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—— Ethyl 2-{2-[(5-{[(4-butoxyphenyl)formamido]methyl}-4-methyl-4H-1,2,4-triazol-3-YL)sulfanyl]acetamido}-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate —— C28H35N5O5S2
Ethyl 2-{2-[(5-{[(4-butoxyphenyl)formamido]methyl}-4-methyl-4H-1,2,4-triazol-3-YL)sulfanyl]acetamido}-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
—— (E)-3-(4-fluorophenyl)-N-[(2R)-1-hydroxypropan-2-yl]prop-2-enamide —— C12H14FNO2
(E)-3-(4-fluorophenyl)-N-[(2R)-1-hydroxypropan-2-yl]prop-2-enamide
—— (E)-3-(5-bromothiophen-2-yl)-N-[(2R)-1-hydroxypropan-2-yl]prop-2-enamide —— C10H12BrNO2S
(E)-3-(5-bromothiophen-2-yl)-N-[(2R)-1-hydroxypropan-2-yl]prop-2-enamide
—— (E)-N-[(2R)-1-hydroxypropan-2-yl]-3-(1,3,5-trimethylpyrazol-4-yl)prop-2-enamide —— C12H19N3O2
(E)-N-[(2R)-1-hydroxypropan-2-yl]-3-(1,3,5-trimethylpyrazol-4-yl)prop-2-enamide
—— (E)-N-[(2R)-1-hydroxypropan-2-yl]-3-(4-nitrophenyl)prop-2-enamide —— C12H14N2O4
(E)-N-[(2R)-1-hydroxypropan-2-yl]-3-(4-nitrophenyl)prop-2-enamide
—— (E)-3-(3-chloro-4-fluorophenyl)-N-[(2R)-1-hydroxypropan-2-yl]prop-2-enamide —— C12H13ClFNO2
(E)-3-(3-chloro-4-fluorophenyl)-N-[(2R)-1-hydroxypropan-2-yl]prop-2-enamide
—— (E)-N-[(2R)-1-hydroxypropan-2-yl]-3-(4-methylphenyl)prop-2-enamide —— C13H17NO2
(E)-N-[(2R)-1-hydroxypropan-2-yl]-3-(4-methylphenyl)prop-2-enamide
—— Ethyl 2-(2-{[4-(2,5-dimethylphenyl)-5-{[(thiophen-2-YL)formamido]methyl}-4H-1,2,4-triazol-3-YL]sulfanyl}propanamido)-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate —— C30H33N5O4S3
Ethyl 2-(2-{[4-(2,5-dimethylphenyl)-5-{[(thiophen-2-YL)formamido]methyl}-4H-1,2,4-triazol-3-YL]sulfanyl}propanamido)-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
—— (E)-N-[(2R)-1-hydroxypropan-2-yl]-3-(3-methoxyphenyl)prop-2-enamide —— C13H17NO3
(E)-N-[(2R)-1-hydroxypropan-2-yl]-3-(3-methoxyphenyl)prop-2-enamide
—— ethyl N-[6-acetyl-2-[[4-[benzyl(methyl)sulfamoyl]benzoyl]amino]-5,7-dihydro-4H-thieno[2,3-c]pyridine-3-carbonyl]carbamate —— C28H30N4O7S2
ethyl N-[6-acetyl-2-[[4-[benzyl(methyl)sulfamoyl]benzoyl]amino]-5,7-dihydro-4H-thieno[2,3-c]pyridine-3-carbonyl]carbamate
—— (E)-3-(5-chloro-1,3-dimethylpyrazol-4-yl)-N-[(2R)-1-hydroxypropan-2-yl]prop-2-enamide —— C11H16ClN3O2
(E)-3-(5-chloro-1,3-dimethylpyrazol-4-yl)-N-[(2R)-1-hydroxypropan-2-yl]prop-2-enamide
—— (E)-3-(3-fluorophenyl)-N-[(2R)-1-hydroxypropan-2-yl]prop-2-enamide —— C12H14FNO2
(E)-3-(3-fluorophenyl)-N-[(2R)-1-hydroxypropan-2-yl]prop-2-enamide
—— Ethyl 3-[(5-formyl-2-methoxyphenyl)methoxy]benzoate —— C18H18O5
Ethyl 3-[(5-formyl-2-methoxyphenyl)methoxy]benzoate
—— (E)-N-[(2R)-1-hydroxypropan-2-yl]-3-(3-methylphenyl)prop-2-enamide —— C13H17NO2
(E)-N-[(2R)-1-hydroxypropan-2-yl]-3-(3-methylphenyl)prop-2-enamide
—— (E)-3-(6-chloroimidazo[2,1-b][1,3]thiazol-5-yl)-N-[(2R)-1-hydroxypropan-2-yl]prop-2-enamide —— C11H12ClN3O2S
(E)-3-(6-chloroimidazo[2,1-b][1,3]thiazol-5-yl)-N-[(2R)-1-hydroxypropan-2-yl]prop-2-enamide
—— (E)-3-(4-ethylphenyl)-N-[(2R)-1-hydroxypropan-2-yl]prop-2-enamide —— C14H19NO2
(E)-3-(4-ethylphenyl)-N-[(2R)-1-hydroxypropan-2-yl]prop-2-enamide
—— (E)-N-[(2S)-1-hydroxypropan-2-yl]-3-[5-[(1R,2R)-2-methylcyclopropyl]furan-2-yl]prop-2-enamide —— C14H19NO3
(E)-N-[(2S)-1-hydroxypropan-2-yl]-3-[5-[(1R,2R)-2-methylcyclopropyl]furan-2-yl]prop-2-enamide
—— (E)-3-[4-(dimethylamino)phenyl]-N-[(2R)-1-hydroxypropan-2-yl]prop-2-enamide —— C14H20N2O2
(E)-3-[4-(dimethylamino)phenyl]-N-[(2R)-1-hydroxypropan-2-yl]prop-2-enamide
—— Ethyl 4-[[2-(methylamino)benzoyl]amino]benzoate —— C17H18N2O3
Ethyl 4-[[2-(methylamino)benzoyl]amino]benzoate
—— Ethyl 2-[[4-[butyl(ethyl)sulfamoyl]benzoyl]amino]-4-phenyl-1,3-thiazole-5-carboxylate —— C25H29N3O5S2
Ethyl 2-[[4-[butyl(ethyl)sulfamoyl]benzoyl]amino]-4-phenyl-1,3-thiazole-5-carboxylate
—— (E)-N-[(2R)-1-hydroxypropan-2-yl]-3-(2-methoxy-5-methylphenyl)prop-2-enamide —— C14H19NO3
(E)-N-[(2R)-1-hydroxypropan-2-yl]-3-(2-methoxy-5-methylphenyl)prop-2-enamide
—— (E)-3-(3,4-dichlorophenyl)-N-[(2R)-1-hydroxypropan-2-yl]prop-2-enamide —— C12H13Cl2NO2
(E)-3-(3,4-dichlorophenyl)-N-[(2R)-1-hydroxypropan-2-yl]prop-2-enamide
—— (E)-N-[(2R)-1-hydroxypropan-2-yl]-3-(4-methoxyphenyl)prop-2-enamide —— C13H17NO3
(E)-N-[(2R)-1-hydroxypropan-2-yl]-3-(4-methoxyphenyl)prop-2-enamide
—— (E)-3-(5-bromo-2-fluorophenyl)-N-[(2R)-1-hydroxypropan-2-yl]prop-2-enamide —— C12H13BrFNO2
(E)-3-(5-bromo-2-fluorophenyl)-N-[(2R)-1-hydroxypropan-2-yl]prop-2-enamide
—— (E)-3-(1,3-benzodioxol-5-yl)-N-[(2R)-1-hydroxypropan-2-yl]prop-2-enamide —— C13H15NO4
(E)-3-(1,3-benzodioxol-5-yl)-N-[(2R)-1-hydroxypropan-2-yl]prop-2-enamide
—— (E)-3-(2,4-dichlorophenyl)-N-[(2R)-1-hydroxypropan-2-yl]prop-2-enamide —— C12H13Cl2NO2
(E)-3-(2,4-dichlorophenyl)-N-[(2R)-1-hydroxypropan-2-yl]prop-2-enamide
—— (E)-3-(2-ethoxyphenyl)-N-[(2R)-1-hydroxypropan-2-yl]prop-2-enamide —— C14H19NO3
(E)-3-(2-ethoxyphenyl)-N-[(2R)-1-hydroxypropan-2-yl]prop-2-enamide
—— Ethyl 2-{2-[(5-{[(3,5-dimethoxyphenyl)formamido]methyl}-4-(4-ethoxyphenyl)-4H-1,2,4-triazol-3-YL)sulfanyl]propanamido}-4H,5H,6H-cyclopenta[B]thiophene-3-carboxylate —— C33H37N5O7S2
Ethyl 2-{2-[(5-{[(3,5-dimethoxyphenyl)formamido]methyl}-4-(4-ethoxyphenyl)-4H-1,2,4-triazol-3-YL)sulfanyl]propanamido}-4H,5H,6H-cyclopenta[B]thiophene-3-carboxylate
—— (E)-3-(4-cyanophenyl)-N-[(2R)-1-hydroxypropan-2-yl]prop-2-enamide —— C13H14N2O2
(E)-3-(4-cyanophenyl)-N-[(2R)-1-hydroxypropan-2-yl]prop-2-enamide
—— Ethyl 4-[(5-chloro-2-methoxybenzoyl)-[(2-oxopyrrolidin-1-yl)methyl]amino]benzoate —— C22H23ClN2O5
Ethyl 4-[(5-chloro-2-methoxybenzoyl)-[(2-oxopyrrolidin-1-yl)methyl]amino]benzoate
—— (E)-3-(2,3-dichlorophenyl)-N-[(2R)-1-hydroxypropan-2-yl]prop-2-enamide —— C12H13Cl2NO2
(E)-3-(2,3-dichlorophenyl)-N-[(2R)-1-hydroxypropan-2-yl]prop-2-enamide
—— (E)-3-(2,5-dichlorophenyl)-N-[(2R)-1-hydroxypropan-2-yl]prop-2-enamide —— C12H13Cl2NO2
(E)-3-(2,5-dichlorophenyl)-N-[(2R)-1-hydroxypropan-2-yl]prop-2-enamide
—— (E)-3-(4-chlorophenyl)-N-[(2R)-1-hydroxypropan-2-yl]prop-2-enamide —— C12H14ClNO2
(E)-3-(4-chlorophenyl)-N-[(2R)-1-hydroxypropan-2-yl]prop-2-enamide
—— (E)-N-[(2S)-1-hydroxypropan-2-yl]-3-[5-[(1R,2S)-2-methylcyclopropyl]furan-2-yl]prop-2-enamide —— C14H19NO3
(E)-N-[(2S)-1-hydroxypropan-2-yl]-3-[5-[(1R,2S)-2-methylcyclopropyl]furan-2-yl]prop-2-enamide
—— Ethyl 4-[[2-oxo-1-(piperidin-1-ylmethyl)indol-3-ylidene]amino]benzoate —— C23H25N3O3
Ethyl 4-[[2-oxo-1-(piperidin-1-ylmethyl)indol-3-ylidene]amino]benzoate
—— Ethyl 2-[2-({1-[(3-fluorophenyl)methyl]-1H-indol-3-YL}sulfanyl)acetamido]-4H,5H,6H-cyclopenta[B]thiophene-3-carboxylate —— C27H25FN2O3S2
Ethyl 2-[2-({1-[(3-fluorophenyl)methyl]-1H-indol-3-YL}sulfanyl)acetamido]-4H,5H,6H-cyclopenta[B]thiophene-3-carboxylate
—— (E)-3-(2-chloro-6-fluorophenyl)-N-[(2R)-1-hydroxypropan-2-yl]prop-2-enamide —— C12H13ClFNO2
(E)-3-(2-chloro-6-fluorophenyl)-N-[(2R)-1-hydroxypropan-2-yl]prop-2-enamide
—— (E)-N-[(2R)-1-hydroxybutan-2-yl]-3-(4-methylphenyl)prop-2-enamide —— C14H19NO2
(E)-N-[(2R)-1-hydroxybutan-2-yl]-3-(4-methylphenyl)prop-2-enamide
—— (E)-3-(3-chlorophenyl)-N-[(2R)-1-hydroxybutan-2-yl]prop-2-enamide —— C13H16ClNO2
(E)-3-(3-chlorophenyl)-N-[(2R)-1-hydroxybutan-2-yl]prop-2-enamide
—— (E)-1-[(3S)-3-hydroxypiperidin-1-yl]-3-(2-methylpyrazol-3-yl)prop-2-en-1-one —— C12H17N3O2
(E)-1-[(3S)-3-hydroxypiperidin-1-yl]-3-(2-methylpyrazol-3-yl)prop-2-en-1-one
—— (E)-3-(5-bromo-2-fluorophenyl)-N-[(2S)-1-hydroxybutan-2-yl]prop-2-enamide —— C13H15BrFNO2
(E)-3-(5-bromo-2-fluorophenyl)-N-[(2S)-1-hydroxybutan-2-yl]prop-2-enamide
—— (E)-N-[(2S)-1-hydroxybutan-2-yl]-3-(4-methylphenyl)prop-2-enamide —— C14H19NO2
(E)-N-[(2S)-1-hydroxybutan-2-yl]-3-(4-methylphenyl)prop-2-enamide
—— (E)-3-(2,3-dichlorophenyl)-N-[(2R)-1-hydroxybutan-2-yl]prop-2-enamide —— C13H15Cl2NO2
(E)-3-(2,3-dichlorophenyl)-N-[(2R)-1-hydroxybutan-2-yl]prop-2-enamide
—— (E)-3-(5-chloro-1,3-dimethylpyrazol-4-yl)-N-[(2S)-1-hydroxybutan-2-yl]prop-2-enamide —— C12H18ClN3O2
(E)-3-(5-chloro-1,3-dimethylpyrazol-4-yl)-N-[(2S)-1-hydroxybutan-2-yl]prop-2-enamide
—— (E)-N-[(2R)-1-hydroxybutan-2-yl]-3-(2-methylphenyl)prop-2-enamide —— C14H19NO2
(E)-N-[(2R)-1-hydroxybutan-2-yl]-3-(2-methylphenyl)prop-2-enamide
—— (E)-3-(2-chloro-6-fluorophenyl)-N-[(2R)-1-hydroxybutan-2-yl]prop-2-enamide —— C13H15ClFNO2
(E)-3-(2-chloro-6-fluorophenyl)-N-[(2R)-1-hydroxybutan-2-yl]prop-2-enamide
—— (E)-3-(3-fluoro-4-methoxyphenyl)-N-[(2R)-1-hydroxybutan-2-yl]prop-2-enamide —— C14H18FNO3
(E)-3-(3-fluoro-4-methoxyphenyl)-N-[(2R)-1-hydroxybutan-2-yl]prop-2-enamide
—— (E)-3-[4-(dimethylamino)phenyl]-N-[(2R)-1-hydroxybutan-2-yl]prop-2-enamide —— C15H22N2O2
(E)-3-[4-(dimethylamino)phenyl]-N-[(2R)-1-hydroxybutan-2-yl]prop-2-enamide
—— (E)-3-(5-chloro-1,3-dimethylpyrazol-4-yl)-N-[(2R)-1-hydroxybutan-2-yl]prop-2-enamide —— C12H18ClN3O2
(E)-3-(5-chloro-1,3-dimethylpyrazol-4-yl)-N-[(2R)-1-hydroxybutan-2-yl]prop-2-enamide
—— ethyl (2Z,5S)-5-(4-chlorophenyl)-2-[(4-hydroxy-3-methoxy-5-prop-2-enylphenyl)methylidene]-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C27H25ClN2O5S
ethyl (2Z,5S)-5-(4-chlorophenyl)-2-[(4-hydroxy-3-methoxy-5-prop-2-enylphenyl)methylidene]-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate