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—— ethyl (6R)-4-[[4-(cyclopropanecarbonyl)-1,4-diazepan-1-yl]methyl]-6-(2,3-dichlorophenyl)-3-ethyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate —— C25H32Cl2N4O4
ethyl (6R)-4-[[4-(cyclopropanecarbonyl)-1,4-diazepan-1-yl]methyl]-6-(2,3-dichlorophenyl)-3-ethyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6S)-6-(3,5-dimethoxyphenyl)-3-ethyl-4-[[4-(ethylcarbamoyl)-1,4-diazepan-1-yl]methyl]-2-oxo-1,6-dihydropyrimidine-5-carboxylate —— C26H39N5O6
ethyl (6S)-6-(3,5-dimethoxyphenyl)-3-ethyl-4-[[4-(ethylcarbamoyl)-1,4-diazepan-1-yl]methyl]-2-oxo-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6S)-6-(3-chlorophenyl)-3-ethyl-2-oxo-4-[[4-(propylcarbamoyl)-1,4-diazepan-1-yl]methyl]-1,6-dihydropyrimidine-5-carboxylate —— C25H36ClN5O4
ethyl (6S)-6-(3-chlorophenyl)-3-ethyl-2-oxo-4-[[4-(propylcarbamoyl)-1,4-diazepan-1-yl]methyl]-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6R)-4-[[(3R)-4-(cyclobutanecarbonyl)-3-methylpiperazin-1-yl]methyl]-2-oxo-3-prop-2-enyl-6-thiophen-3-yl-1,6-dihydropyrimidine-5-carboxylate —— C25H34N4O4S
ethyl (6R)-4-[[(3R)-4-(cyclobutanecarbonyl)-3-methylpiperazin-1-yl]methyl]-2-oxo-3-prop-2-enyl-6-thiophen-3-yl-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6R)-4-[[(3R)-4-(tert-butylcarbamoyl)-3-methylpiperazin-1-yl]methyl]-3-ethyl-2-oxo-6-thiophen-3-yl-1,6-dihydropyrimidine-5-carboxylate —— C24H37N5O4S
ethyl (6R)-4-[[(3R)-4-(tert-butylcarbamoyl)-3-methylpiperazin-1-yl]methyl]-3-ethyl-2-oxo-6-thiophen-3-yl-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6S)-4-[[(3R)-4-(cyclobutanecarbonyl)-3-methylpiperazin-1-yl]methyl]-2-oxo-3-prop-2-enyl-6-thiophen-3-yl-1,6-dihydropyrimidine-5-carboxylate —— C25H34N4O4S
ethyl (6S)-4-[[(3R)-4-(cyclobutanecarbonyl)-3-methylpiperazin-1-yl]methyl]-2-oxo-3-prop-2-enyl-6-thiophen-3-yl-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6S)-4-[[(3R)-4-(tert-butylcarbamoyl)-3-methylpiperazin-1-yl]methyl]-3-ethyl-2-oxo-6-thiophen-3-yl-1,6-dihydropyrimidine-5-carboxylate —— C24H37N5O4S
ethyl (6S)-4-[[(3R)-4-(tert-butylcarbamoyl)-3-methylpiperazin-1-yl]methyl]-3-ethyl-2-oxo-6-thiophen-3-yl-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6R)-3-ethyl-6-(3-methoxyphenyl)-4-[[4-(2-methylpropanoyl)piperazin-1-yl]methyl]-2-oxo-1,6-dihydropyrimidine-5-carboxylate —— C25H36N4O5
ethyl (6R)-3-ethyl-6-(3-methoxyphenyl)-4-[[4-(2-methylpropanoyl)piperazin-1-yl]methyl]-2-oxo-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6R)-3-ethyl-4-[[(3R)-3-methyl-4-(propylcarbamoyl)piperazin-1-yl]methyl]-2-oxo-6-thiophen-3-yl-1,6-dihydropyrimidine-5-carboxylate —— C23H35N5O4S
ethyl (6R)-3-ethyl-4-[[(3R)-3-methyl-4-(propylcarbamoyl)piperazin-1-yl]methyl]-2-oxo-6-thiophen-3-yl-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6S)-3-ethyl-4-[[(3R)-4-(ethylcarbamoyl)-3-methylpiperazin-1-yl]methyl]-6-(2-methoxyphenyl)-2-oxo-1,6-dihydropyrimidine-5-carboxylate —— C25H37N5O5
ethyl (6S)-3-ethyl-4-[[(3R)-4-(ethylcarbamoyl)-3-methylpiperazin-1-yl]methyl]-6-(2-methoxyphenyl)-2-oxo-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6S)-6-(3,4-dimethoxyphenyl)-3-ethyl-2-oxo-4-[[4-(propan-2-ylcarbamoyl)-1,4-diazepan-1-yl]methyl]-1,6-dihydropyrimidine-5-carboxylate —— C27H41N5O6
ethyl (6S)-6-(3,4-dimethoxyphenyl)-3-ethyl-2-oxo-4-[[4-(propan-2-ylcarbamoyl)-1,4-diazepan-1-yl]methyl]-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6R)-4-[[(3R)-4-(tert-butylcarbamoyl)-3-methylpiperazin-1-yl]methyl]-2-oxo-3-prop-2-enyl-6-thiophen-3-yl-1,6-dihydropyrimidine-5-carboxylate —— C25H37N5O4S
ethyl (6R)-4-[[(3R)-4-(tert-butylcarbamoyl)-3-methylpiperazin-1-yl]methyl]-2-oxo-3-prop-2-enyl-6-thiophen-3-yl-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6R)-6-(2,5-dimethylphenyl)-3-ethyl-2-oxo-4-[(4-propanoyl-1,4-diazepan-1-yl)methyl]-1,6-dihydropyrimidine-5-carboxylate —— C26H38N4O4
ethyl (6R)-6-(2,5-dimethylphenyl)-3-ethyl-2-oxo-4-[(4-propanoyl-1,4-diazepan-1-yl)methyl]-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6S)-6-(2,4-dimethoxyphenyl)-3-ethyl-4-[[(3R)-4-(ethylcarbamoyl)-3-methylpiperazin-1-yl]methyl]-2-oxo-1,6-dihydropyrimidine-5-carboxylate —— C26H39N5O6
ethyl (6S)-6-(2,4-dimethoxyphenyl)-3-ethyl-4-[[(3R)-4-(ethylcarbamoyl)-3-methylpiperazin-1-yl]methyl]-2-oxo-1,6-dihydropyrimidine-5-carboxylate
—— ethyl 1-[(2R)-2-[[5-(2,5-dimethoxyphenyl)-1,2-oxazole-3-carbonyl]amino]propanoyl]piperidine-4-carboxylate —— C23H29N3O7
ethyl 1-[(2R)-2-[[5-(2,5-dimethoxyphenyl)-1,2-oxazole-3-carbonyl]amino]propanoyl]piperidine-4-carboxylate
—— ethyl (6R)-4-[(4-benzoylpiperazin-1-yl)methyl]-3-ethyl-2-oxo-6-thiophen-3-yl-1,6-dihydropyrimidine-5-carboxylate —— C25H30N4O4S
ethyl (6R)-4-[(4-benzoylpiperazin-1-yl)methyl]-3-ethyl-2-oxo-6-thiophen-3-yl-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6S)-6-(3,5-dimethoxyphenyl)-3-ethyl-4-[[(3R)-4-(ethylcarbamoyl)-3-methylpiperazin-1-yl]methyl]-2-oxo-1,6-dihydropyrimidine-5-carboxylate —— C26H39N5O6
ethyl (6S)-6-(3,5-dimethoxyphenyl)-3-ethyl-4-[[(3R)-4-(ethylcarbamoyl)-3-methylpiperazin-1-yl]methyl]-2-oxo-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6S)-6-(3-chlorophenyl)-3-ethyl-4-[[(3R)-4-(ethylcarbamoyl)-3-methylpiperazin-1-yl]methyl]-2-oxo-1,6-dihydropyrimidine-5-carboxylate —— C24H34ClN5O4
ethyl (6S)-6-(3-chlorophenyl)-3-ethyl-4-[[(3R)-4-(ethylcarbamoyl)-3-methylpiperazin-1-yl]methyl]-2-oxo-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6R)-6-(3-chlorophenyl)-3-ethyl-2-oxo-4-[[4-(propan-2-ylcarbamoyl)piperazin-1-yl]methyl]-1,6-dihydropyrimidine-5-carboxylate —— C24H34ClN5O4
ethyl (6R)-6-(3-chlorophenyl)-3-ethyl-2-oxo-4-[[4-(propan-2-ylcarbamoyl)piperazin-1-yl]methyl]-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (3S)-1-[3-[2-methoxyethyl-[5-(2,4,6-trimethylphenyl)-1,2-oxazole-3-carbonyl]amino]propanoyl]piperidine-3-carboxylate —— C27H37N3O6
ethyl (3S)-1-[3-[2-methoxyethyl-[5-(2,4,6-trimethylphenyl)-1,2-oxazole-3-carbonyl]amino]propanoyl]piperidine-3-carboxylate
—— ethyl (6R)-4-[[4-(ethylcarbamoyl)piperazin-1-yl]methyl]-2-oxo-3-prop-2-enyl-6-thiophen-3-yl-1,6-dihydropyrimidine-5-carboxylate —— C22H31N5O4S
ethyl (6R)-4-[[4-(ethylcarbamoyl)piperazin-1-yl]methyl]-2-oxo-3-prop-2-enyl-6-thiophen-3-yl-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6R)-3-ethyl-2-oxo-4-[[4-(propan-2-ylcarbamoyl)piperazin-1-yl]methyl]-6-thiophen-3-yl-1,6-dihydropyrimidine-5-carboxylate —— C22H33N5O4S
ethyl (6R)-3-ethyl-2-oxo-4-[[4-(propan-2-ylcarbamoyl)piperazin-1-yl]methyl]-6-thiophen-3-yl-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6R)-4-[[(3R)-4-(tert-butylcarbamoyl)-3-methylpiperazin-1-yl]methyl]-6-(3-chlorophenyl)-3-ethyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate —— C26H38ClN5O4
ethyl (6R)-4-[[(3R)-4-(tert-butylcarbamoyl)-3-methylpiperazin-1-yl]methyl]-6-(3-chlorophenyl)-3-ethyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate
—— Ethyl 2-amino-3-(5-bromothiophen-2-yl)propanoate —— C9H12BrNO2S
Ethyl 2-amino-3-(5-bromothiophen-2-yl)propanoate
—— ethyl (6S)-6-(3,5-dimethoxyphenyl)-3-ethyl-4-[[(3S)-4-(ethylcarbamoyl)-3-methylpiperazin-1-yl]methyl]-2-oxo-1,6-dihydropyrimidine-5-carboxylate —— C26H39N5O6
ethyl (6S)-6-(3,5-dimethoxyphenyl)-3-ethyl-4-[[(3S)-4-(ethylcarbamoyl)-3-methylpiperazin-1-yl]methyl]-2-oxo-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6R)-3-ethyl-4-[[(3R)-4-(ethylcarbamoyl)-3-methylpiperazin-1-yl]methyl]-2-oxo-6-thiophen-3-yl-1,6-dihydropyrimidine-5-carboxylate —— C22H33N5O4S
ethyl (6R)-3-ethyl-4-[[(3R)-4-(ethylcarbamoyl)-3-methylpiperazin-1-yl]methyl]-2-oxo-6-thiophen-3-yl-1,6-dihydropyrimidine-5-carboxylate
—— ethyl 2-[[2-(4-tert-butylcyclohexanecarbonyl)oxyacetyl]amino]-5,6-dihydro-4H-cyclopenta[b]thiophene-3-carboxylate —— C23H33NO5S
ethyl 2-[[2-(4-tert-butylcyclohexanecarbonyl)oxyacetyl]amino]-5,6-dihydro-4H-cyclopenta[b]thiophene-3-carboxylate
—— Ethyl 1-[2-[[5-benzyl-4-[3-(trifluoromethyl)phenyl]-1,2,4-triazol-3-yl]sulfanylmethyl]-1,3-oxazole-4-carbonyl]piperidine-3-carboxylate —— C29H28F3N5O4S
Ethyl 1-[2-[[5-benzyl-4-[3-(trifluoromethyl)phenyl]-1,2,4-triazol-3-yl]sulfanylmethyl]-1,3-oxazole-4-carbonyl]piperidine-3-carboxylate
—— ethyl 1-[(2S)-2-[[5-(2,5-dimethoxyphenyl)-1,2-oxazole-3-carbonyl]amino]propanoyl]piperidine-4-carboxylate —— C23H29N3O7
ethyl 1-[(2S)-2-[[5-(2,5-dimethoxyphenyl)-1,2-oxazole-3-carbonyl]amino]propanoyl]piperidine-4-carboxylate
—— ethyl (6S)-4-[[4-(tert-butylcarbamoyl)-1,4-diazepan-1-yl]methyl]-3-ethyl-6-(2-methoxyphenyl)-2-oxo-1,6-dihydropyrimidine-5-carboxylate —— C27H41N5O5
ethyl (6S)-4-[[4-(tert-butylcarbamoyl)-1,4-diazepan-1-yl]methyl]-3-ethyl-6-(2-methoxyphenyl)-2-oxo-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6S)-6-(2,4-dichlorophenyl)-3-ethyl-4-[[4-(2-methylpropanoyl)piperazin-1-yl]methyl]-2-oxo-1,6-dihydropyrimidine-5-carboxylate —— C24H32Cl2N4O4
ethyl (6S)-6-(2,4-dichlorophenyl)-3-ethyl-4-[[4-(2-methylpropanoyl)piperazin-1-yl]methyl]-2-oxo-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (3R)-1-[3-[[(2S)-oxolan-2-yl]methyl-[5-(2,4,6-trimethylphenyl)-1,2-oxazole-3-carbonyl]amino]propanoyl]piperidine-3-carboxylate —— C29H39N3O6
ethyl (3R)-1-[3-[[(2S)-oxolan-2-yl]methyl-[5-(2,4,6-trimethylphenyl)-1,2-oxazole-3-carbonyl]amino]propanoyl]piperidine-3-carboxylate
—— ethyl (3R)-1-[3-[[(2R)-oxolan-2-yl]methyl-[5-(2,4,6-trimethylphenyl)-1,2-oxazole-3-carbonyl]amino]propanoyl]piperidine-3-carboxylate —— C29H39N3O6
ethyl (3R)-1-[3-[[(2R)-oxolan-2-yl]methyl-[5-(2,4,6-trimethylphenyl)-1,2-oxazole-3-carbonyl]amino]propanoyl]piperidine-3-carboxylate
—— ethyl 1-[3-[[5-(2,5-dimethylphenyl)-1,2-oxazole-3-carbonyl]-[[(2S)-oxolan-2-yl]methyl]amino]propanoyl]piperidine-4-carboxylate —— C28H37N3O6
ethyl 1-[3-[[5-(2,5-dimethylphenyl)-1,2-oxazole-3-carbonyl]-[[(2S)-oxolan-2-yl]methyl]amino]propanoyl]piperidine-4-carboxylate
—— ethyl 1-[(2R)-2-[[5-(2,5-dimethylphenyl)-1,2-oxazole-3-carbonyl]amino]-3-methylbutanoyl]piperidine-4-carboxylate —— C25H33N3O5
ethyl 1-[(2R)-2-[[5-(2,5-dimethylphenyl)-1,2-oxazole-3-carbonyl]amino]-3-methylbutanoyl]piperidine-4-carboxylate
—— Ethyl 2-[[2-(4-bromo-2,6-dimethylphenoxy)acetyl]amino]-6-methyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate —— C22H26BrNO4S
Ethyl 2-[[2-(4-bromo-2,6-dimethylphenoxy)acetyl]amino]-6-methyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
—— ethyl (6R)-4-[[4-(cyclopropanecarbonyl)piperazin-1-yl]methyl]-2-oxo-3-prop-2-enyl-6-thiophen-3-yl-1,6-dihydropyrimidine-5-carboxylate —— C23H30N4O4S
ethyl (6R)-4-[[4-(cyclopropanecarbonyl)piperazin-1-yl]methyl]-2-oxo-3-prop-2-enyl-6-thiophen-3-yl-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6R)-6-(3,5-dimethoxyphenyl)-3-ethyl-4-[[4-(ethylcarbamoyl)-1,4-diazepan-1-yl]methyl]-2-oxo-1,6-dihydropyrimidine-5-carboxylate —— C26H39N5O6
ethyl (6R)-6-(3,5-dimethoxyphenyl)-3-ethyl-4-[[4-(ethylcarbamoyl)-1,4-diazepan-1-yl]methyl]-2-oxo-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6R)-6-(2,4-dichlorophenyl)-3-ethyl-4-[[4-(2-methylpropanoyl)piperazin-1-yl]methyl]-2-oxo-1,6-dihydropyrimidine-5-carboxylate —— C24H32Cl2N4O4
ethyl (6R)-6-(2,4-dichlorophenyl)-3-ethyl-4-[[4-(2-methylpropanoyl)piperazin-1-yl]methyl]-2-oxo-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6R)-4-[[(3R)-4-(tert-butylcarbamoyl)-3-methylpiperazin-1-yl]methyl]-3-ethyl-6-(2-methoxyphenyl)-2-oxo-1,6-dihydropyrimidine-5-carboxylate —— C27H41N5O5
ethyl (6R)-4-[[(3R)-4-(tert-butylcarbamoyl)-3-methylpiperazin-1-yl]methyl]-3-ethyl-6-(2-methoxyphenyl)-2-oxo-1,6-dihydropyrimidine-5-carboxylate
—— Ethyl 2,2,2-trichloro-1-{[(2,4-dibromo-5-methylanilino)carbothioyl]amino}ethylcarbamate —— C13H14Br2Cl3N3O2S
Ethyl 2,2,2-trichloro-1-{[(2,4-dibromo-5-methylanilino)carbothioyl]amino}ethylcarbamate
—— ethyl (3R)-1-(1-benzyl-5-phenylpyrazole-4-carbonyl)piperidine-3-carboxylate —— C25H27N3O3
ethyl (3R)-1-(1-benzyl-5-phenylpyrazole-4-carbonyl)piperidine-3-carboxylate
—— ethyl (6R)-4-[[(3R)-4-(ethylcarbamoyl)-3-methylpiperazin-1-yl]methyl]-2-oxo-3-prop-2-enyl-6-thiophen-3-yl-1,6-dihydropyrimidine-5-carboxylate —— C23H33N5O4S
ethyl (6R)-4-[[(3R)-4-(ethylcarbamoyl)-3-methylpiperazin-1-yl]methyl]-2-oxo-3-prop-2-enyl-6-thiophen-3-yl-1,6-dihydropyrimidine-5-carboxylate
—— Ethyl 2-[3-(4-butoxyphenyl)prop-2-enoylamino]-4,5-dimethylthiophene-3-carboxylate —— C22H27NO4S
Ethyl 2-[3-(4-butoxyphenyl)prop-2-enoylamino]-4,5-dimethylthiophene-3-carboxylate
—— ethyl (6S)-6-(2,4-dimethoxyphenyl)-3-ethyl-2-oxo-4-[[4-(propylcarbamoyl)-1,4-diazepan-1-yl]methyl]-1,6-dihydropyrimidine-5-carboxylate —— C27H41N5O6
ethyl (6S)-6-(2,4-dimethoxyphenyl)-3-ethyl-2-oxo-4-[[4-(propylcarbamoyl)-1,4-diazepan-1-yl]methyl]-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6S)-4-[(4-benzoylpiperazin-1-yl)methyl]-3-ethyl-2-oxo-6-thiophen-3-yl-1,6-dihydropyrimidine-5-carboxylate —— C25H30N4O4S
ethyl (6S)-4-[(4-benzoylpiperazin-1-yl)methyl]-3-ethyl-2-oxo-6-thiophen-3-yl-1,6-dihydropyrimidine-5-carboxylate
—— Ethyl 2-[[2-(2-ethylphenoxy)acetyl]amino]-6-methyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate —— C22H27NO4S
Ethyl 2-[[2-(2-ethylphenoxy)acetyl]amino]-6-methyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
—— ethyl (3S)-1-[3-[[(2S)-oxolan-2-yl]methyl-[5-(2,4,6-trimethylphenyl)-1,2-oxazole-3-carbonyl]amino]propanoyl]piperidine-3-carboxylate —— C29H39N3O6
ethyl (3S)-1-[3-[[(2S)-oxolan-2-yl]methyl-[5-(2,4,6-trimethylphenyl)-1,2-oxazole-3-carbonyl]amino]propanoyl]piperidine-3-carboxylate
—— ethyl (3R)-1-[3-[cyclopropyl-[5-(2,4,6-trimethylphenyl)-1,2-oxazole-3-carbonyl]amino]propanoyl]piperidine-3-carboxylate —— C27H35N3O5
ethyl (3R)-1-[3-[cyclopropyl-[5-(2,4,6-trimethylphenyl)-1,2-oxazole-3-carbonyl]amino]propanoyl]piperidine-3-carboxylate
—— ethyl (6S)-6-(3-chlorophenyl)-3-ethyl-4-[[(3S)-4-(ethylcarbamoyl)-3-methylpiperazin-1-yl]methyl]-2-oxo-1,6-dihydropyrimidine-5-carboxylate —— C24H34ClN5O4
ethyl (6S)-6-(3-chlorophenyl)-3-ethyl-4-[[(3S)-4-(ethylcarbamoyl)-3-methylpiperazin-1-yl]methyl]-2-oxo-1,6-dihydropyrimidine-5-carboxylate