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中文名称 英文名称 CAS号 化学式 结构式图片
—— 5-tert-butyl-N-[(4R)-4,5,6,7-tetrahydro-1-benzofuran-4-yl]-1H-pyrazole-3-carboxamide —— C16H21N3O2
5-tert-butyl-N-[(4R)-4,5,6,7-tetrahydro-1-benzofuran-4-yl]-1H-pyrazole-3-carboxamide
—— 5-tert-butyl-N-[(1R)-1-(2-methoxyphenyl)ethyl]-1H-pyrazole-3-carboxamide —— C17H23N3O2
5-tert-butyl-N-[(1R)-1-(2-methoxyphenyl)ethyl]-1H-pyrazole-3-carboxamide
—— 5-tert-butyl-N-[(4S)-3,4-dihydro-2H-chromen-4-yl]-1H-pyrazole-3-carboxamide —— C17H21N3O2
5-tert-butyl-N-[(4S)-3,4-dihydro-2H-chromen-4-yl]-1H-pyrazole-3-carboxamide
—— 5-(2-methylpropyl)-N-[(4R)-4,5,6,7-tetrahydro-1-benzofuran-4-yl]-1H-pyrazole-3-carboxamide —— C16H21N3O2
5-(2-methylpropyl)-N-[(4R)-4,5,6,7-tetrahydro-1-benzofuran-4-yl]-1H-pyrazole-3-carboxamide
—— 5-tert-butyl-N-[(4S)-4,5,6,7-tetrahydro-1-benzofuran-4-yl]-1H-pyrazole-3-carboxamide —— C16H21N3O2
5-tert-butyl-N-[(4S)-4,5,6,7-tetrahydro-1-benzofuran-4-yl]-1H-pyrazole-3-carboxamide
—— 5-(2-methylpropyl)-N-[(4S)-4,5,6,7-tetrahydro-1-benzofuran-4-yl]-1H-pyrazole-3-carboxamide —— C16H21N3O2
5-(2-methylpropyl)-N-[(4S)-4,5,6,7-tetrahydro-1-benzofuran-4-yl]-1H-pyrazole-3-carboxamide
—— 5-tert-butyl-N-[(1S)-1-(2,4-difluorophenyl)ethyl]-1H-pyrazole-3-carboxamide —— C16H19F2N3O
5-tert-butyl-N-[(1S)-1-(2,4-difluorophenyl)ethyl]-1H-pyrazole-3-carboxamide
—— 5-tert-butyl-N-[(1R)-1-(2,4-difluorophenyl)ethyl]-1H-pyrazole-3-carboxamide —— C16H19F2N3O
5-tert-butyl-N-[(1R)-1-(2,4-difluorophenyl)ethyl]-1H-pyrazole-3-carboxamide
—— 5-[[(3S)-3-methyl-2,3-dihydroindol-1-yl]methyl]-3-phenyl-1,2,4-oxadiazole —— C18H17N3O
5-[[(3S)-3-methyl-2,3-dihydroindol-1-yl]methyl]-3-phenyl-1,2,4-oxadiazole
—— 5-tert-butyl-N-methyl-N-[(1S)-1-thiophen-2-ylethyl]-1H-pyrazole-3-carboxamide —— C15H21N3OS
5-tert-butyl-N-methyl-N-[(1S)-1-thiophen-2-ylethyl]-1H-pyrazole-3-carboxamide
—— 5-tert-butyl-N-[(2R)-2-(dimethylamino)-3-phenylpropyl]-1H-pyrazole-3-carboxamide —— C19H28N4O
5-tert-butyl-N-[(2R)-2-(dimethylamino)-3-phenylpropyl]-1H-pyrazole-3-carboxamide
—— 5-tert-butyl-N-[(1S)-1-(3-fluoro-4-methoxyphenyl)ethyl]-1H-pyrazole-3-carboxamide —— C17H22FN3O2
5-tert-butyl-N-[(1S)-1-(3-fluoro-4-methoxyphenyl)ethyl]-1H-pyrazole-3-carboxamide
—— 5-tert-butyl-N-[(2S)-2-(dimethylamino)-3-phenylpropyl]-1H-pyrazole-3-carboxamide —— C19H28N4O
5-tert-butyl-N-[(2S)-2-(dimethylamino)-3-phenylpropyl]-1H-pyrazole-3-carboxamide
—— 5-[[(3R)-3-methyl-2,3-dihydroindol-1-yl]methyl]-3-phenyl-1,2,4-oxadiazole —— C18H17N3O
5-[[(3R)-3-methyl-2,3-dihydroindol-1-yl]methyl]-3-phenyl-1,2,4-oxadiazole
—— 5-tert-butyl-N-[(1R)-2-(dimethylamino)-1-phenylethyl]-1H-pyrazole-3-carboxamide —— C18H26N4O
5-tert-butyl-N-[(1R)-2-(dimethylamino)-1-phenylethyl]-1H-pyrazole-3-carboxamide
—— 5-[(1R)-1-[4-(5-bromopyridin-2-yl)piperazin-1-yl]ethyl]-3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazole —— C20H21BrFN5O
5-[(1R)-1-[4-(5-bromopyridin-2-yl)piperazin-1-yl]ethyl]-3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazole
—— 5-tert-butyl-N-[(1S)-2-(dimethylamino)-1-phenylethyl]-1H-pyrazole-3-carboxamide —— C18H26N4O
5-tert-butyl-N-[(1S)-2-(dimethylamino)-1-phenylethyl]-1H-pyrazole-3-carboxamide
—— 5-[(1S)-1-(6,7-dihydro-4H-thieno[3,2-c]pyridin-5-yl)ethyl]-3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazole —— C18H18FN3OS
5-[(1S)-1-(6,7-dihydro-4H-thieno[3,2-c]pyridin-5-yl)ethyl]-3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazole
—— 5-[(1R)-1-(4-cyclopentylpiperazin-1-yl)ethyl]-3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazole —— C20H27FN4O
5-[(1R)-1-(4-cyclopentylpiperazin-1-yl)ethyl]-3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazole
—— 5-[(1S)-1-(6,7-dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)ethyl]-3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazole —— C22H24FN3O3
5-[(1S)-1-(6,7-dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)ethyl]-3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazole
—— 5-[(1S)-1-(4-cyclopentylpiperazin-1-yl)ethyl]-3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazole —— C20H27FN4O
5-[(1S)-1-(4-cyclopentylpiperazin-1-yl)ethyl]-3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazole
—— 5-[(1R)-1-(6,7-dihydro-4H-thieno[3,2-c]pyridin-5-yl)ethyl]-3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazole —— C18H18FN3OS
5-[(1R)-1-(6,7-dihydro-4H-thieno[3,2-c]pyridin-5-yl)ethyl]-3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazole
—— 5-[(1R)-1-(6,7-dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)ethyl]-3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazole —— C22H24FN3O3
5-[(1R)-1-(6,7-dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)ethyl]-3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazole
—— 5-[(1S)-1-[4-(5-bromopyridin-2-yl)piperazin-1-yl]ethyl]-3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazole —— C20H21BrFN5O
5-[(1S)-1-[4-(5-bromopyridin-2-yl)piperazin-1-yl]ethyl]-3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazole
—— 5-[(1S)-1-[4-(2-ethoxyphenyl)piperazin-1-yl]ethyl]-3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazole —— C23H27FN4O2
5-[(1S)-1-[4-(2-ethoxyphenyl)piperazin-1-yl]ethyl]-3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazole
—— [(5S)-9-(1H-imidazol-2-ylmethyl)-3-(thiophen-3-ylmethyl)-3,9-diazaspiro[5.5]undecan-5-yl]methanol —— C19H28N4OS
