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—— (5aR)-3-[4-(2-ethoxyphenyl)piperazine-1-carbonyl]-5-methyl-6,7,8,9-tetrahydro-5aH-pyrido[2,1-b]quinazolin-11-one —— C26H32N4O3
(5aR)-3-[4-(2-ethoxyphenyl)piperazine-1-carbonyl]-5-methyl-6,7,8,9-tetrahydro-5aH-pyrido[2,1-b]quinazolin-11-one
—— (5aS)-3-[4-(2-ethoxyphenyl)piperazine-1-carbonyl]-5-methyl-6,7,8,9-tetrahydro-5aH-pyrido[2,1-b]quinazolin-11-one —— C26H32N4O3
(5aS)-3-[4-(2-ethoxyphenyl)piperazine-1-carbonyl]-5-methyl-6,7,8,9-tetrahydro-5aH-pyrido[2,1-b]quinazolin-11-one
—— (5aS)-N-(3-cyanophenyl)-5-ethyl-11-oxo-6,7,8,9-tetrahydro-5aH-pyrido[2,1-b]quinazoline-3-carboxamide —— C22H22N4O2
(5aS)-N-(3-cyanophenyl)-5-ethyl-11-oxo-6,7,8,9-tetrahydro-5aH-pyrido[2,1-b]quinazoline-3-carboxamide
—— (5aR)-5-ethyl-N-[(3-methylphenyl)methyl]-11-oxo-6,7,8,9-tetrahydro-5aH-pyrido[2,1-b]quinazoline-3-carboxamide —— C23H27N3O2
(5aR)-5-ethyl-N-[(3-methylphenyl)methyl]-11-oxo-6,7,8,9-tetrahydro-5aH-pyrido[2,1-b]quinazoline-3-carboxamide
—— 5(4-Meo-PH)-2-PH-2H-pyrazole-3-carboxylic acid (1-(4-CL-PH)-ethylidene)hydrazide —— C25H21ClN4O2
5(4-Meo-PH)-2-PH-2H-pyrazole-3-carboxylic acid (1-(4-CL-PH)-ethylidene)hydrazide
—— (5aR)-N-(4-chlorophenyl)-5-ethyl-11-oxo-6,7,8,9-tetrahydro-5aH-pyrido[2,1-b]quinazoline-3-carboxamide —— C21H22ClN3O2
(5aR)-N-(4-chlorophenyl)-5-ethyl-11-oxo-6,7,8,9-tetrahydro-5aH-pyrido[2,1-b]quinazoline-3-carboxamide
—— 5-[(4-Chlorobenzoyl)oxy]-2-((E)-{[(4-ethylanilino)(oxo)acetyl]hydrazono}methyl)phenyl 4-chlorobenzoate —— C31H23Cl2N3O6
5-[(4-Chlorobenzoyl)oxy]-2-((E)-{[(4-ethylanilino)(oxo)acetyl]hydrazono}methyl)phenyl 4-chlorobenzoate
—— (5aR)-5-ethyl-11-oxo-N-[4-(trifluoromethoxy)phenyl]-6,7,8,9-tetrahydro-5aH-pyrido[2,1-b]quinazoline-3-carboxamide —— C22H22F3N3O3
(5aR)-5-ethyl-11-oxo-N-[4-(trifluoromethoxy)phenyl]-6,7,8,9-tetrahydro-5aH-pyrido[2,1-b]quinazoline-3-carboxamide
—— (5aR)-5-methyl-N-[(2-methylphenyl)methyl]-11-oxo-6,7,8,9-tetrahydro-5aH-pyrido[2,1-b]quinazoline-3-carboxamide —— C22H25N3O2
(5aR)-5-methyl-N-[(2-methylphenyl)methyl]-11-oxo-6,7,8,9-tetrahydro-5aH-pyrido[2,1-b]quinazoline-3-carboxamide
