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—— cyclobutyl{5-[4-methyl-6-(methylamino)pyrimidin-2-yl]-5,6,7,8-tetrahydro-4H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methanol —— C18H26N6O
cyclobutyl{5-[4-methyl-6-(methylamino)pyrimidin-2-yl]-5,6,7,8-tetrahydro-4H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methanol
—— cis-3-[5-{[4-(methoxyacetyl)-1,4-diazepan-1-yl]methyl}-4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]cyclobutanamine —— C18H32N6O3
cis-3-[5-{[4-(methoxyacetyl)-1,4-diazepan-1-yl]methyl}-4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]cyclobutanamine
—— (cis-3-{4-(2-methoxyethyl)-5-[(4-pyrimidin-2-ylpiperazin-1-yl)methyl]-4H-1,2,4-triazol-3-yl}cyclobutyl)amine —— C18H28N8O
(cis-3-{4-(2-methoxyethyl)-5-[(4-pyrimidin-2-ylpiperazin-1-yl)methyl]-4H-1,2,4-triazol-3-yl}cyclobutyl)amine
—— (cis-3-{2-Methyl-6-[4-(3-methylpyridin-4-yl)-1,4-diazepan-1-yl]pyrimidin-4-yl}cyclobutyl)amine —— C20H28N6
(cis-3-{2-Methyl-6-[4-(3-methylpyridin-4-yl)-1,4-diazepan-1-yl]pyrimidin-4-yl}cyclobutyl)amine
—— cyclopropyl(5-{[(3-methoxyphenyl)thio]acetyl}-5,6,7,8-tetrahydro-4H-pyrazolo[1,5-a][1,4]diazepin-2-yl)methanol —— C20H25N3O3S
cyclopropyl(5-{[(3-methoxyphenyl)thio]acetyl}-5,6,7,8-tetrahydro-4H-pyrazolo[1,5-a][1,4]diazepin-2-yl)methanol
—— [cis-3-(5-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-4-ethyl-4H-1,2,4-triazol-3-yl)cyclobutyl]amine —— C15H27N5O
[cis-3-(5-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-4-ethyl-4H-1,2,4-triazol-3-yl)cyclobutyl]amine
—— cis-3-(5-{[(cyclopentylmethyl)(methyl)amino]methyl}-4-ethyl-4H-1,2,4-triazol-3-yl)cyclobutanamine —— C16H29N5
cis-3-(5-{[(cyclopentylmethyl)(methyl)amino]methyl}-4-ethyl-4H-1,2,4-triazol-3-yl)cyclobutanamine
—— cis-3-[6-(2-Azaspiro[4.4]non-2-yl)pyrimidin-4-yl]cyclobutanamine —— C16H24N4
cis-3-[6-(2-Azaspiro[4.4]non-2-yl)pyrimidin-4-yl]cyclobutanamine
—— cis-3-[6-(4-Phenylpiperidin-1-yl)pyrimidin-4-yl]cyclobutanamine —— C19H24N4
cis-3-[6-(4-Phenylpiperidin-1-yl)pyrimidin-4-yl]cyclobutanamine
—— Cyclopropyl(5-{5-[(methylthio)methyl]-2-furoyl}-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-2-yl)methanol —— C17H21N3O3S
Cyclopropyl(5-{5-[(methylthio)methyl]-2-furoyl}-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-2-yl)methanol
—— (cis-3-{4-ethyl-5-[(3-morpholin-4-ylphenoxy)methyl]-4H-1,2,4-triazol-3-yl}cyclobutyl)amine —— C19H27N5O2
(cis-3-{4-ethyl-5-[(3-morpholin-4-ylphenoxy)methyl]-4H-1,2,4-triazol-3-yl}cyclobutyl)amine
—— {[cis-3-({[3-(5-methyl-2-thienyl)-1H-pyrazol-5-yl]carbonyl}amino)tetrahydro-2H-pyran-4-yl]oxy}acetic acid —— C16H19N3O5S
{[cis-3-({[3-(5-methyl-2-thienyl)-1H-pyrazol-5-yl]carbonyl}amino)tetrahydro-2H-pyran-4-yl]oxy}acetic acid
—— cyclopropyl[5-(2-ethyl-6-methylpyrimidin-4-yl)-5,6,7,8-tetrahydro-4H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methanol —— C18H25N5O
cyclopropyl[5-(2-ethyl-6-methylpyrimidin-4-yl)-5,6,7,8-tetrahydro-4H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methanol
—— [(cis-3-{[(2,8-dimethylquinolin-3-yl)carbonyl]amino}tetrahydro-2H-pyran-4-yl)oxy]acetic acid —— C19H22N2O5
[(cis-3-{[(2,8-dimethylquinolin-3-yl)carbonyl]amino}tetrahydro-2H-pyran-4-yl)oxy]acetic acid
—— [cis-3-(4-ethyl-5-{[4-(piperidin-1-ylmethyl)piperidin-1-yl]methyl}-4H-1,2,4-triazol-3-yl)cyclobutyl]amine —— C20H36N6
[cis-3-(4-ethyl-5-{[4-(piperidin-1-ylmethyl)piperidin-1-yl]methyl}-4H-1,2,4-triazol-3-yl)cyclobutyl]amine
—— cis-3-[6-[(9aS)-hexahydro-1H-pyrrolo[1,2-a][1,4]diazepin-2(3H)-yl]-2-(methoxymethyl)pyrimidin-4-yl]cyclobutanamine —— C18H29N5O
cis-3-[6-[(9aS)-hexahydro-1H-pyrrolo[1,2-a][1,4]diazepin-2(3H)-yl]-2-(methoxymethyl)pyrimidin-4-yl]cyclobutanamine
—— cis-3-[4-cyclopropyl-5-({methyl[(5-methyl-2-thienyl)methyl]amino}methyl)-4H-1,2,4-triazol-3-yl]cyclobutanamine —— C17H25N5S
cis-3-[4-cyclopropyl-5-({methyl[(5-methyl-2-thienyl)methyl]amino}methyl)-4H-1,2,4-triazol-3-yl]cyclobutanamine
—— cis-3-[6-(4-Methylpiperidin-1-yl)pyrimidin-4-yl]cyclobutanamine —— C14H22N4
cis-3-[6-(4-Methylpiperidin-1-yl)pyrimidin-4-yl]cyclobutanamine
—— [cis-3-(5-{[4-(4-fluorophenyl)piperazin-1-yl]methyl}-4-methyl-4H-1,2,4-triazol-3-yl)cyclobutyl]amine —— C18H25FN6
[cis-3-(5-{[4-(4-fluorophenyl)piperazin-1-yl]methyl}-4-methyl-4H-1,2,4-triazol-3-yl)cyclobutyl]amine
—— cis-3-[4-ethyl-5-({[(2E)-3-phenylprop-2-en-1-yl]amino}methyl)-4H-1,2,4-triazol-3-yl]cyclobutanamine —— C18H25N5
cis-3-[4-ethyl-5-({[(2E)-3-phenylprop-2-en-1-yl]amino}methyl)-4H-1,2,4-triazol-3-yl]cyclobutanamine
—— cis-3-(4-cyclopropyl-5-{[(5,6,7,8-tetrahydronaphthalen-2-ylmethyl)amino]methyl}-4H-1,2,4-triazol-3-yl)cyclobutanamine —— C21H29N5
cis-3-(4-cyclopropyl-5-{[(5,6,7,8-tetrahydronaphthalen-2-ylmethyl)amino]methyl}-4H-1,2,4-triazol-3-yl)cyclobutanamine
—— cis-3-[5-({[(5-benzyl-1,2,4-oxadiazol-3-yl)methyl]amino}methyl)-4-methyl-4H-1,2,4-triazol-3-yl]cyclobutanamine —— C18H23N7O
cis-3-[5-({[(5-benzyl-1,2,4-oxadiazol-3-yl)methyl]amino}methyl)-4-methyl-4H-1,2,4-triazol-3-yl]cyclobutanamine
—— cis-3-hydroxy-N-{2-[5-(hydroxymethyl)-1,2,4-oxadiazol-3-yl]ethyl}cyclohexanecarboxamide —— C12H19N3O4
cis-3-hydroxy-N-{2-[5-(hydroxymethyl)-1,2,4-oxadiazol-3-yl]ethyl}cyclohexanecarboxamide
—— [cis-3-(4-ethyl-5-{[4-(3-furoyl)-1,4-diazepan-1-yl]methyl}-4H-1,2,4-triazol-3-yl)cyclobutyl]amine —— C19H28N6O2
[cis-3-(4-ethyl-5-{[4-(3-furoyl)-1,4-diazepan-1-yl]methyl}-4H-1,2,4-triazol-3-yl)cyclobutyl]amine
—— [cis-3-(4-cyclopropyl-5-{[4-(3,4-dimethylphenyl)piperazin-1-yl]methyl}-4H-1,2,4-triazol-3-yl)cyclobutyl]amine —— C22H32N6
[cis-3-(4-cyclopropyl-5-{[4-(3,4-dimethylphenyl)piperazin-1-yl]methyl}-4H-1,2,4-triazol-3-yl)cyclobutyl]amine
—— cis-3-(4-(2-methoxyethyl)-5-{[(4,5,6,7-tetrahydro-1-benzothien-3-ylmethyl)amino]methyl}-4H-1,2,4-triazol-3-yl)cyclobutanamine —— C19H29N5OS
cis-3-(4-(2-methoxyethyl)-5-{[(4,5,6,7-tetrahydro-1-benzothien-3-ylmethyl)amino]methyl}-4H-1,2,4-triazol-3-yl)cyclobutanamine
—— Cyclopropyl{5-[5-fluoro-2-(trifluoromethyl)benzyl]-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-2-yl}methanol —— C18H19F4N3O
Cyclopropyl{5-[5-fluoro-2-(trifluoromethyl)benzyl]-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-2-yl}methanol
—— cis-3-[5-[(6-methoxy-3,4-dihydroisoquinolin-2(1H)-yl)methyl]-4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]cyclobutanamine —— C20H29N5O2
cis-3-[5-[(6-methoxy-3,4-dihydroisoquinolin-2(1H)-yl)methyl]-4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]cyclobutanamine
—— (cis-3-{4-(2-methoxyethyl)-5-[(4-phenylpiperidin-1-yl)methyl]-4H-1,2,4-triazol-3-yl}cyclobutyl)amine —— C21H31N5O
(cis-3-{4-(2-methoxyethyl)-5-[(4-phenylpiperidin-1-yl)methyl]-4H-1,2,4-triazol-3-yl}cyclobutyl)amine
—— Cyclopropyl[5-(2,4,5-trimethoxybenzyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-2-yl]methanol —— C20H27N3O4
Cyclopropyl[5-(2,4,5-trimethoxybenzyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-2-yl]methanol
—— cis-3-[4-methyl-5-({methyl[2-(methylthio)ethyl]amino}methyl)-4H-1,2,4-triazol-3-yl]cyclobutanamine —— C12H23N5S
cis-3-[4-methyl-5-({methyl[2-(methylthio)ethyl]amino}methyl)-4H-1,2,4-triazol-3-yl]cyclobutanamine
—— (cis-3-{4-methyl-5-[(3-pyridin-4-ylazetidin-1-yl)methyl]-4H-1,2,4-triazol-3-yl}cyclobutyl)amine —— C16H22N6
(cis-3-{4-methyl-5-[(3-pyridin-4-ylazetidin-1-yl)methyl]-4H-1,2,4-triazol-3-yl}cyclobutyl)amine
—— (cis-3-{6-[3-(3-Ethylphenoxy)azetidin-1-yl]pyrimidin-4-yl}cyclobutyl)amine —— C19H24N4O
(cis-3-{6-[3-(3-Ethylphenoxy)azetidin-1-yl]pyrimidin-4-yl}cyclobutyl)amine
—— cis-3-(5-{[(1,3-benzothiazol-2-ylmethyl)(methyl)amino]methyl}-4-ethyl-4H-1,2,4-triazol-3-yl)cyclobutanamine —— C18H24N6S
cis-3-(5-{[(1,3-benzothiazol-2-ylmethyl)(methyl)amino]methyl}-4-ethyl-4H-1,2,4-triazol-3-yl)cyclobutanamine
—— [cis-3-(5-{[2-chloro-5-(trifluoromethyl)phenoxy]methyl}-4-methyl-4H-1,2,4-triazol-3-yl)cyclobutyl]amine —— C15H16ClF3N4O
[cis-3-(5-{[2-chloro-5-(trifluoromethyl)phenoxy]methyl}-4-methyl-4H-1,2,4-triazol-3-yl)cyclobutyl]amine
—— (cis-3-{4-(2-methoxyethyl)-5-[(4-pyrazin-2-ylpiperazin-1-yl)methyl]-4H-1,2,4-triazol-3-yl}cyclobutyl)amine —— C18H28N8O
(cis-3-{4-(2-methoxyethyl)-5-[(4-pyrazin-2-ylpiperazin-1-yl)methyl]-4H-1,2,4-triazol-3-yl}cyclobutyl)amine
—— cis-3-[6-(4-Pyridin-4-ylpiperazin-1-yl)pyrimidin-4-yl]cyclobutanamine —— C17H22N6
cis-3-[6-(4-Pyridin-4-ylpiperazin-1-yl)pyrimidin-4-yl]cyclobutanamine
—— cyclopropyl[5-(pyrazolo[1,5-a]pyrimidin-2-ylcarbonyl)-5,6,7,8-tetrahydro-4H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methanol —— C18H20N6O2
cyclopropyl[5-(pyrazolo[1,5-a]pyrimidin-2-ylcarbonyl)-5,6,7,8-tetrahydro-4H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methanol
—— (cis-3-{4-methyl-5-[(3-phenyl-5,6,8,9-tetrahydro-7H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl)methyl]-4H-1,2,4-triazol-3-yl}cyclobutyl)amine —— C20H26N8
(cis-3-{4-methyl-5-[(3-phenyl-5,6,8,9-tetrahydro-7H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl)methyl]-4H-1,2,4-triazol-3-yl}cyclobutyl)amine
—— (cis-3-{4-(2-methoxyethyl)-5-[(4-pyrimidin-2-yl-1,4-diazepan-1-yl)methyl]-4H-1,2,4-triazol-3-yl}cyclobutyl)amine —— C19H30N8O
(cis-3-{4-(2-methoxyethyl)-5-[(4-pyrimidin-2-yl-1,4-diazepan-1-yl)methyl]-4H-1,2,4-triazol-3-yl}cyclobutyl)amine
—— (cis-3-{2-Methyl-6-[4-(2-morpholin-4-ylethyl)piperazin-1-yl]pyrimidin-4-yl}cyclobutyl)amine —— C19H32N6O
(cis-3-{2-Methyl-6-[4-(2-morpholin-4-ylethyl)piperazin-1-yl]pyrimidin-4-yl}cyclobutyl)amine
—— Cyclopropyl(5-{[4-(methoxymethyl)-5-methylisoxazol-3-yl]carbonyl}-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-2-yl)methanol —— C17H22N4O4
Cyclopropyl(5-{[4-(methoxymethyl)-5-methylisoxazol-3-yl]carbonyl}-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-2-yl)methanol
—— Cinnamyl (4-chlorophenyl)acetate —— C17H15ClO2
Cinnamyl (4-chlorophenyl)acetate
—— [cis-3-(5-{[4-(4-methoxyphenyl)piperazin-1-yl]methyl}-4-methyl-4H-1,2,4-triazol-3-yl)cyclobutyl]amine —— C19H28N6O
[cis-3-(5-{[4-(4-methoxyphenyl)piperazin-1-yl]methyl}-4-methyl-4H-1,2,4-triazol-3-yl)cyclobutyl]amine
—— cyclobutyl[5-(1H-indol-7-ylmethyl)-5,6,7,8-tetrahydro-4H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methanol —— C21H26N4O
cyclobutyl[5-(1H-indol-7-ylmethyl)-5,6,7,8-tetrahydro-4H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methanol
—— cis-3-(4-cyclopropyl-5-{[({3-[(methylthio)methyl]-1,2,4-oxadiazol-5-yl}methyl)amino]methyl}-4H-1,2,4-triazol-3-yl)cyclobutanamine —— C15H23N7OS
cis-3-(4-cyclopropyl-5-{[({3-[(methylthio)methyl]-1,2,4-oxadiazol-5-yl}methyl)amino]methyl}-4H-1,2,4-triazol-3-yl)cyclobutanamine
—— cyclobutyl[5-(4,6-dimethylquinolin-2-yl)-5,6,7,8-tetrahydro-4H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methanol —— C23H28N4O
cyclobutyl[5-(4,6-dimethylquinolin-2-yl)-5,6,7,8-tetrahydro-4H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methanol
—— Cyclopropyl{5-[(2,5-dimethyl-1,3-thiazol-4-yl)acetyl]-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-2-yl}methanol —— C17H22N4O2S
Cyclopropyl{5-[(2,5-dimethyl-1,3-thiazol-4-yl)acetyl]-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-2-yl}methanol
—— (cis-3-{2-(Methoxymethyl)-6-[3-(1,3-thiazol-2-yl)azetidin-1-yl]pyrimidin-4-yl}cyclobutyl)amine —— C16H21N5OS
(cis-3-{2-(Methoxymethyl)-6-[3-(1,3-thiazol-2-yl)azetidin-1-yl]pyrimidin-4-yl}cyclobutyl)amine
—— cis-3-[5-[(2-ethyl-1H-imidazol-1-yl)methyl]-4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]cyclobutanamine —— C15H24N6O
cis-3-[5-[(2-ethyl-1H-imidazol-1-yl)methyl]-4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]cyclobutanamine