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—— (6S)-6-[(2S,3R,8aR)-3,8,8-trimethyl-2,3,4,6,7,8a-hexahydro-1H-naphthalen-2-yl]-3-benzylsulfanyl-6,7-dihydro-[1,2,4]triazino[5,6-d][3,1]benzoxazepine —— C30H34N4OS
(6S)-6-[(2S,3R,8aR)-3,8,8-trimethyl-2,3,4,6,7,8a-hexahydro-1H-naphthalen-2-yl]-3-benzylsulfanyl-6,7-dihydro-[1,2,4]triazino[5,6-d][3,1]benzoxazepine
—— (6S)-6-[(1R,6S)-6-methyl-4-(4-methylpent-3-enyl)cyclohex-3-en-1-yl]-3-prop-2-enylsulfanyl-6,7-dihydro-[1,2,4]triazino[5,6-d][3,1]benzoxazepine —— C26H32N4OS
(6S)-6-[(1R,6S)-6-methyl-4-(4-methylpent-3-enyl)cyclohex-3-en-1-yl]-3-prop-2-enylsulfanyl-6,7-dihydro-[1,2,4]triazino[5,6-d][3,1]benzoxazepine
—— (6S)-6-[(2S,3S,8aS)-3,8,8-trimethyl-2,3,4,6,7,8a-hexahydro-1H-naphthalen-2-yl]-3-benzylsulfanyl-6,7-dihydro-[1,2,4]triazino[5,6-d][3,1]benzoxazepine —— C30H34N4OS
(6S)-6-[(2S,3S,8aS)-3,8,8-trimethyl-2,3,4,6,7,8a-hexahydro-1H-naphthalen-2-yl]-3-benzylsulfanyl-6,7-dihydro-[1,2,4]triazino[5,6-d][3,1]benzoxazepine
—— 6-[(5E)-4-oxo-2-sulfanylidene-5-[[3-(trifluoromethyl)phenyl]methylidene]-1,3-thiazolidin-3-yl]hexanoic acid —— C17H16F3NO3S2
6-[(5E)-4-oxo-2-sulfanylidene-5-[[3-(trifluoromethyl)phenyl]methylidene]-1,3-thiazolidin-3-yl]hexanoic acid
—— 6-[(5E)-5-[[2-(difluoromethoxy)phenyl]methylidene]-4-oxo-2-sulfanylidene-1,3-thiazolidin-3-yl]hexanoate —— C17H16F2NO4S2-
6-[(5E)-5-[[2-(difluoromethoxy)phenyl]methylidene]-4-oxo-2-sulfanylidene-1,3-thiazolidin-3-yl]hexanoate
—— 6-[(5Z)-5-[[2,5-dimethyl-1-(2-methylpropyl)pyrrol-3-yl]methylidene]-4-oxo-2-sulfanylidene-1,3-thiazolidin-3-yl]hexanoate —— C20H27N2O3S2-
6-[(5Z)-5-[[2,5-dimethyl-1-(2-methylpropyl)pyrrol-3-yl]methylidene]-4-oxo-2-sulfanylidene-1,3-thiazolidin-3-yl]hexanoate
—— 6-[(5E)-5-[[2-(difluoromethoxy)phenyl]methylidene]-4-oxo-2-sulfanylidene-1,3-thiazolidin-3-yl]hexanoic acid —— C17H17F2NO4S2
6-[(5E)-5-[[2-(difluoromethoxy)phenyl]methylidene]-4-oxo-2-sulfanylidene-1,3-thiazolidin-3-yl]hexanoic acid
—— (6-Ethyl-7-hydroxy-2-oxochromen-4-yl)methyl 2-(2-methoxy-5-methylphenyl)acetate —— C22H22O6
(6-Ethyl-7-hydroxy-2-oxochromen-4-yl)methyl 2-(2-methoxy-5-methylphenyl)acetate
—— (6E)-5-imino-2-(2-morpholin-4-yl-2-oxoethyl)-6-[[4-[(2-nitrophenyl)methoxy]phenyl]methylidene]-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C25H22N6O6S
(6E)-5-imino-2-(2-morpholin-4-yl-2-oxoethyl)-6-[[4-[(2-nitrophenyl)methoxy]phenyl]methylidene]-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— (6-Methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl 2-(2,4-dichlorophenoxy)acetate —— C18H14Cl2N2O4
(6-Methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl 2-(2,4-dichlorophenoxy)acetate
—— 6-(4-benzylpiperidin-1-yl)-1,4-dimethyl-2-oxo-5-[(E)-[4-oxo-3-[[(2R)-oxolan-2-yl]methyl]-2-sulfanylidene-1,3-thiazolidin-5-ylidene]methyl]pyridine-3-carbonitrile —— C29H32N4O3S2
6-(4-benzylpiperidin-1-yl)-1,4-dimethyl-2-oxo-5-[(E)-[4-oxo-3-[[(2R)-oxolan-2-yl]methyl]-2-sulfanylidene-1,3-thiazolidin-5-ylidene]methyl]pyridine-3-carbonitrile
