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—— (6E)-6-[(2,5-dimethoxyphenyl)methylidene]-2-heptyl-5-imino-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C21H26N4O3S
(6E)-6-[(2,5-dimethoxyphenyl)methylidene]-2-heptyl-5-imino-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— (6E)-5-imino-6-[[2-[2-(3-methoxyphenoxy)ethoxy]-5-nitrophenyl]methylidene]-2-propan-2-yl-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C24H23N5O6S
(6E)-5-imino-6-[[2-[2-(3-methoxyphenoxy)ethoxy]-5-nitrophenyl]methylidene]-2-propan-2-yl-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— (6E)-5-imino-6-[[3-methoxy-4-[(1S)-1-phenylethoxy]phenyl]methylidene]-2-propyl-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C24H24N4O3S
(6E)-5-imino-6-[[3-methoxy-4-[(1S)-1-phenylethoxy]phenyl]methylidene]-2-propyl-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— (6E)-6-benzylidene-2-heptyl-5-imino-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C19H22N4OS
(6E)-6-benzylidene-2-heptyl-5-imino-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— (6E)-5-imino-6-[[3-methoxy-4-(2-phenoxyethoxy)phenyl]methylidene]-2-propyl-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C24H24N4O4S
(6E)-5-imino-6-[[3-methoxy-4-(2-phenoxyethoxy)phenyl]methylidene]-2-propyl-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— (6E)-5-imino-6-[[3-methoxy-4-[2-(2-prop-2-enylphenoxy)ethoxy]phenyl]methylidene]-2-propan-2-yl-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C27H28N4O4S
(6E)-5-imino-6-[[3-methoxy-4-[2-(2-prop-2-enylphenoxy)ethoxy]phenyl]methylidene]-2-propan-2-yl-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— (6E)-5-imino-6-[[4-[2-(4-nitrophenoxy)ethoxy]phenyl]methylidene]-2-propan-2-yl-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C23H21N5O5S
(6E)-5-imino-6-[[4-[2-(4-nitrophenoxy)ethoxy]phenyl]methylidene]-2-propan-2-yl-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— (6E)-6-[[4-[2-(4-bromophenoxy)ethoxy]-3-methoxyphenyl]methylidene]-5-imino-2-propan-2-yl-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C24H23BrN4O4S
(6E)-6-[[4-[2-(4-bromophenoxy)ethoxy]-3-methoxyphenyl]methylidene]-5-imino-2-propan-2-yl-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— (6E)-6-[[4-[2-[4-[(2S)-butan-2-yl]phenoxy]ethoxy]-3-methoxyphenyl]methylidene]-5-imino-2-propyl-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C28H32N4O4S
(6E)-6-[[4-[2-[4-[(2S)-butan-2-yl]phenoxy]ethoxy]-3-methoxyphenyl]methylidene]-5-imino-2-propyl-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— (6E)-6-[[2-[2-(4-bromophenoxy)ethoxy]phenyl]methylidene]-5-imino-2-propyl-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C23H21BrN4O3S
(6E)-6-[[2-[2-(4-bromophenoxy)ethoxy]phenyl]methylidene]-5-imino-2-propyl-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— 6-[[(1R,5R)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl]sulfonyl]-1H-benzo[cd]indol-2-one —— C21H24N2O3S
6-[[(1R,5R)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl]sulfonyl]-1H-benzo[cd]indol-2-one
—— 6-[[(E)-3-(3-bromophenyl)-2-(furan-2-carbonylamino)prop-2-enoyl]amino]hexanoic acid —— C20H21BrN2O5
6-[[(E)-3-(3-bromophenyl)-2-(furan-2-carbonylamino)prop-2-enoyl]amino]hexanoic acid