—— (5-chlorothiophen-2-yl)-[(3S)-3-[2-(4-methoxyphenyl)imidazo[4,5-b]pyridin-3-yl]pyrrolidin-1-yl]methanone —— C22H19ClN4O2S
(5-chlorothiophen-2-yl)-[(3S)-3-[2-(4-methoxyphenyl)imidazo[4,5-b]pyridin-3-yl]pyrrolidin-1-yl]methanone
—— (5-chlorothiophen-2-yl)-[(3R)-3-[2-(4-methoxyphenyl)imidazo[4,5-b]pyridin-3-yl]pyrrolidin-1-yl]methanone —— C22H19ClN4O2S
(5-chlorothiophen-2-yl)-[(3R)-3-[2-(4-methoxyphenyl)imidazo[4,5-b]pyridin-3-yl]pyrrolidin-1-yl]methanone
—— (5aR)-N-(3,5-dimethoxyphenyl)-5-ethyl-11-oxo-6,7,8,9-tetrahydro-5aH-pyrido[2,1-b]quinazoline-3-carboxamide —— C23H27N3O4
(5aR)-N-(3,5-dimethoxyphenyl)-5-ethyl-11-oxo-6,7,8,9-tetrahydro-5aH-pyrido[2,1-b]quinazoline-3-carboxamide
—— (5aS)-5-methyl-N-[(2-methylphenyl)methyl]-11-oxo-6,7,8,9-tetrahydro-5aH-pyrido[2,1-b]quinazoline-3-carboxamide —— C22H25N3O2
(5aS)-5-methyl-N-[(2-methylphenyl)methyl]-11-oxo-6,7,8,9-tetrahydro-5aH-pyrido[2,1-b]quinazoline-3-carboxamide
—— (5aS)-N-[(3-fluorophenyl)methyl]-5-methyl-11-oxo-6,7,8,9-tetrahydro-5aH-pyrido[2,1-b]quinazoline-3-carboxamide —— C21H22FN3O2
(5aS)-N-[(3-fluorophenyl)methyl]-5-methyl-11-oxo-6,7,8,9-tetrahydro-5aH-pyrido[2,1-b]quinazoline-3-carboxamide
—— (5aR)-5-ethyl-11-oxo-N-(4-propan-2-ylphenyl)-6,7,8,9-tetrahydro-5aH-pyrido[2,1-b]quinazoline-3-carboxamide —— C24H29N3O2
(5aR)-5-ethyl-11-oxo-N-(4-propan-2-ylphenyl)-6,7,8,9-tetrahydro-5aH-pyrido[2,1-b]quinazoline-3-carboxamide
—— (5aR)-N-[(2-chloro-4-fluorophenyl)methyl]-5-ethyl-11-oxo-6,7,8,9-tetrahydro-5aH-pyrido[2,1-b]quinazoline-3-carboxamide —— C22H23ClFN3O2
(5aR)-N-[(2-chloro-4-fluorophenyl)methyl]-5-ethyl-11-oxo-6,7,8,9-tetrahydro-5aH-pyrido[2,1-b]quinazoline-3-carboxamide
—— (5aR)-N-[(3-fluorophenyl)methyl]-5-methyl-11-oxo-6,7,8,9-tetrahydro-5aH-pyrido[2,1-b]quinazoline-3-carboxamide —— C21H22FN3O2
(5aR)-N-[(3-fluorophenyl)methyl]-5-methyl-11-oxo-6,7,8,9-tetrahydro-5aH-pyrido[2,1-b]quinazoline-3-carboxamide
—— (5aR)-N-(3-cyanophenyl)-5-ethyl-11-oxo-6,7,8,9-tetrahydro-5aH-pyrido[2,1-b]quinazoline-3-carboxamide —— C22H22N4O2
(5aR)-N-(3-cyanophenyl)-5-ethyl-11-oxo-6,7,8,9-tetrahydro-5aH-pyrido[2,1-b]quinazoline-3-carboxamide
—— (5E)-5-[(2,5-dichloro-3-phenylimidazol-4-yl)methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one —— C13H7Cl2N3OS2
