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—— (5-methylthiophen-2-yl)-[(3S)-3-(3-propylimidazo[4,5-b]pyridin-2-yl)pyrrolidin-1-yl]methanone —— C19H22N4OS
(5-methylthiophen-2-yl)-[(3S)-3-(3-propylimidazo[4,5-b]pyridin-2-yl)pyrrolidin-1-yl]methanone
—— (5aS)-5-methyl-N-[(4-methylphenyl)methyl]-11-oxo-6,7,8,9-tetrahydro-5aH-pyrido[2,1-b]quinazoline-3-carboxamide —— C22H25N3O2
(5aS)-5-methyl-N-[(4-methylphenyl)methyl]-11-oxo-6,7,8,9-tetrahydro-5aH-pyrido[2,1-b]quinazoline-3-carboxamide
—— (5aS)-5-ethyl-11-oxo-N-(pyridin-4-ylmethyl)-6,7,8,9-tetrahydro-5aH-pyrido[2,1-b]quinazoline-3-carboxamide —— C21H24N4O2
(5aS)-5-ethyl-11-oxo-N-(pyridin-4-ylmethyl)-6,7,8,9-tetrahydro-5aH-pyrido[2,1-b]quinazoline-3-carboxamide
—— 5-[[(2S)-4-methyl-2-propan-2-ylpiperazin-1-yl]methyl]furan-2-carbonitrile —— C14H21N3O
5-[[(2S)-4-methyl-2-propan-2-ylpiperazin-1-yl]methyl]furan-2-carbonitrile
—— 5-{N'-[(E)-(3-bromophenyl)methylidene]hydrazinecarbonyl}-N-(prop-2-en-1-yl)pentanamide —— C16H20BrN3O2
5-{N'-[(E)-(3-bromophenyl)methylidene]hydrazinecarbonyl}-N-(prop-2-en-1-yl)pentanamide
—— (5R)-3-[(4-chlorophenyl)methyl]-9-(3,5-dimethylbenzoyl)-1,3,9-triazaspiro[4.5]decane-2,4-dione —— C23H24ClN3O3
(5R)-3-[(4-chlorophenyl)methyl]-9-(3,5-dimethylbenzoyl)-1,3,9-triazaspiro[4.5]decane-2,4-dione
—— (5aR)-5-ethyl-11-oxo-N-(pyridin-4-ylmethyl)-6,7,8,9-tetrahydro-5aH-pyrido[2,1-b]quinazoline-3-carboxamide —— C21H24N4O2
(5aR)-5-ethyl-11-oxo-N-(pyridin-4-ylmethyl)-6,7,8,9-tetrahydro-5aH-pyrido[2,1-b]quinazoline-3-carboxamide
—— (5aS)-3-[4-(4-methoxyphenyl)piperazine-1-carbonyl]-5-methyl-6,7,8,9-tetrahydro-5aH-pyrido[2,1-b]quinazolin-11-one —— C25H30N4O3
(5aS)-3-[4-(4-methoxyphenyl)piperazine-1-carbonyl]-5-methyl-6,7,8,9-tetrahydro-5aH-pyrido[2,1-b]quinazolin-11-one
—— (5aS)-3-[4-(2-fluorophenyl)piperazine-1-carbonyl]-5-methyl-6,7,8,9-tetrahydro-5aH-pyrido[2,1-b]quinazolin-11-one —— C24H27FN4O2
(5aS)-3-[4-(2-fluorophenyl)piperazine-1-carbonyl]-5-methyl-6,7,8,9-tetrahydro-5aH-pyrido[2,1-b]quinazolin-11-one
—— (5-methylthiophen-2-yl)-[(3R)-3-(3-propylimidazo[4,5-b]pyridin-2-yl)pyrrolidin-1-yl]methanone —— C19H22N4OS
(5-methylthiophen-2-yl)-[(3R)-3-(3-propylimidazo[4,5-b]pyridin-2-yl)pyrrolidin-1-yl]methanone
—— 5-[[(2R)-4-methyl-2-propan-2-ylpiperazin-1-yl]methyl]thiophene-3-carbonitrile —— C14H21N3S
5-[[(2R)-4-methyl-2-propan-2-ylpiperazin-1-yl]methyl]thiophene-3-carbonitrile
—— (5aS)-N-(3,4-dimethoxyphenyl)-5-methyl-11-oxo-6,7,8,9-tetrahydro-5aH-pyrido[2,1-b]quinazoline-3-carboxamide —— C22H25N3O4
(5aS)-N-(3,4-dimethoxyphenyl)-5-methyl-11-oxo-6,7,8,9-tetrahydro-5aH-pyrido[2,1-b]quinazoline-3-carboxamide
—— (5aR)-5-methyl-N-[(4-methylphenyl)methyl]-11-oxo-6,7,8,9-tetrahydro-5aH-pyrido[2,1-b]quinazoline-3-carboxamide —— C22H25N3O2
(5aR)-5-methyl-N-[(4-methylphenyl)methyl]-11-oxo-6,7,8,9-tetrahydro-5aH-pyrido[2,1-b]quinazoline-3-carboxamide
—— 5-[[(2R)-4-methyl-2-propan-2-ylpiperazin-1-yl]methyl]furan-2-carbonitrile —— C14H21N3O
5-[[(2R)-4-methyl-2-propan-2-ylpiperazin-1-yl]methyl]furan-2-carbonitrile
—— (5-methylthiophen-2-yl)-[4-[(6R)-6-phenyl-6,7-dihydro-4H-triazolo[5,1-c][1,4]oxazine-3-carbonyl]piperazin-1-yl]methanone —— C22H23N5O3S
(5-methylthiophen-2-yl)-[4-[(6R)-6-phenyl-6,7-dihydro-4H-triazolo[5,1-c][1,4]oxazine-3-carbonyl]piperazin-1-yl]methanone
—— 5-[[(2S)-2-(2-methylphenyl)-3-oxopiperazin-1-yl]methyl]thiophene-3-carboxamide —— C17H19N3O2S
5-[[(2S)-2-(2-methylphenyl)-3-oxopiperazin-1-yl]methyl]thiophene-3-carboxamide
—— (5aS)-N-[(2,4-dimethoxyphenyl)methyl]-5-methyl-11-oxo-6,7,8,9-tetrahydro-5aH-pyrido[2,1-b]quinazoline-3-carboxamide —— C23H27N3O4
(5aS)-N-[(2,4-dimethoxyphenyl)methyl]-5-methyl-11-oxo-6,7,8,9-tetrahydro-5aH-pyrido[2,1-b]quinazoline-3-carboxamide
—— 5-[(2E)-2-[(3-bromophenyl)methylidene]hydrazinyl]-2-chlorobenzoic acid —— C14H10BrClN2O2
5-[(2E)-2-[(3-bromophenyl)methylidene]hydrazinyl]-2-chlorobenzoic acid
—— (5aR)-3-[4-(4-methoxyphenyl)piperazine-1-carbonyl]-5-methyl-6,7,8,9-tetrahydro-5aH-pyrido[2,1-b]quinazolin-11-one —— C25H30N4O3
(5aR)-3-[4-(4-methoxyphenyl)piperazine-1-carbonyl]-5-methyl-6,7,8,9-tetrahydro-5aH-pyrido[2,1-b]quinazolin-11-one
—— 5-chloro-N-{4-[N-(4-fluorobenzoyl)ethanehydrazonoyl]phenyl}-2-thiophenecarboxamide —— C20H15ClFN3O2S
5-chloro-N-{4-[N-(4-fluorobenzoyl)ethanehydrazonoyl]phenyl}-2-thiophenecarboxamide
—— (5-methylthiophen-2-yl)-[4-[(6S)-6-phenyl-6,7-dihydro-4H-triazolo[5,1-c][1,4]oxazine-3-carbonyl]piperazin-1-yl]methanone —— C22H23N5O3S
