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—— [cis-3-(4-cyclopropyl-5-{[3-(trifluoromethyl)phenoxy]methyl}-4H-1,2,4-triazol-3-yl)cyclobutyl]amine —— C17H19F3N4O
[cis-3-(4-cyclopropyl-5-{[3-(trifluoromethyl)phenoxy]methyl}-4H-1,2,4-triazol-3-yl)cyclobutyl]amine
—— (cis-3-{6-[3-(1,3-Thiazol-2-yl)azetidin-1-yl]pyrimidin-4-yl}cyclobutyl)amine —— C14H17N5S
(cis-3-{6-[3-(1,3-Thiazol-2-yl)azetidin-1-yl]pyrimidin-4-yl}cyclobutyl)amine
—— cis-3-(5-{[[2-(3,4-dimethoxyphenyl)ethyl](methyl)amino]methyl}-4-methyl-4H-1,2,4-triazol-3-yl)cyclobutanamine —— C19H29N5O2
cis-3-(5-{[[2-(3,4-dimethoxyphenyl)ethyl](methyl)amino]methyl}-4-methyl-4H-1,2,4-triazol-3-yl)cyclobutanamine
—— [cis-3-(4-ethyl-5-{[4-(2-furylmethyl)piperazin-1-yl]methyl}-4H-1,2,4-triazol-3-yl)cyclobutyl]amine —— C18H28N6O
[cis-3-(4-ethyl-5-{[4-(2-furylmethyl)piperazin-1-yl]methyl}-4H-1,2,4-triazol-3-yl)cyclobutyl]amine
—— [cis-3-(5-{[4-(cyclobutylcarbonyl)piperazin-1-yl]methyl}-4-ethyl-4H-1,2,4-triazol-3-yl)cyclobutyl]amine —— C18H30N6O
[cis-3-(5-{[4-(cyclobutylcarbonyl)piperazin-1-yl]methyl}-4-ethyl-4H-1,2,4-triazol-3-yl)cyclobutyl]amine
—— cis-3-[5-({[(3,5-dimethylisoxazol-4-yl)methyl]amino}methyl)-4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]cyclobutanamine —— C16H26N6O2
cis-3-[5-({[(3,5-dimethylisoxazol-4-yl)methyl]amino}methyl)-4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]cyclobutanamine
—— Cyclopropyl{5-[2-(3,4-dimethylphenoxy)ethyl]-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-2-yl}methanol —— C20H27N3O2
Cyclopropyl{5-[2-(3,4-dimethylphenoxy)ethyl]-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-2-yl}methanol
—— [cis-3-(4-cyclopropyl-5-{[(1,2-dimethyl-1H-indol-5-yl)oxy]methyl}-4H-1,2,4-triazol-3-yl)cyclobutyl]amine —— C20H25N5O
[cis-3-(4-cyclopropyl-5-{[(1,2-dimethyl-1H-indol-5-yl)oxy]methyl}-4H-1,2,4-triazol-3-yl)cyclobutyl]amine
—— cis-3-(5-{[[(4,6-dimethylpyridin-2-yl)methyl](methyl)amino]methyl}-4-ethyl-4H-1,2,4-triazol-3-yl)cyclobutanamine —— C18H28N6
cis-3-(5-{[[(4,6-dimethylpyridin-2-yl)methyl](methyl)amino]methyl}-4-ethyl-4H-1,2,4-triazol-3-yl)cyclobutanamine
—— [cis-3-(4-cyclopropyl-5-{[4-(4-fluorobenzyl)piperazin-1-yl]methyl}-4H-1,2,4-triazol-3-yl)cyclobutyl]amine —— C21H29FN6
[cis-3-(4-cyclopropyl-5-{[4-(4-fluorobenzyl)piperazin-1-yl]methyl}-4H-1,2,4-triazol-3-yl)cyclobutyl]amine
—— [cis-3-(5-{[4-(2-chlorophenyl)piperazin-1-yl]methyl}-4-ethyl-4H-1,2,4-triazol-3-yl)cyclobutyl]amine —— C19H27ClN6
[cis-3-(5-{[4-(2-chlorophenyl)piperazin-1-yl]methyl}-4-ethyl-4H-1,2,4-triazol-3-yl)cyclobutyl]amine
—— cis-3-(5-{[(3-furylmethyl)(methyl)amino]methyl}-4-methyl-4H-1,2,4-triazol-3-yl)cyclobutanamine —— C14H21N5O
cis-3-(5-{[(3-furylmethyl)(methyl)amino]methyl}-4-methyl-4H-1,2,4-triazol-3-yl)cyclobutanamine
—— [cis-3-(4-(2-methoxyethyl)-5-{[(2,4,6-trimethylpyrimidin-5-yl)oxy]methyl}-4H-1,2,4-triazol-3-yl)cyclobutyl]amine —— C17H26N6O2
[cis-3-(4-(2-methoxyethyl)-5-{[(2,4,6-trimethylpyrimidin-5-yl)oxy]methyl}-4H-1,2,4-triazol-3-yl)cyclobutyl]amine
—— (cis-3-{6-[4-(3,6-Dimethylpyrazin-2-yl)piperazin-1-yl]pyrimidin-4-yl}cyclobutyl)amine —— C18H25N7
(cis-3-{6-[4-(3,6-Dimethylpyrazin-2-yl)piperazin-1-yl]pyrimidin-4-yl}cyclobutyl)amine
—— cis-3-[5-{[(2-fluorobenzyl)(methyl)amino]methyl}-4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]cyclobutanamine —— C18H26FN5O
cis-3-[5-{[(2-fluorobenzyl)(methyl)amino]methyl}-4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]cyclobutanamine
—— Cyclopropyl{5-[2-(2,4-dimethylphenoxy)ethyl]-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-2-yl}methanol —— C20H27N3O2
Cyclopropyl{5-[2-(2,4-dimethylphenoxy)ethyl]-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-2-yl}methanol
—— cis-3-[5-{[(cyclopentylmethyl)(methyl)amino]methyl}-4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]cyclobutanamine —— C17H31N5O
cis-3-[5-{[(cyclopentylmethyl)(methyl)amino]methyl}-4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]cyclobutanamine
—— Cyclopropyl(5-{[2-(methylamino)pyridin-3-yl]methyl}-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-2-yl)methanol —— C17H23N5O
Cyclopropyl(5-{[2-(methylamino)pyridin-3-yl]methyl}-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-2-yl)methanol
—— cis-3-{6-[3-(2,6-Dimethylphenoxy)azetidin-1-yl]pyrimidin-4-yl}cyclobutanol —— C19H23N3O2
cis-3-{6-[3-(2,6-Dimethylphenoxy)azetidin-1-yl]pyrimidin-4-yl}cyclobutanol
—— cis-3-[4-cyclopropyl-5-({4-[(methylthio)methyl]piperidin-1-yl}methyl)-4H-1,2,4-triazol-3-yl]cyclobutanamine —— C17H29N5S
cis-3-[4-cyclopropyl-5-({4-[(methylthio)methyl]piperidin-1-yl}methyl)-4H-1,2,4-triazol-3-yl]cyclobutanamine
—— (cis-3-{4-(2-methoxyethyl)-5-[(4-pyridin-3-ylpiperazin-1-yl)methyl]-4H-1,2,4-triazol-3-yl}cyclobutyl)amine —— C19H29N7O
(cis-3-{4-(2-methoxyethyl)-5-[(4-pyridin-3-ylpiperazin-1-yl)methyl]-4H-1,2,4-triazol-3-yl}cyclobutyl)amine
—— [cis-3-(6-{4-[5-(Trifluoromethyl)-1,3,4-thiadiazol-2-yl]piperazin-1-yl}pyrimidin-4-yl)cyclobutyl]amine —— C15H18F3N7S
[cis-3-(6-{4-[5-(Trifluoromethyl)-1,3,4-thiadiazol-2-yl]piperazin-1-yl}pyrimidin-4-yl)cyclobutyl]amine
—— [cis-3-(4-cyclopropyl-5-{[4-(4H-1,2,4-triazol-4-yl)piperidin-1-yl]methyl}-4H-1,2,4-triazol-3-yl)cyclobutyl]amine —— C17H26N8
[cis-3-(4-cyclopropyl-5-{[4-(4H-1,2,4-triazol-4-yl)piperidin-1-yl]methyl}-4H-1,2,4-triazol-3-yl)cyclobutyl]amine
—— [cis-3-(4-cyclopropyl-5-{[4-(2-methylpyridin-4-yl)piperazin-1-yl]methyl}-4H-1,2,4-triazol-3-yl)cyclobutyl]amine —— C20H29N7
[cis-3-(4-cyclopropyl-5-{[4-(2-methylpyridin-4-yl)piperazin-1-yl]methyl}-4H-1,2,4-triazol-3-yl)cyclobutyl]amine
—— Cyclopropyl[5-(4-methoxypyrimidin-2-yl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-2-yl]methanol —— C15H19N5O2
Cyclopropyl[5-(4-methoxypyrimidin-2-yl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-2-yl]methanol
—— cis-3-[5-({[3-(3,4-dihydroquinolin-1(2H)-yl)propyl]amino}methyl)-4-methyl-4H-1,2,4-triazol-3-yl]cyclobutanamine —— C20H30N6
cis-3-[5-({[3-(3,4-dihydroquinolin-1(2H)-yl)propyl]amino}methyl)-4-methyl-4H-1,2,4-triazol-3-yl]cyclobutanamine
—— [cis-3-(4-cyclopropyl-5-{[4-(2-methoxyphenyl)piperazin-1-yl]methyl}-4H-1,2,4-triazol-3-yl)cyclobutyl]amine —— C21H30N6O
[cis-3-(4-cyclopropyl-5-{[4-(2-methoxyphenyl)piperazin-1-yl]methyl}-4H-1,2,4-triazol-3-yl)cyclobutyl]amine
—— {[cis-3-({5-[(methylthio)methyl]-2-furoyl}amino)tetrahydro-2H-pyran-4-yl]oxy}acetic acid —— C14H19NO6S
{[cis-3-({5-[(methylthio)methyl]-2-furoyl}amino)tetrahydro-2H-pyran-4-yl]oxy}acetic acid
—— cyclopropyl[5-(4,5,6,7-tetrahydro-1-benzothien-2-ylcarbonyl)-5,6,7,8-tetrahydro-4H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methanol —— C20H25N3O2S
cyclopropyl[5-(4,5,6,7-tetrahydro-1-benzothien-2-ylcarbonyl)-5,6,7,8-tetrahydro-4H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methanol
—— (cis-3-{4-methyl-5-[(4-phenylpiperidin-1-yl)methyl]-4H-1,2,4-triazol-3-yl}cyclobutyl)amine —— C19H27N5
(cis-3-{4-methyl-5-[(4-phenylpiperidin-1-yl)methyl]-4H-1,2,4-triazol-3-yl}cyclobutyl)amine
—— cis-3-{4-methyl-5-[({[5-(2-thienylmethyl)-1,2,4-oxadiazol-3-yl]methyl}amino)methyl]-4H-1,2,4-triazol-3-yl}cyclobutanamine —— C16H21N7OS
cis-3-{4-methyl-5-[({[5-(2-thienylmethyl)-1,2,4-oxadiazol-3-yl]methyl}amino)methyl]-4H-1,2,4-triazol-3-yl}cyclobutanamine
—— (cis-3-{5-[(4-chloro-2-methoxyphenoxy)methyl]-4-ethyl-4H-1,2,4-triazol-3-yl}cyclobutyl)amine —— C16H21ClN4O2
(cis-3-{5-[(4-chloro-2-methoxyphenoxy)methyl]-4-ethyl-4H-1,2,4-triazol-3-yl}cyclobutyl)amine
—— cis-3-[4-ethyl-5-({[(2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl)methyl]amino}methyl)-4H-1,2,4-triazol-3-yl]cyclobutanamine —— C15H22N8S
cis-3-[4-ethyl-5-({[(2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl)methyl]amino}methyl)-4H-1,2,4-triazol-3-yl]cyclobutanamine
—— cis-3-(4-methyl-5-{[methyl(quinoxalin-2-ylmethyl)amino]methyl}-4H-1,2,4-triazol-3-yl)cyclobutanamine —— C18H23N7
cis-3-(4-methyl-5-{[methyl(quinoxalin-2-ylmethyl)amino]methyl}-4H-1,2,4-triazol-3-yl)cyclobutanamine
—— cis-3-(4-cyclopropyl-5-{[methyl(pyridin-3-ylmethyl)amino]methyl}-4H-1,2,4-triazol-3-yl)cyclobutanamine —— C17H24N6
cis-3-(4-cyclopropyl-5-{[methyl(pyridin-3-ylmethyl)amino]methyl}-4H-1,2,4-triazol-3-yl)cyclobutanamine
—— (cis-3-{2-Cyclopropyl-6-[4-(methylsulfonyl)piperazin-1-yl]pyrimidin-4-yl}cyclobutyl)amine —— C16H25N5O2S
(cis-3-{2-Cyclopropyl-6-[4-(methylsulfonyl)piperazin-1-yl]pyrimidin-4-yl}cyclobutyl)amine
—— cis-3-[4-methyl-5-({[2-(4-methyl-1H-1,2,3-triazol-1-yl)ethyl]amino}methyl)-4H-1,2,4-triazol-3-yl]cyclobutanamine —— C13H22N8
cis-3-[4-methyl-5-({[2-(4-methyl-1H-1,2,3-triazol-1-yl)ethyl]amino}methyl)-4H-1,2,4-triazol-3-yl]cyclobutanamine
