butoxy)-2-(2-((4-fluoro-2-(methylsulfonyl)benzyl)carbamoyl)-7-(8-fluoro-5-methylchroman-6-yl)-5-methylpyrazolo[1,5-a]pyrimidin-6-yl)acetic acid 1423741-36-9 C32H34F2N4O7S
(2S)-2-(tert-butoxy)-2-(2-((4-fluoro-2-(methylsulfonyl)benzyl)carbamoyl)-7-(8-fluoro-5-methylchroman-6-yl)-5-methylpyrazolo[1,5-a]pyrimidin-6-yl)acetic acid
—— (2S)-2-(tert-butoxy)-2-(2-((4-fluoro-2-methoxybenzyl)carbamoyl)-7-(8-fluoro-5-methylchroman-6-yl)-5-methylpyrazolo[1,5-a]pyrimidin-6-yl)acetic acid 1423741-37-0 C32H34F2N4O6
(2S)-2-(tert-butoxy)-2-(2-((4-fluoro-2-methoxybenzyl)carbamoyl)-7-(8-fluoro-5-methylchroman-6-yl)-5-methylpyrazolo[1,5-a]pyrimidin-6-yl)acetic acid
—— (2S)-2-(tert-butoxy)-2-(2-((3-cyclopropyl-4-fluorobenzyl)carbamoyl)-7-(8-fluoro-5-methylchroman-6-yl)-5-methylpyrazolo[1,5-a]pyrimidin-6-yl)acetic acid 1423741-32-5 C34H36F2N4O5
(2S)-2-(tert-butoxy)-2-(2-((3-cyclopropyl-4-fluorobenzyl)carbamoyl)-7-(8-fluoro-5-methylchroman-6-yl)-5-methylpyrazolo[1,5-a]pyrimidin-6-yl)acetic acid
—— (2S)-2-(tert-butoxy)-2-(2-((4-fluoro-2-(2-oxopyrrolidin-1-yl)benzyl)carbamoyl)-7-(8-fluoro-5-methylchroman-6-yl)-5-methylpyrazolo[1,5-a]pyrimidin-6-yl)acetic acid 1423741-18-7 C35H37F2N5O6
(2S)-2-(tert-butoxy)-2-(2-((4-fluoro-2-(2-oxopyrrolidin-1-yl)benzyl)carbamoyl)-7-(8-fluoro-5-methylchroman-6-yl)-5-methylpyrazolo[1,5-a]pyrimidin-6-yl)acetic acid
—— (S)-6-(1-(tert-butoxy)-2-ethoxy-2-oxoethyl)-7-(4,4-dimethylpiperidin-1-yl)-5-methylpyrazolo[1,5-a]pyrimidine-2-carboxylic acid 1423742-86-2 C23H34N4O5
(S)-6-(1-(tert-butoxy)-2-ethoxy-2-oxoethyl)-7-(4,4-dimethylpiperidin-1-yl)-5-methylpyrazolo[1,5-a]pyrimidine-2-carboxylic acid
—— (2S)-ethyl 2-(tert-butoxy)-2-(2-((4-fluoro-3-methylbenzyl)carbamoyl)-7-(8-fluoro-5-methylchroman-6-yl)-5-methylpyrazolo[1,5-a]pyrimidin-6-yl)acetate 1423742-87-3 C34H38F2N4O5
(2S)-ethyl 2-(tert-butoxy)-2-(2-((4-fluoro-3-methylbenzyl)carbamoyl)-7-(8-fluoro-5-methylchroman-6-yl)-5-methylpyrazolo[1,5-a]pyrimidin-6-yl)acetate
—— 6-((S)-1-(tert-butoxy)-2-ethoxy-2-oxoethyl)-7-(8-fluoro-5-methylchroman-6-yl)-5-methylpyrazolo[1,5-a]pyrimidine-2-carboxylate 1423742-72-6 C28H34FN3O6
6-((S)-1-(tert-butoxy)-2-ethoxy-2-oxoethyl)-7-(8-fluoro-5-methylchroman-6-yl)-5-methylpyrazolo[1,5-a]pyrimidine-2-carboxylate
—— ethyl 7-chloro-6-(2-ethoxy-2-oxoethyl)-5-methylpyrazolo[1,5-a]pyrimidine-2-carboxylate 1423742-66-8 C14H16ClN3O4
ethyl 7-chloro-6-(2-ethoxy-2-oxoethyl)-5-methylpyrazolo[1,5-a]pyrimidine-2-carboxylate
—— d<sub>3</sub>-N-(1,3-dioxo-1,3-dihydroisobenzofuran-4-yl)acetamide 1258598-10-5 C10H7NO4
d<sub>3</sub>-N-(1,3-dioxo-1,3-dihydroisobenzofuran-4-yl)acetamide
—— 3,3-difluoropiperidin-4-ol hydrochloride 1334416-77-1 C5H9F2NO*ClH
3,3-difluoropiperidin-4-ol hydrochloride
—— (S)-1-(6-bromo-1-methyl-1H-pyrrolo[3,2-b]pyridin-5-yl)ethanamine 1537208-12-0 C10H12BrN3
(S)-1-(6-bromo-1-methyl-1H-pyrrolo[3,2-b]pyridin-5-yl)ethanamine
—— (2,2-difluoroethoxy)benzene 1309602-18-3 C8H8F2O
(2,2-difluoroethoxy)benzene
—— 1-[5-(tetrahydro-pyran-2-yloxymethyl)-furan-2-yl]-ethanol 1256277-91-4 C12H18O4
1-[5-(tetrahydro-pyran-2-yloxymethyl)-furan-2-yl]-ethanol
—— 5-(octyloxymethyl)-2-furoic acid 1039853-28-5 C14H22O4
5-(octyloxymethyl)-2-furoic acid
—— 4-(4-chlorophenyl)-3-(pyridin-4-yl)furan-2(5H)-one 1494217-90-1 C15H10ClNO2
4-(4-chlorophenyl)-3-(pyridin-4-yl)furan-2(5H)-one
—— (R)-2-amino-3-(4-ethoxyphenyl)propionic acid hydrochloride 1417694-04-2 C11H15NO3*ClH
(R)-2-amino-3-(4-ethoxyphenyl)propionic acid hydrochloride
—— 1-bromo-4-(difluoromethoxy)-2-methylbenzene 1021172-76-8 C8H7BrF2O
1-bromo-4-(difluoromethoxy)-2-methylbenzene
—— sodium dibenzyldithiocarbamate hydrate 1082663-31-7 C15H14NS2*H2O*Na
sodium dibenzyldithiocarbamate hydrate
—— (S)-5-[3,5-bis(trifluoromethyl)benzyl]-2,3,4,5-tetrahydro-3-methyl-6-oxo-7-phenyl-6H-pyrido[2,3-b][1,5]oxazocine 183550-59-6 C25H20F6N2O2
(S)-5-[3,5-bis(trifluoromethyl)benzyl]-2,3,4,5-tetrahydro-3-methyl-6-oxo-7-phenyl-6H-pyrido[2,3-b][1,5]oxazocine
—— 4-amino-2,2-dimethyl-butan-1-ol 179419-04-6 C6H15NO
4-amino-2,2-dimethyl-butan-1-ol
—— 1-(difluoromethyl)-1H-pyrazole-4-carbaldehyde 1216244-84-6 C5H4F2N2O
1-(difluoromethyl)-1H-pyrazole-4-carbaldehyde
—— 2-(difluoromethoxy)-5-fluorobenzaldehyde 1214326-36-9 C8H5F3O2
2-(difluoromethoxy)-5-fluorobenzaldehyde
—— 1-(2-(difluoromethoxy)-5-fluorophenyl)ethan-1-one 1214338-07-4 C9H7F3O2
1-(2-(difluoromethoxy)-5-fluorophenyl)ethan-1-one
—— ethyl 3-hydroxy-8-thia-4,6-diazatricyclo[7.4.0.0[2,7]]trideca-1(9),2(7),3,5,10,12-hexaene-12-carboxylate 1537184-71-6 C13H10N2O3S
ethyl 3-hydroxy-8-thia-4,6-diazatricyclo[7.4.0.0[2,7]]trideca-1(9),2(7),3,5,10,12-hexaene-12-carboxylate
—— ethyl 4-hydroxy-5,6,7,8-tetrahydrobenzo[4,5]thieno[2,3-d]pyrimidine-6-carboxylate 1447956-28-6 C13H14N2O3S
ethyl 4-hydroxy-5,6,7,8-tetrahydrobenzo[4,5]thieno[2,3-d]pyrimidine-6-carboxylate