(5-methylthiophen-2-yl)-[4-[(6S)-6-phenyl-6,7-dihydro-4H-triazolo[5,1-c][1,4]oxazine-3-carbonyl]piperazin-1-yl]methanone
—— (5aR)-N-(4-bromo-3-methylphenyl)-5-ethyl-11-oxo-6,7,8,9-tetrahydro-5aH-pyrido[2,1-b]quinazoline-3-carboxamide —— C22H24BrN3O2
(5aR)-N-(4-bromo-3-methylphenyl)-5-ethyl-11-oxo-6,7,8,9-tetrahydro-5aH-pyrido[2,1-b]quinazoline-3-carboxamide
—— 5-[(2E)-2-[1-(5-bromothiophen-2-yl)ethylidene]hydrazinyl]-2-chlorobenzoic acid —— C13H10BrClN2O2S
5-[(2E)-2-[1-(5-bromothiophen-2-yl)ethylidene]hydrazinyl]-2-chlorobenzoic acid
—— (5aR)-N-(3,4-dimethoxyphenyl)-5-methyl-11-oxo-6,7,8,9-tetrahydro-5aH-pyrido[2,1-b]quinazoline-3-carboxamide —— C22H25N3O4
(5aR)-N-(3,4-dimethoxyphenyl)-5-methyl-11-oxo-6,7,8,9-tetrahydro-5aH-pyrido[2,1-b]quinazoline-3-carboxamide
—— (5aS)-N-(4-bromo-3-methylphenyl)-5-ethyl-11-oxo-6,7,8,9-tetrahydro-5aH-pyrido[2,1-b]quinazoline-3-carboxamide —— C22H24BrN3O2
(5aS)-N-(4-bromo-3-methylphenyl)-5-ethyl-11-oxo-6,7,8,9-tetrahydro-5aH-pyrido[2,1-b]quinazoline-3-carboxamide
—— (5aS)-N-[(3-chloro-4-fluorophenyl)methyl]-5-methyl-11-oxo-6,7,8,9-tetrahydro-5aH-pyrido[2,1-b]quinazoline-3-carboxamide —— C21H21ClFN3O2
(5aS)-N-[(3-chloro-4-fluorophenyl)methyl]-5-methyl-11-oxo-6,7,8,9-tetrahydro-5aH-pyrido[2,1-b]quinazoline-3-carboxamide
—— 5-[(2E)-2-[(3,4-diethoxyphenyl)methylidene]hydrazinyl]-2-methyl-1,3-oxazole-4-carbonitrile —— C16H18N4O3
5-[(2E)-2-[(3,4-diethoxyphenyl)methylidene]hydrazinyl]-2-methyl-1,3-oxazole-4-carbonitrile
—— (5aR)-N-[(3-chloro-4-fluorophenyl)methyl]-5-methyl-11-oxo-6,7,8,9-tetrahydro-5aH-pyrido[2,1-b]quinazoline-3-carboxamide —— C21H21ClFN3O2
(5aR)-N-[(3-chloro-4-fluorophenyl)methyl]-5-methyl-11-oxo-6,7,8,9-tetrahydro-5aH-pyrido[2,1-b]quinazoline-3-carboxamide
—— 5-[(2E)-2-[[3-(3-chloro-4-methoxyphenyl)-1-phenylpyrazol-4-yl]methylidene]hydrazinyl]-2-methyl-1,3-oxazole-4-carbonitrile —— C22H17ClN6O2
5-[(2E)-2-[[3-(3-chloro-4-methoxyphenyl)-1-phenylpyrazol-4-yl]methylidene]hydrazinyl]-2-methyl-1,3-oxazole-4-carbonitrile
—— (5aS)-N-(3,5-dimethylphenyl)-5-ethyl-11-oxo-6,7,8,9-tetrahydro-5aH-pyrido[2,1-b]quinazoline-3-carboxamide —— C23H27N3O2
(5aS)-N-(3,5-dimethylphenyl)-5-ethyl-11-oxo-6,7,8,9-tetrahydro-5aH-pyrido[2,1-b]quinazoline-3-carboxamide
—— (5aR)-N-(3,5-dimethylphenyl)-5-ethyl-11-oxo-6,7,8,9-tetrahydro-5aH-pyrido[2,1-b]quinazoline-3-carboxamide —— C23H27N3O2
(5aR)-N-(3,5-dimethylphenyl)-5-ethyl-11-oxo-6,7,8,9-tetrahydro-5aH-pyrido[2,1-b]quinazoline-3-carboxamide
—— 5-[[2,5-dimethyl-3-[[(3S)-3-methylpiperidin-1-yl]methyl]phenyl]methyl]-3,4,6,7-tetrahydroimidazo[4,5-c]pyridine —— C22H32N4
5-[[2,5-dimethyl-3-[[(3S)-3-methylpiperidin-1-yl]methyl]phenyl]methyl]-3,4,6,7-tetrahydroimidazo[4,5-c]pyridine
—— 5-[(2E)-2-[(4-hexoxyphenyl)methylidene]hydrazinyl]-2-propan-2-yl-1,3-oxazole-4-carbonitrile —— C20H26N4O2
5-[(2E)-2-[(4-hexoxyphenyl)methylidene]hydrazinyl]-2-propan-2-yl-1,3-oxazole-4-carbonitrile
—— 5-[(2E)-2-[[3-(3-bromo-4-methoxyphenyl)-1-phenylpyrazol-4-yl]methylidene]hydrazinyl]-2-propan-2-yl-1,3-oxazole-4-carbonitrile —— C24H21BrN6O2
5-[(2E)-2-[[3-(3-bromo-4-methoxyphenyl)-1-phenylpyrazol-4-yl]methylidene]hydrazinyl]-2-propan-2-yl-1,3-oxazole-4-carbonitrile
—— 5-[(2E)-2-[[4-(3-methylbutoxy)phenyl]methylidene]hydrazinyl]-2-propan-2-yl-1,3-oxazole-4-carbonitrile —— C19H24N4O2
5-[(2E)-2-[[4-(3-methylbutoxy)phenyl]methylidene]hydrazinyl]-2-propan-2-yl-1,3-oxazole-4-carbonitrile
—— 5-[(2E)-2-[(2-methyl-2H-chromen-3-yl)methylidene]hydrazinyl]-2-propan-2-yl-1,3-oxazole-4-carbonitrile —— C18H18N4O2
5-[(2E)-2-[(2-methyl-2H-chromen-3-yl)methylidene]hydrazinyl]-2-propan-2-yl-1,3-oxazole-4-carbonitrile
—— (5S)-3-methyl-2-oxo-N-(2-phenylpyrazol-3-yl)-1-oxa-3,9-diazaspiro[4.6]undecane-9-carboxamide —— C19H23N5O3
(5S)-3-methyl-2-oxo-N-(2-phenylpyrazol-3-yl)-1-oxa-3,9-diazaspiro[4.6]undecane-9-carboxamide
—— 5-[(2E)-2-[(3,4-diethoxyphenyl)methylidene]hydrazinyl]-2-propan-2-yl-1,3-oxazole-4-carbonitrile —— C18H22N4O3
5-[(2E)-2-[(3,4-diethoxyphenyl)methylidene]hydrazinyl]-2-propan-2-yl-1,3-oxazole-4-carbonitrile
—— 5-[[2,5-dimethyl-3-[[(3R)-3-methylpiperidin-1-yl]methyl]phenyl]methyl]-3,4,6,7-tetrahydroimidazo[4,5-c]pyridine —— C22H32N4
5-[[2,5-dimethyl-3-[[(3R)-3-methylpiperidin-1-yl]methyl]phenyl]methyl]-3,4,6,7-tetrahydroimidazo[4,5-c]pyridine
—— 5-[(2E)-2-[(3-ethoxy-4-propoxyphenyl)methylidene]hydrazinyl]-2-propan-2-yl-1,3-oxazole-4-carbonitrile —— C19H24N4O3
5-[(2E)-2-[(3-ethoxy-4-propoxyphenyl)methylidene]hydrazinyl]-2-propan-2-yl-1,3-oxazole-4-carbonitrile
—— 5-[(2E)-2-[[3-(4-morpholin-4-ylsulfonylphenyl)-1-phenylpyrazol-4-yl]methylidene]hydrazinyl]-2-propan-2-yl-1,3-oxazole-4-carbonitrile —— C27H27N7O4S
5-[(2E)-2-[[3-(4-morpholin-4-ylsulfonylphenyl)-1-phenylpyrazol-4-yl]methylidene]hydrazinyl]-2-propan-2-yl-1,3-oxazole-4-carbonitrile
—— 5-[(2E)-2-[(4-ethylphenyl)methylidene]hydrazinyl]-2-propan-2-yl-1,3-oxazole-4-carbonitrile —— C16H18N4O
5-[(2E)-2-[(4-ethylphenyl)methylidene]hydrazinyl]-2-propan-2-yl-1,3-oxazole-4-carbonitrile
—— 5-pyridin-2-yl-N-[(1S)-1-[4-(triazol-1-yl)phenyl]ethyl]-1,3,4-thiadiazol-2-amine —— C17H15N7S
5-pyridin-2-yl-N-[(1S)-1-[4-(triazol-1-yl)phenyl]ethyl]-1,3,4-thiadiazol-2-amine
—— (5R)-3-methyl-2-oxo-N-(2-phenylpyrazol-3-yl)-1-oxa-3,9-diazaspiro[4.6]undecane-9-carboxamide —— C19H23N5O3
(5R)-3-methyl-2-oxo-N-(2-phenylpyrazol-3-yl)-1-oxa-3,9-diazaspiro[4.6]undecane-9-carboxamide
—— 5-pyridin-2-yl-N-[(1R)-1-[4-(triazol-1-yl)phenyl]ethyl]-1,3,4-thiadiazol-2-amine —— C17H15N7S
5-pyridin-2-yl-N-[(1R)-1-[4-(triazol-1-yl)phenyl]ethyl]-1,3,4-thiadiazol-2-amine
—— 5-{(2E)-2-[(6-chloro-4-oxo-4H-chromen-3-yl)methylidene]hydrazinyl}-2-(propan-2-yl)-1,3-oxazole-4-carbonitrile —— C17H13ClN4O3
5-{(2E)-2-[(6-chloro-4-oxo-4H-chromen-3-yl)methylidene]hydrazinyl}-2-(propan-2-yl)-1,3-oxazole-4-carbonitrile
—— 5-(2-chlorophenyl)-N-[[(2R)-1,1-dioxothiolan-2-yl]methyl]-1,3,4-thiadiazol-2-amine —— C13H14ClN3O2S2
5-(2-chlorophenyl)-N-[[(2R)-1,1-dioxothiolan-2-yl]methyl]-1,3,4-thiadiazol-2-amine
—— 5-(2-chlorophenyl)-N-[[(2S)-1,1-dioxothiolan-2-yl]methyl]-1,3,4-thiadiazol-2-amine —— C13H14ClN3O2S2
5-(2-chlorophenyl)-N-[[(2S)-1,1-dioxothiolan-2-yl]methyl]-1,3,4-thiadiazol-2-amine
—— 5-(2-chlorophenyl)-N-[(2R)-4-methylsulfonylbutan-2-yl]-1,3,4-thiadiazol-2-amine —— C13H16ClN3O2S2
5-(2-chlorophenyl)-N-[(2R)-4-methylsulfonylbutan-2-yl]-1,3,4-thiadiazol-2-amine
—— 5-[(2E)-2-[(4-hexoxyphenyl)methylidene]hydrazinyl]-2-methyl-1,3-oxazole-4-carbonitrile —— C18H22N4O2
5-[(2E)-2-[(4-hexoxyphenyl)methylidene]hydrazinyl]-2-methyl-1,3-oxazole-4-carbonitrile