—— cyclobutyl{5-[3-(1,2-oxazinan-2-yl)propanoyl]-5,6,7,8-tetrahydro-4H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methanol —— C19H30N4O3
cyclobutyl{5-[3-(1,2-oxazinan-2-yl)propanoyl]-5,6,7,8-tetrahydro-4H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methanol
—— [cis-3-(4-ethyl-5-{[4-(2-oxo-2-piperidin-1-ylethyl)piperazin-1-yl]methyl}-4H-1,2,4-triazol-3-yl)cyclobutyl]amine —— C20H35N7O
[cis-3-(4-ethyl-5-{[4-(2-oxo-2-piperidin-1-ylethyl)piperazin-1-yl]methyl}-4H-1,2,4-triazol-3-yl)cyclobutyl]amine
—— cis-3-(4-cyclopropyl-5-{[methyl(3-pyrrolidin-1-ylpropyl)amino]methyl}-4H-1,2,4-triazol-3-yl)cyclobutanamine —— C18H32N6
cis-3-(4-cyclopropyl-5-{[methyl(3-pyrrolidin-1-ylpropyl)amino]methyl}-4H-1,2,4-triazol-3-yl)cyclobutanamine
—— Cyclopropyl{5-[(3,5-difluorophenyl)acetyl]-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-2-yl}methanol —— C18H19F2N3O2
Cyclopropyl{5-[(3,5-difluorophenyl)acetyl]-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-2-yl}methanol
—— [cis-3-(4-(2-methoxyethyl)-5-{[3-(trifluoromethyl)-1H-1,2,4-triazol-1-yl]methyl}-4H-1,2,4-triazol-3-yl)cyclobutyl]amine —— C13H18F3N7O
[cis-3-(4-(2-methoxyethyl)-5-{[3-(trifluoromethyl)-1H-1,2,4-triazol-1-yl]methyl}-4H-1,2,4-triazol-3-yl)cyclobutyl]amine
—— cyclopropyl{5-[3-(1H-tetrazol-1-yl)propanoyl]-5,6,7,8-tetrahydro-4H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methanol —— C15H21N7O2
cyclopropyl{5-[3-(1H-tetrazol-1-yl)propanoyl]-5,6,7,8-tetrahydro-4H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methanol
—— cis-3-[4-methyl-5-({methyl[(3-methylpyridin-2-yl)methyl]amino}methyl)-4H-1,2,4-triazol-3-yl]cyclobutanamine —— C16H24N6
cis-3-[4-methyl-5-({methyl[(3-methylpyridin-2-yl)methyl]amino}methyl)-4H-1,2,4-triazol-3-yl]cyclobutanamine
—— (cis-3-{2-(Methoxymethyl)-6-[4-(methylsulfonyl)piperazin-1-yl]pyrimidin-4-yl}cyclobutyl)amine —— C15H25N5O3S
(cis-3-{2-(Methoxymethyl)-6-[4-(methylsulfonyl)piperazin-1-yl]pyrimidin-4-yl}cyclobutyl)amine
—— (cis-3-{6-[4-(Pyrrolidin-1-ylcarbonyl)piperidin-1-yl]pyrimidin-4-yl}cyclobutyl)amine —— C18H27N5O
(cis-3-{6-[4-(Pyrrolidin-1-ylcarbonyl)piperidin-1-yl]pyrimidin-4-yl}cyclobutyl)amine
—— (cis-3-{4-methyl-5-[(3-morpholin-4-ylphenoxy)methyl]-4H-1,2,4-triazol-3-yl}cyclobutyl)amine —— C18H25N5O2
(cis-3-{4-methyl-5-[(3-morpholin-4-ylphenoxy)methyl]-4H-1,2,4-triazol-3-yl}cyclobutyl)amine
—— Cyclopropyl[5-(quinolin-6-ylcarbonyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-2-yl]methanol —— C20H20N4O2
Cyclopropyl[5-(quinolin-6-ylcarbonyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-2-yl]methanol
—— cyanomethyl (E)-3-(3-chloro-4,5-dimethoxyphenyl)prop-2-enoate —— C13H12ClNO4
cyanomethyl (E)-3-(3-chloro-4,5-dimethoxyphenyl)prop-2-enoate
—— cis-3-[2-Methyl-6-(4-thiomorpholin-4-ylpiperidin-1-yl)pyrimidin-4-yl]cyclobutanol —— C18H28N4OS
cis-3-[2-Methyl-6-(4-thiomorpholin-4-ylpiperidin-1-yl)pyrimidin-4-yl]cyclobutanol