—— 6-[2-(3,4-difluorophenyl)sulfanylacetyl]-3,4-dihydro-1H-quinolin-2-one —— C17H13F2NO2S
6-[2-(3,4-difluorophenyl)sulfanylacetyl]-3,4-dihydro-1H-quinolin-2-one
—— (6-Methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl 3-(furan-2-carbonylamino)-4-methylbenzoate —— C23H19N3O5
(6-Methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl 3-(furan-2-carbonylamino)-4-methylbenzoate
—— 6-(4-benzylpiperidin-1-yl)-1,4-dimethyl-2-oxo-5-[(E)-[4-oxo-3-[[(2S)-oxolan-2-yl]methyl]-2-sulfanylidene-1,3-thiazolidin-5-ylidene]methyl]pyridine-3-carbonitrile —— C29H32N4O3S2
6-(4-benzylpiperidin-1-yl)-1,4-dimethyl-2-oxo-5-[(E)-[4-oxo-3-[[(2S)-oxolan-2-yl]methyl]-2-sulfanylidene-1,3-thiazolidin-5-ylidene]methyl]pyridine-3-carbonitrile
—— (6R)-2-amino-N-ethyl-6-propyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide —— C14H22N2OS
(6R)-2-amino-N-ethyl-6-propyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide
—— (6R)-2-amino-N-cyclopropyl-6-propyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide —— C15H22N2OS
(6R)-2-amino-N-cyclopropyl-6-propyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide
—— (6S)-2-amino-N-propan-2-yl-6-propyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide —— C15H24N2OS
(6S)-2-amino-N-propan-2-yl-6-propyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide
—— (6R)-2-amino-N,N-dimethyl-6-propyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide —— C14H22N2OS
(6R)-2-amino-N,N-dimethyl-6-propyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide
—— (6E)-5-imino-2-(2-morpholin-4-yl-2-oxoethyl)-6-[[5-(4-nitrophenyl)furan-2-yl]methylidene]-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C22H18N6O6S
(6E)-5-imino-2-(2-morpholin-4-yl-2-oxoethyl)-6-[[5-(4-nitrophenyl)furan-2-yl]methylidene]-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— (6R)-2-amino-N,6-dipropyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide —— C15H24N2OS
(6R)-2-amino-N,6-dipropyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide
—— (6-Methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl 2-(4-ethylphenoxy)acetate —— C20H20N2O4
(6-Methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl 2-(4-ethylphenoxy)acetate
—— (6S)-2-amino-N-ethyl-6-propyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide —— C14H22N2OS
(6S)-2-amino-N-ethyl-6-propyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide
—— (6S)-2-amino-N,N-dimethyl-6-propyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide —— C14H22N2OS
(6S)-2-amino-N,N-dimethyl-6-propyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide
—— (6S)-2-amino-N-methyl-6-propyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide —— C13H20N2OS
(6S)-2-amino-N-methyl-6-propyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide
—— (6S)-2-amino-N-cyclopropyl-6-propyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide —— C15H22N2OS
(6S)-2-amino-N-cyclopropyl-6-propyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide
—— (6R)-2-amino-N-methyl-6-propyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide —— C13H20N2OS
(6R)-2-amino-N-methyl-6-propyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide
—— (6S)-2-amino-N,6-dipropyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide —— C15H24N2OS
(6S)-2-amino-N,6-dipropyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide
—— 6-imidazol-1-yl-N-[(1S,2R,4R)-1,7,7-trimethyl-2-bicyclo[2.2.1]heptanyl]pyridine-3-carboxamide —— C19H24N4O
6-imidazol-1-yl-N-[(1S,2R,4R)-1,7,7-trimethyl-2-bicyclo[2.2.1]heptanyl]pyridine-3-carboxamide
—— 6-amino-5-[(2S)-2-[5-(4-fluorophenyl)-3-(2-methoxyethyl)-4-oxothieno[2,3-d]pyrimidin-2-yl]sulfanylpropanoyl]-1,3-dimethylpyrimidine-2,4-dione —— C24H24FN5O5S2
6-amino-5-[(2S)-2-[5-(4-fluorophenyl)-3-(2-methoxyethyl)-4-oxothieno[2,3-d]pyrimidin-2-yl]sulfanylpropanoyl]-1,3-dimethylpyrimidine-2,4-dione
—— 6-amino-5-[(2R)-2-[5-(4-fluorophenyl)-3-(2-methoxyethyl)-4-oxothieno[2,3-d]pyrimidin-2-yl]sulfanylpropanoyl]-1,3-dimethylpyrimidine-2,4-dione —— C24H24FN5O5S2
6-amino-5-[(2R)-2-[5-(4-fluorophenyl)-3-(2-methoxyethyl)-4-oxothieno[2,3-d]pyrimidin-2-yl]sulfanylpropanoyl]-1,3-dimethylpyrimidine-2,4-dione
—— (6-nitro-4H-1,3-benzodioxin-8-yl)methyl (2S,3R)-2-(3,4-dimethoxyphenyl)-1-(4-methylphenyl)-6-oxopiperidine-3-carboxylate —— C30H30N2O9
(6-nitro-4H-1,3-benzodioxin-8-yl)methyl (2S,3R)-2-(3,4-dimethoxyphenyl)-1-(4-methylphenyl)-6-oxopiperidine-3-carboxylate
—— (6-Methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl 2,5-dimethylfuran-3-carboxylate —— C17H16N2O4
(6-Methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl 2,5-dimethylfuran-3-carboxylate
—— 6-[(2R,6R)-2,6-dimethylmorpholine-4-carbonyl]-2-phenyl-4,5-dihydropyridazin-3-one —— C17H21N3O3
6-[(2R,6R)-2,6-dimethylmorpholine-4-carbonyl]-2-phenyl-4,5-dihydropyridazin-3-one
—— 6-(4-benzylpiperidin-1-yl)-5-[(E)-[3-(furan-2-ylmethyl)-4-oxo-2-sulfanylidene-1,3-thiazolidin-5-ylidene]methyl]-1,4-dimethyl-2-oxopyridine-3-carbonitrile —— C29H28N4O3S2
6-(4-benzylpiperidin-1-yl)-5-[(E)-[3-(furan-2-ylmethyl)-4-oxo-2-sulfanylidene-1,3-thiazolidin-5-ylidene]methyl]-1,4-dimethyl-2-oxopyridine-3-carbonitrile
—— (6-nitro-4H-1,3-benzodioxin-8-yl)methyl (2S,3S)-2-(3,4-dimethoxyphenyl)-1-(4-methylphenyl)-6-oxopiperidine-3-carboxylate —— C30H30N2O9
(6-nitro-4H-1,3-benzodioxin-8-yl)methyl (2S,3S)-2-(3,4-dimethoxyphenyl)-1-(4-methylphenyl)-6-oxopiperidine-3-carboxylate
—— 6-(4-benzylpiperazin-1-yl)-1,4-dimethyl-5-[(E)-[3-[(4-methylphenyl)methyl]-4-oxo-2-sulfanylidene-1,3-thiazolidin-5-ylidene]methyl]-2-oxopyridine-3-carbonitrile —— C31H31N5O2S2
6-(4-benzylpiperazin-1-yl)-1,4-dimethyl-5-[(E)-[3-[(4-methylphenyl)methyl]-4-oxo-2-sulfanylidene-1,3-thiazolidin-5-ylidene]methyl]-2-oxopyridine-3-carbonitrile
—— (6-chloro-4H-1,3-benzodioxin-8-yl)methyl (2R)-2-(3-methylphenoxy)propanoate —— C19H19ClO5
(6-chloro-4H-1,3-benzodioxin-8-yl)methyl (2R)-2-(3-methylphenoxy)propanoate
—— (6E)-5-imino-6-[[4-[(2-nitrophenyl)methoxy]phenyl]methylidene]-2-(2-oxo-2-pyrrolidin-1-ylethyl)-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C25H22N6O5S
(6E)-5-imino-6-[[4-[(2-nitrophenyl)methoxy]phenyl]methylidene]-2-(2-oxo-2-pyrrolidin-1-ylethyl)-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— (6-nitro-4H-1,3-benzodioxin-8-yl)methyl (2R,3R)-2-(3,4-dimethoxyphenyl)-1-(4-methylphenyl)-6-oxopiperidine-3-carboxylate —— C30H30N2O9
(6-nitro-4H-1,3-benzodioxin-8-yl)methyl (2R,3R)-2-(3,4-dimethoxyphenyl)-1-(4-methylphenyl)-6-oxopiperidine-3-carboxylate
—— (6-Methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl 1-oxidopyridin-1-ium-4-carboxylate —— C16H13N3O4
(6-Methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl 1-oxidopyridin-1-ium-4-carboxylate
—— 6-amino-5-[(2R)-2-[[5-[(5S)-5-tert-butyl-4,5,6,7-tetrahydro-1-benzothiophen-2-yl]-4-prop-2-enyl-1,2,4-triazol-3-yl]sulfanyl]propanoyl]-1,3-dimethylpyrimidine-2,4-dione —— C26H34N6O3S2
6-amino-5-[(2R)-2-[[5-[(5S)-5-tert-butyl-4,5,6,7-tetrahydro-1-benzothiophen-2-yl]-4-prop-2-enyl-1,2,4-triazol-3-yl]sulfanyl]propanoyl]-1,3-dimethylpyrimidine-2,4-dione
—— (6-Methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl 2,3-dihydro-1,4-benzodioxine-6-carboxylate —— C19H16N2O5
(6-Methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl 2,3-dihydro-1,4-benzodioxine-6-carboxylate
—— (6-Methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl 2-benzylbenzoate —— C24H20N2O3
(6-Methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl 2-benzylbenzoate
—— (6-chloro-7-methyl-2-oxochromen-4-yl)methyl (E)-3-(1,3-benzoxazol-2-yl)prop-2-enoate —— C21H14ClNO5
(6-chloro-7-methyl-2-oxochromen-4-yl)methyl (E)-3-(1,3-benzoxazol-2-yl)prop-2-enoate
—— (6-Methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl 4-tert-butylcyclohexane-1-carboxylate —— C21H28N2O3
(6-Methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl 4-tert-butylcyclohexane-1-carboxylate
—— (6-Methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl 3-chloro-1-benzothiophene-2-carboxylate —— C19H13ClN2O3S
(6-Methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl 3-chloro-1-benzothiophene-2-carboxylate
—— (6-Methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl 3,4-dimethylbenzoate —— C19H18N2O3
(6-Methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl 3,4-dimethylbenzoate
—— (6R)-6-[4-(4-methoxyphenyl)piperazine-1-carbonyl]-2-methylsulfanylthieno[2,3-d]pyrimidin-5-one —— C19H20N4O3S2
(6R)-6-[4-(4-methoxyphenyl)piperazine-1-carbonyl]-2-methylsulfanylthieno[2,3-d]pyrimidin-5-one
—— (6-Methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl 2-(2-methylphenoxy)acetate —— C19H18N2O4
(6-Methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl 2-(2-methylphenoxy)acetate
—— 6-Amino-5-[2-[1-(3,4-dimethylphenyl)imidazol-2-yl]sulfanylacetyl]-1-propylpyrimidine-2,4-dione —— C20H23N5O3S
6-Amino-5-[2-[1-(3,4-dimethylphenyl)imidazol-2-yl]sulfanylacetyl]-1-propylpyrimidine-2,4-dione