—— 6-Chloro-7-[[4-(difluoromethoxy)-3-methoxyphenyl]methoxy]-4-methylchromen-2-one —— C19H15ClF2O5
6-Chloro-7-[[4-(difluoromethoxy)-3-methoxyphenyl]methoxy]-4-methylchromen-2-one
—— (6R)-2-[(3-fluorophenyl)sulfonylamino]-6-methyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide —— C16H17FN2O3S2
(6R)-2-[(3-fluorophenyl)sulfonylamino]-6-methyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide
—— (6S)-2-[(4-fluorophenyl)sulfonylamino]-6-methyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide —— C16H17FN2O3S2
(6S)-2-[(4-fluorophenyl)sulfonylamino]-6-methyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide
—— 6-Chloro-4-methyl-7-[2-(5-methylthiophen-2-yl)-2-oxoethoxy]chromen-2-one —— C17H13ClO4S
6-Chloro-4-methyl-7-[2-(5-methylthiophen-2-yl)-2-oxoethoxy]chromen-2-one
—— (6S)-2-[(2-chlorophenyl)sulfonylamino]-6-methyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide —— C16H17ClN2O3S2
(6S)-2-[(2-chlorophenyl)sulfonylamino]-6-methyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide
—— (6R)-2-[(3-acetylphenyl)sulfonylamino]-6-methyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide —— C18H20N2O4S2
(6R)-2-[(3-acetylphenyl)sulfonylamino]-6-methyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide
—— (6S)-2-[(3-chloro-4-fluorophenyl)sulfonylamino]-6-methyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide —— C16H16ClFN2O3S2
(6S)-2-[(3-chloro-4-fluorophenyl)sulfonylamino]-6-methyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide
—— (6S)-2-[(4-acetylphenyl)sulfonylamino]-6-methyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide —— C18H20N2O4S2
(6S)-2-[(4-acetylphenyl)sulfonylamino]-6-methyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide
—— (6R)-6-methyl-2-(thiophen-2-ylsulfonylamino)-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide —— C14H16N2O3S3
(6R)-6-methyl-2-(thiophen-2-ylsulfonylamino)-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide
—— 6-[(Z)-3-(dimethylamino)prop-2-enoyl]-7-hydroxy-4,8-dimethylchromen-2-one —— C16H17NO4
6-[(Z)-3-(dimethylamino)prop-2-enoyl]-7-hydroxy-4,8-dimethylchromen-2-one
—— (6S,9S)-5-[(4-chlorophenyl)methyl]-6,9-bis(furan-2-yl)-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one —— C28H23ClN2O3
(6S,9S)-5-[(4-chlorophenyl)methyl]-6,9-bis(furan-2-yl)-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one
—— (6S,9S)-6-(4-chlorophenyl)-5-[(4-chlorophenyl)methyl]-9-(furan-2-yl)-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one —— C30H24Cl2N2O2
(6S,9S)-6-(4-chlorophenyl)-5-[(4-chlorophenyl)methyl]-9-(furan-2-yl)-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one
—— 6-[(Z)-3-(dimethylamino)prop-2-enoyl]-7-hydroxy-3,4,8-trimethylchromen-2-one —— C17H19NO4
6-[(Z)-3-(dimethylamino)prop-2-enoyl]-7-hydroxy-3,4,8-trimethylchromen-2-one
—— (6E)-6-[[3-bromo-4-[2-[4-[(2S)-butan-2-yl]phenoxy]ethoxy]-5-ethoxyphenyl]methylidene]-2-ethyl-5-imino-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C28H31BrN4O4S
(6E)-6-[[3-bromo-4-[2-[4-[(2S)-butan-2-yl]phenoxy]ethoxy]-5-ethoxyphenyl]methylidene]-2-ethyl-5-imino-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— (6E)-2-ethyl-6-[[1-[2-(4-hexoxyphenoxy)ethyl]indol-3-yl]methylidene]-5-imino-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C30H33N5O3S