(5E)-5-[(2,5-dichloro-3-phenylimidazol-4-yl)methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one
—— 5-methyl-4-nitro-N-[(1S)-1-pyridin-3-ylethyl]thiophene-2-sulfonamide —— C12H13N3O4S2
5-methyl-4-nitro-N-[(1S)-1-pyridin-3-ylethyl]thiophene-2-sulfonamide
—— (5aR)-N-(3-fluorophenyl)-5-methyl-11-oxo-6,7,8,9-tetrahydro-5aH-pyrido[2,1-b]quinazoline-3-carboxamide —— C20H20FN3O2
(5aR)-N-(3-fluorophenyl)-5-methyl-11-oxo-6,7,8,9-tetrahydro-5aH-pyrido[2,1-b]quinazoline-3-carboxamide
—— 5-chloro-2-hydroxy-N-[(E)-[5-(2-methyl-3-nitrophenyl)furan-2-yl]methylideneamino]benzamide —— C19H14ClN3O5
5-chloro-2-hydroxy-N-[(E)-[5-(2-methyl-3-nitrophenyl)furan-2-yl]methylideneamino]benzamide
—— (5aS)-N-(3-fluorophenyl)-5-methyl-11-oxo-6,7,8,9-tetrahydro-5aH-pyrido[2,1-b]quinazoline-3-carboxamide —— C20H20FN3O2
(5aS)-N-(3-fluorophenyl)-5-methyl-11-oxo-6,7,8,9-tetrahydro-5aH-pyrido[2,1-b]quinazoline-3-carboxamide
—— 5-bromo-N'-[(E)-{3-ethoxy-4-[2-(morpholin-4-yl)ethoxy]phenyl}methylidene]furan-2-carbohydrazide —— C20H24BrN3O5
5-bromo-N'-[(E)-{3-ethoxy-4-[2-(morpholin-4-yl)ethoxy]phenyl}methylidene]furan-2-carbohydrazide
—— (5aS)-5-ethyl-11-oxo-N-(4-propan-2-ylphenyl)-6,7,8,9-tetrahydro-5aH-pyrido[2,1-b]quinazoline-3-carboxamide —— C24H29N3O2
(5aS)-5-ethyl-11-oxo-N-(4-propan-2-ylphenyl)-6,7,8,9-tetrahydro-5aH-pyrido[2,1-b]quinazoline-3-carboxamide
—— (5aS)-N-(3,5-dimethoxyphenyl)-5-ethyl-11-oxo-6,7,8,9-tetrahydro-5aH-pyrido[2,1-b]quinazoline-3-carboxamide —— C23H27N3O4
(5aS)-N-(3,5-dimethoxyphenyl)-5-ethyl-11-oxo-6,7,8,9-tetrahydro-5aH-pyrido[2,1-b]quinazoline-3-carboxamide
—— 5-(methoxymethyl)-N-[(1R)-1-(2-methoxyphenyl)ethyl]-N-methylfuran-2-carboxamide —— C17H21NO4
5-(methoxymethyl)-N-[(1R)-1-(2-methoxyphenyl)ethyl]-N-methylfuran-2-carboxamide
—— 5-(methoxymethyl)-N-[(1S)-1-(2-methoxyphenyl)ethyl]-N-methylfuran-2-carboxamide —— C17H21NO4
5-(methoxymethyl)-N-[(1S)-1-(2-methoxyphenyl)ethyl]-N-methylfuran-2-carboxamide
—— 5-methyl-1-(3-nitrophenyl)-N-[(1R)-1-(4-propan-2-yloxyphenyl)ethyl]triazole-4-carboxamide —— C21H23N5O4
5-methyl-1-(3-nitrophenyl)-N-[(1R)-1-(4-propan-2-yloxyphenyl)ethyl]triazole-4-carboxamide
