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—— ethyl (6S)-6-(2,3-dimethoxyphenyl)-3-ethyl-2-oxo-4-[[4-(propan-2-ylcarbamoyl)piperazin-1-yl]methyl]-1,6-dihydropyrimidine-5-carboxylate —— C26H39N5O6
ethyl (6S)-6-(2,3-dimethoxyphenyl)-3-ethyl-2-oxo-4-[[4-(propan-2-ylcarbamoyl)piperazin-1-yl]methyl]-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6S)-6-(2,3-dimethoxyphenyl)-3-ethyl-4-[[(3S)-4-(ethylcarbamoyl)-3-methylpiperazin-1-yl]methyl]-2-oxo-1,6-dihydropyrimidine-5-carboxylate —— C26H39N5O6
ethyl (6S)-6-(2,3-dimethoxyphenyl)-3-ethyl-4-[[(3S)-4-(ethylcarbamoyl)-3-methylpiperazin-1-yl]methyl]-2-oxo-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6S)-6-(2,5-dimethylphenyl)-3-ethyl-2-oxo-4-[[4-(propylcarbamoyl)piperazin-1-yl]methyl]-1,6-dihydropyrimidine-5-carboxylate —— C26H39N5O4
ethyl (6S)-6-(2,5-dimethylphenyl)-3-ethyl-2-oxo-4-[[4-(propylcarbamoyl)piperazin-1-yl]methyl]-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6R)-2-oxo-6-phenyl-4-[(4-propanoyl-1,4-diazepan-1-yl)methyl]-3-prop-2-enyl-1,6-dihydropyrimidine-5-carboxylate —— C25H34N4O4
ethyl (6R)-2-oxo-6-phenyl-4-[(4-propanoyl-1,4-diazepan-1-yl)methyl]-3-prop-2-enyl-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6S)-6-(2,5-dimethoxyphenyl)-3-ethyl-2-oxo-4-[(4-propanoyl-1,4-diazepan-1-yl)methyl]-1,6-dihydropyrimidine-5-carboxylate —— C26H38N4O6
ethyl (6S)-6-(2,5-dimethoxyphenyl)-3-ethyl-2-oxo-4-[(4-propanoyl-1,4-diazepan-1-yl)methyl]-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6R)-6-(2,5-dimethylphenyl)-3-ethyl-2-oxo-4-[[4-(propylcarbamoyl)-1,4-diazepan-1-yl]methyl]-1,6-dihydropyrimidine-5-carboxylate —— C27H41N5O4
ethyl (6R)-6-(2,5-dimethylphenyl)-3-ethyl-2-oxo-4-[[4-(propylcarbamoyl)-1,4-diazepan-1-yl]methyl]-1,6-dihydropyrimidine-5-carboxylate
—— Ethyl 2-[2-[4-(trifluoromethyl)benzoyl]oxypropanoylamino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate —— C22H22F3NO5S
Ethyl 2-[2-[4-(trifluoromethyl)benzoyl]oxypropanoylamino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
—— ethyl 2-[[3-ethoxy-4-[(4-fluorophenyl)methoxy]phenyl]methylidene]-5-(4-methoxyphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C33H31FN2O6S
ethyl 2-[[3-ethoxy-4-[(4-fluorophenyl)methoxy]phenyl]methylidene]-5-(4-methoxyphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (3S)-1-[1-(3-chlorophenyl)-3,5-di(propan-2-yl)pyrazole-4-carbonyl]piperidine-3-carboxylate —— C24H32ClN3O3
ethyl (3S)-1-[1-(3-chlorophenyl)-3,5-di(propan-2-yl)pyrazole-4-carbonyl]piperidine-3-carboxylate
—— ethyl (6R)-4-[(4-benzoylpiperazin-1-yl)methyl]-3-ethyl-6-(3-methoxyphenyl)-2-oxo-1,6-dihydropyrimidine-5-carboxylate —— C28H34N4O5
ethyl (6R)-4-[(4-benzoylpiperazin-1-yl)methyl]-3-ethyl-6-(3-methoxyphenyl)-2-oxo-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6S)-2-oxo-6-phenyl-4-[(4-propanoyl-1,4-diazepan-1-yl)methyl]-3-prop-2-enyl-1,6-dihydropyrimidine-5-carboxylate —— C25H34N4O4