(6E)-2-ethyl-6-[[1-[2-(4-hexoxyphenoxy)ethyl]indol-3-yl]methylidene]-5-imino-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— (6E)-6-[[5-bromo-2-[2-(4-tert-butylphenoxy)ethoxy]phenyl]methylidene]-2-ethyl-5-imino-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C26H27BrN4O3S
(6E)-6-[[5-bromo-2-[2-(4-tert-butylphenoxy)ethoxy]phenyl]methylidene]-2-ethyl-5-imino-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— (6R,9S)-5-[(4-chlorophenyl)methyl]-6,9-bis(furan-2-yl)-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one —— C28H23ClN2O3
(6R,9S)-5-[(4-chlorophenyl)methyl]-6,9-bis(furan-2-yl)-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one
—— (6E)-6-[[4-[2-(4-chlorophenyl)sulfanylethoxy]phenyl]methylidene]-2-ethyl-5-imino-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C22H19ClN4O2S2
(6E)-6-[[4-[2-(4-chlorophenyl)sulfanylethoxy]phenyl]methylidene]-2-ethyl-5-imino-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— 6,7,8,9-Tetrahydrodibenzofuran-2-yl 2-(2-cyanophenoxy)acetate —— C21H17NO4
6,7,8,9-Tetrahydrodibenzofuran-2-yl 2-(2-cyanophenoxy)acetate
—— (6E)-6-[[5-chloro-2-[2-(3,4-dimethylphenoxy)ethoxy]phenyl]methylidene]-2-ethyl-5-imino-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C24H23ClN4O3S
(6E)-6-[[5-chloro-2-[2-(3,4-dimethylphenoxy)ethoxy]phenyl]methylidene]-2-ethyl-5-imino-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— (6R,9S)-6-(4-chlorophenyl)-5-[(4-chlorophenyl)methyl]-9-(furan-2-yl)-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one —— C30H24Cl2N2O2
(6R,9S)-6-(4-chlorophenyl)-5-[(4-chlorophenyl)methyl]-9-(furan-2-yl)-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one
—— (6E)-6-[[3-chloro-5-ethoxy-4-[2-(2-prop-2-enylphenoxy)ethoxy]phenyl]methylidene]-2-ethyl-5-imino-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C27H27ClN4O4S
(6E)-6-[[3-chloro-5-ethoxy-4-[2-(2-prop-2-enylphenoxy)ethoxy]phenyl]methylidene]-2-ethyl-5-imino-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— (6E)-6-[[3-bromo-5-ethoxy-4-[2-(3-ethyl-5-methylphenoxy)ethoxy]phenyl]methylidene]-2-ethyl-5-imino-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C27H29BrN4O4S
(6E)-6-[[3-bromo-5-ethoxy-4-[2-(3-ethyl-5-methylphenoxy)ethoxy]phenyl]methylidene]-2-ethyl-5-imino-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— (6E)-6-[[3-[2-(3,4-dimethylphenoxy)ethoxy]phenyl]methylidene]-2-ethyl-5-imino-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C24H24N4O3S
(6E)-6-[[3-[2-(3,4-dimethylphenoxy)ethoxy]phenyl]methylidene]-2-ethyl-5-imino-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— (6-anilinopyridin-3-yl)-[(2S)-4-(2-nitrophenyl)-2-phenylpiperazin-1-yl]methanone —— C28H25N5O3
(6-anilinopyridin-3-yl)-[(2S)-4-(2-nitrophenyl)-2-phenylpiperazin-1-yl]methanone
—— (6E)-6-[[2-[2-(4-bromophenoxy)ethoxy]phenyl]methylidene]-2-ethyl-5-imino-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C22H19BrN4O3S
(6E)-6-[[2-[2-(4-bromophenoxy)ethoxy]phenyl]methylidene]-2-ethyl-5-imino-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— (6E)-6-[[5-chloro-2-[2-(5-methyl-2-propan-2-ylphenoxy)ethoxy]phenyl]methylidene]-2-ethyl-5-imino-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C26H27ClN4O3S
(6E)-6-[[5-chloro-2-[2-(5-methyl-2-propan-2-ylphenoxy)ethoxy]phenyl]methylidene]-2-ethyl-5-imino-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— (6E)-6-[[3-[2-(4-bromophenoxy)ethoxy]phenyl]methylidene]-2-ethyl-5-imino-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C22H19BrN4O3S
(6E)-6-[[3-[2-(4-bromophenoxy)ethoxy]phenyl]methylidene]-2-ethyl-5-imino-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— (6E)-6-[[3-ethoxy-4-[2-(4-methylphenyl)sulfanylethoxy]phenyl]methylidene]-2-ethyl-5-imino-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C25H26N4O3S2
(6E)-6-[[3-ethoxy-4-[2-(4-methylphenyl)sulfanylethoxy]phenyl]methylidene]-2-ethyl-5-imino-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— (6-anilinopyridin-3-yl)-[(2R)-4-(2-nitrophenyl)-2-phenylpiperazin-1-yl]methanone —— C28H25N5O3
(6-anilinopyridin-3-yl)-[(2R)-4-(2-nitrophenyl)-2-phenylpiperazin-1-yl]methanone
—— (6-anilinopyridin-3-yl)-[(2S)-2-(4-fluorophenyl)-4-(2-nitrophenyl)piperazin-1-yl]methanone —— C28H24FN5O3
(6-anilinopyridin-3-yl)-[(2S)-2-(4-fluorophenyl)-4-(2-nitrophenyl)piperazin-1-yl]methanone
—— 6-bromo-3-[(Z)-3-(6-bromo-2,3-dihydro-1,4-benzodioxin-7-yl)prop-2-enoyl]-4-phenyl-1H-quinolin-2-one —— C26H17Br2NO4
6-bromo-3-[(Z)-3-(6-bromo-2,3-dihydro-1,4-benzodioxin-7-yl)prop-2-enoyl]-4-phenyl-1H-quinolin-2-one
—— (6-anilinopyridin-3-yl)-[(2R)-2-(4-fluorophenyl)-4-(2-nitrophenyl)piperazin-1-yl]methanone —— C28H24FN5O3
(6-anilinopyridin-3-yl)-[(2R)-2-(4-fluorophenyl)-4-(2-nitrophenyl)piperazin-1-yl]methanone
—— 6-[(1S,2R,9S,10S,11S,12R,16S)-9-(4-hydroxyphenyl)-6,13,15-trioxo-3,7-dithia-5,14-diazapentacyclo[9.5.1.02,10.04,8.012,16]heptadec-4(8)-en-14-yl]hexanoic acid —— C25H26N2O6S2
6-[(1S,2R,9S,10S,11S,12R,16S)-9-(4-hydroxyphenyl)-6,13,15-trioxo-3,7-dithia-5,14-diazapentacyclo[9.5.1.02,10.04,8.012,16]heptadec-4(8)-en-14-yl]hexanoic acid
—— 6-[(1S,2R,9S,10S,11S,12S,16R)-9-(4-hydroxyphenyl)-6,13,15-trioxo-3,7-dithia-5,14-diazapentacyclo[9.5.1.02,10.04,8.012,16]heptadec-4(8)-en-14-yl]hexanoic acid —— C25H26N2O6S2
6-[(1S,2R,9S,10S,11S,12S,16R)-9-(4-hydroxyphenyl)-6,13,15-trioxo-3,7-dithia-5,14-diazapentacyclo[9.5.1.02,10.04,8.012,16]heptadec-4(8)-en-14-yl]hexanoic acid
—— 6-[(1S,2R,9S,10S,11S,12R,16R)-9-(4-hydroxyphenyl)-6,13,15-trioxo-3,7-dithia-5,14-diazapentacyclo[9.5.1.02,10.04,8.012,16]heptadec-4(8)-en-14-yl]hexanoic acid —— C25H26N2O6S2
6-[(1S,2R,9S,10S,11S,12R,16R)-9-(4-hydroxyphenyl)-6,13,15-trioxo-3,7-dithia-5,14-diazapentacyclo[9.5.1.02,10.04,8.012,16]heptadec-4(8)-en-14-yl]hexanoic acid
—— 6-[(1S,2R,9S,10S,11S,12S,16S)-9-(4-hydroxyphenyl)-6,13,15-trioxo-3,7-dithia-5,14-diazapentacyclo[9.5.1.02,10.04,8.012,16]heptadec-4(8)-en-14-yl]hexanoic acid —— C25H26N2O6S2
6-[(1S,2R,9S,10S,11S,12S,16S)-9-(4-hydroxyphenyl)-6,13,15-trioxo-3,7-dithia-5,14-diazapentacyclo[9.5.1.02,10.04,8.012,16]heptadec-4(8)-en-14-yl]hexanoic acid
—— 6-phenyl-1-propan-2-yl-N-(1,3-thiazol-2-yl)pyrazolo[3,4-b]pyridine-4-carboxamide —— C19H17N5OS
6-phenyl-1-propan-2-yl-N-(1,3-thiazol-2-yl)pyrazolo[3,4-b]pyridine-4-carboxamide