[(5S)-9-(1H-imidazol-2-ylmethyl)-3-(thiophen-3-ylmethyl)-3,9-diazaspiro[5.5]undecan-5-yl]methanol
—— 5-[(1R)-1-[4-(2-ethoxyphenyl)piperazin-1-yl]ethyl]-3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazole —— C23H27FN4O2
5-[(1R)-1-[4-(2-ethoxyphenyl)piperazin-1-yl]ethyl]-3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazole
—— [(5R)-3-(1-phenylpiperidin-4-yl)-9-propyl-3,9-diazaspiro[5.5]undecan-5-yl]methanol —— C24H39N3O
[(5R)-3-(1-phenylpiperidin-4-yl)-9-propyl-3,9-diazaspiro[5.5]undecan-5-yl]methanol
—— [(5S)-3-(1-phenylpiperidin-4-yl)-9-propyl-3,9-diazaspiro[5.5]undecan-5-yl]methanol —— C24H39N3O
[(5S)-3-(1-phenylpiperidin-4-yl)-9-propyl-3,9-diazaspiro[5.5]undecan-5-yl]methanol
—— [(5S)-9-[(3-fluorophenyl)methyl]-3-(3-methylsulfanylpropyl)-3,9-diazaspiro[5.5]undecan-5-yl]methanol —— C21H33FN2OS
[(5S)-9-[(3-fluorophenyl)methyl]-3-(3-methylsulfanylpropyl)-3,9-diazaspiro[5.5]undecan-5-yl]methanol
—— [(5R)-9-[(3-fluorophenyl)methyl]-3-(3-methylsulfanylpropyl)-3,9-diazaspiro[5.5]undecan-5-yl]methanol —— C21H33FN2OS
[(5R)-9-[(3-fluorophenyl)methyl]-3-(3-methylsulfanylpropyl)-3,9-diazaspiro[5.5]undecan-5-yl]methanol
—— (5Z)-3-anilino-5-[(4-methoxyphenyl)methylidene]-2-(4-methylphenyl)imidazol-4-one —— C24H21N3O2
(5Z)-3-anilino-5-[(4-methoxyphenyl)methylidene]-2-(4-methylphenyl)imidazol-4-one
—— 5-methyl-3-[(2S)-1-[(E)-3-phenylprop-2-enyl]pyrrolidin-2-yl]-1H-1,2,4-triazole —— C16H20N4
5-methyl-3-[(2S)-1-[(E)-3-phenylprop-2-enyl]pyrrolidin-2-yl]-1H-1,2,4-triazole
—— 5-[(2S)-1-[[1-(2-chlorophenyl)pyrazol-4-yl]methyl]pyrrolidin-2-yl]-3-methyl-1,2-oxazole —— C18H19ClN4O
5-[(2S)-1-[[1-(2-chlorophenyl)pyrazol-4-yl]methyl]pyrrolidin-2-yl]-3-methyl-1,2-oxazole
—— 5-[[(3R)-3-methoxypiperidin-1-yl]methyl]-2-oxo-1,3-dihydroimidazole-4-carboxylic acid —— C11H17N3O4
5-[[(3R)-3-methoxypiperidin-1-yl]methyl]-2-oxo-1,3-dihydroimidazole-4-carboxylic acid
—— 5-cyclopropyl-3-[4-[5-[(3R)-oxolan-3-yl]-1H-1,2,4-triazol-3-yl]phenyl]-1,2,4-oxadiazole —— C17H17N5O2
5-cyclopropyl-3-[4-[5-[(3R)-oxolan-3-yl]-1H-1,2,4-triazol-3-yl]phenyl]-1,2,4-oxadiazole
—— 5-[[(3S)-3-methoxypiperidin-1-yl]methyl]-2-oxo-1,3-dihydroimidazole-4-carboxylic acid —— C11H17N3O4
5-[[(3S)-3-methoxypiperidin-1-yl]methyl]-2-oxo-1,3-dihydroimidazole-4-carboxylic acid
—— 5-cyclopropyl-3-[4-[5-[(3S)-oxolan-3-yl]-1H-1,2,4-triazol-3-yl]phenyl]-1,2,4-oxadiazole —— C17H17N5O2
5-cyclopropyl-3-[4-[5-[(3S)-oxolan-3-yl]-1H-1,2,4-triazol-3-yl]phenyl]-1,2,4-oxadiazole
—— 5-[(1R)-1-[4-(benzenesulfonyl)piperazin-1-yl]ethyl]-3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazole —— C21H23FN4O3S
5-[(1R)-1-[4-(benzenesulfonyl)piperazin-1-yl]ethyl]-3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazole
—— 5-[(2R)-1-[[1-(2-chlorophenyl)pyrazol-4-yl]methyl]pyrrolidin-2-yl]-3-methyl-1,2-oxazole —— C18H19ClN4O
5-[(2R)-1-[[1-(2-chlorophenyl)pyrazol-4-yl]methyl]pyrrolidin-2-yl]-3-methyl-1,2-oxazole
—— 5-[(1S)-1-(3,4-dihydro-1H-isoquinolin-2-yl)ethyl]-3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazole —— C20H20FN3O
5-[(1S)-1-(3,4-dihydro-1H-isoquinolin-2-yl)ethyl]-3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazole
—— 5-[(1S)-1-[4-[(3,5-dimethyl-1,2-oxazol-4-yl)sulfonyl]piperazin-1-yl]ethyl]-3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazole —— C20H24FN5O4S
5-[(1S)-1-[4-[(3,5-dimethyl-1,2-oxazol-4-yl)sulfonyl]piperazin-1-yl]ethyl]-3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazole
—— 5-methyl-3-[(2R)-1-[(E)-3-phenylprop-2-enyl]pyrrolidin-2-yl]-1H-1,2,4-triazole —— C16H20N4
5-methyl-3-[(2R)-1-[(E)-3-phenylprop-2-enyl]pyrrolidin-2-yl]-1H-1,2,4-triazole
—— 5-[(1S)-1-[4-(benzenesulfonyl)piperazin-1-yl]ethyl]-3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazole —— C21H23FN4O3S
5-[(1S)-1-[4-(benzenesulfonyl)piperazin-1-yl]ethyl]-3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazole
—— 5-[[(2R)-5-ethoxy-2-methyl-2,3-dihydro-1-benzofuran-6-yl]methyl]-1-(2-nitrophenyl)pyrazolo[3,4-d]pyrimidin-4-one —— C23H21N5O5
5-[[(2R)-5-ethoxy-2-methyl-2,3-dihydro-1-benzofuran-6-yl]methyl]-1-(2-nitrophenyl)pyrazolo[3,4-d]pyrimidin-4-one
—— 5-[(1R)-1-(3,4-dihydro-1H-isoquinolin-2-yl)ethyl]-3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazole —— C20H20FN3O
5-[(1R)-1-(3,4-dihydro-1H-isoquinolin-2-yl)ethyl]-3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazole
—— 5-[(1R)-1-[4-[(3,5-dimethyl-1,2-oxazol-4-yl)sulfonyl]piperazin-1-yl]ethyl]-3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazole —— C20H24FN5O4S
5-[(1R)-1-[4-[(3,5-dimethyl-1,2-oxazol-4-yl)sulfonyl]piperazin-1-yl]ethyl]-3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazole
—— 5-[(Z)-3-(furan-2-yl)-2-methylprop-2-enyl]-N,N-dimethyl-1-(3,3,3-trifluoropropyl)-6,7-dihydro-4H-pyrazolo[4,3-c]pyridine-3-carboxamide —— C20H25F3N4O2
5-[(Z)-3-(furan-2-yl)-2-methylprop-2-enyl]-N,N-dimethyl-1-(3,3,3-trifluoropropyl)-6,7-dihydro-4H-pyrazolo[4,3-c]pyridine-3-carboxamide
—— 5-(methoxymethyl)-N-[[6-[(2R)-2-methylmorpholin-4-yl]pyridin-3-yl]methyl]furan-2-carboxamide —— C18H23N3O4
5-(methoxymethyl)-N-[[6-[(2R)-2-methylmorpholin-4-yl]pyridin-3-yl]methyl]furan-2-carboxamide
—— 5-(methoxymethyl)-N-[[6-[(2S)-2-methylmorpholin-4-yl]pyridin-3-yl]methyl]furan-2-carboxamide —— C18H23N3O4
5-(methoxymethyl)-N-[[6-[(2S)-2-methylmorpholin-4-yl]pyridin-3-yl]methyl]furan-2-carboxamide