ethyl (6S)-2-oxo-6-phenyl-4-[(4-propanoyl-1,4-diazepan-1-yl)methyl]-3-prop-2-enyl-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6S)-4-[[4-(cyclopropanecarbonyl)-1,4-diazepan-1-yl]methyl]-6-(2,3-dichlorophenyl)-3-ethyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate —— C25H32Cl2N4O4
ethyl (6S)-4-[[4-(cyclopropanecarbonyl)-1,4-diazepan-1-yl]methyl]-6-(2,3-dichlorophenyl)-3-ethyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6R)-6-(2,3-dimethoxyphenyl)-3-ethyl-2-oxo-4-[[4-(propan-2-ylcarbamoyl)-1,4-diazepan-1-yl]methyl]-1,6-dihydropyrimidine-5-carboxylate —— C27H41N5O6
ethyl (6R)-6-(2,3-dimethoxyphenyl)-3-ethyl-2-oxo-4-[[4-(propan-2-ylcarbamoyl)-1,4-diazepan-1-yl]methyl]-1,6-dihydropyrimidine-5-carboxylate
—— ethyl 1-[(3S)-8-methyl-4-(3-methylbenzoyl)-1-oxa-4-azaspiro[4.5]decane-3-carbonyl]piperidine-4-carboxylate —— C26H36N2O5
ethyl 1-[(3S)-8-methyl-4-(3-methylbenzoyl)-1-oxa-4-azaspiro[4.5]decane-3-carbonyl]piperidine-4-carboxylate
—— ethyl (6R)-6-(2,3-dimethoxyphenyl)-3-ethyl-4-[[(3R)-3-methyl-4-(propan-2-ylcarbamoyl)piperazin-1-yl]methyl]-2-oxo-1,6-dihydropyrimidine-5-carboxylate —— C27H41N5O6
ethyl (6R)-6-(2,3-dimethoxyphenyl)-3-ethyl-4-[[(3R)-3-methyl-4-(propan-2-ylcarbamoyl)piperazin-1-yl]methyl]-2-oxo-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6S)-3-ethyl-6-(2-methoxyphenyl)-4-[[(3S)-3-methyl-4-(propylcarbamoyl)piperazin-1-yl]methyl]-2-oxo-1,6-dihydropyrimidine-5-carboxylate —— C26H39N5O5
ethyl (6S)-3-ethyl-6-(2-methoxyphenyl)-4-[[(3S)-3-methyl-4-(propylcarbamoyl)piperazin-1-yl]methyl]-2-oxo-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6S)-4-[[4-(cyclopropanecarbonyl)piperazin-1-yl]methyl]-2-oxo-3-prop-2-enyl-6-thiophen-3-yl-1,6-dihydropyrimidine-5-carboxylate —— C23H30N4O4S
ethyl (6S)-4-[[4-(cyclopropanecarbonyl)piperazin-1-yl]methyl]-2-oxo-3-prop-2-enyl-6-thiophen-3-yl-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6R)-6-(2,5-dimethoxyphenyl)-3-ethyl-4-[[4-(ethylcarbamoyl)-1,4-diazepan-1-yl]methyl]-2-oxo-1,6-dihydropyrimidine-5-carboxylate —— C26H39N5O6
ethyl (6R)-6-(2,5-dimethoxyphenyl)-3-ethyl-4-[[4-(ethylcarbamoyl)-1,4-diazepan-1-yl]methyl]-2-oxo-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6R)-6-(2,5-dimethoxyphenyl)-3-ethyl-2-oxo-4-[(4-propanoyl-1,4-diazepan-1-yl)methyl]-1,6-dihydropyrimidine-5-carboxylate —— C26H38N4O6
ethyl (6R)-6-(2,5-dimethoxyphenyl)-3-ethyl-2-oxo-4-[(4-propanoyl-1,4-diazepan-1-yl)methyl]-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (3S)-1-(1-benzyl-5-phenylpyrazole-4-carbonyl)piperidine-3-carboxylate —— C25H27N3O3
ethyl (3S)-1-(1-benzyl-5-phenylpyrazole-4-carbonyl)piperidine-3-carboxylate
—— ethyl (6R)-4-[[(3R)-4-benzoyl-3-methylpiperazin-1-yl]methyl]-3-ethyl-6-(3-methoxyphenyl)-2-oxo-1,6-dihydropyrimidine-5-carboxylate —— C29H36N4O5
