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—— ethyl (6R)-4-[[4-(ethylcarbamoyl)-1,4-diazepan-1-yl]methyl]-6-(4-methoxyphenyl)-3-methyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate —— C24H35N5O5
ethyl (6R)-4-[[4-(ethylcarbamoyl)-1,4-diazepan-1-yl]methyl]-6-(4-methoxyphenyl)-3-methyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6R)-6-(4-chlorophenyl)-4-[[4-(cyclobutanecarbonyl)piperazin-1-yl]methyl]-2-oxo-3-prop-2-enyl-1,6-dihydropyrimidine-5-carboxylate —— C26H33ClN4O4
ethyl (6R)-6-(4-chlorophenyl)-4-[[4-(cyclobutanecarbonyl)piperazin-1-yl]methyl]-2-oxo-3-prop-2-enyl-1,6-dihydropyrimidine-5-carboxylate
—— ethyl 4-[(2R)-2-[acetyl(2-methylpropyl)amino]propanoyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate —— C18H28N2O4
ethyl 4-[(2R)-2-[acetyl(2-methylpropyl)amino]propanoyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate
—— ethyl 4-[(2R)-2-[(4-fluorophenyl)methyl-(4-methylbenzoyl)amino]propanoyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate —— C27H29FN2O4
ethyl 4-[(2R)-2-[(4-fluorophenyl)methyl-(4-methylbenzoyl)amino]propanoyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate
—— ethyl 2-[5-(3-ethoxycarbonyl-5-formyl-4-propyl-1H-pyrrol-2-yl)-1H-pyrrol-2-yl]-5-formyl-4-propyl-1H-pyrrole-3-carboxylate —— C26H31N3O6
ethyl 2-[5-(3-ethoxycarbonyl-5-formyl-4-propyl-1H-pyrrol-2-yl)-1H-pyrrol-2-yl]-5-formyl-4-propyl-1H-pyrrole-3-carboxylate
—— ethyl 4-[(2S)-2-[(4-fluorophenyl)methyl-(furan-2-carbonyl)amino]propanoyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate —— C24H25FN2O5
ethyl 4-[(2S)-2-[(4-fluorophenyl)methyl-(furan-2-carbonyl)amino]propanoyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate
—— ethyl (6R)-4-[[4-(4-chlorobenzoyl)piperazin-1-yl]methyl]-3-methyl-6-(4-methylphenyl)-2-oxo-1,6-dihydropyrimidine-5-carboxylate —— C27H31ClN4O4
ethyl (6R)-4-[[4-(4-chlorobenzoyl)piperazin-1-yl]methyl]-3-methyl-6-(4-methylphenyl)-2-oxo-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6S)-4-[[4-(ethylcarbamoyl)-1,4-diazepan-1-yl]methyl]-6-(4-methoxyphenyl)-3-methyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate —— C24H35N5O5
ethyl (6S)-4-[[4-(ethylcarbamoyl)-1,4-diazepan-1-yl]methyl]-6-(4-methoxyphenyl)-3-methyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6R)-4-[[4-(ethylcarbamoyl)piperazin-1-yl]methyl]-3-methyl-6-(4-methylphenyl)-2-oxo-1,6-dihydropyrimidine-5-carboxylate —— C23H33N5O4
ethyl (6R)-4-[[4-(ethylcarbamoyl)piperazin-1-yl]methyl]-3-methyl-6-(4-methylphenyl)-2-oxo-1,6-dihydropyrimidine-5-carboxylate
