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—— ethyl (6R)-3-methyl-4-[[(3R)-3-methyl-4-(3-methylbutanoyl)piperazin-1-yl]methyl]-6-(2-methylphenyl)-2-oxo-1,6-dihydropyrimidine-5-carboxylate —— C26H38N4O4
ethyl (6R)-3-methyl-4-[[(3R)-3-methyl-4-(3-methylbutanoyl)piperazin-1-yl]methyl]-6-(2-methylphenyl)-2-oxo-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6S)-3-methyl-6-(2-methylphenyl)-2-oxo-4-[[4-(propan-2-ylcarbamoyl)-1,4-diazepan-1-yl]methyl]-1,6-dihydropyrimidine-5-carboxylate —— C25H37N5O4
ethyl (6S)-3-methyl-6-(2-methylphenyl)-2-oxo-4-[[4-(propan-2-ylcarbamoyl)-1,4-diazepan-1-yl]methyl]-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (3R)-1-[4-[[(5-methyl-1,2-oxazole-3-carbonyl)amino]methyl]benzoyl]piperidine-3-carboxylate —— C21H25N3O5
ethyl (3R)-1-[4-[[(5-methyl-1,2-oxazole-3-carbonyl)amino]methyl]benzoyl]piperidine-3-carboxylate
—— ethyl (6S)-6-(4-chlorophenyl)-4-[[4-(ethylcarbamoyl)-1,4-diazepan-1-yl]methyl]-3-methyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate —— C23H32ClN5O4
ethyl (6S)-6-(4-chlorophenyl)-4-[[4-(ethylcarbamoyl)-1,4-diazepan-1-yl]methyl]-3-methyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6R)-6-(4-chlorophenyl)-4-[[(3R)-4-(2-fluorobenzoyl)-3-methylpiperazin-1-yl]methyl]-3-methyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate —— C27H30ClFN4O4
ethyl (6R)-6-(4-chlorophenyl)-4-[[(3R)-4-(2-fluorobenzoyl)-3-methylpiperazin-1-yl]methyl]-3-methyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (3S)-1-(2-phenyl-4-thiomorpholin-4-ylpyrimidine-5-carbonyl)piperidine-3-carboxylate —— C23H28N4O3S
ethyl (3S)-1-(2-phenyl-4-thiomorpholin-4-ylpyrimidine-5-carbonyl)piperidine-3-carboxylate
—— ethyl (6S)-4-[[4-(tert-butylcarbamoyl)-1,4-diazepan-1-yl]methyl]-6-(4-chlorophenyl)-3-methyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate —— C25H36ClN5O4
ethyl (6S)-4-[[4-(tert-butylcarbamoyl)-1,4-diazepan-1-yl]methyl]-6-(4-chlorophenyl)-3-methyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6S)-4-[[(3R)-4-(ethylcarbamoyl)-3-methylpiperazin-1-yl]methyl]-6-(3-fluorophenyl)-3-methyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate —— C23H32FN5O4
ethyl (6S)-4-[[(3R)-4-(ethylcarbamoyl)-3-methylpiperazin-1-yl]methyl]-6-(3-fluorophenyl)-3-methyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6R)-6-(4-chlorophenyl)-4-[[(3R)-4-(cyclopropanecarbonyl)-3-methylpiperazin-1-yl]methyl]-3-methyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate —— C24H31ClN4O4
ethyl (6R)-6-(4-chlorophenyl)-4-[[(3R)-4-(cyclopropanecarbonyl)-3-methylpiperazin-1-yl]methyl]-3-methyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6R)-3-methyl-6-(2-methylphenyl)-2-oxo-4-[[4-(propylcarbamoyl)-1,4-diazepan-1-yl]methyl]-1,6-dihydropyrimidine-5-carboxylate —— C25H37N5O4
ethyl (6R)-3-methyl-6-(2-methylphenyl)-2-oxo-4-[[4-(propylcarbamoyl)-1,4-diazepan-1-yl]methyl]-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6S)-3-methyl-4-[[4-(3-methylbutanoyl)-1,4-diazepan-1-yl]methyl]-6-(2-methylphenyl)-2-oxo-1,6-dihydropyrimidine-5-carboxylate —— C26H38N4O4
ethyl (6S)-3-methyl-4-[[4-(3-methylbutanoyl)-1,4-diazepan-1-yl]methyl]-6-(2-methylphenyl)-2-oxo-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (3R)-1-[3-[2-methoxyethyl-[5-(2-methoxyphenyl)-1,2-oxazole-3-carbonyl]amino]propanoyl]piperidine-3-carboxylate —— C25H33N3O7
ethyl (3R)-1-[3-[2-methoxyethyl-[5-(2-methoxyphenyl)-1,2-oxazole-3-carbonyl]amino]propanoyl]piperidine-3-carboxylate
—— ethyl (6S)-6-(3-fluorophenyl)-3-methyl-4-[[(3R)-3-methyl-4-(phenylcarbamoyl)piperazin-1-yl]methyl]-2-oxo-1,6-dihydropyrimidine-5-carboxylate —— C27H32FN5O4
ethyl (6S)-6-(3-fluorophenyl)-3-methyl-4-[[(3R)-3-methyl-4-(phenylcarbamoyl)piperazin-1-yl]methyl]-2-oxo-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6S)-6-(3-fluorophenyl)-4-[[4-[(2-methoxyphenyl)carbamoyl]piperazin-1-yl]methyl]-3-methyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate —— C27H32FN5O5
ethyl (6S)-6-(3-fluorophenyl)-4-[[4-[(2-methoxyphenyl)carbamoyl]piperazin-1-yl]methyl]-3-methyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6S)-6-(4-chlorophenyl)-4-[[(3R)-4-(furan-2-carbonyl)-3-methylpiperazin-1-yl]methyl]-3-methyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate —— C25H29ClN4O5
ethyl (6S)-6-(4-chlorophenyl)-4-[[(3R)-4-(furan-2-carbonyl)-3-methylpiperazin-1-yl]methyl]-3-methyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6S)-4-[[4-(benzenesulfonyl)-1,4-diazepan-1-yl]methyl]-3-methyl-6-(2-methylphenyl)-2-oxo-1,6-dihydropyrimidine-5-carboxylate —— C27H34N4O5S
ethyl (6S)-4-[[4-(benzenesulfonyl)-1,4-diazepan-1-yl]methyl]-3-methyl-6-(2-methylphenyl)-2-oxo-1,6-dihydropyrimidine-5-carboxylate
—— Ethyl 2-[2-bromo-4-[[2-(4-bromo-3-methylphenyl)-5-oxo-1,3-oxazol-4-ylidene]methyl]-6-methoxyphenoxy]acetate —— C22H19Br2NO6
Ethyl 2-[2-bromo-4-[[2-(4-bromo-3-methylphenyl)-5-oxo-1,3-oxazol-4-ylidene]methyl]-6-methoxyphenoxy]acetate
—— Ethyl 4-[[3-(1,3-benzodioxol-5-ylmethyl)-4-oxo-6-[(4-propoxyphenyl)carbamoyl]-1,3-thiazinan-2-ylidene]amino]benzoate —— C31H31N3O7S
Ethyl 4-[[3-(1,3-benzodioxol-5-ylmethyl)-4-oxo-6-[(4-propoxyphenyl)carbamoyl]-1,3-thiazinan-2-ylidene]amino]benzoate
—— ethyl (6R)-4-[[(3R)-4-(3-fluorobenzoyl)-3-methylpiperazin-1-yl]methyl]-3-methyl-6-(2-methylphenyl)-2-oxo-1,6-dihydropyrimidine-5-carboxylate —— C28H33FN4O4
ethyl (6R)-4-[[(3R)-4-(3-fluorobenzoyl)-3-methylpiperazin-1-yl]methyl]-3-methyl-6-(2-methylphenyl)-2-oxo-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6R)-6-(2-chlorophenyl)-3-methyl-2-oxo-4-[(4-propanoylpiperazin-1-yl)methyl]-1,6-dihydropyrimidine-5-carboxylate —— C22H29ClN4O4
ethyl (6R)-6-(2-chlorophenyl)-3-methyl-2-oxo-4-[(4-propanoylpiperazin-1-yl)methyl]-1,6-dihydropyrimidine-5-carboxylate
—— ethyl 4-[(2R)-2-[2-methoxyethyl(3-methylbutanoyl)amino]propanoyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate —— C20H32N2O5
ethyl 4-[(2R)-2-[2-methoxyethyl(3-methylbutanoyl)amino]propanoyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate
—— ethyl (6S)-4-[[4-(cyclopropanecarbonyl)piperazin-1-yl]methyl]-6-(3-fluorophenyl)-3-methyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate —— C23H29FN4O4
ethyl (6S)-4-[[4-(cyclopropanecarbonyl)piperazin-1-yl]methyl]-6-(3-fluorophenyl)-3-methyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6S)-6-(3-fluorophenyl)-4-[[4-(furan-2-carbonyl)piperazin-1-yl]methyl]-3-methyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate —— C24H27FN4O5
ethyl (6S)-6-(3-fluorophenyl)-4-[[4-(furan-2-carbonyl)piperazin-1-yl]methyl]-3-methyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6S)-6-(2-chlorophenyl)-4-[[4-(cyclobutanecarbonyl)piperazin-1-yl]methyl]-3-methyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate —— C24H31ClN4O4
ethyl (6S)-6-(2-chlorophenyl)-4-[[4-(cyclobutanecarbonyl)piperazin-1-yl]methyl]-3-methyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6S)-4-[[(3S)-4-(ethylcarbamoyl)-3-methylpiperazin-1-yl]methyl]-3-methyl-6-(2-methylphenyl)-2-oxo-1,6-dihydropyrimidine-5-carboxylate —— C24H35N5O4
ethyl (6S)-4-[[(3S)-4-(ethylcarbamoyl)-3-methylpiperazin-1-yl]methyl]-3-methyl-6-(2-methylphenyl)-2-oxo-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6R)-4-[[4-(cyclobutanecarbonyl)piperazin-1-yl]methyl]-6-(3-fluorophenyl)-3-methyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate —— C24H31FN4O4
ethyl (6R)-4-[[4-(cyclobutanecarbonyl)piperazin-1-yl]methyl]-6-(3-fluorophenyl)-3-methyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6S)-6-(3-fluorophenyl)-4-[[(3R)-4-(2-methoxyacetyl)-3-methylpiperazin-1-yl]methyl]-3-methyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate —— C23H31FN4O5
ethyl (6S)-6-(3-fluorophenyl)-4-[[(3R)-4-(2-methoxyacetyl)-3-methylpiperazin-1-yl]methyl]-3-methyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6R)-6-(4-chlorophenyl)-3-methyl-4-[[(3R)-3-methyl-4-(propan-2-ylcarbamoyl)piperazin-1-yl]methyl]-2-oxo-1,6-dihydropyrimidine-5-carboxylate —— C24H34ClN5O4
ethyl (6R)-6-(4-chlorophenyl)-3-methyl-4-[[(3R)-3-methyl-4-(propan-2-ylcarbamoyl)piperazin-1-yl]methyl]-2-oxo-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6S)-4-[[(3R)-4-(2-chlorobenzoyl)-3-methylpiperazin-1-yl]methyl]-3-ethyl-2-oxo-6-phenyl-1,6-dihydropyrimidine-5-carboxylate —— C28H33ClN4O4
ethyl (6S)-4-[[(3R)-4-(2-chlorobenzoyl)-3-methylpiperazin-1-yl]methyl]-3-ethyl-2-oxo-6-phenyl-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6S)-3-methyl-6-(2-methylphenyl)-4-[[(3S)-3-methyl-4-(propylcarbamoyl)piperazin-1-yl]methyl]-2-oxo-1,6-dihydropyrimidine-5-carboxylate —— C25H37N5O4
ethyl (6S)-3-methyl-6-(2-methylphenyl)-4-[[(3S)-3-methyl-4-(propylcarbamoyl)piperazin-1-yl]methyl]-2-oxo-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6S)-6-(3-fluorophenyl)-3-methyl-4-[[(3S)-3-methyl-4-(propylcarbamoyl)piperazin-1-yl]methyl]-2-oxo-1,6-dihydropyrimidine-5-carboxylate —— C24H34FN5O4
ethyl (6S)-6-(3-fluorophenyl)-3-methyl-4-[[(3S)-3-methyl-4-(propylcarbamoyl)piperazin-1-yl]methyl]-2-oxo-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (3S)-1-[3-[cyclopropyl-[5-(4-methoxyphenyl)-1,2-oxazole-3-carbonyl]amino]propanoyl]piperidine-3-carboxylate —— C25H31N3O6
ethyl (3S)-1-[3-[cyclopropyl-[5-(4-methoxyphenyl)-1,2-oxazole-3-carbonyl]amino]propanoyl]piperidine-3-carboxylate
—— ethyl (3S)-1-[(3R)-1-[5-(2-methoxyphenyl)-1,2-oxazole-3-carbonyl]piperidine-3-carbonyl]piperidine-3-carboxylate —— C25H31N3O6
ethyl (3S)-1-[(3R)-1-[5-(2-methoxyphenyl)-1,2-oxazole-3-carbonyl]piperidine-3-carbonyl]piperidine-3-carboxylate
—— ethyl (6R)-4-[[(3R)-4-benzoyl-3-methylpiperazin-1-yl]methyl]-3-ethyl-2-oxo-6-phenyl-1,6-dihydropyrimidine-5-carboxylate —— C28H34N4O4
ethyl (6R)-4-[[(3R)-4-benzoyl-3-methylpiperazin-1-yl]methyl]-3-ethyl-2-oxo-6-phenyl-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6S)-6-(3-fluorophenyl)-3-methyl-4-[[4-(4-methylbenzoyl)piperazin-1-yl]methyl]-2-oxo-1,6-dihydropyrimidine-5-carboxylate —— C27H31FN4O4
ethyl (6S)-6-(3-fluorophenyl)-3-methyl-4-[[4-(4-methylbenzoyl)piperazin-1-yl]methyl]-2-oxo-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6R)-4-[[4-(benzenesulfonyl)-1,4-diazepan-1-yl]methyl]-3-methyl-6-(2-methylphenyl)-2-oxo-1,6-dihydropyrimidine-5-carboxylate —— C27H34N4O5S
ethyl (6R)-4-[[4-(benzenesulfonyl)-1,4-diazepan-1-yl]methyl]-3-methyl-6-(2-methylphenyl)-2-oxo-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6R)-6-(2-chlorophenyl)-3-methyl-2-oxo-4-[[4-(phenylcarbamoyl)piperazin-1-yl]methyl]-1,6-dihydropyrimidine-5-carboxylate —— C26H30ClN5O4
ethyl (6R)-6-(2-chlorophenyl)-3-methyl-2-oxo-4-[[4-(phenylcarbamoyl)piperazin-1-yl]methyl]-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6S)-3-methyl-6-(2-methylphenyl)-2-oxo-4-[(4-propanoyl-1,4-diazepan-1-yl)methyl]-1,6-dihydropyrimidine-5-carboxylate —— C24H34N4O4
ethyl (6S)-3-methyl-6-(2-methylphenyl)-2-oxo-4-[(4-propanoyl-1,4-diazepan-1-yl)methyl]-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6S)-4-[[4-(4-chlorobenzoyl)-1,4-diazepan-1-yl]methyl]-3-methyl-6-(2-methylphenyl)-2-oxo-1,6-dihydropyrimidine-5-carboxylate —— C28H33ClN4O4
ethyl (6S)-4-[[4-(4-chlorobenzoyl)-1,4-diazepan-1-yl]methyl]-3-methyl-6-(2-methylphenyl)-2-oxo-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6S)-4-[[4-[(2-methoxyphenyl)carbamoyl]-1,4-diazepan-1-yl]methyl]-3-methyl-6-(2-methylphenyl)-2-oxo-1,6-dihydropyrimidine-5-carboxylate —— C29H37N5O5
ethyl (6S)-4-[[4-[(2-methoxyphenyl)carbamoyl]-1,4-diazepan-1-yl]methyl]-3-methyl-6-(2-methylphenyl)-2-oxo-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6R)-4-[[4-(tert-butylcarbamoyl)-1,4-diazepan-1-yl]methyl]-6-(4-chlorophenyl)-3-methyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate —— C25H36ClN5O4
ethyl (6R)-4-[[4-(tert-butylcarbamoyl)-1,4-diazepan-1-yl]methyl]-6-(4-chlorophenyl)-3-methyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6S)-6-(4-chlorophenyl)-3-methyl-2-oxo-4-[(4-propanoyl-1,4-diazepan-1-yl)methyl]-1,6-dihydropyrimidine-5-carboxylate —— C23H31ClN4O4
ethyl (6S)-6-(4-chlorophenyl)-3-methyl-2-oxo-4-[(4-propanoyl-1,4-diazepan-1-yl)methyl]-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6S)-3-ethyl-4-[[(3R)-4-(4-fluorobenzoyl)-3-methylpiperazin-1-yl]methyl]-2-oxo-6-phenyl-1,6-dihydropyrimidine-5-carboxylate —— C28H33FN4O4
ethyl (6S)-3-ethyl-4-[[(3R)-4-(4-fluorobenzoyl)-3-methylpiperazin-1-yl]methyl]-2-oxo-6-phenyl-1,6-dihydropyrimidine-5-carboxylate
—— ethyl 4-[(2S)-2-[tert-butylcarbamoyl(2-methoxyethyl)amino]propanoyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate —— C20H33N3O5
ethyl 4-[(2S)-2-[tert-butylcarbamoyl(2-methoxyethyl)amino]propanoyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate
—— ethyl 4-[(2R)-2-[2-methoxyethyl(propan-2-ylcarbamoyl)amino]propanoyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate —— C19H31N3O5
ethyl 4-[(2R)-2-[2-methoxyethyl(propan-2-ylcarbamoyl)amino]propanoyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate
—— ethyl (6S)-6-(2-chlorophenyl)-3-methyl-4-[[4-(4-methylbenzoyl)piperazin-1-yl]methyl]-2-oxo-1,6-dihydropyrimidine-5-carboxylate —— C27H31ClN4O4
ethyl (6S)-6-(2-chlorophenyl)-3-methyl-4-[[4-(4-methylbenzoyl)piperazin-1-yl]methyl]-2-oxo-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6R)-6-(4-chlorophenyl)-4-[[4-(cyclobutanecarbonyl)-1,4-diazepan-1-yl]methyl]-3-methyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate —— C25H33ClN4O4
ethyl (6R)-6-(4-chlorophenyl)-4-[[4-(cyclobutanecarbonyl)-1,4-diazepan-1-yl]methyl]-3-methyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6R)-3-methyl-6-(2-methylphenyl)-2-oxo-4-[[4-(propan-2-ylcarbamoyl)-1,4-diazepan-1-yl]methyl]-1,6-dihydropyrimidine-5-carboxylate —— C25H37N5O4
ethyl (6R)-3-methyl-6-(2-methylphenyl)-2-oxo-4-[[4-(propan-2-ylcarbamoyl)-1,4-diazepan-1-yl]methyl]-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6R)-6-(3-fluorophenyl)-3-methyl-4-[[(3R)-3-methyl-4-(3-methylbutanoyl)piperazin-1-yl]methyl]-2-oxo-1,6-dihydropyrimidine-5-carboxylate —— C25H35FN4O4
ethyl (6R)-6-(3-fluorophenyl)-3-methyl-4-[[(3R)-3-methyl-4-(3-methylbutanoyl)piperazin-1-yl]methyl]-2-oxo-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6R)-6-(3-fluorophenyl)-4-[[(3R)-4-(furan-2-carbonyl)-3-methylpiperazin-1-yl]methyl]-3-methyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate —— C25H29FN4O5
ethyl (6R)-6-(3-fluorophenyl)-4-[[(3R)-4-(furan-2-carbonyl)-3-methylpiperazin-1-yl]methyl]-3-methyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate