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—— 3-{4-methyl-5-[(1R)-1-(2-(3-methylphenyl)-2H-tetrazol-5-yl)-ethoxy]-4H-[1,2,4]triazol-3-yl}-pyridine 1144034-01-4 C18H18N8O
3-{4-methyl-5-[(1R)-1-(2-(3-methylphenyl)-2H-tetrazol-5-yl)-ethoxy]-4H-[1,2,4]triazol-3-yl}-pyridine
—— N-((1R)-phenylethyl)-3-dichloromethyl-5-methylhexanamide 1144854-26-1 C16H23Cl2NO
N-((1R)-phenylethyl)-3-dichloromethyl-5-methylhexanamide
—— (2-amino-4-(3-methoxyphenyl)thiophen-3-yl)(phenyl)methanone 1146188-38-6 C18H15NO2S
(2-amino-4-(3-methoxyphenyl)thiophen-3-yl)(phenyl)methanone
—— (2-amino-4-(3-bromophenyl)thiophen-3-yl)(phenyl)methanone 1146188-29-5 C17H12BrNOS
(2-amino-4-(3-bromophenyl)thiophen-3-yl)(phenyl)methanone
—— 2-[4-methyl-5-(methylsulfonyl)-4H-1,2,4-triazol-3-yl]pyrimidine 1144033-87-3 C8H9N5O2S
2-[4-methyl-5-(methylsulfonyl)-4H-1,2,4-triazol-3-yl]pyrimidine
—— [(4-{[(3-cyano-furoxan-4-yl)methyl]thio}benzoyl)oxy]methyl 2-(acetyloxy)benzoate 1144618-72-3 C21H15N3O8S
[(4-{[(3-cyano-furoxan-4-yl)methyl]thio}benzoyl)oxy]methyl 2-(acetyloxy)benzoate
—— 4-(5-acetyl-4,5,6,7-tetrahydrothieno[3,2-c]pyridin-2-yl)-N-[4-(4-methylpiperazin-1-yl)phenyl]-7H-pyrrolo[2,3-d]pyrimidin-2-amine 1142946-94-8 C26H29N7OS
4-(5-acetyl-4,5,6,7-tetrahydrothieno[3,2-c]pyridin-2-yl)-N-[4-(4-methylpiperazin-1-yl)phenyl]-7H-pyrrolo[2,3-d]pyrimidin-2-amine
—— 3-{3-[(2,2,2-trifluoro-ethyl)-ureido]-imidazo[1,2-a]pyridine-7-[3-(1H-imidazol-4-yl)]}-propanamide 1141505-15-8 C23H22F3N7O2
3-{3-[(2,2,2-trifluoro-ethyl)-ureido]-imidazo[1,2-a]pyridine-7-[3-(1H-imidazol-4-yl)]}-propanamide
—— 1-[4-hydroxy-6-(4-methyl-1-piperazinyl)-1,3,5-triazin-2-yl]-N-{[2-(trifluoromethyl)phenyl]methyl}-4-piperidinecarboxamide 1141895-07-9 C22H28F3N7O2
1-[4-hydroxy-6-(4-methyl-1-piperazinyl)-1,3,5-triazin-2-yl]-N-{[2-(trifluoromethyl)phenyl]methyl}-4-piperidinecarboxamide
—— 2-(2-(4-(morpholinomethyl)phenylamino)-7H-pyrrolo[2,3-d]pyrimidin-4-yl)benzo[b]thiophene-6-carbonitrile 1142946-59-5 C26H22N6OS
2-(2-(4-(morpholinomethyl)phenylamino)-7H-pyrrolo[2,3-d]pyrimidin-4-yl)benzo[b]thiophene-6-carbonitrile
—— 2-[5-(2,6-difluoro-pyridin-4-yl)-4'-trifluoromethyl-biphenyl-3-yl]-4-methyl-pentanoic acid 1146595-02-9 C24H20F5NO2
2-[5-(2,6-difluoro-pyridin-4-yl)-4'-trifluoromethyl-biphenyl-3-yl]-4-methyl-pentanoic acid
—— (S)-2-[5-(3,5-difluoro-benzyloxy)-4'-trifluoromethyl-biphenyl-3-yl]-4-methyl-pentanoic acid 1144592-94-8 C26H23F5O3
(S)-2-[5-(3,5-difluoro-benzyloxy)-4'-trifluoromethyl-biphenyl-3-yl]-4-methyl-pentanoic acid
—— 5-amino-1-N,3-N-bis(3-ethynylphenyl)benzene-1,3-dicarboxamide;hydrochloride 1135615-30-3 C24H17N3O2*ClH
5-amino-1-N,3-N-bis(3-ethynylphenyl)benzene-1,3-dicarboxamide;hydrochloride
—— 4-(5-methylbenzo[b]thiophen-2-yl)-N-(4-(morpholinomethyl)phenyl)-7H-pyrrolo[2,3-d]pyrimidin-2-amine 1142946-60-8 C26H25N5OS
4-(5-methylbenzo[b]thiophen-2-yl)-N-(4-(morpholinomethyl)phenyl)-7H-pyrrolo[2,3-d]pyrimidin-2-amine
—— 4-[(1R)-1-(4-{[4-(trifluoromethyl)-1,3-thiazol-2-yl]amino}phenyl)ethyl]-1,2,5-oxadiazol-3-ol 1144016-07-8 C14H11F3N4O2S
4-[(1R)-1-(4-{[4-(trifluoromethyl)-1,3-thiazol-2-yl]amino}phenyl)ethyl]-1,2,5-oxadiazol-3-ol
—— 5-(1H-1,3-benzodiazol-1-yl)-3-[(2-methoxyphenyl)methoxy]thiophene-2-carboxamide 1135118-99-8 C20H17N3O3S
5-(1H-1,3-benzodiazol-1-yl)-3-[(2-methoxyphenyl)methoxy]thiophene-2-carboxamide
—— 3-(cyclopentylmethoxy)-5-(5,6-dimethoxy-1H-1,3-benzodiazol-1-yl)thiophene-2-carboxamide 1135121-07-1 C20H23N3O4S
3-(cyclopentylmethoxy)-5-(5,6-dimethoxy-1H-1,3-benzodiazol-1-yl)thiophene-2-carboxamide
—— (2-amino-4-(4-methoxyphenyl)thiophen-3-yl)(phenyl)methanone 1146188-36-4 C18H15NO2S
(2-amino-4-(4-methoxyphenyl)thiophen-3-yl)(phenyl)methanone
—— (2-amino-4-(4-nitrophenyl)thiophen-3-yl)(phenyl)methanone 1146188-41-1 C17H12N2O3S
(2-amino-4-(4-nitrophenyl)thiophen-3-yl)(phenyl)methanone
—— (2R,3R)-3-[tert-butyl(dimethyl)silyl]oxy-N-[3-[(2R,3S,6S,8S)-8-[(E,3S,6S)-6-[tert-butyl(dimethyl)silyl]oxy-3,5-dimethylhept-4-enyl]-3-methyl-1,7-dioxaspiro[5.5]undecan-2-yl]propyl]-2-methyl-4-[[2-[(2S,3R,6S)-3-methyl-6-[(E)-2-oxopent-3-enyl]oxan-2-yl]acetyl]amino]butanamide 1126107-83-2 C52H96N2O8Si2
(2R,3R)-3-[tert-butyl(dimethyl)silyl]oxy-N-[3-[(2R,3S,6S,8S)-8-[(E,3S,6S)-6-[tert-butyl(dimethyl)silyl]oxy-3,5-dimethylhept-4-enyl]-3-methyl-1,7-dioxaspiro[5.5]undecan-2-yl]propyl]-2-methyl-4-[[2-[(2S,3R,6S)-3-methyl-6-[(E)-2-oxopent-3-enyl]oxan-2-yl]acetyl]amino]butanamide
—— 5-(1H-1,3-benzodiazol-1-yl)-3-[(4-methoxyphenyl)methoxy]thiophene-2-carboxamide 1135119-04-8 C20H17N3O3S
5-(1H-1,3-benzodiazol-1-yl)-3-[(4-methoxyphenyl)methoxy]thiophene-2-carboxamide
—— 2,4-diamino-6-ethyl-5-(3-(7-fluoro-2-methylquinolin-4-yloxy)propoxy)pyrimidine 1142407-75-7 C19H22FN5O2
2,4-diamino-6-ethyl-5-(3-(7-fluoro-2-methylquinolin-4-yloxy)propoxy)pyrimidine
—— Anthranilic acid deriv., 5 1066821-75-7 C23H19BrN2O5S
Anthranilic acid deriv., 5
—— 5-tert-butyl-2-benzyl-N-(3-(aminosulfonyl)phenyl)-2H-1,2,4-triazole-3-carboxamide 1143504-09-9 C20H23N5O3S
5-tert-butyl-2-benzyl-N-(3-(aminosulfonyl)phenyl)-2H-1,2,4-triazole-3-carboxamide
—— (8-Ethynyl-6-phenyl-4H-benzo[f]imidazo[1,5-a][1,4]diazepin-3-yl)(4-methylpiperazin-1-yl)methanone 1140967-62-9 C25H23N5O
(8-Ethynyl-6-phenyl-4H-benzo[f]imidazo[1,5-a][1,4]diazepin-3-yl)(4-methylpiperazin-1-yl)methanone
—— 2-(2-(3-(4-methylpiperazin-1-yl)phenylamino)-7H-pyrrolo[2,3-d]pyrimidin-4-yl)benzo[b]thiophene-6-carbonitrile 1142947-47-4 C26H23N7S
2-(2-(3-(4-methylpiperazin-1-yl)phenylamino)-7H-pyrrolo[2,3-d]pyrimidin-4-yl)benzo[b]thiophene-6-carbonitrile
—— 3-[4-({[4-(1-methylethyl)phenyl]carbonyl}amino)butyl]-1-(2-pyridinyl)-1H-indole-5-carboxylic acid 1144523-08-9 C28H29N3O3
3-[4-({[4-(1-methylethyl)phenyl]carbonyl}amino)butyl]-1-(2-pyridinyl)-1H-indole-5-carboxylic acid
—— 3-[(2-bromopyridin-4-yl)methoxy]-5-(5,6-dimethoxy-1H-1,3-benzodiazol-1-yl)thiophene-2-carboxamide 1135121-30-0 C20H17BrN4O4S
3-[(2-bromopyridin-4-yl)methoxy]-5-(5,6-dimethoxy-1H-1,3-benzodiazol-1-yl)thiophene-2-carboxamide
—— (3R,5S)-5-{2-[4-({3-chloro-4-[(3-fluorophenyl)methoxy]phenyl}amino)thieno[3,2-d]pyrimidin-6-yl]ethynyl}pyrrolidin-3-yl N-ethyl-N-methylcarbamate 1120371-57-4 C29H27ClFN5O3S
(3R,5S)-5-{2-[4-({3-chloro-4-[(3-fluorophenyl)methoxy]phenyl}amino)thieno[3,2-d]pyrimidin-6-yl]ethynyl}pyrrolidin-3-yl N-ethyl-N-methylcarbamate
—— 2,4-diamino-6-ethyl-5-(3-(6-chloro-quinolin-4-yloxy)propoxy)pyrimidine 1142407-68-8 C18H20ClN5O2
2,4-diamino-6-ethyl-5-(3-(6-chloro-quinolin-4-yloxy)propoxy)pyrimidine
—— 2-(4-Cyclopropanesulfonylphenyl)-2-(2,4-difluoro-phenoxy)-N-thiazol-2-yl-acetamide 1143512-16-6 C20H16F2N2O4S2
2-(4-Cyclopropanesulfonylphenyl)-2-(2,4-difluoro-phenoxy)-N-thiazol-2-yl-acetamide
—— 3-[3-(3-pyrazol-1-yl-phenyl)-imidazo[1,2-a]pyridin-7-yl]-benzoic acid ethyl ester 1146612-35-2 C25H20N4O2
3-[3-(3-pyrazol-1-yl-phenyl)-imidazo[1,2-a]pyridin-7-yl]-benzoic acid ethyl ester
—— (2R)-3-methyl-2-{8-oxatricyclo[7.4.0.0^{2,7}]trideca-1(13),2,4,6,9,11-hexaene-4-sulfonamido}butanoic acid 1140632-75-2 C17H17NO5S
(2R)-3-methyl-2-{8-oxatricyclo[7.4.0.0^{2,7}]trideca-1(13),2,4,6,9,11-hexaene-4-sulfonamido}butanoic acid
—— 5-(1H-1,3-benzodiazol-1-yl)-3-[(2-bromophenyl)methoxy]thiophene-2-carboxamide 1135119-15-1 C19H14BrN3O2S
5-(1H-1,3-benzodiazol-1-yl)-3-[(2-bromophenyl)methoxy]thiophene-2-carboxamide
—— N-cyclohexyl-2-(3,4-dimethoxyphenyl)-4-(4-fluorobenzyl)-5-oxo-3,4-dihydrobenzo[e][1,4]diazepine-3-carboxamide 1123339-45-6 C31H32FN3O4
N-cyclohexyl-2-(3,4-dimethoxyphenyl)-4-(4-fluorobenzyl)-5-oxo-3,4-dihydrobenzo[e][1,4]diazepine-3-carboxamide
—— 5-tert-butyl-N-(3-sulfamoylphenyl)-1,3,4-thiadiazole-2-carboxamide 1143504-06-6 C13H16N4O3S2
5-tert-butyl-N-(3-sulfamoylphenyl)-1,3,4-thiadiazole-2-carboxamide
—— N-methyl-3-[3-(3-pyrazol-1-yl-phenyl)-imidazo[1,2-a]pyridin-7-yl]-benzamide 1146613-28-6 C24H19N5O
N-methyl-3-[3-(3-pyrazol-1-yl-phenyl)-imidazo[1,2-a]pyridin-7-yl]-benzamide
—— 1-[4-(methoxy)-6-(4-methyl-1-piperazinyl)-1,3,5-triazin-2-yl]-N-{[2-(trifluoromethyl)phenyl]methyl}-4-piperidinecarboxamide 1141895-09-1 C23H30F3N7O2
1-[4-(methoxy)-6-(4-methyl-1-piperazinyl)-1,3,5-triazin-2-yl]-N-{[2-(trifluoromethyl)phenyl]methyl}-4-piperidinecarboxamide
—— 3-[(3-cyanophenyl)methoxy]-5-(5,6-dimethoxy-1H-1,3-benzodiazol-1-yl)thiophene-2-carboxamide 1135120-60-3 C22H18N4O4S
3-[(3-cyanophenyl)methoxy]-5-(5,6-dimethoxy-1H-1,3-benzodiazol-1-yl)thiophene-2-carboxamide
—— 3-[(3-{4-chloro-3-[2-methyl-8-(trifluoromethyl)quinazolin-4-yl]phenoxy}-phenyl)sulfonyl]propan-1-ol 1112985-95-1 C25H20ClF3N2O4S
3-[(3-{4-chloro-3-[2-methyl-8-(trifluoromethyl)quinazolin-4-yl]phenoxy}-phenyl)sulfonyl]propan-1-ol
—— 4-(4-methylthiophen-2-yl)-N-(4-(1-morpholinoethyl)phenyl)-7H-pyrrolo[2,3-d]pyrimidin-2-amine 1143018-48-7 C23H25N5OS
4-(4-methylthiophen-2-yl)-N-(4-(1-morpholinoethyl)phenyl)-7H-pyrrolo[2,3-d]pyrimidin-2-amine
—— N-[4-(4-methylpiperazin-1-yl)phenyl]-4-[4-(3-morpholin-4-ylsulfonylphenyl)thiophen-2-yl]-7H-pyrrolo[2,3-d]pyrimidin-2-amine 1142947-26-9 C31H33N7O3S2
N-[4-(4-methylpiperazin-1-yl)phenyl]-4-[4-(3-morpholin-4-ylsulfonylphenyl)thiophen-2-yl]-7H-pyrrolo[2,3-d]pyrimidin-2-amine
—— 4-(4-ethylthiophen-2-yl)-N-(4-(morpholinomethyl)phenyl)-7H-pyrrolo[2,3-d]pyrimidin-2-amine 1142946-76-6 C23H25N5OS
4-(4-ethylthiophen-2-yl)-N-(4-(morpholinomethyl)phenyl)-7H-pyrrolo[2,3-d]pyrimidin-2-amine
—— 1-(2-(2-(4-(2-(pyrrolidin-1-yl)ethoxy)phenylamino)-7H-pyrrolo[2,3-d]pyrimidin-4-yl)benzo[b]thiophen-5-yl)pentan-1-one 1142947-54-3 C31H33N5O2S
1-(2-(2-(4-(2-(pyrrolidin-1-yl)ethoxy)phenylamino)-7H-pyrrolo[2,3-d]pyrimidin-4-yl)benzo[b]thiophen-5-yl)pentan-1-one
—— 1-[4-(4-methyl-1-piperazinyl)-6-(methylthio)-1,3,5-triazin-2-yl]-N-{[2-(trifluoromethyl)phenyl]methyl}-4-piperidinecarboxamide 1141895-10-4 C23H30F3N7OS
1-[4-(4-methyl-1-piperazinyl)-6-(methylthio)-1,3,5-triazin-2-yl]-N-{[2-(trifluoromethyl)phenyl]methyl}-4-piperidinecarboxamide
—— (8-ethynyl-6-phenyl-4H-benzo[f]imidazo[1,5-a][1,4]diazepin-3-yl)(morpholino)methanone 1140967-64-1 C24H20N4O2
(8-ethynyl-6-phenyl-4H-benzo[f]imidazo[1,5-a][1,4]diazepin-3-yl)(morpholino)methanone
—— (S)-2-[6-(4-trifluoromethylphenyl)-1H-benzoimidazol-2-yl]pyrrolidine-1-carboxylic acid benzyl ester 1031746-80-1 C26H22F3N3O2
(S)-2-[6-(4-trifluoromethylphenyl)-1H-benzoimidazol-2-yl]pyrrolidine-1-carboxylic acid benzyl ester
—— 2,4-diamino-6-ethyl-5-(3-(quinolin-4-yloxy)propoxy)pyrimidine 1142407-67-7 C18H21N5O2
2,4-diamino-6-ethyl-5-(3-(quinolin-4-yloxy)propoxy)pyrimidine
—— 3-(1-(3-(biphenyl-4-ylamino)-3-oxopropyl)-1H-1,2,3-triazol-4-yl)-6-hydroxy-1-methyl-2-phenyl-1H-indole-5-carboxylic acid 1143579-78-5 C33H27N5O4
3-(1-(3-(biphenyl-4-ylamino)-3-oxopropyl)-1H-1,2,3-triazol-4-yl)-6-hydroxy-1-methyl-2-phenyl-1H-indole-5-carboxylic acid
—— 2-(2-(4-(4-methylpiperazin-1-yl)phenylamino)-7H-pyrrolo[2,3-d]pyrimidin-4-yl)thiophene-3-carbonitrile 1142946-54-0 C22H21N7S
2-(2-(4-(4-methylpiperazin-1-yl)phenylamino)-7H-pyrrolo[2,3-d]pyrimidin-4-yl)thiophene-3-carbonitrile