—— ethyl 4-[(2S)-2-[(4-fluorophenyl)methyl-(3-methylbutanoyl)amino]propanoyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate —— C24H31FN2O4
ethyl 4-[(2S)-2-[(4-fluorophenyl)methyl-(3-methylbutanoyl)amino]propanoyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate
—— ethyl (6R)-3-methyl-6-(4-methylphenyl)-2-oxo-4-[[4-(thiophene-2-carbonyl)piperazin-1-yl]methyl]-1,6-dihydropyrimidine-5-carboxylate —— C25H30N4O4S
ethyl (6R)-3-methyl-6-(4-methylphenyl)-2-oxo-4-[[4-(thiophene-2-carbonyl)piperazin-1-yl]methyl]-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6S)-3-ethyl-6-(4-methylphenyl)-2-oxo-4-[(4-propanoylpiperazin-1-yl)methyl]-1,6-dihydropyrimidine-5-carboxylate —— C24H34N4O4
ethyl (6S)-3-ethyl-6-(4-methylphenyl)-2-oxo-4-[(4-propanoylpiperazin-1-yl)methyl]-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6R)-3-ethyl-6-(2-methylphenyl)-2-oxo-4-[[4-(propan-2-ylcarbamoyl)piperazin-1-yl]methyl]-1,6-dihydropyrimidine-5-carboxylate —— C25H37N5O4
ethyl (6R)-3-ethyl-6-(2-methylphenyl)-2-oxo-4-[[4-(propan-2-ylcarbamoyl)piperazin-1-yl]methyl]-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6S)-3-methyl-6-(4-methylphenyl)-2-oxo-4-[[4-(propan-2-ylcarbamoyl)piperazin-1-yl]methyl]-1,6-dihydropyrimidine-5-carboxylate —— C24H35N5O4
ethyl (6S)-3-methyl-6-(4-methylphenyl)-2-oxo-4-[[4-(propan-2-ylcarbamoyl)piperazin-1-yl]methyl]-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6R)-3-ethyl-4-[[4-(4-methoxybenzoyl)piperazin-1-yl]methyl]-6-(2-methylphenyl)-2-oxo-1,6-dihydropyrimidine-5-carboxylate —— C29H36N4O5
ethyl (6R)-3-ethyl-4-[[4-(4-methoxybenzoyl)piperazin-1-yl]methyl]-6-(2-methylphenyl)-2-oxo-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6S)-4-[[4-(2-fluorobenzoyl)piperazin-1-yl]methyl]-3-methyl-6-(4-methylphenyl)-2-oxo-1,6-dihydropyrimidine-5-carboxylate —— C27H31FN4O4
ethyl (6S)-4-[[4-(2-fluorobenzoyl)piperazin-1-yl]methyl]-3-methyl-6-(4-methylphenyl)-2-oxo-1,6-dihydropyrimidine-5-carboxylate
—— ethyl 4-[(2R)-2-[3-methoxypropyl-(4-methylbenzoyl)amino]propanoyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate —— C24H32N2O5
ethyl 4-[(2R)-2-[3-methoxypropyl-(4-methylbenzoyl)amino]propanoyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate
—— ethyl (6R)-3-methyl-4-[[4-(4-methylbenzoyl)-1,4-diazepan-1-yl]methyl]-6-(3-methylphenyl)-2-oxo-1,6-dihydropyrimidine-5-carboxylate —— C29H36N4O4
ethyl (6R)-3-methyl-4-[[4-(4-methylbenzoyl)-1,4-diazepan-1-yl]methyl]-6-(3-methylphenyl)-2-oxo-1,6-dihydropyrimidine-5-carboxylate
—— ethyl 4-[(2R)-2-[3-methoxypropyl(2-methylpropanoyl)amino]propanoyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate —— C20H32N2O5
ethyl 4-[(2R)-2-[3-methoxypropyl(2-methylpropanoyl)amino]propanoyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate
—— ethyl (6R)-6-(4-methoxyphenyl)-3-methyl-2-oxo-4-[[4-(propan-2-ylcarbamoyl)-1,4-diazepan-1-yl]methyl]-1,6-dihydropyrimidine-5-carboxylate —— C25H37N5O5
ethyl (6R)-6-(4-methoxyphenyl)-3-methyl-2-oxo-4-[[4-(propan-2-ylcarbamoyl)-1,4-diazepan-1-yl]methyl]-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6R)-3-ethyl-6-(4-methylphenyl)-4-[[4-(2-methylpropanoyl)piperazin-1-yl]methyl]-2-oxo-1,6-dihydropyrimidine-5-carboxylate —— C25H36N4O4
ethyl (6R)-3-ethyl-6-(4-methylphenyl)-4-[[4-(2-methylpropanoyl)piperazin-1-yl]methyl]-2-oxo-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (3R)-1-[4-(4-ethylpiperazin-1-yl)-2-(4-fluorophenyl)pyrimidine-5-carbonyl]piperidine-3-carboxylate —— C25H32FN5O3
ethyl (3R)-1-[4-(4-ethylpiperazin-1-yl)-2-(4-fluorophenyl)pyrimidine-5-carbonyl]piperidine-3-carboxylate
—— ethyl (3R)-1-[2-(4-fluorophenyl)-4-(N-methylanilino)pyrimidine-5-carbonyl]piperidine-3-carboxylate —— C26H27FN4O3
ethyl (3R)-1-[2-(4-fluorophenyl)-4-(N-methylanilino)pyrimidine-5-carbonyl]piperidine-3-carboxylate
—— ethyl (3S)-1-[3-[2-methoxyethyl-[5-(3-methoxyphenyl)-1,2-oxazole-3-carbonyl]amino]propanoyl]piperidine-3-carboxylate —— C25H33N3O7
ethyl (3S)-1-[3-[2-methoxyethyl-[5-(3-methoxyphenyl)-1,2-oxazole-3-carbonyl]amino]propanoyl]piperidine-3-carboxylate
—— Ethyl 4-phenyl-2-[(4-propan-2-yloxybenzoyl)amino]-1,3-thiazole-5-carboxylate —— C22H22N2O4S
Ethyl 4-phenyl-2-[(4-propan-2-yloxybenzoyl)amino]-1,3-thiazole-5-carboxylate
—— ethyl (6R)-4-[[4-(2-fluorobenzoyl)-1,4-diazepan-1-yl]methyl]-3-methyl-6-(3-methylphenyl)-2-oxo-1,6-dihydropyrimidine-5-carboxylate —— C28H33FN4O4
ethyl (6R)-4-[[4-(2-fluorobenzoyl)-1,4-diazepan-1-yl]methyl]-3-methyl-6-(3-methylphenyl)-2-oxo-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (3S)-1-[4-(4-benzylpiperidin-1-yl)-2-(4-fluorophenyl)pyrimidine-5-carbonyl]piperidine-3-carboxylate —— C31H35FN4O3
ethyl (3S)-1-[4-(4-benzylpiperidin-1-yl)-2-(4-fluorophenyl)pyrimidine-5-carbonyl]piperidine-3-carboxylate
—— ethyl (6S)-4-[[4-(ethylcarbamoyl)-1,4-diazepan-1-yl]methyl]-3-methyl-2-oxo-6-(3-phenoxyphenyl)-1,6-dihydropyrimidine-5-carboxylate —— C29H37N5O5
ethyl (6S)-4-[[4-(ethylcarbamoyl)-1,4-diazepan-1-yl]methyl]-3-methyl-2-oxo-6-(3-phenoxyphenyl)-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (3R)-1-[4-[benzyl(methyl)amino]-2-(4-fluorophenyl)pyrimidine-5-carbonyl]piperidine-3-carboxylate —— C27H29FN4O3
ethyl (3R)-1-[4-[benzyl(methyl)amino]-2-(4-fluorophenyl)pyrimidine-5-carbonyl]piperidine-3-carboxylate
—— ethyl (6S)-4-[[4-(tert-butylcarbamoyl)-1,4-diazepan-1-yl]methyl]-3-ethyl-2-oxo-6-phenyl-1,6-dihydropyrimidine-5-carboxylate —— C26H39N5O4
ethyl (6S)-4-[[4-(tert-butylcarbamoyl)-1,4-diazepan-1-yl]methyl]-3-ethyl-2-oxo-6-phenyl-1,6-dihydropyrimidine-5-carboxylate
—— (E)-2-chloro-N-(3-ethyl-4-methoxybenzo[d]thiazol-2(3H)-ylidene)benzamide —— C17H15ClN2O2S
(E)-2-chloro-N-(3-ethyl-4-methoxybenzo[d]thiazol-2(3H)-ylidene)benzamide
—— ethyl (6S)-3-ethyl-4-[[4-(4-methoxybenzoyl)piperazin-1-yl]methyl]-6-(2-methylphenyl)-2-oxo-1,6-dihydropyrimidine-5-carboxylate —— C29H36N4O5
ethyl (6S)-3-ethyl-4-[[4-(4-methoxybenzoyl)piperazin-1-yl]methyl]-6-(2-methylphenyl)-2-oxo-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (3S)-1-[4-(4-ethylpiperazin-1-yl)-2-(4-fluorophenyl)pyrimidine-5-carbonyl]piperidine-3-carboxylate —— C25H32FN5O3
ethyl (3S)-1-[4-(4-ethylpiperazin-1-yl)-2-(4-fluorophenyl)pyrimidine-5-carbonyl]piperidine-3-carboxylate
—— ethyl (3R)-1-[4-(4-benzylpiperidin-1-yl)-2-(4-fluorophenyl)pyrimidine-5-carbonyl]piperidine-3-carboxylate —— C31H35FN4O3
ethyl (3R)-1-[4-(4-benzylpiperidin-1-yl)-2-(4-fluorophenyl)pyrimidine-5-carbonyl]piperidine-3-carboxylate
—— ethyl (6R)-6-(4-methoxyphenyl)-3-methyl-2-oxo-4-[[4-(propylcarbamoyl)piperazin-1-yl]methyl]-1,6-dihydropyrimidine-5-carboxylate —— C24H35N5O5
ethyl (6R)-6-(4-methoxyphenyl)-3-methyl-2-oxo-4-[[4-(propylcarbamoyl)piperazin-1-yl]methyl]-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (3S)-1-[(2S)-2-[[5-(3-methoxyphenyl)-1,2-oxazole-3-carbonyl]amino]-3-methylbutanoyl]piperidine-3-carboxylate —— C24H31N3O6
ethyl (3S)-1-[(2S)-2-[[5-(3-methoxyphenyl)-1,2-oxazole-3-carbonyl]amino]-3-methylbutanoyl]piperidine-3-carboxylate
—— ethyl (3S)-1-[2-(4-fluorophenyl)-4-[(2S)-2-methylpiperidin-1-yl]pyrimidine-5-carbonyl]piperidine-3-carboxylate —— C25H31FN4O3
ethyl (3S)-1-[2-(4-fluorophenyl)-4-[(2S)-2-methylpiperidin-1-yl]pyrimidine-5-carbonyl]piperidine-3-carboxylate
—— ethyl (3S)-1-[4-(dimethylamino)-2-(4-fluorophenyl)pyrimidine-5-carbonyl]piperidine-3-carboxylate —— C21H25FN4O3
ethyl (3S)-1-[4-(dimethylamino)-2-(4-fluorophenyl)pyrimidine-5-carbonyl]piperidine-3-carboxylate
—— ethyl (3R)-1-[(2S)-2-[[5-(3-methoxyphenyl)-1,2-oxazole-3-carbonyl]amino]-3-methylbutanoyl]piperidine-3-carboxylate —— C24H31N3O6
ethyl (3R)-1-[(2S)-2-[[5-(3-methoxyphenyl)-1,2-oxazole-3-carbonyl]amino]-3-methylbutanoyl]piperidine-3-carboxylate
—— Ethyl 1-[3-(tert-butylcarbamoyl)phenyl]-2-methyl-5-phenyl-1H-pyrrole-3-carboxylate —— C25H28N2O3
Ethyl 1-[3-(tert-butylcarbamoyl)phenyl]-2-methyl-5-phenyl-1H-pyrrole-3-carboxylate
—— ethyl 2-[(2-chlorophenyl)methylsulfanyl]-5-(2-methoxyphenyl)-4-oxo-7-phenyl-5,8-dihydro-3H-pyrido[2,3-d]pyrimidine-6-carboxylate —— C30H26ClN3O4S
ethyl 2-[(2-chlorophenyl)methylsulfanyl]-5-(2-methoxyphenyl)-4-oxo-7-phenyl-5,8-dihydro-3H-pyrido[2,3-d]pyrimidine-6-carboxylate
—— ethyl (3S)-1-[3-[[5-(3-methoxyphenyl)-1,2-oxazole-3-carbonyl]-[[(2R)-oxolan-2-yl]methyl]amino]propanoyl]piperidine-3-carboxylate —— C27H35N3O7
ethyl (3S)-1-[3-[[5-(3-methoxyphenyl)-1,2-oxazole-3-carbonyl]-[[(2R)-oxolan-2-yl]methyl]amino]propanoyl]piperidine-3-carboxylate
—— ethyl (3R)-1-[(2R)-2-[[5-(3-methoxyphenyl)-1,2-oxazole-3-carbonyl]amino]-3-methylbutanoyl]piperidine-3-carboxylate —— C24H31N3O6
ethyl (3R)-1-[(2R)-2-[[5-(3-methoxyphenyl)-1,2-oxazole-3-carbonyl]amino]-3-methylbutanoyl]piperidine-3-carboxylate
—— ethyl 1-[3-[[5-(3-chlorophenyl)-1,2-oxazole-3-carbonyl]-[[(2S)-oxolan-2-yl]methyl]amino]propanoyl]piperidine-4-carboxylate —— C26H32ClN3O6
ethyl 1-[3-[[5-(3-chlorophenyl)-1,2-oxazole-3-carbonyl]-[[(2S)-oxolan-2-yl]methyl]amino]propanoyl]piperidine-4-carboxylate
—— ethyl 1-[3-[[5-(3-methoxyphenyl)-1,2-oxazole-3-carbonyl]-[[(2R)-oxolan-2-yl]methyl]amino]propanoyl]piperidine-4-carboxylate —— C27H35N3O7
ethyl 1-[3-[[5-(3-methoxyphenyl)-1,2-oxazole-3-carbonyl]-[[(2R)-oxolan-2-yl]methyl]amino]propanoyl]piperidine-4-carboxylate
—— ethyl (3R)-1-[3-[[5-(3-methoxyphenyl)-1,2-oxazole-3-carbonyl]-[[(2R)-oxolan-2-yl]methyl]amino]propanoyl]piperidine-3-carboxylate —— C27H35N3O7
ethyl (3R)-1-[3-[[5-(3-methoxyphenyl)-1,2-oxazole-3-carbonyl]-[[(2R)-oxolan-2-yl]methyl]amino]propanoyl]piperidine-3-carboxylate
—— ethyl 1-[(2S)-2-[[5-(3-methoxyphenyl)-1,2-oxazole-3-carbonyl]amino]-3-methylbutanoyl]piperidine-4-carboxylate —— C24H31N3O6
ethyl 1-[(2S)-2-[[5-(3-methoxyphenyl)-1,2-oxazole-3-carbonyl]amino]-3-methylbutanoyl]piperidine-4-carboxylate
—— ethyl (3R)-1-[2-(4-fluorophenyl)-4-[(2S)-2-methylpiperidin-1-yl]pyrimidine-5-carbonyl]piperidine-3-carboxylate —— C25H31FN4O3
ethyl (3R)-1-[2-(4-fluorophenyl)-4-[(2S)-2-methylpiperidin-1-yl]pyrimidine-5-carbonyl]piperidine-3-carboxylate
—— ethyl 1-[3-[[5-(3-methoxyphenyl)-1,2-oxazole-3-carbonyl]-[[(2S)-oxolan-2-yl]methyl]amino]propanoyl]piperidine-4-carboxylate —— C27H35N3O7
ethyl 1-[3-[[5-(3-methoxyphenyl)-1,2-oxazole-3-carbonyl]-[[(2S)-oxolan-2-yl]methyl]amino]propanoyl]piperidine-4-carboxylate
—— ethyl (6S)-4-[[4-(2-chlorobenzoyl)piperazin-1-yl]methyl]-3-methyl-6-(4-methylphenyl)-2-oxo-1,6-dihydropyrimidine-5-carboxylate —— C27H31ClN4O4
ethyl (6S)-4-[[4-(2-chlorobenzoyl)piperazin-1-yl]methyl]-3-methyl-6-(4-methylphenyl)-2-oxo-1,6-dihydropyrimidine-5-carboxylate