ethyl (6R)-4-[[(3R)-4-benzoyl-3-methylpiperazin-1-yl]methyl]-3-ethyl-6-(3-methoxyphenyl)-2-oxo-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6S)-4-[[(3R)-4-(tert-butylcarbamoyl)-3-methylpiperazin-1-yl]methyl]-2-oxo-3-prop-2-enyl-6-thiophen-3-yl-1,6-dihydropyrimidine-5-carboxylate —— C25H37N5O4S
ethyl (6S)-4-[[(3R)-4-(tert-butylcarbamoyl)-3-methylpiperazin-1-yl]methyl]-2-oxo-3-prop-2-enyl-6-thiophen-3-yl-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6S)-3-ethyl-4-[[4-(ethylcarbamoyl)-1,4-diazepan-1-yl]methyl]-6-(2-methoxyphenyl)-2-oxo-1,6-dihydropyrimidine-5-carboxylate —— C25H37N5O5
ethyl (6S)-3-ethyl-4-[[4-(ethylcarbamoyl)-1,4-diazepan-1-yl]methyl]-6-(2-methoxyphenyl)-2-oxo-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6S)-6-(2,5-dimethylphenyl)-3-ethyl-2-oxo-4-[(4-propanoyl-1,4-diazepan-1-yl)methyl]-1,6-dihydropyrimidine-5-carboxylate —— C26H38N4O4
ethyl (6S)-6-(2,5-dimethylphenyl)-3-ethyl-2-oxo-4-[(4-propanoyl-1,4-diazepan-1-yl)methyl]-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6S)-6-(3-chlorophenyl)-3-ethyl-4-[[4-(ethylcarbamoyl)-1,4-diazepan-1-yl]methyl]-2-oxo-1,6-dihydropyrimidine-5-carboxylate —— C24H34ClN5O4
ethyl (6S)-6-(3-chlorophenyl)-3-ethyl-4-[[4-(ethylcarbamoyl)-1,4-diazepan-1-yl]methyl]-2-oxo-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6R)-6-(3,4-dichlorophenyl)-3-ethyl-4-[[4-(ethylcarbamoyl)-1,4-diazepan-1-yl]methyl]-2-oxo-1,6-dihydropyrimidine-5-carboxylate —— C24H33Cl2N5O4
ethyl (6R)-6-(3,4-dichlorophenyl)-3-ethyl-4-[[4-(ethylcarbamoyl)-1,4-diazepan-1-yl]methyl]-2-oxo-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6S)-3-ethyl-2-oxo-4-[[4-(propan-2-ylcarbamoyl)piperazin-1-yl]methyl]-6-thiophen-3-yl-1,6-dihydropyrimidine-5-carboxylate —— C22H33N5O4S
ethyl (6S)-3-ethyl-2-oxo-4-[[4-(propan-2-ylcarbamoyl)piperazin-1-yl]methyl]-6-thiophen-3-yl-1,6-dihydropyrimidine-5-carboxylate
—— Ethyl 3-amino-3-(4-methoxy-2-propan-2-ylphenyl)propanoate —— C15H23NO3
Ethyl 3-amino-3-(4-methoxy-2-propan-2-ylphenyl)propanoate
—— ethyl (6R)-6-(2,4-dimethoxyphenyl)-3-ethyl-4-[[(3R)-3-methyl-4-(propan-2-ylcarbamoyl)piperazin-1-yl]methyl]-2-oxo-1,6-dihydropyrimidine-5-carboxylate —— C27H41N5O6
ethyl (6R)-6-(2,4-dimethoxyphenyl)-3-ethyl-4-[[(3R)-3-methyl-4-(propan-2-ylcarbamoyl)piperazin-1-yl]methyl]-2-oxo-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6S)-6-(3-chlorophenyl)-3-ethyl-2-oxo-4-[[4-(propan-2-ylcarbamoyl)piperazin-1-yl]methyl]-1,6-dihydropyrimidine-5-carboxylate —— C24H34ClN5O4
ethyl (6S)-6-(3-chlorophenyl)-3-ethyl-2-oxo-4-[[4-(propan-2-ylcarbamoyl)piperazin-1-yl]methyl]-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6S)-4-[[(3R)-3-methyl-4-(propan-2-ylcarbamoyl)piperazin-1-yl]methyl]-2-oxo-3-prop-2-enyl-6-thiophen-3-yl-1,6-dihydropyrimidine-5-carboxylate —— C24H35N5O4S
ethyl (6S)-4-[[(3R)-3-methyl-4-(propan-2-ylcarbamoyl)piperazin-1-yl]methyl]-2-oxo-3-prop-2-enyl-6-thiophen-3-yl-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6R)-3-ethyl-4-[[4-(ethylcarbamoyl)-1,4-diazepan-1-yl]methyl]-6-(2-methoxyphenyl)-2-oxo-1,6-dihydropyrimidine-5-carboxylate —— C25H37N5O5
ethyl (6R)-3-ethyl-4-[[4-(ethylcarbamoyl)-1,4-diazepan-1-yl]methyl]-6-(2-methoxyphenyl)-2-oxo-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6R)-3-ethyl-4-[[(3S)-4-(ethylcarbamoyl)-3-methylpiperazin-1-yl]methyl]-2-oxo-6-thiophen-3-yl-1,6-dihydropyrimidine-5-carboxylate —— C22H33N5O4S
ethyl (6R)-3-ethyl-4-[[(3S)-4-(ethylcarbamoyl)-3-methylpiperazin-1-yl]methyl]-2-oxo-6-thiophen-3-yl-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6R)-6-(3-chlorophenyl)-3-ethyl-4-[[4-(ethylcarbamoyl)piperazin-1-yl]methyl]-2-oxo-1,6-dihydropyrimidine-5-carboxylate —— C23H32ClN5O4
ethyl (6R)-6-(3-chlorophenyl)-3-ethyl-4-[[4-(ethylcarbamoyl)piperazin-1-yl]methyl]-2-oxo-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6S)-3-ethyl-6-(2-methoxyphenyl)-4-[[(3R)-3-methyl-4-(propylcarbamoyl)piperazin-1-yl]methyl]-2-oxo-1,6-dihydropyrimidine-5-carboxylate —— C26H39N5O5
ethyl (6S)-3-ethyl-6-(2-methoxyphenyl)-4-[[(3R)-3-methyl-4-(propylcarbamoyl)piperazin-1-yl]methyl]-2-oxo-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6R)-4-[[4-(2-methylpropanoyl)piperazin-1-yl]methyl]-2-oxo-6-phenyl-3-prop-2-enyl-1,6-dihydropyrimidine-5-carboxylate —— C25H34N4O4
ethyl (6R)-4-[[4-(2-methylpropanoyl)piperazin-1-yl]methyl]-2-oxo-6-phenyl-3-prop-2-enyl-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6R)-4-[[4-(tert-butylcarbamoyl)-1,4-diazepan-1-yl]methyl]-3-ethyl-6-(2-methoxyphenyl)-2-oxo-1,6-dihydropyrimidine-5-carboxylate —— C27H41N5O5
ethyl (6R)-4-[[4-(tert-butylcarbamoyl)-1,4-diazepan-1-yl]methyl]-3-ethyl-6-(2-methoxyphenyl)-2-oxo-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6R)-6-(3-chlorophenyl)-3-ethyl-4-[[4-(ethylcarbamoyl)-1,4-diazepan-1-yl]methyl]-2-oxo-1,6-dihydropyrimidine-5-carboxylate —— C24H34ClN5O4
ethyl (6R)-6-(3-chlorophenyl)-3-ethyl-4-[[4-(ethylcarbamoyl)-1,4-diazepan-1-yl]methyl]-2-oxo-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6R)-4-[[4-(tert-butylcarbamoyl)piperazin-1-yl]methyl]-2-oxo-3-prop-2-enyl-6-thiophen-3-yl-1,6-dihydropyrimidine-5-carboxylate —— C24H35N5O4S
ethyl (6R)-4-[[4-(tert-butylcarbamoyl)piperazin-1-yl]methyl]-2-oxo-3-prop-2-enyl-6-thiophen-3-yl-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6S)-6-(3,5-dimethoxyphenyl)-3-ethyl-2-oxo-4-[[4-(propylcarbamoyl)-1,4-diazepan-1-yl]methyl]-1,6-dihydropyrimidine-5-carboxylate —— C27H41N5O6
ethyl (6S)-6-(3,5-dimethoxyphenyl)-3-ethyl-2-oxo-4-[[4-(propylcarbamoyl)-1,4-diazepan-1-yl]methyl]-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6R)-6-(2,4-dichlorophenyl)-3-ethyl-4-[[4-(ethylcarbamoyl)piperazin-1-yl]methyl]-2-oxo-1,6-dihydropyrimidine-5-carboxylate —— C23H31Cl2N5O4
ethyl (6R)-6-(2,4-dichlorophenyl)-3-ethyl-4-[[4-(ethylcarbamoyl)piperazin-1-yl]methyl]-2-oxo-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6R)-6-(2,4-dimethoxyphenyl)-3-ethyl-2-oxo-4-[[4-(propan-2-ylcarbamoyl)-1,4-diazepan-1-yl]methyl]-1,6-dihydropyrimidine-5-carboxylate —— C27H41N5O6
ethyl (6R)-6-(2,4-dimethoxyphenyl)-3-ethyl-2-oxo-4-[[4-(propan-2-ylcarbamoyl)-1,4-diazepan-1-yl]methyl]-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6S)-6-(2,5-dimethylphenyl)-3-ethyl-4-[[(3R)-4-(4-fluorobenzoyl)-3-methylpiperazin-1-yl]methyl]-2-oxo-1,6-dihydropyrimidine-5-carboxylate —— C30H37FN4O4
ethyl (6S)-6-(2,5-dimethylphenyl)-3-ethyl-4-[[(3R)-4-(4-fluorobenzoyl)-3-methylpiperazin-1-yl]methyl]-2-oxo-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6R)-6-(3,5-dimethoxyphenyl)-3-ethyl-4-[[4-(ethylcarbamoyl)piperazin-1-yl]methyl]-2-oxo-1,6-dihydropyrimidine-5-carboxylate —— C25H37N5O6
ethyl (6R)-6-(3,5-dimethoxyphenyl)-3-ethyl-4-[[4-(ethylcarbamoyl)piperazin-1-yl]methyl]-2-oxo-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6S)-3-ethyl-2-oxo-4-[(4-propanoylpiperazin-1-yl)methyl]-6-thiophen-3-yl-1,6-dihydropyrimidine-5-carboxylate —— C21H30N4O4S
ethyl (6S)-3-ethyl-2-oxo-4-[(4-propanoylpiperazin-1-yl)methyl]-6-thiophen-3-yl-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6S)-3-ethyl-4-[[(3S)-4-(ethylcarbamoyl)-3-methylpiperazin-1-yl]methyl]-6-(2-methoxyphenyl)-2-oxo-1,6-dihydropyrimidine-5-carboxylate —— C25H37N5O5
ethyl (6S)-3-ethyl-4-[[(3S)-4-(ethylcarbamoyl)-3-methylpiperazin-1-yl]methyl]-6-(2-methoxyphenyl)-2-oxo-1,6-dihydropyrimidine-5-carboxylate
—— ethyl 1-[(2S)-2-[[5-(2,5-dimethylphenyl)-1,2-oxazole-3-carbonyl]amino]-3-methylbutanoyl]piperidine-4-carboxylate —— C25H33N3O5
ethyl 1-[(2S)-2-[[5-(2,5-dimethylphenyl)-1,2-oxazole-3-carbonyl]amino]-3-methylbutanoyl]piperidine-4-carboxylate
—— ethyl (6R)-3-ethyl-2-oxo-4-[[4-(propylcarbamoyl)piperazin-1-yl]methyl]-6-thiophen-3-yl-1,6-dihydropyrimidine-5-carboxylate —— C22H33N5O4S
ethyl (6R)-3-ethyl-2-oxo-4-[[4-(propylcarbamoyl)piperazin-1-yl]methyl]-6-thiophen-3-yl-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6S)-6-(2,4-dimethoxyphenyl)-3-ethyl-4-[[(3R)-3-methyl-4-(propan-2-ylcarbamoyl)piperazin-1-yl]methyl]-2-oxo-1,6-dihydropyrimidine-5-carboxylate —— C27H41N5O6
ethyl (6S)-6-(2,4-dimethoxyphenyl)-3-ethyl-4-[[(3R)-3-methyl-4-(propan-2-ylcarbamoyl)piperazin-1-yl]methyl]-2-oxo-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6R)-4-[[4-(cyclobutanecarbonyl)-1,4-diazepan-1-yl]methyl]-6-(2,5-dimethylphenyl)-3-ethyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate —— C28H40N4O4
ethyl (6R)-4-[[4-(cyclobutanecarbonyl)-1,4-diazepan-1-yl]methyl]-6-(2,5-dimethylphenyl)-3-ethyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate