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—— (5-aminothiadiazol-4-yl)-[(3S)-3-(1-propan-2-ylbenzimidazol-2-yl)piperidin-1-yl]methanone —— C18H22N6OS
(5-aminothiadiazol-4-yl)-[(3S)-3-(1-propan-2-ylbenzimidazol-2-yl)piperidin-1-yl]methanone
—— (5R)-4-benzyl-5-methyl-1-[[(3R)-piperidin-3-yl]methyl]-1,4-diazepane —— C19H31N3
(5R)-4-benzyl-5-methyl-1-[[(3R)-piperidin-3-yl]methyl]-1,4-diazepane
—— (5-aminothiadiazol-4-yl)-[(3R)-3-(1-propan-2-ylbenzimidazol-2-yl)piperidin-1-yl]methanone —— C18H22N6OS
(5-aminothiadiazol-4-yl)-[(3R)-3-(1-propan-2-ylbenzimidazol-2-yl)piperidin-1-yl]methanone
—— (5R)-5-[[(2S)-4-(2-fluorophenyl)butan-2-yl]amino]-1-methylpiperidin-2-one —— C16H23FN2O
(5R)-5-[[(2S)-4-(2-fluorophenyl)butan-2-yl]amino]-1-methylpiperidin-2-one
—— (5S)-5-[[(2R)-4-(2-fluorophenyl)butan-2-yl]amino]-1-methylpiperidin-2-one —— C16H23FN2O
(5S)-5-[[(2R)-4-(2-fluorophenyl)butan-2-yl]amino]-1-methylpiperidin-2-one
—— (5S)-5-[[(2S)-4-(2-fluorophenyl)butan-2-yl]amino]-1-methylpiperidin-2-one —— C16H23FN2O
(5S)-5-[[(2S)-4-(2-fluorophenyl)butan-2-yl]amino]-1-methylpiperidin-2-one
—— (5R)-5-[[(2R)-4-(2-fluorophenyl)butan-2-yl]amino]-1-methylpiperidin-2-one —— C16H23FN2O
(5R)-5-[[(2R)-4-(2-fluorophenyl)butan-2-yl]amino]-1-methylpiperidin-2-one
—— 5-[(2S)-2-thiophen-2-ylmorpholin-4-yl]pyridine-2-carbonitrile —— C14H13N3OS
5-[(2S)-2-thiophen-2-ylmorpholin-4-yl]pyridine-2-carbonitrile
—— (5S)-N-[2-(cyclopropylmethyl)-4-methylpyrazol-3-yl]-2-oxa-7-azaspiro[4.4]nonane-7-carboxamide —— C16H24N4O2
(5S)-N-[2-(cyclopropylmethyl)-4-methylpyrazol-3-yl]-2-oxa-7-azaspiro[4.4]nonane-7-carboxamide
—— [(5S,7R)-5,7-dimethyl-6,7-dihydro-5H-pyrazolo[1,5-a]pyrimidin-4-yl]-(4-fluoro-2-nitrophenyl)methanone —— C15H15FN4O3
[(5S,7R)-5,7-dimethyl-6,7-dihydro-5H-pyrazolo[1,5-a]pyrimidin-4-yl]-(4-fluoro-2-nitrophenyl)methanone
—— 5-tert-butyl-3-[[(S)-(1-phenylpyrazol-4-yl)methylsulfinyl]methyl]-1,2,4-oxadiazole —— C17H20N4O2S
5-tert-butyl-3-[[(S)-(1-phenylpyrazol-4-yl)methylsulfinyl]methyl]-1,2,4-oxadiazole
—— 5-tert-butyl-3-[[(R)-(1-phenylpyrazol-4-yl)methylsulfinyl]methyl]-1,2,4-oxadiazole —— C17H20N4O2S
5-tert-butyl-3-[[(R)-(1-phenylpyrazol-4-yl)methylsulfinyl]methyl]-1,2,4-oxadiazole
—— (5R)-N-[2-(cyclopropylmethyl)-4-methylpyrazol-3-yl]-2-oxa-7-azaspiro[4.4]nonane-7-carboxamide —— C16H24N4O2
(5R)-N-[2-(cyclopropylmethyl)-4-methylpyrazol-3-yl]-2-oxa-7-azaspiro[4.4]nonane-7-carboxamide
—— [(5R,7R)-5,7-dimethyl-6,7-dihydro-5H-pyrazolo[1,5-a]pyrimidin-4-yl]-(4-fluoro-2-nitrophenyl)methanone —— C15H15FN4O3
[(5R,7R)-5,7-dimethyl-6,7-dihydro-5H-pyrazolo[1,5-a]pyrimidin-4-yl]-(4-fluoro-2-nitrophenyl)methanone
—— [(5R,7S)-5,7-dimethyl-6,7-dihydro-5H-pyrazolo[1,5-a]pyrimidin-4-yl]-(4-fluoro-2-nitrophenyl)methanone —— C15H15FN4O3
[(5R,7S)-5,7-dimethyl-6,7-dihydro-5H-pyrazolo[1,5-a]pyrimidin-4-yl]-(4-fluoro-2-nitrophenyl)methanone
—— 5-[(3R)-3-(3,5-dimethoxyanilino)piperidin-1-yl]pyridine-2-carbonitrile —— C19H22N4O2
5-[(3R)-3-(3,5-dimethoxyanilino)piperidin-1-yl]pyridine-2-carbonitrile
—— 5-[(3S)-3-(3,5-dimethoxyanilino)piperidin-1-yl]pyridine-2-carbonitrile —— C19H22N4O2
5-[(3S)-3-(3,5-dimethoxyanilino)piperidin-1-yl]pyridine-2-carbonitrile
—— 5-[(1R,6S)-9-propan-2-yl-3,9-diazabicyclo[4.2.1]nonan-3-yl]pyridine-2-carbonitrile —— C16H22N4
5-[(1R,6S)-9-propan-2-yl-3,9-diazabicyclo[4.2.1]nonan-3-yl]pyridine-2-carbonitrile
—— 5-[(2R)-2-thiophen-2-ylmorpholin-4-yl]pyridine-2-carbonitrile —— C14H13N3OS
5-[(2R)-2-thiophen-2-ylmorpholin-4-yl]pyridine-2-carbonitrile
—— 5-[(1R,6S)-9-methyl-3,9-diazabicyclo[4.2.1]nonan-3-yl]pyridine-2-carbonitrile —— C14H18N4
5-[(1R,6S)-9-methyl-3,9-diazabicyclo[4.2.1]nonan-3-yl]pyridine-2-carbonitrile
—— 5-[(3R)-3-hydroxy-3-(trifluoromethyl)pyrrolidin-1-yl]pentanenitrile —— C10H15F3N2O
5-[(3R)-3-hydroxy-3-(trifluoromethyl)pyrrolidin-1-yl]pentanenitrile
—— 5-[4-[[3-[(1R)-1-ethoxyethyl]-1,2,4-oxadiazol-5-yl]methyl]piperazin-1-yl]pyridine-2-carbonitrile —— C17H22N6O2
5-[4-[[3-[(1R)-1-ethoxyethyl]-1,2,4-oxadiazol-5-yl]methyl]piperazin-1-yl]pyridine-2-carbonitrile
—— [(5S,7S)-5,7-dimethyl-6,7-dihydro-5H-pyrazolo[1,5-a]pyrimidin-4-yl]-(4-fluoro-2-nitrophenyl)methanone —— C15H15FN4O3
[(5S,7S)-5,7-dimethyl-6,7-dihydro-5H-pyrazolo[1,5-a]pyrimidin-4-yl]-(4-fluoro-2-nitrophenyl)methanone
—— 5-[4-[[3-[(1S)-1-ethoxyethyl]-1,2,4-oxadiazol-5-yl]methyl]piperazin-1-yl]pyridine-2-carbonitrile —— C17H22N6O2
5-[4-[[3-[(1S)-1-ethoxyethyl]-1,2,4-oxadiazol-5-yl]methyl]piperazin-1-yl]pyridine-2-carbonitrile
—— 5,6-dimethyl-N-[(E)-5-methylhexan-2-ylideneamino]thieno[2,3-d]pyrimidin-4-amine —— C15H22N4S
5,6-dimethyl-N-[(E)-5-methylhexan-2-ylideneamino]thieno[2,3-d]pyrimidin-4-amine
—— 5,6-dimethyl-N-[(E)-1-(5-methylfuran-2-yl)ethylideneamino]thieno[2,3-d]pyrimidin-4-amine —— C15H16N4OS
5,6-dimethyl-N-[(E)-1-(5-methylfuran-2-yl)ethylideneamino]thieno[2,3-d]pyrimidin-4-amine
—— 5,6-dimethyl-N-[(E)-1-phenylpropylideneamino]thieno[2,3-d]pyrimidin-4-amine —— C17H18N4S
5,6-dimethyl-N-[(E)-1-phenylpropylideneamino]thieno[2,3-d]pyrimidin-4-amine
—— 5,6-dimethyl-N-[(E)-1-(3-nitrophenyl)ethylideneamino]thieno[2,3-d]pyrimidin-4-amine —— C16H15N5O2S
5,6-dimethyl-N-[(E)-1-(3-nitrophenyl)ethylideneamino]thieno[2,3-d]pyrimidin-4-amine
—— 5,6-dimethyl-N-[(E)-(4-methylsulfanylphenyl)methylideneamino]thieno[2,3-d]pyrimidin-4-amine —— C16H16N4S2
5,6-dimethyl-N-[(E)-(4-methylsulfanylphenyl)methylideneamino]thieno[2,3-d]pyrimidin-4-amine
—— 5,6-dimethyl-N-[(E)-(2,3,4,5,6-pentafluorophenyl)methylideneamino]thieno[2,3-d]pyrimidin-4-amine —— C15H9F5N4S
5,6-dimethyl-N-[(E)-(2,3,4,5,6-pentafluorophenyl)methylideneamino]thieno[2,3-d]pyrimidin-4-amine
—— 5-[[(2S)-2-methyl-4-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]piperazin-1-yl]methyl]-3-phenyl-1,2,4-oxadiazole —— C23H24N6O2
5-[[(2S)-2-methyl-4-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]piperazin-1-yl]methyl]-3-phenyl-1,2,4-oxadiazole
—— 5-[[(2R)-2-methyl-4-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]piperazin-1-yl]methyl]-3-phenyl-1,2,4-oxadiazole —— C23H24N6O2
5-[[(2R)-2-methyl-4-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]piperazin-1-yl]methyl]-3-phenyl-1,2,4-oxadiazole
—— 5-ethyl-N-[(1S)-1-(4-propan-2-yloxyphenyl)ethyl]-1H-pyrazole-3-carboxamide —— C17H23N3O2
5-ethyl-N-[(1S)-1-(4-propan-2-yloxyphenyl)ethyl]-1H-pyrazole-3-carboxamide
—— (5-ethyl-1H-pyrazol-3-yl)-[4-[(S)-hydroxy(phenyl)methyl]piperidin-1-yl]methanone —— C18H23N3O2
(5-ethyl-1H-pyrazol-3-yl)-[4-[(S)-hydroxy(phenyl)methyl]piperidin-1-yl]methanone
—— 5-ethyl-N-[(1S)-1-phenyl-2-pyrrolidin-1-ylethyl]-1H-pyrazole-3-carboxamide —— C18H24N4O
5-ethyl-N-[(1S)-1-phenyl-2-pyrrolidin-1-ylethyl]-1H-pyrazole-3-carboxamide
—— (5-bromo-1H-indol-2-yl)-[(2R)-2-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-3-yl)pyrrolidin-1-yl]methanone —— C20H22BrN5O
(5-bromo-1H-indol-2-yl)-[(2R)-2-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-3-yl)pyrrolidin-1-yl]methanone
—— 5-(methoxymethyl)-N-[3-[(2R)-4-methyl-2-phenylpiperazin-1-yl]propyl]furan-2-carboxamide —— C21H29N3O3
5-(methoxymethyl)-N-[3-[(2R)-4-methyl-2-phenylpiperazin-1-yl]propyl]furan-2-carboxamide
—— 5-ethyl-N-[(1S)-1-(4-methylphenyl)ethyl]-1H-pyrazole-3-carboxamide —— C15H19N3O
5-ethyl-N-[(1S)-1-(4-methylphenyl)ethyl]-1H-pyrazole-3-carboxamide
—— (5-ethyl-1H-pyrazol-3-yl)-[4-[(R)-hydroxy(phenyl)methyl]piperidin-1-yl]methanone —— C18H23N3O2
(5-ethyl-1H-pyrazol-3-yl)-[4-[(R)-hydroxy(phenyl)methyl]piperidin-1-yl]methanone
—— 5-ethyl-N-[(1R)-1-(4-propan-2-yloxyphenyl)ethyl]-1H-pyrazole-3-carboxamide —— C17H23N3O2
5-ethyl-N-[(1R)-1-(4-propan-2-yloxyphenyl)ethyl]-1H-pyrazole-3-carboxamide
—— 5-ethyl-N-[(1R)-1-(furan-2-yl)ethyl]-N-methyl-1H-pyrazole-3-carboxamide —— C13H17N3O2
5-ethyl-N-[(1R)-1-(furan-2-yl)ethyl]-N-methyl-1H-pyrazole-3-carboxamide
—— 5-ethyl-N-[(1S)-1-(furan-2-yl)ethyl]-N-methyl-1H-pyrazole-3-carboxamide —— C13H17N3O2
5-ethyl-N-[(1S)-1-(furan-2-yl)ethyl]-N-methyl-1H-pyrazole-3-carboxamide
—— 5-ethyl-N-[(2R)-1-methoxypropan-2-yl]-1H-pyrazole-3-carboxamide —— C10H17N3O2
5-ethyl-N-[(2R)-1-methoxypropan-2-yl]-1H-pyrazole-3-carboxamide
—— 5-ethyl-N-[(S)-(4-methoxyphenyl)-phenylmethyl]-1H-pyrazole-3-carboxamide —— C20H21N3O2
5-ethyl-N-[(S)-(4-methoxyphenyl)-phenylmethyl]-1H-pyrazole-3-carboxamide
—— 5-ethyl-N-[(S)-(2-methoxyphenyl)-(1-methylimidazol-2-yl)methyl]-1H-pyrazole-3-carboxamide —— C18H21N5O2
5-ethyl-N-[(S)-(2-methoxyphenyl)-(1-methylimidazol-2-yl)methyl]-1H-pyrazole-3-carboxamide
—— 5-ethyl-N-[(4S)-4,5,6,7-tetrahydro-1-benzofuran-4-yl]-1H-pyrazole-3-carboxamide —— C14H17N3O2
5-ethyl-N-[(4S)-4,5,6,7-tetrahydro-1-benzofuran-4-yl]-1H-pyrazole-3-carboxamide
—— (5-ethyl-1H-pyrazol-3-yl)-[(2S)-4-methyl-2-phenylpiperazin-1-yl]methanone —— C17H22N4O
(5-ethyl-1H-pyrazol-3-yl)-[(2S)-4-methyl-2-phenylpiperazin-1-yl]methanone
—— (5-ethyl-1H-pyrazol-3-yl)-[(2R)-4-methyl-2-phenylpiperazin-1-yl]methanone —— C17H22N4O
(5-ethyl-1H-pyrazol-3-yl)-[(2R)-4-methyl-2-phenylpiperazin-1-yl]methanone
—— 5-ethyl-N-[(1S)-3-methylsulfanyl-1-([1,2,4]triazolo[4,3-a]pyridin-3-yl)propyl]-1H-pyrazole-3-carboxamide —— C16H20N6OS
5-ethyl-N-[(1S)-3-methylsulfanyl-1-([1,2,4]triazolo[4,3-a]pyridin-3-yl)propyl]-1H-pyrazole-3-carboxamide
—— 5-ethyl-N-[(4R)-4,5,6,7-tetrahydro-1-benzofuran-4-yl]-1H-pyrazole-3-carboxamide —— C14H17N3O2
5-ethyl-N-[(4R)-4,5,6,7-tetrahydro-1-benzofuran-4-yl]-1H-pyrazole-3-carboxamide