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—— ethyl (3S)-1-[(3S)-1-[5-(3-methoxyphenyl)-1,2-oxazole-3-carbonyl]piperidine-3-carbonyl]piperidine-3-carboxylate —— C25H31N3O6
ethyl (3S)-1-[(3S)-1-[5-(3-methoxyphenyl)-1,2-oxazole-3-carbonyl]piperidine-3-carbonyl]piperidine-3-carboxylate
—— ethyl 1-[(2S)-2-[[5-(4-methylphenyl)-1,2-oxazole-3-carbonyl]amino]propanoyl]piperidine-4-carboxylate —— C22H27N3O5
ethyl 1-[(2S)-2-[[5-(4-methylphenyl)-1,2-oxazole-3-carbonyl]amino]propanoyl]piperidine-4-carboxylate
—— ethyl (6R)-4-[[(3R)-4-(benzenesulfonyl)-3-methylpiperazin-1-yl]methyl]-3-ethyl-2-oxo-6-phenyl-1,6-dihydropyrimidine-5-carboxylate —— C27H34N4O5S
ethyl (6R)-4-[[(3R)-4-(benzenesulfonyl)-3-methylpiperazin-1-yl]methyl]-3-ethyl-2-oxo-6-phenyl-1,6-dihydropyrimidine-5-carboxylate
—— Ethyl 2-methyl-5-phenyl-1-[3-(1,3-thiazol-2-ylcarbamoyl)phenyl]pyrrole-3-carboxylate —— C24H21N3O3S
Ethyl 2-methyl-5-phenyl-1-[3-(1,3-thiazol-2-ylcarbamoyl)phenyl]pyrrole-3-carboxylate
—— ethyl (6R)-3-ethyl-4-[[4-(ethylcarbamoyl)piperazin-1-yl]methyl]-2-oxo-6-phenyl-1,6-dihydropyrimidine-5-carboxylate —— C23H33N5O4
ethyl (6R)-3-ethyl-4-[[4-(ethylcarbamoyl)piperazin-1-yl]methyl]-2-oxo-6-phenyl-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6R)-3-methyl-2-oxo-4-[[4-(propan-2-ylcarbamoyl)-1,4-diazepan-1-yl]methyl]-6-[4-(trifluoromethyl)phenyl]-1,6-dihydropyrimidine-5-carboxylate —— C25H34F3N5O4
ethyl (6R)-3-methyl-2-oxo-4-[[4-(propan-2-ylcarbamoyl)-1,4-diazepan-1-yl]methyl]-6-[4-(trifluoromethyl)phenyl]-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6S)-3-ethyl-4-[[(3R)-3-methyl-4-(propylcarbamoyl)piperazin-1-yl]methyl]-2-oxo-6-phenyl-1,6-dihydropyrimidine-5-carboxylate —— C25H37N5O4
ethyl (6S)-3-ethyl-4-[[(3R)-3-methyl-4-(propylcarbamoyl)piperazin-1-yl]methyl]-2-oxo-6-phenyl-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6S)-3-ethyl-4-[[4-(ethylcarbamoyl)piperazin-1-yl]methyl]-2-oxo-6-phenyl-1,6-dihydropyrimidine-5-carboxylate —— C23H33N5O4
ethyl (6S)-3-ethyl-4-[[4-(ethylcarbamoyl)piperazin-1-yl]methyl]-2-oxo-6-phenyl-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6S)-3-ethyl-4-[[(3R)-3-methyl-4-(4-methylbenzoyl)piperazin-1-yl]methyl]-2-oxo-6-phenyl-1,6-dihydropyrimidine-5-carboxylate —— C29H36N4O4
ethyl (6S)-3-ethyl-4-[[(3R)-3-methyl-4-(4-methylbenzoyl)piperazin-1-yl]methyl]-2-oxo-6-phenyl-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6S)-3-ethyl-4-[[(3R)-4-(2-methoxyacetyl)-3-methylpiperazin-1-yl]methyl]-2-oxo-6-phenyl-1,6-dihydropyrimidine-5-carboxylate —— C24H34N4O5
ethyl (6S)-3-ethyl-4-[[(3R)-4-(2-methoxyacetyl)-3-methylpiperazin-1-yl]methyl]-2-oxo-6-phenyl-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (3R)-1-[4-(4-benzylpiperidin-1-yl)-2-phenylpyrimidine-5-carbonyl]piperidine-3-carboxylate —— C31H36N4O3
ethyl (3R)-1-[4-(4-benzylpiperidin-1-yl)-2-phenylpyrimidine-5-carbonyl]piperidine-3-carboxylate
—— Ethyl 2-methyl-1-{3-[(4-methylphenyl)carbamoyl]phenyl}-5-phenyl-1H-pyrrole-3-carboxylate —— C28H26N2O3
Ethyl 2-methyl-1-{3-[(4-methylphenyl)carbamoyl]phenyl}-5-phenyl-1H-pyrrole-3-carboxylate
—— ethyl (6S)-3-methyl-4-[[(3R)-3-methyl-4-(3-methylbutanoyl)piperazin-1-yl]methyl]-2-oxo-6-thiophen-3-yl-1,6-dihydropyrimidine-5-carboxylate —— C23H34N4O4S
ethyl (6S)-3-methyl-4-[[(3R)-3-methyl-4-(3-methylbutanoyl)piperazin-1-yl]methyl]-2-oxo-6-thiophen-3-yl-1,6-dihydropyrimidine-5-carboxylate
—— ethyl 1-[(2R)-2-[[5-(4-methylphenyl)-1,2-oxazole-3-carbonyl]amino]propanoyl]piperidine-4-carboxylate —— C22H27N3O5
ethyl 1-[(2R)-2-[[5-(4-methylphenyl)-1,2-oxazole-3-carbonyl]amino]propanoyl]piperidine-4-carboxylate
—— ethyl (6R)-3-ethyl-4-[[(3R)-4-(3-fluorobenzoyl)-3-methylpiperazin-1-yl]methyl]-6-(3-methylphenyl)-2-oxo-1,6-dihydropyrimidine-5-carboxylate —— C29H35FN4O4
ethyl (6R)-3-ethyl-4-[[(3R)-4-(3-fluorobenzoyl)-3-methylpiperazin-1-yl]methyl]-6-(3-methylphenyl)-2-oxo-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (3R)-1-[3-[[5-(3-methoxyphenyl)-1,2-oxazole-3-carbonyl]-[[(2S)-oxolan-2-yl]methyl]amino]propanoyl]piperidine-3-carboxylate —— C27H35N3O7
ethyl (3R)-1-[3-[[5-(3-methoxyphenyl)-1,2-oxazole-3-carbonyl]-[[(2S)-oxolan-2-yl]methyl]amino]propanoyl]piperidine-3-carboxylate
—— Ethyl 1-{2-[(3,4-dimethylphenyl)carbamoyl]ethyl}-2-methyl-5-phenyl-1H-pyrrole-3-carboxylate —— C25H28N2O3
Ethyl 1-{2-[(3,4-dimethylphenyl)carbamoyl]ethyl}-2-methyl-5-phenyl-1H-pyrrole-3-carboxylate
—— ethyl (6S)-4-[[4-(benzenesulfonyl)piperazin-1-yl]methyl]-6-(3-fluorophenyl)-3-methyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate —— C25H29FN4O5S
ethyl (6S)-4-[[4-(benzenesulfonyl)piperazin-1-yl]methyl]-6-(3-fluorophenyl)-3-methyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (3S)-1-[3-[benzyl-[5-(3-methoxyphenyl)-1,2-oxazole-3-carbonyl]amino]propanoyl]piperidine-3-carboxylate —— C29H33N3O6
ethyl (3S)-1-[3-[benzyl-[5-(3-methoxyphenyl)-1,2-oxazole-3-carbonyl]amino]propanoyl]piperidine-3-carboxylate
—— ethyl (6S)-3-ethyl-4-[[(3R)-4-(3-fluorobenzoyl)-3-methylpiperazin-1-yl]methyl]-2-oxo-6-phenyl-1,6-dihydropyrimidine-5-carboxylate —— C28H33FN4O4
ethyl (6S)-3-ethyl-4-[[(3R)-4-(3-fluorobenzoyl)-3-methylpiperazin-1-yl]methyl]-2-oxo-6-phenyl-1,6-dihydropyrimidine-5-carboxylate
—— Ethyl 1-(2-{[(2H-1,3-benzodioxol-5-YL)methyl]carbamoyl}ethyl)-2-methyl-5-phenyl-1H-pyrrole-3-carboxylate —— C25H26N2O5
