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—— ethyl (6S)-4-[[4-(cyclopentanecarbonyl)piperazin-1-yl]methyl]-6-(2,4-dimethylphenyl)-3-ethyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate —— C28H40N4O4
ethyl (6S)-4-[[4-(cyclopentanecarbonyl)piperazin-1-yl]methyl]-6-(2,4-dimethylphenyl)-3-ethyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6S)-6-(2,4-dichlorophenyl)-3-methyl-2-oxo-4-[[4-(propylcarbamoyl)piperazin-1-yl]methyl]-1,6-dihydropyrimidine-5-carboxylate —— C23H31Cl2N5O4
ethyl (6S)-6-(2,4-dichlorophenyl)-3-methyl-2-oxo-4-[[4-(propylcarbamoyl)piperazin-1-yl]methyl]-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6R)-3-methyl-2-oxo-6-(4-propan-2-ylphenyl)-4-[[4-(thiophene-2-carbonyl)piperazin-1-yl]methyl]-1,6-dihydropyrimidine-5-carboxylate —— C27H34N4O4S
ethyl (6R)-3-methyl-2-oxo-6-(4-propan-2-ylphenyl)-4-[[4-(thiophene-2-carbonyl)piperazin-1-yl]methyl]-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6R)-6-(2,5-dimethylphenyl)-3-methyl-2-oxo-4-[[4-(propan-2-ylcarbamoyl)-1,4-diazepan-1-yl]methyl]-1,6-dihydropyrimidine-5-carboxylate —— C26H39N5O4
ethyl (6R)-6-(2,5-dimethylphenyl)-3-methyl-2-oxo-4-[[4-(propan-2-ylcarbamoyl)-1,4-diazepan-1-yl]methyl]-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6S)-6-(4-tert-butylphenyl)-4-[[(3R)-4-(2-methoxyacetyl)-3-methylpiperazin-1-yl]methyl]-3-methyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate —— C27H40N4O5
ethyl (6S)-6-(4-tert-butylphenyl)-4-[[(3R)-4-(2-methoxyacetyl)-3-methylpiperazin-1-yl]methyl]-3-methyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6S)-4-[[(3R)-4-(cyclopropanecarbonyl)-3-methylpiperazin-1-yl]methyl]-6-(2,3-dichlorophenyl)-3-methyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate —— C24H30Cl2N4O4
ethyl (6S)-4-[[(3R)-4-(cyclopropanecarbonyl)-3-methylpiperazin-1-yl]methyl]-6-(2,3-dichlorophenyl)-3-methyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6R)-4-[[4-(4-chlorobenzoyl)piperazin-1-yl]methyl]-6-(2,5-dimethylphenyl)-3-methyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate —— C28H33ClN4O4
ethyl (6R)-4-[[4-(4-chlorobenzoyl)piperazin-1-yl]methyl]-6-(2,5-dimethylphenyl)-3-methyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6S)-6-(4-tert-butylphenyl)-4-[[4-(2-fluorobenzoyl)piperazin-1-yl]methyl]-3-methyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate —— C30H37FN4O4
ethyl (6S)-6-(4-tert-butylphenyl)-4-[[4-(2-fluorobenzoyl)piperazin-1-yl]methyl]-3-methyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6S)-6-(4-tert-butylphenyl)-4-[[(3R)-4-(ethylcarbamoyl)-3-methylpiperazin-1-yl]methyl]-3-methyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate —— C27H41N5O4
ethyl (6S)-6-(4-tert-butylphenyl)-4-[[(3R)-4-(ethylcarbamoyl)-3-methylpiperazin-1-yl]methyl]-3-methyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6S)-6-(4-tert-butylphenyl)-4-[[4-(ethylcarbamoyl)piperazin-1-yl]methyl]-3-methyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate —— C26H39N5O4
ethyl (6S)-6-(4-tert-butylphenyl)-4-[[4-(ethylcarbamoyl)piperazin-1-yl]methyl]-3-methyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (3R)-1-[3-[[5-(2-chlorophenyl)-1,2-oxazole-3-carbonyl]-(2-methylpropyl)amino]propanoyl]piperidine-3-carboxylate —— C25H32ClN3O5
ethyl (3R)-1-[3-[[5-(2-chlorophenyl)-1,2-oxazole-3-carbonyl]-(2-methylpropyl)amino]propanoyl]piperidine-3-carboxylate
—— ethyl (6R)-4-[[4-(tert-butylcarbamoyl)piperazin-1-yl]methyl]-3-methyl-2-oxo-6-[2-(trifluoromethyl)phenyl]-1,6-dihydropyrimidine-5-carboxylate —— C25H34F3N5O4
ethyl (6R)-4-[[4-(tert-butylcarbamoyl)piperazin-1-yl]methyl]-3-methyl-2-oxo-6-[2-(trifluoromethyl)phenyl]-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6S)-6-(2,5-dimethylphenyl)-3-methyl-4-[[(3S)-3-methyl-4-propanoylpiperazin-1-yl]methyl]-2-oxo-1,6-dihydropyrimidine-5-carboxylate —— C25H36N4O4
ethyl (6S)-6-(2,5-dimethylphenyl)-3-methyl-4-[[(3S)-3-methyl-4-propanoylpiperazin-1-yl]methyl]-2-oxo-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6R)-6-(2,4-dichlorophenyl)-3-methyl-2-oxo-4-[[4-(propylcarbamoyl)piperazin-1-yl]methyl]-1,6-dihydropyrimidine-5-carboxylate —— C23H31Cl2N5O4
ethyl (6R)-6-(2,4-dichlorophenyl)-3-methyl-2-oxo-4-[[4-(propylcarbamoyl)piperazin-1-yl]methyl]-1,6-dihydropyrimidine-5-carboxylate
—— ethyl 1-ethyl-4-[(2S)-2-[(4-fluorophenyl)methyl-(3-methylbutanoyl)amino]propanoyl]-3,5-dimethylpyrrole-2-carboxylate —— C26H35FN2O4
ethyl 1-ethyl-4-[(2S)-2-[(4-fluorophenyl)methyl-(3-methylbutanoyl)amino]propanoyl]-3,5-dimethylpyrrole-2-carboxylate
—— ethyl (6R)-6-(2,5-dimethylphenyl)-4-[[4-(4-fluorobenzoyl)piperazin-1-yl]methyl]-3-methyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate —— C28H33FN4O4
ethyl (6R)-6-(2,5-dimethylphenyl)-4-[[4-(4-fluorobenzoyl)piperazin-1-yl]methyl]-3-methyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6S)-6-(2,4-dimethylphenyl)-3-methyl-4-[[4-(3-methylbutanoyl)-1,4-diazepan-1-yl]methyl]-2-oxo-1,6-dihydropyrimidine-5-carboxylate —— C27H40N4O4
ethyl (6S)-6-(2,4-dimethylphenyl)-3-methyl-4-[[4-(3-methylbutanoyl)-1,4-diazepan-1-yl]methyl]-2-oxo-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6S)-6-(2,4-dimethylphenyl)-4-[[4-(2-methoxyacetyl)-1,4-diazepan-1-yl]methyl]-3-methyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate —— C25H36N4O5
ethyl (6S)-6-(2,4-dimethylphenyl)-4-[[4-(2-methoxyacetyl)-1,4-diazepan-1-yl]methyl]-3-methyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6S)-4-[[4-(cyclopentanecarbonyl)piperazin-1-yl]methyl]-3-methyl-2-oxo-6-(4-propan-2-ylphenyl)-1,6-dihydropyrimidine-5-carboxylate —— C28H40N4O4
ethyl (6S)-4-[[4-(cyclopentanecarbonyl)piperazin-1-yl]methyl]-3-methyl-2-oxo-6-(4-propan-2-ylphenyl)-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6R)-6-(2,3-dichlorophenyl)-3-methyl-2-oxo-4-[[4-(propan-2-ylcarbamoyl)piperazin-1-yl]methyl]-1,6-dihydropyrimidine-5-carboxylate —— C23H31Cl2N5O4
ethyl (6R)-6-(2,3-dichlorophenyl)-3-methyl-2-oxo-4-[[4-(propan-2-ylcarbamoyl)piperazin-1-yl]methyl]-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6S)-6-(2-chlorophenyl)-3-ethyl-2-oxo-4-[[4-(propan-2-ylcarbamoyl)piperazin-1-yl]methyl]-1,6-dihydropyrimidine-5-carboxylate —— C24H34ClN5O4
ethyl (6S)-6-(2-chlorophenyl)-3-ethyl-2-oxo-4-[[4-(propan-2-ylcarbamoyl)piperazin-1-yl]methyl]-1,6-dihydropyrimidine-5-carboxylate
—— ethyl 6-[5-({[3-cyano-4,6-bis(4-methoxyphenyl)-2-pyridinyl]thio}methyl)-2-oxo-2,3-dihydro-1H-imidazol-4-yl]-6-oxohexanoate —— C32H32N4O6S
ethyl 6-[5-({[3-cyano-4,6-bis(4-methoxyphenyl)-2-pyridinyl]thio}methyl)-2-oxo-2,3-dihydro-1H-imidazol-4-yl]-6-oxohexanoate
—— ethyl (6R)-4-[[4-(tert-butylcarbamoyl)piperazin-1-yl]methyl]-6-(2,4-dichlorophenyl)-3-methyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate —— C24H33Cl2N5O4
ethyl (6R)-4-[[4-(tert-butylcarbamoyl)piperazin-1-yl]methyl]-6-(2,4-dichlorophenyl)-3-methyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6R)-4-[[4-(tert-butylcarbamoyl)piperazin-1-yl]methyl]-6-(4-tert-butylphenyl)-3-methyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate —— C28H43N5O4
ethyl (6R)-4-[[4-(tert-butylcarbamoyl)piperazin-1-yl]methyl]-6-(4-tert-butylphenyl)-3-methyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate
—— ethyl 4-[(2R)-2-[(2-chlorobenzoyl)-[(4-fluorophenyl)methyl]amino]propanoyl]-1-ethyl-3,5-dimethylpyrrole-2-carboxylate —— C28H30ClFN2O4
ethyl 4-[(2R)-2-[(2-chlorobenzoyl)-[(4-fluorophenyl)methyl]amino]propanoyl]-1-ethyl-3,5-dimethylpyrrole-2-carboxylate
—— ethyl 4-[(2S)-2-[(2-chlorobenzoyl)-(pyridin-2-ylmethyl)amino]propanoyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate —— C25H26ClN3O4
ethyl 4-[(2S)-2-[(2-chlorobenzoyl)-(pyridin-2-ylmethyl)amino]propanoyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate
—— ethyl (6S)-6-(2-chlorophenyl)-3-ethyl-4-[[(3R)-3-methyl-4-(thiophene-2-carbonyl)piperazin-1-yl]methyl]-2-oxo-1,6-dihydropyrimidine-5-carboxylate —— C26H31ClN4O4S
ethyl (6S)-6-(2-chlorophenyl)-3-ethyl-4-[[(3R)-3-methyl-4-(thiophene-2-carbonyl)piperazin-1-yl]methyl]-2-oxo-1,6-dihydropyrimidine-5-carboxylate
—— ethyl 4-[(2R)-2-[cyclopropanecarbonyl(furan-2-ylmethyl)amino]propanoyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate —— C21H26N2O5
ethyl 4-[(2R)-2-[cyclopropanecarbonyl(furan-2-ylmethyl)amino]propanoyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate
—— ethyl 4-[(2S)-2-[cyclopropyl-(3-fluorobenzoyl)amino]propanoyl]-1-ethyl-3,5-dimethylpyrrole-2-carboxylate —— C24H29FN2O4
ethyl 4-[(2S)-2-[cyclopropyl-(3-fluorobenzoyl)amino]propanoyl]-1-ethyl-3,5-dimethylpyrrole-2-carboxylate
—— ethyl 1-ethyl-3,5-dimethyl-4-[(2R)-2-[2-methylpropanoyl(2-methylpropyl)amino]propanoyl]pyrrole-2-carboxylate —— C22H36N2O4
ethyl 1-ethyl-3,5-dimethyl-4-[(2R)-2-[2-methylpropanoyl(2-methylpropyl)amino]propanoyl]pyrrole-2-carboxylate
—— Ethyl 3-methyl-2-[2-[2-oxo-2-(1,3-thiazol-2-ylamino)ethyl]sulfonylacetyl]imino-1,3-benzothiazole-6-carboxylate —— C18H18N4O6S3
Ethyl 3-methyl-2-[2-[2-oxo-2-(1,3-thiazol-2-ylamino)ethyl]sulfonylacetyl]imino-1,3-benzothiazole-6-carboxylate
—— ethyl (6R)-4-[[(3R)-4-(cyclopropanecarbonyl)-3-methylpiperazin-1-yl]methyl]-3-ethyl-2-oxo-6-[2-(trifluoromethyl)phenyl]-1,6-dihydropyrimidine-5-carboxylate —— C26H33F3N4O4
ethyl (6R)-4-[[(3R)-4-(cyclopropanecarbonyl)-3-methylpiperazin-1-yl]methyl]-3-ethyl-2-oxo-6-[2-(trifluoromethyl)phenyl]-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6S)-4-[[(3R)-4-(cyclopropanecarbonyl)-3-methylpiperazin-1-yl]methyl]-3-ethyl-2-oxo-6-[2-(trifluoromethyl)phenyl]-1,6-dihydropyrimidine-5-carboxylate —— C26H33F3N4O4
ethyl (6S)-4-[[(3R)-4-(cyclopropanecarbonyl)-3-methylpiperazin-1-yl]methyl]-3-ethyl-2-oxo-6-[2-(trifluoromethyl)phenyl]-1,6-dihydropyrimidine-5-carboxylate
—— Ethyl 2-[2-(4-chlorobenzoyl)imino-6-sulfamoyl-1,3-benzothiazol-3-yl]acetate —— C18H16ClN3O5S2
Ethyl 2-[2-(4-chlorobenzoyl)imino-6-sulfamoyl-1,3-benzothiazol-3-yl]acetate
—— ethyl 4-[(2S)-2-[(2-chlorobenzoyl)-(3-ethoxypropyl)amino]propanoyl]-1-ethyl-3,5-dimethylpyrrole-2-carboxylate —— C26H35ClN2O5
ethyl 4-[(2S)-2-[(2-chlorobenzoyl)-(3-ethoxypropyl)amino]propanoyl]-1-ethyl-3,5-dimethylpyrrole-2-carboxylate
—— ethyl (6R)-6-(2,4-dichlorophenyl)-3-methyl-4-[[(3R)-3-methyl-4-(propan-2-ylcarbamoyl)piperazin-1-yl]methyl]-2-oxo-1,6-dihydropyrimidine-5-carboxylate —— C24H33Cl2N5O4
ethyl (6R)-6-(2,4-dichlorophenyl)-3-methyl-4-[[(3R)-3-methyl-4-(propan-2-ylcarbamoyl)piperazin-1-yl]methyl]-2-oxo-1,6-dihydropyrimidine-5-carboxylate
—— ethyl 1-ethyl-4-[(2R)-2-[(4-fluorophenyl)methyl-(3-methylbutanoyl)amino]propanoyl]-3,5-dimethylpyrrole-2-carboxylate —— C26H35FN2O4
ethyl 1-ethyl-4-[(2R)-2-[(4-fluorophenyl)methyl-(3-methylbutanoyl)amino]propanoyl]-3,5-dimethylpyrrole-2-carboxylate
—— ethyl (6S)-4-[[4-(cyclopropanecarbonyl)-1,4-diazepan-1-yl]methyl]-3-methyl-2-oxo-6-(4-propan-2-ylphenyl)-1,6-dihydropyrimidine-5-carboxylate —— C27H38N4O4
ethyl (6S)-4-[[4-(cyclopropanecarbonyl)-1,4-diazepan-1-yl]methyl]-3-methyl-2-oxo-6-(4-propan-2-ylphenyl)-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6R)-6-(4-tert-butylphenyl)-4-[[4-(ethylcarbamoyl)piperazin-1-yl]methyl]-3-methyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate —— C26H39N5O4
ethyl (6R)-6-(4-tert-butylphenyl)-4-[[4-(ethylcarbamoyl)piperazin-1-yl]methyl]-3-methyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6S)-4-[[4-(tert-butylcarbamoyl)piperazin-1-yl]methyl]-3-methyl-2-oxo-6-[2-(trifluoromethyl)phenyl]-1,6-dihydropyrimidine-5-carboxylate —— C25H34F3N5O4
ethyl (6S)-4-[[4-(tert-butylcarbamoyl)piperazin-1-yl]methyl]-3-methyl-2-oxo-6-[2-(trifluoromethyl)phenyl]-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6R)-6-(4-tert-butylphenyl)-4-[[(3R)-4-(cyclopentanecarbonyl)-3-methylpiperazin-1-yl]methyl]-3-methyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate —— C30H44N4O4
ethyl (6R)-6-(4-tert-butylphenyl)-4-[[(3R)-4-(cyclopentanecarbonyl)-3-methylpiperazin-1-yl]methyl]-3-methyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate
—— ethyl 1-ethyl-3,5-dimethyl-4-[(2S)-2-[prop-2-enyl(thiophene-2-carbonyl)amino]propanoyl]pyrrole-2-carboxylate —— C22H28N2O4S
ethyl 1-ethyl-3,5-dimethyl-4-[(2S)-2-[prop-2-enyl(thiophene-2-carbonyl)amino]propanoyl]pyrrole-2-carboxylate
—— ethyl (6R)-4-[[4-(cyclobutanecarbonyl)piperazin-1-yl]methyl]-6-(2,3-dichlorophenyl)-3-methyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate —— C24H30Cl2N4O4
ethyl (6R)-4-[[4-(cyclobutanecarbonyl)piperazin-1-yl]methyl]-6-(2,3-dichlorophenyl)-3-methyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6S)-4-[[4-(cyclopropanecarbonyl)piperazin-1-yl]methyl]-3-methyl-2-oxo-6-(4-propan-2-ylphenyl)-1,6-dihydropyrimidine-5-carboxylate —— C26H36N4O4
ethyl (6S)-4-[[4-(cyclopropanecarbonyl)piperazin-1-yl]methyl]-3-methyl-2-oxo-6-(4-propan-2-ylphenyl)-1,6-dihydropyrimidine-5-carboxylate
—— Ethyl 2-(2-amino-1,3-thiazol-3-ium-4-yl)acetate —— C7H11N2O2S+
Ethyl 2-(2-amino-1,3-thiazol-3-ium-4-yl)acetate
—— ethyl (6S)-4-[[4-(cyclobutanecarbonyl)-1,4-diazepan-1-yl]methyl]-6-(2,5-dimethylphenyl)-3-methyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate —— C27H38N4O4
ethyl (6S)-4-[[4-(cyclobutanecarbonyl)-1,4-diazepan-1-yl]methyl]-6-(2,5-dimethylphenyl)-3-methyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6R)-6-(2,5-dimethylphenyl)-3-methyl-4-[[4-(4-methylbenzoyl)piperazin-1-yl]methyl]-2-oxo-1,6-dihydropyrimidine-5-carboxylate —— C29H36N4O4
ethyl (6R)-6-(2,5-dimethylphenyl)-3-methyl-4-[[4-(4-methylbenzoyl)piperazin-1-yl]methyl]-2-oxo-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6S)-6-(4-tert-butylphenyl)-3-methyl-4-[[(3S)-3-methyl-4-propanoylpiperazin-1-yl]methyl]-2-oxo-1,6-dihydropyrimidine-5-carboxylate —— C27H40N4O4
ethyl (6S)-6-(4-tert-butylphenyl)-3-methyl-4-[[(3S)-3-methyl-4-propanoylpiperazin-1-yl]methyl]-2-oxo-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6R)-4-[[(3R)-4-(tert-butylcarbamoyl)-3-methylpiperazin-1-yl]methyl]-3-methyl-2-oxo-6-(4-propan-2-ylphenyl)-1,6-dihydropyrimidine-5-carboxylate —— C28H43N5O4
ethyl (6R)-4-[[(3R)-4-(tert-butylcarbamoyl)-3-methylpiperazin-1-yl]methyl]-3-methyl-2-oxo-6-(4-propan-2-ylphenyl)-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6R)-6-(4-tert-butylphenyl)-4-[[4-(2-fluorobenzoyl)piperazin-1-yl]methyl]-3-methyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate —— C30H37FN4O4
ethyl (6R)-6-(4-tert-butylphenyl)-4-[[4-(2-fluorobenzoyl)piperazin-1-yl]methyl]-3-methyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate