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—— (E)-3-[4-(cyanomethoxy)-3-methoxyphenyl]-N-[(1S)-2-(2-oxopyrrolidin-1-yl)-1-phenylethyl]prop-2-enamide —— C24H25N3O4
(E)-3-[4-(cyanomethoxy)-3-methoxyphenyl]-N-[(1S)-2-(2-oxopyrrolidin-1-yl)-1-phenylethyl]prop-2-enamide
—— (E)-3-(5-methylthiophen-2-yl)-N-[(1S)-2-(2-oxopyrrolidin-1-yl)-1-phenylethyl]prop-2-enamide —— C20H22N2O2S
(E)-3-(5-methylthiophen-2-yl)-N-[(1S)-2-(2-oxopyrrolidin-1-yl)-1-phenylethyl]prop-2-enamide
—— ethyl N-[(3-chlorobenzoyl)-[1-(3-methoxyphenyl)-2,5-dioxopyrrolidin-3-yl]amino]carbamate —— C21H20ClN3O6
ethyl N-[(3-chlorobenzoyl)-[1-(3-methoxyphenyl)-2,5-dioxopyrrolidin-3-yl]amino]carbamate
—— Ethyl 1-[3-[(2,5-dimethylfuran-3-carbonyl)-hexylamino]propanoyl]piperidine-4-carboxylate —— C24H38N2O5
Ethyl 1-[3-[(2,5-dimethylfuran-3-carbonyl)-hexylamino]propanoyl]piperidine-4-carboxylate
—— (E)-3-(4-ethoxyphenyl)-N-[(1R)-2-(2-oxopyrrolidin-1-yl)-1-phenylethyl]prop-2-enamide —— C23H26N2O3
(E)-3-(4-ethoxyphenyl)-N-[(1R)-2-(2-oxopyrrolidin-1-yl)-1-phenylethyl]prop-2-enamide
—— Ethyl 4-phenyl-2-[[2-(1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl)acetyl]amino]thiophene-3-carboxylate —— C25H32N2O3S
Ethyl 4-phenyl-2-[[2-(1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl)acetyl]amino]thiophene-3-carboxylate
—— Ethyl 2-[[2-(2-methylpiperidin-1-ium-1-yl)acetyl]amino]-4-phenylthiophene-3-carboxylate —— C21H27N2O3S+
Ethyl 2-[[2-(2-methylpiperidin-1-ium-1-yl)acetyl]amino]-4-phenylthiophene-3-carboxylate
—— Ethyl 2-[[2-methylpropyl-[2-[(5-methyl-1,3-thiazol-2-yl)amino]-2-oxoethyl]carbamoyl]amino]acetate —— C15H24N4O4S
Ethyl 2-[[2-methylpropyl-[2-[(5-methyl-1,3-thiazol-2-yl)amino]-2-oxoethyl]carbamoyl]amino]acetate
—— (E)-3-(2-fluorophenyl)-N-(pyridin-4-ylmethyl)but-2-enamide —— C16H15FN2O
(E)-3-(2-fluorophenyl)-N-(pyridin-4-ylmethyl)but-2-enamide
—— Ethyl 6-ethyl-2-[[5-(5-ethylthiophen-2-yl)-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidine-2-carbonyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate —— C27H27F3N4O3S2
Ethyl 6-ethyl-2-[[5-(5-ethylthiophen-2-yl)-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidine-2-carbonyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
—— (E)-3-(2-cyanophenyl)-N-[(1R)-2-(2-oxopyrrolidin-1-yl)-1-phenylethyl]prop-2-enamide —— C22H21N3O2
(E)-3-(2-cyanophenyl)-N-[(1R)-2-(2-oxopyrrolidin-1-yl)-1-phenylethyl]prop-2-enamide
—— (E)-3-(3-fluoro-4-methoxyphenyl)-N-[(1R)-2-(2-oxopyrrolidin-1-yl)-1-phenylethyl]prop-2-enamide —— C22H23FN2O3
(E)-3-(3-fluoro-4-methoxyphenyl)-N-[(1R)-2-(2-oxopyrrolidin-1-yl)-1-phenylethyl]prop-2-enamide
—— (E)-3-(3-fluoro-4-methoxyphenyl)-N-[(1S)-2-(2-oxopyrrolidin-1-yl)-1-phenylethyl]prop-2-enamide —— C22H23FN2O3
(E)-3-(3-fluoro-4-methoxyphenyl)-N-[(1S)-2-(2-oxopyrrolidin-1-yl)-1-phenylethyl]prop-2-enamide
—— Ethyl 4-[[4-[5-[(4-chlorophenyl)methyl]-2,6-dimethylpyrimidin-4-yl]-1,4-diazepane-1-carbonyl]amino]benzoate —— C28H32ClN5O3
Ethyl 4-[[4-[5-[(4-chlorophenyl)methyl]-2,6-dimethylpyrimidin-4-yl]-1,4-diazepane-1-carbonyl]amino]benzoate
—— (E)-N-[(2R)-2-cyanopropyl]-N-ethyl-2-phenylethenesulfonamide —— C14H18N2O2S
(E)-N-[(2R)-2-cyanopropyl]-N-ethyl-2-phenylethenesulfonamide
—— (E)-3-[4-(cyanomethoxy)-3-methoxyphenyl]-N-[(1R)-2-(2-oxopyrrolidin-1-yl)-1-phenylethyl]prop-2-enamide —— C24H25N3O4
(E)-3-[4-(cyanomethoxy)-3-methoxyphenyl]-N-[(1R)-2-(2-oxopyrrolidin-1-yl)-1-phenylethyl]prop-2-enamide
—— (E)-3-(2-cyanophenyl)-N-[(1S)-2-(2-oxopyrrolidin-1-yl)-1-phenylethyl]prop-2-enamide —— C22H21N3O2
(E)-3-(2-cyanophenyl)-N-[(1S)-2-(2-oxopyrrolidin-1-yl)-1-phenylethyl]prop-2-enamide
—— (E)-3-(2-fluorophenyl)-N-pyridin-4-ylbut-2-enamide —— C15H13FN2O
(E)-3-(2-fluorophenyl)-N-pyridin-4-ylbut-2-enamide
—— (E)-N-[[6-(azepan-1-yl)pyridin-3-yl]methyl]-2-methylpent-2-enamide —— C18H27N3O
(E)-N-[[6-(azepan-1-yl)pyridin-3-yl]methyl]-2-methylpent-2-enamide
—— Ethyl 1-[2-(4-chlorophenyl)-5-phenylpyrazole-3-carbonyl]piperidine-4-carboxylate —— C24H24ClN3O3
Ethyl 1-[2-(4-chlorophenyl)-5-phenylpyrazole-3-carbonyl]piperidine-4-carboxylate
—— ethyl (3S)-1-(4-methoxypyrimidin-2-yl)piperidine-3-carboxylate —— C13H19N3O3
ethyl (3S)-1-(4-methoxypyrimidin-2-yl)piperidine-3-carboxylate
—— ethyl (3R)-1-(4-methoxypyrimidin-2-yl)piperidine-3-carboxylate —— C13H19N3O3
ethyl (3R)-1-(4-methoxypyrimidin-2-yl)piperidine-3-carboxylate
—— (E)-2-methyl-1-[4-[3-(trifluoromethyl)benzoyl]piperazin-1-yl]pent-2-en-1-one —— C18H21F3N2O2
(E)-2-methyl-1-[4-[3-(trifluoromethyl)benzoyl]piperazin-1-yl]pent-2-en-1-one
—— Ethyl 4-[2-(5-bromothiophen-2-yl)-4-oxo-1,3-thiazolidin-3-yl]butanoate —— C13H16BrNO3S2
Ethyl 4-[2-(5-bromothiophen-2-yl)-4-oxo-1,3-thiazolidin-3-yl]butanoate
—— ethyl 2-[[(5R)-5-phenyl-4,5-dihydro-1,2-oxazole-3-carbonyl]amino]acetate —— C14H16N2O4
ethyl 2-[[(5R)-5-phenyl-4,5-dihydro-1,2-oxazole-3-carbonyl]amino]acetate
—— Ethyl 5-[2-[1-[2-(3,4-difluorophenyl)acetyl]piperidin-4-yl]-1,3-thiazol-4-yl]-1,2-oxazole-3-carboxylate —— C22H21F2N3O4S
Ethyl 5-[2-[1-[2-(3,4-difluorophenyl)acetyl]piperidin-4-yl]-1,3-thiazol-4-yl]-1,2-oxazole-3-carboxylate
—— Ethyl 3-phenyl-2-[[4-[[2-[3-[3-(trifluoromethyl)phenyl]pyrazol-1-yl]acetyl]amino]piperidine-4-carbonyl]amino]propanoate —— C29H32F3N5O4
Ethyl 3-phenyl-2-[[4-[[2-[3-[3-(trifluoromethyl)phenyl]pyrazol-1-yl]acetyl]amino]piperidine-4-carbonyl]amino]propanoate
—— ethyl 6-fluoro-2-methyl-3,4-dihydroquinoline-1(2H)-carboxylate —— C13H16FNO2
ethyl 6-fluoro-2-methyl-3,4-dihydroquinoline-1(2H)-carboxylate
—— Ethyl 4-[[4-[4-[4-(5-methyl-3-phenyl-1,2-oxazol-4-yl)-1,3-thiazol-2-yl]piperidin-1-yl]-4-oxobut-2-enoyl]amino]benzoate —— C31H30N4O5S
Ethyl 4-[[4-[4-[4-(5-methyl-3-phenyl-1,2-oxazol-4-yl)-1,3-thiazol-2-yl]piperidin-1-yl]-4-oxobut-2-enoyl]amino]benzoate
—— Ethyl 4-[[2-(2-methylphenyl)sulfanylacetyl]amino]benzoate —— C18H19NO3S
Ethyl 4-[[2-(2-methylphenyl)sulfanylacetyl]amino]benzoate
—— ethyl 2-[[2-[[5-(2-chlorophenyl)-1,3,4-oxadiazol-2-yl]sulfonyl]acetyl]amino]-5,6,7,8-tetrahydro-4H-cyclohepta[b]thiophene-3-carboxylate —— C22H22ClN3O6S2
ethyl 2-[[2-[[5-(2-chlorophenyl)-1,3,4-oxadiazol-2-yl]sulfonyl]acetyl]amino]-5,6,7,8-tetrahydro-4H-cyclohepta[b]thiophene-3-carboxylate
—— Ethyl 2-amino-1-[4-(aminosulfonyl)phenyl]-5-oxo-4-(3-pyridinyl)-1,4,5,6,7,8-hexahydro-3-quinolinecarboxylate —— C23H24N4O5S
Ethyl 2-amino-1-[4-(aminosulfonyl)phenyl]-5-oxo-4-(3-pyridinyl)-1,4,5,6,7,8-hexahydro-3-quinolinecarboxylate
—— ethyl 5-(2,4-dimethoxyphenyl)-7-methyl-2-[(1-methylpyrrol-2-yl)methylidene]-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C24H25N3O5S
ethyl 5-(2,4-dimethoxyphenyl)-7-methyl-2-[(1-methylpyrrol-2-yl)methylidene]-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl 2-[[5-[(2-fluoro-5-nitrophenoxy)methyl]furan-2-yl]methylidene]-7-methyl-3-oxo-5-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C28H22FN3O7S
ethyl 2-[[5-[(2-fluoro-5-nitrophenoxy)methyl]furan-2-yl]methylidene]-7-methyl-3-oxo-5-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— Ethyl 2-[[2-[4-[4-[4-(hydroxymethyl)phenyl]-5-methyl-6-[(1-oxidopyridin-1-ium-2-yl)sulfanylmethyl]-1,3-dioxan-2-yl]phenyl]phenyl]methylcarbamoylamino]acetate —— C36H39N3O7S
Ethyl 2-[[2-[4-[4-[4-(hydroxymethyl)phenyl]-5-methyl-6-[(1-oxidopyridin-1-ium-2-yl)sulfanylmethyl]-1,3-dioxan-2-yl]phenyl]phenyl]methylcarbamoylamino]acetate
—— Ethyl 2-[4-[(9,10-dioxoanthracen-2-yl)sulfonylamino]phenyl]acetate —— C24H19NO6S
Ethyl 2-[4-[(9,10-dioxoanthracen-2-yl)sulfonylamino]phenyl]acetate
—— ethyl 3-amino-3-(furan-2-ylmethylamino)-2-(4-methoxybenzoyl)prop-2-enoate —— C18H20N2O5
ethyl 3-amino-3-(furan-2-ylmethylamino)-2-(4-methoxybenzoyl)prop-2-enoate
—— Ethyl 2-[3-(2,6-dichlorophenyl)prop-2-enoylamino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate —— C20H19Cl2NO3S
Ethyl 2-[3-(2,6-dichlorophenyl)prop-2-enoylamino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
—— Ethyl 2-[(8-chloronaphthalen-1-yl)sulfonylamino]hexanoate —— C18H22ClNO4S
Ethyl 2-[(8-chloronaphthalen-1-yl)sulfonylamino]hexanoate
—— Ethyl 3-[[2-(cyclopropanecarbonyl)pyrazolidine-1-carbothioyl]amino]propanoate —— C13H21N3O3S
Ethyl 3-[[2-(cyclopropanecarbonyl)pyrazolidine-1-carbothioyl]amino]propanoate
—— Ethyl 2-[2-[[2-[(7-methyl-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-yl)sulfanyl]acetyl]amino]-1,3-thiazol-4-yl]acetate —— C20H22N4O3S3
Ethyl 2-[2-[[2-[(7-methyl-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-yl)sulfanyl]acetyl]amino]-1,3-thiazol-4-yl]acetate
—— (E)-N-(3-acetamido-4-methylphenyl)-2-methylpent-2-enamide —— C15H20N2O2
(E)-N-(3-acetamido-4-methylphenyl)-2-methylpent-2-enamide
—— ethyl 1-({1-[2-(morpholin-4-yl)ethyl]-1H-pyrrol-2-yl}methyl)piperidine-3-carboxylate —— C19H31N3O3
ethyl 1-({1-[2-(morpholin-4-yl)ethyl]-1H-pyrrol-2-yl}methyl)piperidine-3-carboxylate
—— [(E)-but-2-enyl] (2S)-2-methyl-3-oxo-4H-1,4-benzothiazine-6-carboxylate —— C14H15NO3S
[(E)-but-2-enyl] (2S)-2-methyl-3-oxo-4H-1,4-benzothiazine-6-carboxylate
—— Ethyl 3-[[6-[(5-bromo-2-fluorophenyl)methylamino]-5-nitropyrimidin-4-yl]-(furan-2-ylmethyl)amino]propanoate —— C21H21BrFN5O5
Ethyl 3-[[6-[(5-bromo-2-fluorophenyl)methylamino]-5-nitropyrimidin-4-yl]-(furan-2-ylmethyl)amino]propanoate
—— ethyl 1-benzyl-1-methyl-3,6-dihydro-2H-pyridin-1-ium-4-carboxylate —— C16H22NO2+
ethyl 1-benzyl-1-methyl-3,6-dihydro-2H-pyridin-1-ium-4-carboxylate
—— Ethyl 4-[[2-(3-nitro-1,2,4-triazol-1-yl)acetyl]amino]piperidine-1-carboxylate —— C12H18N6O5
Ethyl 4-[[2-(3-nitro-1,2,4-triazol-1-yl)acetyl]amino]piperidine-1-carboxylate
—— Ethyl 5-(diethylcarbamoyl)-2-[[2-(4-methoxyphenyl)quinoline-4-carbonyl]amino]-4-methylthiophene-3-carboxylate —— C30H31N3O5S
Ethyl 5-(diethylcarbamoyl)-2-[[2-(4-methoxyphenyl)quinoline-4-carbonyl]amino]-4-methylthiophene-3-carboxylate
—— Ethyl 4-[6-methyl-2-[1-(5-nitrothiophene-2-carbonyl)piperidin-4-yl]pyridine-3-carbonyl]piperazine-1-carboxylate —— C24H29N5O6S
Ethyl 4-[6-methyl-2-[1-(5-nitrothiophene-2-carbonyl)piperidin-4-yl]pyridine-3-carbonyl]piperazine-1-carboxylate
—— ethyl 2-[[4-(3,4-dihydro-2H-quinolin-1-ylsulfonyl)benzoyl]amino]-3-(3,5-dimethylpyrazole-1-carbonyl)-5,7-dihydro-4H-thieno[2,3-c]pyridine-6-carboxylate —— C32H33N5O6S2
ethyl 2-[[4-(3,4-dihydro-2H-quinolin-1-ylsulfonyl)benzoyl]amino]-3-(3,5-dimethylpyrazole-1-carbonyl)-5,7-dihydro-4H-thieno[2,3-c]pyridine-6-carboxylate