—— 5-bromo-N-[3-(dimethylamino)propyl]-N-[(3S)-1,1-dioxothiolan-3-yl]furan-3-carboxamide —— C14H21BrN2O4S
5-bromo-N-[3-(dimethylamino)propyl]-N-[(3S)-1,1-dioxothiolan-3-yl]furan-3-carboxamide
—— 5-(methoxymethyl)-N-[(1R)-1-(4-propan-2-yloxyphenyl)ethyl]furan-2-carboxamide —— C18H23NO4
5-(methoxymethyl)-N-[(1R)-1-(4-propan-2-yloxyphenyl)ethyl]furan-2-carboxamide
—— 5-methyl-1-(3-nitrophenyl)-N-[(1S)-1-(4-propan-2-yloxyphenyl)ethyl]triazole-4-carboxamide —— C21H23N5O4
5-methyl-1-(3-nitrophenyl)-N-[(1S)-1-(4-propan-2-yloxyphenyl)ethyl]triazole-4-carboxamide
—— 5-[4-[(1S)-1-(2-chlorophenyl)ethyl]piperazine-1-carbonyl]-2,3-dimethylbenzenesulfonamide —— C21H26ClN3O3S
5-[4-[(1S)-1-(2-chlorophenyl)ethyl]piperazine-1-carbonyl]-2,3-dimethylbenzenesulfonamide
—— 5-(methoxymethyl)-N-[(1S)-1-(4-methylphenyl)ethyl]furan-2-carboxamide —— C16H19NO3
5-(methoxymethyl)-N-[(1S)-1-(4-methylphenyl)ethyl]furan-2-carboxamide
—— 5-[(3aR,4R,6aS)-2-oxo-1,3,3a,4,6,6a-hexahydrothieno[3,4-d]imidazol-4-yl]-N-[4-(2-oxopyrrolidin-1-yl)phenyl]pentanamide —— C20H26N4O3S
5-[(3aR,4R,6aS)-2-oxo-1,3,3a,4,6,6a-hexahydrothieno[3,4-d]imidazol-4-yl]-N-[4-(2-oxopyrrolidin-1-yl)phenyl]pentanamide
—— 5-[(3aS,4S,6aS)-2-oxo-1,3,3a,4,6,6a-hexahydrothieno[3,4-d]imidazol-4-yl]-N-[(2-bromo-5-fluorophenyl)methyl]pentanamide —— C17H21BrFN3O2S
5-[(3aS,4S,6aS)-2-oxo-1,3,3a,4,6,6a-hexahydrothieno[3,4-d]imidazol-4-yl]-N-[(2-bromo-5-fluorophenyl)methyl]pentanamide
—— 5-[(3aR,4R,6aS)-2-oxo-1,3,3a,4,6,6a-hexahydrothieno[3,4-d]imidazol-4-yl]-N-[(2-bromo-5-fluorophenyl)methyl]pentanamide —— C17H21BrFN3O2S
5-[(3aR,4R,6aS)-2-oxo-1,3,3a,4,6,6a-hexahydrothieno[3,4-d]imidazol-4-yl]-N-[(2-bromo-5-fluorophenyl)methyl]pentanamide
—— 5-bromo-N-[3-(dimethylamino)propyl]-N-[(3R)-1,1-dioxothiolan-3-yl]furan-3-carboxamide —— C14H21BrN2O4S
5-bromo-N-[3-(dimethylamino)propyl]-N-[(3R)-1,1-dioxothiolan-3-yl]furan-3-carboxamide
—— 5-[(3aR,4S,6aS)-2-oxo-1,3,3a,4,6,6a-hexahydrothieno[3,4-d]imidazol-4-yl]-N-[(2-bromo-5-fluorophenyl)methyl]pentanamide —— C17H21BrFN3O2S
5-[(3aR,4S,6aS)-2-oxo-1,3,3a,4,6,6a-hexahydrothieno[3,4-d]imidazol-4-yl]-N-[(2-bromo-5-fluorophenyl)methyl]pentanamide
—— 5-[(3aR,4S,6aS)-2-oxo-1,3,3a,4,6,6a-hexahydrothieno[3,4-d]imidazol-4-yl]-N-[4-(2-oxopyrrolidin-1-yl)phenyl]pentanamide —— C20H26N4O3S
5-[(3aR,4S,6aS)-2-oxo-1,3,3a,4,6,6a-hexahydrothieno[3,4-d]imidazol-4-yl]-N-[4-(2-oxopyrrolidin-1-yl)phenyl]pentanamide
—— 5-[(3aS,4R,6aS)-2-oxo-1,3,3a,4,6,6a-hexahydrothieno[3,4-d]imidazol-4-yl]-N-[4-(2-oxopyrrolidin-1-yl)phenyl]pentanamide —— C20H26N4O3S
5-[(3aS,4R,6aS)-2-oxo-1,3,3a,4,6,6a-hexahydrothieno[3,4-d]imidazol-4-yl]-N-[4-(2-oxopyrrolidin-1-yl)phenyl]pentanamide
—— 5-[4-[(1R)-1-(2-chlorophenyl)ethyl]piperazine-1-carbonyl]-2,3-dimethylbenzenesulfonamide —— C21H26ClN3O3S
5-[4-[(1R)-1-(2-chlorophenyl)ethyl]piperazine-1-carbonyl]-2,3-dimethylbenzenesulfonamide
—— 5-[(3S)-1-(cyclopentylmethyl)piperidin-3-yl]-3-methyl-1,2,4-oxadiazole —— C14H23N3O
5-[(3S)-1-(cyclopentylmethyl)piperidin-3-yl]-3-methyl-1,2,4-oxadiazole
—— 5-fluoro-3-methyl-2-[[4-[(3R)-pyrrolidin-3-yl]piperazin-1-yl]methyl]-1H-indole —— C18H25FN4
5-fluoro-3-methyl-2-[[4-[(3R)-pyrrolidin-3-yl]piperazin-1-yl]methyl]-1H-indole
—— [5-(morpholin-4-ylmethyl)furan-3-yl]-[(3R)-3-phenylpiperazin-1-yl]methanone —— C20H25N3O3
[5-(morpholin-4-ylmethyl)furan-3-yl]-[(3R)-3-phenylpiperazin-1-yl]methanone
—— (5S)-5-[4-(4,6-dimethylpyrimidin-2-yl)piperazine-1-carbonyl]-2,2-dimethylthiomorpholin-3-one —— C17H25N5O2S
(5S)-5-[4-(4,6-dimethylpyrimidin-2-yl)piperazine-1-carbonyl]-2,2-dimethylthiomorpholin-3-one
—— (5R)-5-[4-(4,6-dimethylpyrimidin-2-yl)piperazine-1-carbonyl]-2,2-dimethylthiomorpholin-3-one —— C17H25N5O2S
(5R)-5-[4-(4,6-dimethylpyrimidin-2-yl)piperazine-1-carbonyl]-2,2-dimethylthiomorpholin-3-one
—— 5-fluoro-3-methyl-2-[[4-[(3S)-pyrrolidin-3-yl]piperazin-1-yl]methyl]-1H-indole —— C18H25FN4
5-fluoro-3-methyl-2-[[4-[(3S)-pyrrolidin-3-yl]piperazin-1-yl]methyl]-1H-indole
—— [(5S)-9-[(1,3-dimethylpyrazol-4-yl)methyl]-3-(1,3-thiazol-4-ylmethyl)-3,9-diazaspiro[5.5]undecan-5-yl]methanol —— C20H31N5OS
[(5S)-9-[(1,3-dimethylpyrazol-4-yl)methyl]-3-(1,3-thiazol-4-ylmethyl)-3,9-diazaspiro[5.5]undecan-5-yl]methanol
—— 5-ethyl-4-methyl-N-[2-[(3R)-3-(2-methylphenyl)pyrrolidin-1-yl]ethyl]-1H-pyrazole-3-carboxamide —— C20H28N4O
5-ethyl-4-methyl-N-[2-[(3R)-3-(2-methylphenyl)pyrrolidin-1-yl]ethyl]-1H-pyrazole-3-carboxamide