Ethyl 1-(2-{[(2H-1,3-benzodioxol-5-YL)methyl]carbamoyl}ethyl)-2-methyl-5-phenyl-1H-pyrrole-3-carboxylate
—— ethyl (3R)-1-[4-(dimethylamino)-2-(4-fluorophenyl)pyrimidine-5-carbonyl]piperidine-3-carboxylate —— C21H25FN4O3
ethyl (3R)-1-[4-(dimethylamino)-2-(4-fluorophenyl)pyrimidine-5-carbonyl]piperidine-3-carboxylate
—— ethyl (6S)-3-ethyl-4-[[(3R)-4-(ethylcarbamoyl)-3-methylpiperazin-1-yl]methyl]-2-oxo-6-phenyl-1,6-dihydropyrimidine-5-carboxylate —— C24H35N5O4
ethyl (6S)-3-ethyl-4-[[(3R)-4-(ethylcarbamoyl)-3-methylpiperazin-1-yl]methyl]-2-oxo-6-phenyl-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6S)-3-methyl-2-oxo-4-[[4-(propylcarbamoyl)-1,4-diazepan-1-yl]methyl]-6-[4-(trifluoromethyl)phenyl]-1,6-dihydropyrimidine-5-carboxylate —— C25H34F3N5O4
ethyl (6S)-3-methyl-2-oxo-4-[[4-(propylcarbamoyl)-1,4-diazepan-1-yl]methyl]-6-[4-(trifluoromethyl)phenyl]-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6S)-3-ethyl-4-[[(3S)-3-methyl-4-propanoylpiperazin-1-yl]methyl]-2-oxo-6-phenyl-1,6-dihydropyrimidine-5-carboxylate —— C24H34N4O4
ethyl (6S)-3-ethyl-4-[[(3S)-3-methyl-4-propanoylpiperazin-1-yl]methyl]-2-oxo-6-phenyl-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6R)-3-ethyl-4-[[(3R)-4-(2-methoxyacetyl)-3-methylpiperazin-1-yl]methyl]-6-(3-methylphenyl)-2-oxo-1,6-dihydropyrimidine-5-carboxylate —— C25H36N4O5
ethyl (6R)-3-ethyl-4-[[(3R)-4-(2-methoxyacetyl)-3-methylpiperazin-1-yl]methyl]-6-(3-methylphenyl)-2-oxo-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (3S)-1-[(3S)-1-[5-(2-methoxyphenyl)-1,2-oxazole-3-carbonyl]piperidine-3-carbonyl]piperidine-3-carboxylate —— C25H31N3O6
ethyl (3S)-1-[(3S)-1-[5-(2-methoxyphenyl)-1,2-oxazole-3-carbonyl]piperidine-3-carbonyl]piperidine-3-carboxylate
—— ethyl (3R)-1-[2-[[5-(2-methoxyphenyl)-1,2-oxazole-3-carbonyl]amino]acetyl]piperidine-3-carboxylate —— C21H25N3O6
ethyl (3R)-1-[2-[[5-(2-methoxyphenyl)-1,2-oxazole-3-carbonyl]amino]acetyl]piperidine-3-carboxylate
—— ethyl (3R)-1-[3-[2-methoxyethyl-[5-(3-methoxyphenyl)-1,2-oxazole-3-carbonyl]amino]propanoyl]piperidine-3-carboxylate —— C25H33N3O7
ethyl (3R)-1-[3-[2-methoxyethyl-[5-(3-methoxyphenyl)-1,2-oxazole-3-carbonyl]amino]propanoyl]piperidine-3-carboxylate
—— ethyl (3S)-1-[3-[2-methoxyethyl-[5-(2-methoxyphenyl)-1,2-oxazole-3-carbonyl]amino]propanoyl]piperidine-3-carboxylate —— C25H33N3O7
ethyl (3S)-1-[3-[2-methoxyethyl-[5-(2-methoxyphenyl)-1,2-oxazole-3-carbonyl]amino]propanoyl]piperidine-3-carboxylate
—— Ethyl 1-[3-(cycloheptylcarbamoyl)phenyl]-2-methyl-5-phenyl-1H-pyrrole-3-carboxylate —— C28H32N2O3
Ethyl 1-[3-(cycloheptylcarbamoyl)phenyl]-2-methyl-5-phenyl-1H-pyrrole-3-carboxylate
—— ethyl (3S)-1-[(3R)-1-[5-(3-methoxyphenyl)-1,2-oxazole-3-carbonyl]piperidine-3-carbonyl]piperidine-3-carboxylate —— C25H31N3O6
ethyl (3S)-1-[(3R)-1-[5-(3-methoxyphenyl)-1,2-oxazole-3-carbonyl]piperidine-3-carbonyl]piperidine-3-carboxylate
—— ethyl (6S)-3-ethyl-4-[[(3S)-3-methyl-4-(propylcarbamoyl)piperazin-1-yl]methyl]-2-oxo-6-phenyl-1,6-dihydropyrimidine-5-carboxylate —— C25H37N5O4
ethyl (6S)-3-ethyl-4-[[(3S)-3-methyl-4-(propylcarbamoyl)piperazin-1-yl]methyl]-2-oxo-6-phenyl-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6S)-3-ethyl-2-oxo-6-phenyl-4-[[4-(propan-2-ylcarbamoyl)piperazin-1-yl]methyl]-1,6-dihydropyrimidine-5-carboxylate —— C24H35N5O4
ethyl (6S)-3-ethyl-2-oxo-6-phenyl-4-[[4-(propan-2-ylcarbamoyl)piperazin-1-yl]methyl]-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6R)-4-[[4-(ethylcarbamoyl)-1,4-diazepan-1-yl]methyl]-6-(3-fluorophenyl)-3-methyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate —— C23H32FN5O4
ethyl (6R)-4-[[4-(ethylcarbamoyl)-1,4-diazepan-1-yl]methyl]-6-(3-fluorophenyl)-3-methyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate
—— Ethyl 1-(2-{[(4-chlorophenyl)methyl]carbamoyl}ethyl)-2-methyl-5-phenyl-1H-pyrrole-3-carboxylate —— C24H25ClN2O3
Ethyl 1-(2-{[(4-chlorophenyl)methyl]carbamoyl}ethyl)-2-methyl-5-phenyl-1H-pyrrole-3-carboxylate
—— ethyl (3S)-1-[4-(4-benzylpiperidin-1-yl)-2-phenylpyrimidine-5-carbonyl]piperidine-3-carboxylate —— C31H36N4O3
ethyl (3S)-1-[4-(4-benzylpiperidin-1-yl)-2-phenylpyrimidine-5-carbonyl]piperidine-3-carboxylate
—— ethyl (6R)-3-methyl-2-oxo-4-[[4-(propylcarbamoyl)-1,4-diazepan-1-yl]methyl]-6-[4-(trifluoromethyl)phenyl]-1,6-dihydropyrimidine-5-carboxylate —— C25H34F3N5O4
ethyl (6R)-3-methyl-2-oxo-4-[[4-(propylcarbamoyl)-1,4-diazepan-1-yl]methyl]-6-[4-(trifluoromethyl)phenyl]-1,6-dihydropyrimidine-5-carboxylate
—— ethyl 2-[(3-bromo-4-methoxyphenyl)methylidene]-5-(4-methylsulfanylphenyl)-3-oxo-7-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C30H25BrN2O4S2
ethyl 2-[(3-bromo-4-methoxyphenyl)methylidene]-5-(4-methylsulfanylphenyl)-3-oxo-7-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (6R)-3-ethyl-4-[[(3R)-3-methyl-4-(2-methylpropanoyl)piperazin-1-yl]methyl]-2-oxo-6-phenyl-1,6-dihydropyrimidine-5-carboxylate —— C25H36N4O4
ethyl (6R)-3-ethyl-4-[[(3R)-3-methyl-4-(2-methylpropanoyl)piperazin-1-yl]methyl]-2-oxo-6-phenyl-1,6-dihydropyrimidine-5-carboxylate
—— ethyl 1-[3-[[5-(4-methoxyphenyl)-1,2-oxazole-3-carbonyl]-[[(2R)-oxolan-2-yl]methyl]amino]propanoyl]piperidine-4-carboxylate —— C27H35N3O7
ethyl 1-[3-[[5-(4-methoxyphenyl)-1,2-oxazole-3-carbonyl]-[[(2R)-oxolan-2-yl]methyl]amino]propanoyl]piperidine-4-carboxylate
—— ethyl 1-ethyl-4-[2-[(4-methoxybenzoyl)-[[(2S)-oxolan-2-yl]methyl]amino]acetyl]-3,5-dimethylpyrrole-2-carboxylate —— C26H34N2O6
ethyl 1-ethyl-4-[2-[(4-methoxybenzoyl)-[[(2S)-oxolan-2-yl]methyl]amino]acetyl]-3,5-dimethylpyrrole-2-carboxylate
—— ethyl 4-[[[2-[benzyl-[2-(1H-indol-3-yl)ethyl]amino]-2-oxoethyl]-cyclopropylcarbamoyl]amino]benzoate —— C32H34N4O4
ethyl 4-[[[2-[benzyl-[2-(1H-indol-3-yl)ethyl]amino]-2-oxoethyl]-cyclopropylcarbamoyl]amino]benzoate
—— ethyl (3S)-1-[4-[4-(2-methylphenyl)piperazin-1-yl]-2-phenylpyrimidine-5-carbonyl]piperidine-3-carboxylate —— C30H35N5O3
ethyl (3S)-1-[4-[4-(2-methylphenyl)piperazin-1-yl]-2-phenylpyrimidine-5-carbonyl]piperidine-3-carboxylate
—— ethyl (6R)-4-[[4-(cyclopropanecarbonyl)piperazin-1-yl]methyl]-6-(3-fluorophenyl)-3-methyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate —— C23H29FN4O4
ethyl (6R)-4-[[4-(cyclopropanecarbonyl)piperazin-1-yl]methyl]-6-(3-fluorophenyl)-3-methyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6S)-4-[[(3R)-4-(3-fluorobenzoyl)-3-methylpiperazin-1-yl]methyl]-6-(3-fluorophenyl)-3-methyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate —— C27H30F2N4O4
ethyl (6S)-4-[[(3R)-4-(3-fluorobenzoyl)-3-methylpiperazin-1-yl]methyl]-6-(3-fluorophenyl)-3-methyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6R)-6-(3-fluorophenyl)-3-methyl-4-[[(3R)-3-methyl-4-(phenylcarbamoyl)piperazin-1-yl]methyl]-2-oxo-1,6-dihydropyrimidine-5-carboxylate —— C27H32FN5O4
ethyl (6R)-6-(3-fluorophenyl)-3-methyl-4-[[(3R)-3-methyl-4-(phenylcarbamoyl)piperazin-1-yl]methyl]-2-oxo-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6R)-6-(3-fluorophenyl)-4-[[4-(4-methoxybenzoyl)-1,4-diazepan-1-yl]methyl]-3-methyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate —— C28H33FN4O5
ethyl (6R)-6-(3-fluorophenyl)-4-[[4-(4-methoxybenzoyl)-1,4-diazepan-1-yl]methyl]-3-methyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6S)-4-[[(3R)-4-(4-chlorobenzoyl)-3-methylpiperazin-1-yl]methyl]-6-(3-fluorophenyl)-3-methyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate —— C27H30ClFN4O4
ethyl (6S)-4-[[(3R)-4-(4-chlorobenzoyl)-3-methylpiperazin-1-yl]methyl]-6-(3-fluorophenyl)-3-methyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6R)-6-(3-fluorophenyl)-4-[[4-(furan-2-carbonyl)piperazin-1-yl]methyl]-3-methyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate —— C24H27FN4O5
ethyl (6R)-6-(3-fluorophenyl)-4-[[4-(furan-2-carbonyl)piperazin-1-yl]methyl]-3-methyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate